Deutsch English Français

Contact

EP0978512

European procedure

Quick help

Maintenance news

Scheduled maintenance

Regular maintenance outages:
between 05.00 and 05.15 hrs CET (Monday to Sunday).

Other outages
Availability

2022.02.11

More...

News flashes

News Flashes

New version of the European Patent Register – SPC proceedings information in the Unitary Patent Register.

2024-07-24

More...

Extract from the Register of European Patents

EP About this file: EP0978512

EP0978512 - Non-imidazole aryloxy (or arylthio) alkylamines as histamine H3-receptor antagonists and their therapeutic applications [Right-click to bookmark this link]
Status	The application has been withdrawn Status updated on 12.05.2000 Database last updated on 05.12.2024
Most recent event Tooltip	12.05.2000	Withdrawal of application	published on 28.06.2000 [2000/26]
Applicant(s)	For all designated states SOCIETE CIVILE BIOPROJET 30, rue des Francs Bourgeois F-75003 Paris / FR
	[2000/06]
Inventor(s)	01 / Schwartz, Jean-Charles 9, villa Seurat 75014 Paris / FR
	02 / Arrang, Jean-Michel 3, avenue des Acacias 91419 Dourdan / FR
	03 / Garbarg, Monique 26 Boulevard Gouvion Saint Cyr 75017 Paris / FR
	04 / Lecomte, Jeanne-Marie 30 rue des Francs-Bourgeois 75003 Paris / FR
	05 / Ligneau, Xavier 10 rue des Tanneries 75013 Paris / FR
	06 / Schunack, Walter G. Spanische Allee 95 14129 Berlin / DE
	07 / Stark, Holger Lothar-Bucher-Strasse 19 12157 Berlin / DE
	08 / Ganellin, Charon Robin Kinwood Briary Wood End Welwyn, Hert AL6 OTD / GB
	09 / Leurquin, Fabien 49 Chilton Street London E2 6DZ / GB
	10 / Sigurd, Elz Albulaweg 7 a 12107 Berlin / DE
	[2000/06]
Representative(s)	Le Guen, Gérard, et al CABINET LAVOIX 2, place d'Estienne d'Orves 75441 Paris Cédex 09 / FR
	[2000/06]
Application number, filing date	98401944.8	29.07.1998
	[2000/06]
Filing language	EN
Procedural language	EN
Publication	Type:	A1 Application with search report
	No.:	EP0978512
	Date:	09.02.2000
	Language:	EN
	[2000/06]
Search report(s)	(Supplementary) European search report - dispatched on:	EP	29.12.1998
Classification	IPC:	C07D295/088, C07C211/08, C07D211/04, C07D295/185, C07D211/62, C07D211/70, C07D207/20, A61K31/13, A61K31/40, A61K31/445, A61K31/495	[2000/06]
	CPC:	C07D213/74 (EP); C07C215/34 (EP); C07C217/16 (EP); C07C217/20 (EP); C07C217/22 (EP); C07C251/48 (EP); (+) C07C255/54 (EP); C07D207/20 (EP); C07D211/58 (EP); C07D211/60 (EP); C07D211/62 (EP); C07D211/70 (EP); C07D215/38 (EP); C07D215/46 (EP); C07D239/42 (EP); C07D271/06 (EP); C07D277/82 (EP); C07D295/03 (EP); C07D295/088 (EP); C07D295/096 (EP); C07D295/13 (EP); C07D295/185 (EP); C07B2200/07 (EP); C07C2602/10 (EP) (-)
Designated contracting states	AT, BE, CH, CY, DE, DK, ES, FI, FR, GB, GR, IE, IT, LI, LU, MC, NL, PT, SE [2000/06]
Extension states	AL	Not yet paid
	LT	Not yet paid
	LV	Not yet paid
	MK	Not yet paid
	RO	Not yet paid
	SI	Not yet paid
Title	German:	Aryloxy- (oder Arylthio)alkylamine ohne Imidazolring als Histamin-H3-Antagonisten und deren therapeutische Anwendung	[2000/06]
	English:	Non-imidazole aryloxy (or arylthio) alkylamines as histamine H3-receptor antagonists and their therapeutic applications	[2000/06]
	French:	Non-imidazole aryloxy- (ou arylthio)alkylamines comme antagonistes du recepteur H3 et leur application thérapeutique	[2000/06]
Examination procedure	28.04.2000	Application withdrawn by applicant [2000/26]
Opt-out from the exclusive Tooltip competence of the Unified Patent Court	See the Register of the Unified Patent Court for opt-out data
	Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Documents cited:	Search	[X]GB1512880 (MITSUBISHI CHEM IND) [X] 1-24 * example -; table I *;
		[X]DE1269134 (VEB DEUTSCHES HYDRIERWERK RODLEBEN) [X] 1-24 * examples 1-5 *;
		[X]US3947434 (SPENCER CLAUDE F ET AL) [X] 1-24 * examples LXXIXA,B *;
		[X]US4751302 (IBUKI TADAYUKI ET AL) [X] 1-24 * tables 5-2,5-3 *;
		[X]GB924961 (THE WELLCOME FOUNDATION LIMITED) [X] 1-24 * table II *;
		[X]US3312696 (LUIGI TURBANTI) [X] 1-24 * examples 1-20; claim 1 *;
		[X]DE2624261 (BOTTU FA) [X] 1-24 * page 4; example 10 *;
		[X]US2870151 (WRIGHT H.B. AND MOORE M.B.) [X] 1-24 * examples I-XII *;
		[X]DE965813 (ABBOTT LABORATORIES) [X] 1-24 * examples 1-5,7 *;
		[X] - LITTMANN E. R. AND MARVEL C. S., "Cyclic Quaternary Ammonium Salts from Halogenated Aliphatic Tertiary Amines", J.AMER.CHEM.SOC., (1930), vol. 52, pages 287 - 294, XP002084866 [X] 1-24 * page 289 - page 290 * DOI: http://dx.doi.org/10.1021/ja01364a041
		[X] - KIKUMOTO R. ET AL., "Synthesis and Antidepressant Activity of Substituted (gamma-Aminoalkoxy)benzene Derivatives", J.MED.CHEM., (1981), vol. 24, no. 2, pages 145 - 148, XP000565653 [X] 1-26 * table 1 * DOI: http://dx.doi.org/10.1021/jm00134a004
		[X] - SHADBOLT R. S. ET AL., "Some Aryloxyalkylamines, N-Arylethylenediamines and Related Compounds as Anorectic Agents", J.MED.CHEM., (1971), vol. 14, no. 9, pages 836 - 842, XP002084867 [X] 1-24 * table 1 * DOI: http://dx.doi.org/10.1021/jm00291a015
		[X] - WALSH D. A. ET AL., "Synthesis and Antiallergy Activity of 4-(Diarylhydroxymethyl)-1-[3-(aryloxy)propyl]piperidines and Structurally Related Compounds", J.MED.CHEM., (1989), vol. 32, no. 1, pages 105 - 118, XP002084868 [X] 1-24 * tables I-III * DOI: http://dx.doi.org/10.1021/jm00121a022
		[X] - SOHDA T ET AL, "STUDIES ON ANTIDIABETIC AGENTS. SYNTHESIS OF 5- 4-(1-METHYLCYCLOHEXYLMETHOXY)-BENZYL)THIAZOLIDINE-2,4-DIONE (ADD-3878) AND ITS DERIVATIVES", CHEMICAL AND PHARMACEUTICAL BULLETIN, (1982), vol. 30, no. 10, pages 3580 - 3600, XP002046259 [X] 1-24 * table VIII *
		[X] - CHABRIER P. ET AL., "Nouveaux carbamates doués d'activité anesthésique locale", BULL.SOC.CHIM.FR., (1955), pages 1353 - 1357, XP002084869 [X] 1-24 * table IV *
		[X] - MARQUET J. ET AL., "Topologically Controlled Coulombic Interactions, a New Tool in the Developing of Novel Reactivity. Photochemical and Electrochemical Cleavage of Phenyl Alkyl Ethers", J.ORG.CHEM., (1995), vol. 60, no. 12, pages 3814 - 3825, XP002084870 [X] 1-24 * table 1 * DOI: http://dx.doi.org/10.1021/jo00117a037
		[X] - CASANOVAS A.-M. ET AL., "Etude des relations structure-activté d'une série d'anesthésiques locaux", EUR.J.MED.CHEM.-CHIM.THER., (1982), vol. 17, no. 4, pages 333 - 337, XP002084871 [X] 1-24 * page 334 *
		[X] - KIKUMOTO R ET AL, "SYNTHESES AND PLATELET AGGREGATION INHIBITORY AND ANTITHROMBOTIC PROPERTIES OF 2- (OMEGA-AMINOALKOXY)PHENYLETHYLBENZENES", JOURNAL OF MEDICINAL CHEMISTRY, (199006), vol. 33, no. 6, pages 1818 - 1823, XP000673455 [X] 1-24 * tables I-III * DOI: http://dx.doi.org/10.1021/jm00168a043
		[X] - CHENEY L.C. ET AL., "Alkylaminoalkyl Ethers of the Benzylphenols", J.AMER.CHEM.SOC., (1949), vol. 71, pages 60 - 64, XP002086293 [X] 1-26 * page 60; table I * DOI: http://dx.doi.org/10.1021/ja01169a017
		[A] - STARK H. ET AL., "Developments of Histamine H3-receptor Antagonists", DRUGS OF THE FUTURE, (1996), vol. 21, no. 5, pages 507 - 520, XP002084872 [A] 1-34 * page 507 *

The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.

Legal notice
Terms of use
24.2.25; 35p