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EP3953351
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EP Citations: EP3953351
| Cited in | International search | Type: | Patent literature | Publication No.: | WO2009054941
[XI] (MERCK & CO INC [US], et al) [X] 1-5,7-20,22 * step 1, intermediate: 1H-Pyrrolo[2,3-b]pyridine, 5-(1-methyl-1H-pyrazol-4-yl)-1- (phenylsulfonyl)-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-;; example 1 * [I] 6,21; | Type: | Patent literature | Publication No.: | WO2012129338
[XI] (AMGEN INC [US], et al) [X] 1-5,7-20,22 * examples 54b,54 * [I] 6,21; | Type: | Patent literature | Publication No.: | WO2013075785
[XI] (MERCK PATENT GMBH [DE]) [X] 1-5,7-20,22 * Intermediate; page 64 * * claim - * [I] 6,21; | Type: | Patent literature | Publication No.: | WO2014053568
[XI] (SANOFI SA [FR]) [X] 1-5,7-20,22 * stage 5, intermediate; page 119; example 14 * [I] 6,21; | Type: | Patent literature | Publication No.: | WO2014145051
[I] (ZHANG JIAZHONG [US], et al) [I] 1-37 * table - * * page 97 - page 261; example - * * claim - *; | Type: | Patent literature | Publication No.: | WO2014154760
[I] (BOEHRINGER INGELHEIM INT [DE]) [I] 1-37 * example - ** claim - *; | Type: | Patent literature | Publication No.: | WO2017053243
[I] (PLEXXIKON INC [US]) [I] 1-37 * page 49 - page 65; example - * * table - * * claim - *; | Type: | Patent literature | Publication No.: | WO2018175311
[I] (PLEXXIKON INC [US]) [I] 1-37 * the whole document * * example - * * claim - *; | Type: | Patent literature | Publication No.: | WO2019075243
[IP] (PLEXXIKON INC [US]) [IP] 1-37 * the whole document * * example - * * claim - *; | Type: | Non-patent literature | Publication information: | [XI] - ANU J. AIRAKSINEN ET AL, "Radiosynthesis and evaluation of new [alpha]1-adrenoceptor antagonists as PET radioligands for brain imaging", NUCLEAR MEDICINE AND BIOLOGY., US, (20130801), vol. 40, no. 6, doi:10.1016/j.nucmedbio.2013.05.007, ISSN 0969-8051, pages 747 - 754, XP055712575 [X] 1-5,7-20,22-24 * figure 1 * * Scheme 1 * [I] 6,21 | DOI: | http://dx.doi.org/10.1016/j.nucmedbio.2013.05.007 | Type: | Non-patent literature | Publication information: | [XI] - JØRGENSEN MORTEN ET AL, "Discovery of novel [alpha]1-adrenoceptor ligands based on the antipsychotic sertindole suitable for labeling as PET ligands", BIOORGANIC & MEDICINAL CHEMISTRY : A TETRAHEDRON PUBLICATION FOR THE RAPID DISSEMINATION OF FULL ORIGINAL RESEARCH PAPERS AND CRITICAL REVIEWS ON BIOMOLECULAR CHEMISTRY, MEDICINAL CHEMISTRY AND RELATED DISCIPLINES, (20121115), vol. 21, no. 1, doi:10.1016/J.BMC.2012.10.049, ISSN 0968-0896, pages 196 - 204, XP028961411 [X] 1-5,7-20,22-24 * table 1 * * Schemes 3,4 * [I] 6,21 | DOI: | http://dx.doi.org/10.1016/j.bmc.2012.10.049 | Cited in | by applicant | Type: | Patent literature | Publication No.: | US4150949
| Type: | Patent literature | Publication No.: | EP0154734
| Type: | Patent literature | Publication No.: | US4568649
| Type: | Patent literature | Publication No.: | US4626513
| Type: | Patent literature | Publication No.: | US2004077595
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Res., (19950000), vol. 34, pages 220 - 230 | Type: | Non-patent literature | Publication information: | - JERRY MARCH, Advanced Organic Chemistry: Reactions, Mechanisms and Structures, John Wiley & Sons, (19920000), pages 69 - 74 | Type: | Non-patent literature | Publication information: | - VELY F. et al., "BIAcore® analysis to test phosphopeptide-SH2 domain interactions", Methods in Molecular Biology, (20000000), vol. 121, pages 313 - 21 | Type: | Non-patent literature | Publication information: | - LIPAROTO et al., "Biosensor analysis of the interleukin-2 receptor complex", Journal of Molecular Recognition, (19990000), vol. 12, doi:10.1002/(SICI)1099-1352(199909/10)12:5<316::AID-JMR468>3.3.CO;2-T, pages 316 - 21, XP001070799 | DOI: | http://dx.doi.org/10.1002/(SICI)1099-1352(199909/10)12:5<316::AID-JMR468>3.3.CO;2-T | Type: | Non-patent literature | Publication information: | - LIPSCHULTZ et al., "Experimental design for analysis of complex kinetics using surface plasmon resonance", Methods, (20000000), vol. 20, no. 3, doi:10.1006/meth.1999.0924, pages 310 - 8, XP004466887 | DOI: | http://dx.doi.org/10.1006/meth.1999.0924 | Type: | Non-patent literature | Publication information: | - MALMQVIST., "BIACORE: an affinity biosensor system for characterization of biomolecular interactions", Biochemical Society Transactions, (19990000), vol. 27, pages 335 - 40, XP000956194 | Type: | Non-patent literature | Publication information: | - ALFTHAN, "Surface plasmon resonance biosensors as a tool in antibody engineering", Biosensors & Bioelectronics, (19980000), vol. 13, doi:10.1016/S0956-5663(98)00020-7, pages 653 - 63, XP026050117 | DOI: | http://dx.doi.org/10.1016/S0956-5663(98)00020-7 | Type: | Non-patent literature | Publication information: | - FIVASH et al., "BIAcore for macromolecular interaction", Current Opinion in Biotechnology, (19980000), vol. 9, pages 97 - 101 | Type: | Non-patent literature | Publication information: | - PRICE et al., "Summary report on the ISOBM TD-4 Workshop: analysis of 56 monoclonal antibodies against the MUC 1 mucin", Tumour Biology, (19980000), vol. 19, no. 1, pages 1 - 20 | Type: | Non-patent literature | Publication information: | - MALMQVIST et al., "Biomolecular interaction analysis: affinity biosensor technologies for functional analysis of proteins", Current Opinion in Chemical Biology, (19970000), vol. 1, doi:10.1016/S1367-5931(97)80077-4, pages 378 - 83, XP002978720 | DOI: | http://dx.doi.org/10.1016/S1367-5931(97)80077-4 | Type: | Non-patent literature | Publication information: | - O'SHANNESSY et al., "Interpretation of deviations from pseudo-first-order kinetic behavior in the characterization of ligand binding by biosensor technology", Analytical Biochemistry, (19960000), vol. 236, pages 275 - 83 | Type: | Non-patent literature | Publication information: | - MALMBORG et al., "BIAcore as a tool in antibody engineering", Journal of Immunological Methods, (19950000), vol. 183, doi:10.1016/0022-1759(95)00018-6, pages 7 - 13, XP004021020 | DOI: | http://dx.doi.org/10.1016/0022-1759(95)00018-6 | Type: | Non-patent literature | Publication information: | - VAN REGENMORTEL, "Use of biosensors to characterize recombinant proteins", Developments in Biological Standardization, (19940000), vol. 83, pages 143 - 51 | Type: | Non-patent literature | Publication information: | - O'SHANNESSY, "Determination of kinetic rate and equilibrium binding constants for macromolecular interactions: a critique of the surface plasmon resonance literature", Current Opinions in Biotechnology, (19940000), vol. 5, doi:10.1016/S0958-1669(05)80072-2, pages 65 - 71, XP022839327 | DOI: | http://dx.doi.org/10.1016/S0958-1669(05)80072-2 | Type: | Non-patent literature | Publication information: | - GORDON, A. 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