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Extract from the Register of European Patents

EP About this file: EP1145718

EP1145718 - DICARBA-closo-DODECABORANE DERIVATIVES [Right-click to bookmark this link]
Status	The application is deemed to be withdrawn Status updated on 19.01.2004 Database last updated on 30.10.2024
Most recent event Tooltip	19.01.2004	Application deemed to be withdrawn	published on 03.03.2004 [2004/10]
Applicant(s)	For all designated states Institute of Medicinal Molecular Design, Inc. 4th floor Kadokawa-hongo Bldg. 24-5, Hongo 5-chome Bunkyo-ku Tokyo 113-0033 / JP
	[N/P]
Former [2001/42]	For all designated states Institute of Medicinal Molecular Design, Inc. 4th floor Kadokawa-hongo Bldg., 24-5, Hongo 5-chome, Bunkyo-ku Tokyo 113-0033 / JP
Inventor(s)	01 / ENDO, Yasuyuki, Cosmo Chigasaki Belle Seine 2-47-303,Hibarigaoka, Chigaraki-shi Kanagawa 253-0027 / JP
	[2001/42]
Representative(s)	polypatent Patentanwälte An den Gärten 7 51491 Overath / DE
	[N/P]
Former [2001/42]	Sternagel, Fleischer, Godemeyer & Partner Patentanwälte An den Gärten 7 51491 Overath / DE
Application number, filing date	00900863.2	21.01.2000
	[2001/42]
	WO2000JP00285
Priority number, date	JP19990014261	22.01.1999 Original published format: JP 1426199
	JP19990280257	30.09.1999 Original published format: JP 28025799
	[2001/42]
Filing language	JA
Procedural language	EN
Publication	Type:	A1 Application with search report
	No.:	WO0043016
	Date:	27.07.2000
	Language:	EN
	[2000/30]
	Type:	A1 Application with search report
	No.:	EP1145718
	Date:	17.10.2001
	Language:	EN
	The application published by WIPO in one of the EPO official languages on 27.07.2000 takes the place of the publication of the European patent application.
	[2001/42]
Search report(s)	International search report - published on:	JP	27.07.2000
Classification	IPC:	A61K31/69, A61P3/02, A61P3/10, A61P5/30, A61P9/10, A61P29/00, A61P35/00, A61P37/06, C07F5/02	[2001/42]
	CPC:	C07F5/027 (EP,US); A61P15/00 (EP); A61P29/00 (EP); A61P3/02 (EP); A61P3/10 (EP); A61P35/00 (EP); (+) A61P37/06 (EP); A61P5/30 (EP); A61P9/10 (EP) (-)
Designated contracting states	AT, BE, CH, CY, DE, DK, ES, FI, FR, GB, GR, IE, IT, LI, LU, MC, NL, PT, SE [2001/42]
Extension states	AL	Not yet paid
	LT	Not yet paid
	LV	Not yet paid
	MK	Not yet paid
	RO	18.07.2001
	SI	18.07.2001
Title	German:	DICARBA--I(CLOSO)-DODECABORANDERIVATE	[2001/42]
	English:	DICARBA-closo-DODECABORANE DERIVATIVES	[2001/42]
	French:	DERIVES DE DICARBA-closo-DODECABORANE	[2001/42]
Entry into regional phase	18.07.2001	Translation filed
	18.07.2001	National basic fee paid
	18.07.2001	Search fee paid
	18.07.2001	Designation fee(s) paid
	18.07.2001	Examination fee paid
Examination procedure	21.01.2000	Request for preliminary examination filed International Preliminary Examining Authority: JP
	18.07.2001	Examination requested [2001/42]
	01.08.2003	Application deemed to be withdrawn, date of legal effect [2004/10]
	19.09.2003	Despatch of communication that the application is deemed to be withdrawn, reason: renewal fee not paid in time [2004/10]
Fees paid	Renewal fee
	14.01.2002	Renewal fee patent year 03
	Penalty fee
	Additional fee for renewal fee
	31.01.2003	04 M06 Not yet paid
Opt-out from the exclusive Tooltip competence of the Unified Patent Court	See the Register of the Unified Patent Court for opt-out data
	Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Cited in	International search	[A]JPH05163296 (SUNTORY LTD);
		[A]JPS55154982 (SHIONOGI SEIYAKU KK);
		[A]EP0205326 (IMMUNOMEDICS INC [US]);
		[XP] - ENDO Y. ET. AL., "Structure-activity study of estrogenic agonists bearing dicarba-closo dodecaborane, Effect of geometry and separation distance of hydroxyl groups at the ends of molecules", BIOORG. MED. CHEM. LETT., (1999), vol. 9, no. 23, pages 3313 - 3318, XP002928432 DOI: http://dx.doi.org/10.1016/S0960-894X(99)00596-X
		[XP] - ENDO Y- ET- AL., "Estrogenic antagonists bearing dicarba-closo-dodecaborane as a hydrophobic pharmacophore", BIOORG. MED. CHEM. LETT., (1999), vol. 9, no. 24, pages 3387 - 3392, XP002928433 DOI: http://dx.doi.org/10.1016/S0960-894X(99)00579-X
		[XP] - ENDO Y. ET. AL., "Potent estrogenic agonists bearing dicarba-closo-dodecaborane as a hydrophobic pharmacophore", (1999), vol. 42, no. 9, pages 1501 - 1504, XP002928434 DOI: http://dx.doi.org/10.1021/jm9900725
		[XP] - ENDO Y. ET. AL., "Dicarba-closo-dodecaboranes as pharmacophore, Novel potent retinoidal agonists", (1999), vol. 47, no. 4, pages 585 - 587, XP002928435
		[XP] - IIJIMA T. ET. AL., "Dicarba-closo-dodecaboranes as a pharma-cophore, Retinoidal antagonists and potential agonists", CHEM. PHARM. BULL, (1999), vol. 47, no. 3, pages 398 - 404, XP002928436
		[X] - FOX. M. A. ET. AL., "Transmission of electronic effects by icosahedral carboranes; skeletal carbon-13chemical shifts and ultraviolet-visible spectra of substituted aryl-p-carboranes (1,12-dicarba-closo-dodecaboranes", J. CHEM. SOC., DALTON TRANS., (1998), no. 3, pages 401 - 411, XP002928437 DOI: http://dx.doi.org/10.1039/a707154j
		[X] - COLQUHOUN H. M. ET. AL., "Polyetherketones based on para-carborane: synthesis, sulfonation, and membrane-forming characteristics", POLYMER, (1997), vol. 38, no. 17, pages 4539 - 4546, XP002928438 DOI: http://dx.doi.org/10.1016/S0032-3861(96)01016-6
		[X] - PRASHAR J. K. ET. AL., "Synthesis of carboranyl phenylalanine for potential use in neutron capture therapy of melanoma", J. CHEM. SOC. PERKIN. TRANS., (1993), no. 9, pages 1051 - 1053, XP002928439
		[X] - BROWN D. A. ET. AL., "Polymers and ceramics based on icosahedral carboranes, model studies of the formation and hydrolytic stability of aryl ether, ketone, amide and borane linkages between carborane units", J. MATER. CHEM., (1992), vol. 2, no. 8, pages 793 - 804, XP002928440 DOI: http://dx.doi.org/10.1039/jm9920200793
		[X] - NEMOTO H. ET. AL., "The first alkylation of o-carboranes under essentially neutral conditions, Application to the synthesis of 10B carriers", J. ORG. CHEM., (1990), vol. 55, no. 25, pages 6065 - 6066, XP002928441 DOI: http://dx.doi.org/10.1021/jo00312a002
		[X] - KALININ ET. AL., CHEMICAL ABSTRACTS, vol. 89, Database accession no. 196733W, XP002928448
		[X] - KALININ ET. AL., CHEMICAL ABSTRACTS, vol. 89, Database accession no. 6351Z, XP002928449
		[ ] - J. ORGANOMENT, CHEM., (1978), vol. 149, no. 1, pages 9 - 21
		[X] - MATOCHKIN V. S. ET. AL., "Molecular mobility in polyarylates having difenylcarborane fragments in the chain", FASERFORSCH, TEXTILTECH., (1975), vol. 26, no. 6, pages 261 - 265, XP002928446
		[X] - VINOGRADORA ET. AL., CHEMICAL ABSTRACTS, vol. 82, Database accession no. 17164X, XP002928450
		[X] - VALETSKII P. M. ET. AL., "Polyamides of 1,7-bis (p-carboxy-phenyl) carborane", VYSOKOMOL, SOEDIN, SER. A., (1973), vol. 15, no. 6, pages 1227 - 1233, XP002928447
		[X] - DANILOV ET. AL., CHEMICAL ABSTRACTS, vol. 76, Database accession no. 46645M, XP002928451
		[X] - ZAKHARKIN L. I. ET. AL., "ionization constants of 1-(p- and m-carboxyphenyl) -2-substituted o-carboranes", CHEMICAL ABSTRACTS, vol. 75, Database accession no. 98063U, XP002928452
		[ ] - ZH. OBSHCH. KHIM., (1971), vol. 41, no. 6, pages 1300 - 1303
		[X] - STANKO ET. AL., CHEMICAL ABSTRACTS, vol. 71, Database accession no. 39047M, XP002928453
		[X] - ZAKHARKIN ET. AL., CHEMICAL ABSTRACTS, vol. 68, Database accession no. 39684E, XP002928454
		[X] - ZAKHARKIN ET. AL., CHEMICAL ABSTRACTS, vol. 66, Database accession no. 95101R, XP002928455
		[X] - ZAKHARKIN ET. AL., CHEMICAL ABSTRACTS, vol. 65, Database accession no. 16989F-G, XP002928456
		[ ] - IZV. AKAD. NAUK. SSSR. SEV. KHIM, (196607), page 1286
		[X] - ZAKARKIN ET. AL., CHEMICAL ABSTRACTS, vol. 65, Database accession no. 10604G-H, XP002928457
		[X] - ZAKHARKIN ET. AL., CHEMICAL ABSTRACTS, vol. 64, Database accession no. 11235D-H, XP002928458
		[X] - FREDERICK HAWTHORNE ET. AL., CHEMICAL ABSTRACTS, vol. 63, Database accession no. 17865F-H, XP002928459
		[ ] - J. AM. CHEM SOC., (1965), vol. 87, no. 21, pages 4746 - 4750 (ENG)

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