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Extract from the Register of European Patents

EP About this file: EP3027611

EP3027611 - MACROCYCLIC UREA DERIVATIVES AS INHIBITORS OF TAFI A, THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  01.06.2018
Database last updated on 28.09.2024
FormerThe patent has been granted
Status updated on  23.06.2017
FormerGrant of patent is intended
Status updated on  23.02.2017
Most recent event   Tooltip17.07.2020Lapse of the patent in a contracting state
New state(s): AL		published on 19.08.2020  [2020/34]
Applicant(s)For all designated states
SANOFI
54, rue La Boétie
75008 Paris / FR
[2016/23]
Inventor(s)01 / EVERS, Andreas
Sanofi-Aventis Deutschland GmbH
65926 Frankfurt am Main / DE
02 / KALLUS, Christopher
Sanofi-Aventis Deutschland GmbH
65926 Frankfurt am Main / DE
03 / WAGNER, Michael
Sanofi-Aventis Deutschland GmbH
65926 Frankfurt am Main / DE
04 / WEHLAN, Hermut
Sanofi-Aventis Deutschland GmbH
65926 Frankfurt am Main / DE
 [2016/23]
Representative(s)Venne-Dunker, Sabine, et al
Sanofi-Aventis Deutschland GmbH
Global Intellectual Property Department
Industriepark Höchst
Gebäude K 703
65926 Frankfurt am Main / DE
[2016/23]
Application number, filing date14729285.805.06.2014
[2016/23]
WO2014EP61669
Priority number, dateEP2013030577910.06.2013         Original published format: EP 13305779
[2016/23]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2014198620
Date:18.12.2014
Language:EN
[2014/51]
Type: A1 Application with search report 
No.:EP3027611
Date:08.06.2016
Language:EN
The application published by WIPO in one of the EPO official languages on 18.12.2014 takes the place of the publication of the European patent application.
[2016/23]
Type: B1 Patent specification 
No.:EP3027611
Date:26.07.2017
Language:EN
[2017/30]
Search report(s)International search report - published on:EP18.12.2014
ClassificationIPC:C07D413/12, C07D273/01, A61K31/553, A61P7/00, A61K45/06, A61K31/395, A61K31/4427, C07D213/75
[2017/10]
CPC:
C07D273/01 (EP,US); A61K31/395 (EP,US); A61K31/4427 (EP,US);
A61K45/06 (US); A61P11/00 (EP); A61P17/02 (EP);
A61P19/02 (EP); A61P29/00 (EP); A61P3/00 (EP);
A61P3/10 (EP); A61P31/04 (EP); A61P35/00 (EP);
A61P35/04 (EP); A61P7/00 (EP); A61P7/02 (EP);
A61P9/00 (EP); A61P9/10 (EP); C07D213/75 (EP,US);
C07D413/12 (EP,US) (-)
Former IPC [2016/23]C07D413/12, C07D273/01, A61K31/553, A61P7/00
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   RS,   SE,   SI,   SK,   SM,   TR [2016/23]
Extension statesBANot yet paid
MENot yet paid
TitleGerman:MAKROCYCLISCHE HARNSTOFFDERIVATE ALS HEMMER VON TAFIA, DEREN HERSTELLUNG UND DEREN VERWENDUNG ALS PHARMAZEUTIKA[2017/10]
English:MACROCYCLIC UREA DERIVATIVES AS INHIBITORS OF TAFI A, THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS[2016/23]
French:DÉRIVÉS MACROCYCLIQUES D'URÉE EN TANT QU'INHIBITEURS DE TAFIA, LEUR PRÉPARATION ET LEUR UTILISATION COMME PRODUITS PHARMACEUTIQUES[2016/23]
Former [2016/23]MAKROCYCLISCHE HARNSTOFFDERIVATE ALS HEMMER VON TAFI A, DEREN HERSTELLUNG UND DEREN VERWENDUNG ALS PHARMAZEUTIKA
Entry into regional phase11.01.2016National basic fee paid 
11.01.2016Designation fee(s) paid 
11.01.2016Examination fee paid 
Examination procedure11.01.2016Examination requested  [2016/23]
26.07.2016Amendment by applicant (claims and/or description)
24.02.2017Communication of intention to grant the patent
09.05.2017Fee for grant paid
09.05.2017Fee for publishing/printing paid
09.05.2017Receipt of the translation of the claim(s)
Opposition(s)30.04.2018No opposition filed within time limit [2018/27]
Fees paidRenewal fee
10.06.2016Renewal fee patent year 03
16.06.2017Renewal fee patent year 04
Opt-out from the exclusive  Tooltip
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Patent Court		 See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipHU05.06.2014
AL26.07.2017
AT26.07.2017
CY26.07.2017
CZ26.07.2017
DK26.07.2017
EE26.07.2017
ES26.07.2017
FI26.07.2017
HR26.07.2017
IT26.07.2017
LT26.07.2017
LV26.07.2017
MC26.07.2017
MK26.07.2017
NL26.07.2017
PL26.07.2017
PT26.07.2017
RO26.07.2017
RS26.07.2017
SE26.07.2017
SI26.07.2017
SK26.07.2017
SM26.07.2017
TR26.07.2017
BG26.10.2017
NO26.10.2017
GR27.10.2017
IS26.11.2017
[2020/34]
Former [2020/31]HU05.06.2014
AT26.07.2017
CY26.07.2017
CZ26.07.2017
DK26.07.2017
EE26.07.2017
ES26.07.2017
FI26.07.2017
HR26.07.2017
IT26.07.2017
LT26.07.2017
LV26.07.2017
MC26.07.2017
MK26.07.2017
NL26.07.2017
PL26.07.2017
PT26.07.2017
RO26.07.2017
RS26.07.2017
SE26.07.2017
SI26.07.2017
SK26.07.2017
SM26.07.2017
TR26.07.2017
BG26.10.2017
NO26.10.2017
GR27.10.2017
IS26.11.2017
Former [2020/30]HU05.06.2014
AT26.07.2017
CZ26.07.2017
DK26.07.2017
EE26.07.2017
ES26.07.2017
FI26.07.2017
HR26.07.2017
IT26.07.2017
LT26.07.2017
LV26.07.2017
MC26.07.2017
NL26.07.2017
PL26.07.2017
PT26.07.2017
RO26.07.2017
RS26.07.2017
SE26.07.2017
SI26.07.2017
SK26.07.2017
SM26.07.2017
TR26.07.2017
BG26.10.2017
NO26.10.2017
GR27.10.2017
IS26.11.2017
Former [2020/28]AT26.07.2017
CZ26.07.2017
DK26.07.2017
EE26.07.2017
ES26.07.2017
FI26.07.2017
HR26.07.2017
IT26.07.2017
LT26.07.2017
LV26.07.2017
MC26.07.2017
NL26.07.2017
PL26.07.2017
PT26.07.2017
RO26.07.2017
RS26.07.2017
SE26.07.2017
SI26.07.2017
SK26.07.2017
SM26.07.2017
TR26.07.2017
BG26.10.2017
NO26.10.2017
GR27.10.2017
IS26.11.2017
Former [2020/15]AT26.07.2017
CZ26.07.2017
DK26.07.2017
EE26.07.2017
ES26.07.2017
FI26.07.2017
HR26.07.2017
IT26.07.2017
LT26.07.2017
LV26.07.2017
MC26.07.2017
NL26.07.2017
PL26.07.2017
RO26.07.2017
RS26.07.2017
SE26.07.2017
SI26.07.2017
SK26.07.2017
SM26.07.2017
TR26.07.2017
BG26.10.2017
NO26.10.2017
GR27.10.2017
IS26.11.2017
Former [2019/15]AT26.07.2017
CZ26.07.2017
DK26.07.2017
EE26.07.2017
ES26.07.2017
FI26.07.2017
HR26.07.2017
IT26.07.2017
LT26.07.2017
LV26.07.2017
MC26.07.2017
NL26.07.2017
PL26.07.2017
RO26.07.2017
RS26.07.2017
SE26.07.2017
SI26.07.2017
SK26.07.2017
SM26.07.2017
BG26.10.2017
NO26.10.2017
GR27.10.2017
IS26.11.2017
Former [2018/40]AT26.07.2017
CZ26.07.2017
DK26.07.2017
EE26.07.2017
ES26.07.2017
FI26.07.2017
HR26.07.2017
IT26.07.2017
LT26.07.2017
LV26.07.2017
NL26.07.2017
PL26.07.2017
RO26.07.2017
RS26.07.2017
SE26.07.2017
SI26.07.2017
SK26.07.2017
SM26.07.2017
BG26.10.2017
NO26.10.2017
GR27.10.2017
IS26.11.2017
Former [2018/24]AT26.07.2017
CZ26.07.2017
DK26.07.2017
EE26.07.2017
ES26.07.2017
FI26.07.2017
HR26.07.2017
IT26.07.2017
LT26.07.2017
LV26.07.2017
NL26.07.2017
PL26.07.2017
RO26.07.2017
RS26.07.2017
SE26.07.2017
SK26.07.2017
SM26.07.2017
BG26.10.2017
NO26.10.2017
GR27.10.2017
IS26.11.2017
Former [2018/21]AT26.07.2017
CZ26.07.2017
DK26.07.2017
ES26.07.2017
FI26.07.2017
HR26.07.2017
LT26.07.2017
LV26.07.2017
NL26.07.2017
PL26.07.2017
RS26.07.2017
SE26.07.2017
BG26.10.2017
NO26.10.2017
GR27.10.2017
IS26.11.2017
Former [2018/12]AT26.07.2017
ES26.07.2017
FI26.07.2017
HR26.07.2017
LT26.07.2017
LV26.07.2017
NL26.07.2017
PL26.07.2017
RS26.07.2017
SE26.07.2017
BG26.10.2017
NO26.10.2017
GR27.10.2017
IS26.11.2017
Former [2018/11]AT26.07.2017
ES26.07.2017
FI26.07.2017
HR26.07.2017
LT26.07.2017
NL26.07.2017
PL26.07.2017
RS26.07.2017
SE26.07.2017
BG26.10.2017
NO26.10.2017
GR27.10.2017
IS26.11.2017
Former [2018/10]AT26.07.2017
FI26.07.2017
HR26.07.2017
LT26.07.2017
NL26.07.2017
RS26.07.2017
SE26.07.2017
NO26.10.2017
Former [2018/09]FI26.07.2017
LT26.07.2017
NL26.07.2017
SE26.07.2017
NO26.10.2017
Former [2018/08]FI26.07.2017
LT26.07.2017
NL26.07.2017
NO26.10.2017
Former [2018/07]LT26.07.2017
NO26.10.2017
Cited inInternational search[IDA]WO2009146802  (SANOFI AVENTIS [FR], et al) [ID] 1,6-12 * claim 1; compounds 5-2 * [A] 2-5;
 [A]  - VIOLETA IOSUB ET AL, "Enantioselective Synthesis of [alpha]-Quaternary Amino Acid Derivatives by Sequential Enzymatic Desymmetrization and Curtius Rearrangement of [alpha],[alpha]-Disubstituted Malonate Diesters", THE JOURNAL OF ORGANIC CHEMISTRY, (20100305), vol. 75, no. 5, doi:10.1021/jo902584r, ISSN 0022-3263, pages 1612 - 1619, XP055083907 [A] 11,12 * Schemes 2-3;; compounds 5e,6e *

DOI:   http://dx.doi.org/10.1021/jo902584r
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.