blank Quick help
blank Maintenance news

Scheduled maintenance

Regular maintenance outages:
between 05.00 and 05.15 hrs CET (Monday to Sunday).

Other outages
Availability

2022.02.11

More...
blank News flashes

News Flashes

New version of the European Patent Register – SPC proceedings information in the Unitary Patent Register.

2024-07-24

More...
blank Related links

Extract from the Register of European Patents

EP About this file: EP1216980

EP1216980 - CARBOXYLIC ACID DERIVATIVES AND DRUGS CONTAINING THE SAME [Right-click to bookmark this link]
StatusThe application has been withdrawn
Status updated on  21.01.2011
Database last updated on 25.09.2024
Most recent event   Tooltip21.01.2011Withdrawal of applicationpublished on 23.02.2011  [2011/08]
Applicant(s)For all designated states
Eisai R&D Management Co., Ltd.
6-10, Koishikawa 4-chome
Bunkyo-ku
Tokyo 112-8088 / JP
[N/P]
Former [2007/08]For all designated states
Eisai R&D Management Co., Ltd.
6-10, Koishikawa, 4-chome Bunkyo-ku
Tokyo 112-8088 / JP
Former [2002/26]For all designated states
Eisai Co., Ltd.
6-10, Koishikawa 4-chome, Bunkyo-ku
Tokyo 112-8088 / JP
Inventor(s)01 / SHINODA, Masanobu
4-1, Wakaba, Kukizakimachi
Inashiki-gun, Ibaraki 300-1249 / JP
02 / EMORI, Eita
1-8-19-202, Namiki
Tsuchiura-shi, Ibaraki 300-0061 / JP
03 / MATSUURA, Fumiyoshi
3-25-2-205, Matsushiro
Tsukuba-shi, Ibaraki 305-0035 / JP
04 / KANEKO, Toshihiko
1082-70, Taguumachi
Ushiku-shi, Ibaraki 300-1236 / JP
05 / OHI, Norihito
1-12-7, Nanpeidai, Amimachi
Inashiki-gun, Ibaraki 300-0312 / JP
06 / KASAI, Shunji
7-9-11, Matsumaedai, Moriyamachi
Kitasouma-gun, Ibaraki 302-0102 / JP
07 / YOSHITOMI, Hideki
Sorio Hanabatake 202, 2-11-2, Hanabatake
Tsukuba-shi, Ibaraki 300-3261 / JP
08 / YAMAZAKI, Kazuto
3-304, 3-19-1, Azuma
Tsukuba-shi, Ibaraki 305-0031 / JP
09 / MIYASHITA, Sadakazu
1-35-19-2-402, Kannondai
Tsukuba-shi, Ibaraki 305-0856 / JP
10 / HIBARA, Taro
Tsukubanedainiryo 306, 9-7, Inarimae
Tsukuba-shi, Ibaraki 305-0061 / JP
11 / SEIKI, Takashi
Tsukubanedainiryo 406, 9-7, Inarimae
Tsukuba-shi, Ibaraki 305-0061 / JP
12 / CLARK, Richard
2-20-2, Ottominami
Tsuchiura-shi, Ibaraki 300-0845 / JP
13 / HARADA, Hitoshi
2-24-27, Kamikashiwada
Ushiku-shi, Ibaraki 300-1232 / JP
 [2002/35]
Former [2002/26]01 / SHINODA, Masanobu
4-1, Wakaba, Kukizakimachi
Inashiki-gun, Ibaraki 300-1249 / JP
02 / EMORI, Eita
Tsukubanedainiryo 101, 9-7, Inarimae
Tsukuba-shi, Ibaraki 305-0061 / JP
03 / MATSUURA, Fumiyoshi
Green Palace Nakayama 205, 34-6, Higashiarai
Tsukuba-shi, Ibaraki 305-0033 / JP
04 / KANEKO, Toshihiko
1082-70, Taguumachi
Ushiku-shi, Ibaraki 300-1236 / JP
05 / OHI, Norihito
1-12-7, Nanpeidai, Amimachi
Inashiki-gun, Ibaraki 300-0312 / JP
06 / KASAI, Shunji
7-9-11, Matsumaedai, Moriyamachi
Kitasouma-gun, Ibaraki 302-0102 / JP
07 / YOSHITOMI, Hideki
Sorio Hanabatake 202, 2-11-2, Hanabatake
Tsukuba-shi, Ibaraki 300-3261 / JP
08 / YAMAZAKI, Kazuto
3-304, 3-19-1, Azuma
Tsukuba-shi, Ibaraki 305-0031 / JP
09 / MIYASHITA, Sadakazu
1-35-19-2-402, Kannondai
Tsukuba-shi, Ibaraki 305-0856 / JP
10 / HIBARA, Taro
Tsukubanedainiryo 306, 9-7, Inarimae
Tsukuba-shi, Ibaraki 305-0061 / JP
11 / SEIKI, Takashi
Tsukubanedainiryo 406, 9-7, Inarimae
Tsukuba-shi, Ibaraki 305-0061 / JP
12 / CLARK, Richard
2-20-2, Ottominami
Tsuchiura-shi, Ibaraki 300-0845 / JP
13 / HARADA, Hitoshi
2-24-27, Kamikashiwada
Ushiku-shi, Ibaraki 300-1232 / JP
Representative(s)Hoffmann Eitle
Patent- und Rechtsanwälte PartmbB
Arabellastraße 30
81925 München / DE
[N/P]
Former [2008/31]HOFFMANN EITLE
Patent- und Rechtsanwälte Arabellastrasse 4
81925 München / DE
Former [2002/26]HOFFMANN EITLE
Patent- und Rechtsanwälte Arabellastrasse 4
81925 München / DE
Application number, filing date00962993.229.09.2000
[2002/26]
WO2000JP06788
Priority number, dateJP1999028207901.10.1999         Original published format: JP 28207999
JP1999036944227.12.1999         Original published format: JP 36944299
JP2000003879516.02.2000         Original published format: JP 2000038795
JP2000010426006.04.2000         Original published format: JP 2000104260
[2002/26]
Filing languageJA
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO0125181
Date:12.04.2001
Language:EN
[2001/15]
Type: A1 Application with search report 
No.:EP1216980
Date:26.06.2002
Language:EN
The application published by WIPO in one of the EPO official languages on 12.04.2001 takes the place of the publication of the European patent application.
[2002/26]
Search report(s)International search report - published on:JP12.04.2001
(Supplementary) European search report - dispatched on:EP10.11.2010
ClassificationIPC:C07C59/66
[2002/26]
CPC:
C07D213/30 (EP,US); C07D417/12 (EP,KR,US); A61P3/10 (EP);
A61P43/00 (EP); C07C233/51 (EP,US); C07C233/55 (EP,US);
C07C233/87 (EP,US); C07C235/34 (EP,US); C07C235/38 (EP,US);
C07C235/52 (EP,US); C07C235/60 (EP,US); C07C235/78 (EP,US);
C07C235/84 (EP,US); C07C255/57 (EP,US); C07C59/66 (EP,US);
C07C59/68 (EP,US); C07D209/14 (EP,US); C07D209/42 (EP,US);
C07D213/55 (EP,US); C07D213/56 (EP,US); C07D213/81 (EP,KR,US);
C07D213/82 (EP,US); C07D215/04 (EP,KR,US); C07D217/26 (EP,KR,US);
C07D231/14 (EP,KR,US); C07D233/90 (EP,KR,US); C07D239/52 (EP,KR,US);
C07D241/24 (EP,KR,US); C07D261/18 (EP,KR,US); C07D263/26 (EP,KR,US);
C07D263/32 (EP,US); C07D277/20 (EP,KR,US); C07D277/30 (EP,US);
C07D277/34 (EP,US); C07D277/56 (EP,US); C07D307/54 (EP,US);
C07D307/79 (EP,US); C07D333/24 (EP,US); C07D401/04 (EP,US);
C07D417/04 (EP,US); C07D417/14 (EP,US); C07C2601/08 (EP,US);
C07C2601/14 (EP,US) (-)
Designated contracting statesAT,   BE,   CH,   CY,   DE,   DK,   ES,   FI,   FR,   GB,   GR,   IE,   IT,   LI,   LU,   MC,   NL,   PT,   SE [2002/26]
TitleGerman:CARBONSÄUREDERIVATE UND MEDIKAMENTE, DIE DIESE ENTHALTEN[2002/26]
English:CARBOXYLIC ACID DERIVATIVES AND DRUGS CONTAINING THE SAME[2002/26]
French:DERIVES D'ACIDE CARBOXYLIQUE ET MEDICAMENTS LES CONTENANT[2002/26]
Entry into regional phase13.03.2002Translation filed 
13.03.2002National basic fee paid 
13.03.2002Search fee paid 
13.03.2002Designation fee(s) paid 
13.03.2002Examination fee paid 
Examination procedure01.03.2001Request for preliminary examination filed
International Preliminary Examining Authority: JP
13.03.2002Examination requested  [2002/26]
13.06.2002Amendment by applicant (claims and/or description)
14.01.2011Application withdrawn by applicant  [2011/08]
Fees paidRenewal fee
26.09.2002Renewal fee patent year 03
25.09.2003Renewal fee patent year 04
23.09.2004Renewal fee patent year 05
26.09.2005Renewal fee patent year 06
21.09.2006Renewal fee patent year 07
24.09.2007Renewal fee patent year 08
25.09.2008Renewal fee patent year 09
25.09.2009Renewal fee patent year 10
22.09.2010Renewal fee patent year 11
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court
See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Documents cited:Search[X]WO9920275  (RHONE POULENC RORER PHARMA [US], et al) [X] 1-4,6-9,11-17 * page 2, line 31 - page 4, line 13; page 16, line 11 - page page 18, line 3; page 99, 1st compound *;
 [X]WO9736862  (SEARLE & CO [US], et al) [X] 1,2,4-8,10,11 * page 4, line 18 - page 11, line 7; examples 1, 2, 4-10, 12-16, 19-26, 28-44, 46-51, 53-65, 67, 69, 70, 75-84, 90, 91, 94, 95, 97-99, 102 *;
 [X]DE3026402  (SYNTEX CORP [US]) [X] 1-4,6,9,11 * page 6, line 27 - page 7, line 20; page 8, lines 4, 14, 29, 34 *;
 JPS5764655  [ ] (NIPPON ZOKI PHARMACEUTICAL CO);
 [X]EP0516069  (SUMITOMO PHARMA [JP]) [X] 1,2,4-7,10,11 * page 3, line 40 - page 5, line 16; examples 2-8, 13, 15-23, 25-32, 35, 37-41, 43-50, 53-70, 73-82, 85-100, 103-112, 117-120, 122-125, 127-139 *;
 [X]GB1465661  (TAISHO PHARMA CO LTD) [X] 1-4,6,9,11 * the whole document *;
 [X]WO9919300  (PFIZER [US], et al) [X] 1-4,6-9,11 * page 4, line 1 - page 8, line 24; page 21, line 29 - page 26, line 4; examples 1b-1w, 1ad-1am, 2-2c, 9-9c, 11a-11b, 11d-11e, 11h, 11m-11z, 12a-12b, 12f-12z, 15a-15b, 15d-15g, 16a *;
 [X]WO9631492  (TEXAS BIOTECHNOLOGY CORP [US], et al) [X] 1,2,4,5,8,11 * page 20, line 1 - page 21, line 26; page 262, lines 27-29; page 265, lines 10-11 *;
 [X]EP0763524  (SANKYO CO [JP]) [X] 1,4-7,10,11 * page 3, line 29 - page 6, line 30; table 1, e.g. compounds 38-45 *;
 [X]CH480070  (EPROVA AG [CH]) [X] 1-7,9,10 * column 9, lines 21-22; column 10, lines 29-30, 63-64; column 11, lines 30-31; column 12, lines 1-2, column 14, lines 44-45 *;
 [Y]EP0846693  (KYORIN SEIYAKU KK [JP]) [Y] 1-7,9-17 * page 2, lines 5-49; examples 14-51 *;
 WO9638428  [ ] (KYORIN SEIYAKU KK [JP], et al);
 [E]EP1213287  (KYORIN SEIYAKU KK [JP]) [E] 1,4-8,10-17 * page 3, lines 10-31; examples 5, 6, 23 *;
 [E]EP1184366  (KYORIN SEIYAKU KK [JP]) [E] 1-6,9-17 * the whole document, in particular examples 8-46, 49-141, 152-153, 158-159, 161, 174-197 *
 [X]  - CAPLUS, CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US, (1982), Database accession no. 1982:491971, URL: STN, XP002602130 [X] 1-7,9-11 * abstract; RN 64198-92-1, 82693-43-4, 82693-44-5, 82693-45-6, 82693-49-0, 82693-50-3, 82693-52-5 *
 [X]  - CAPLUS, CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US, (1963), Database accession no. 1963:435633, URL: STN, XP002602131 [X] 1-5,7,9,11 * abstract; RN 100087-40-9, 100173-40-8, 100089-37-0, 100149-63-1 *
    [ ] - H. BOJARSKA-DAHLIG ET AL, CONGR. SCI. FARM., CONF COMMUN., 21, PISA, (1962), pages 203 - 209
 [X]  - CAPLUS, CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US, (1987), Database accession no. 1987:477384, URL: STN, XP002602132 [X] 1-5,9-11 * abstract; RN 22161-81-5, 109679-89-2, 109679-90-5, 109679-85-8, 109679-86-9, 109718-57-2, 109718-58-3, 47087-07-0, 56105-81-8, 22071-15-4 *
    [ ] - J.W. KIM ET AL, ARCHIVES OF PHARMACAL RESEARCH, (1987), vol. 10, no. 1, pages 25 - 28
 [X]  - CAPLUS, CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US, (1995), Database accession no. 1995:478516, URL: STN, XP002602133 [X] 1-6,9,10 * abstract; RN 163433-43-0, 163433-44-1, 163433-45-2, 163433-46-3 *
    [ ] - H.D. CHOI ET AL, YAKHAK HOECHI, (1994), vol. 38, no. 5, pages 504 - 510
 [X]  - CAPLUS, CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US, (1991), Database accession no. 1991:622671, URL: STN, XP002602389 [X] 1,4,6-8 * RN 137103-47-0 *
    [ ] - H.G. FOUDA ET AL, XENOBIOTICA, (1991), vol. 21, no. 7, pages 925 - 934
 [YD]  - D.R. BUCKLE ET AL, BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, (19960903), vol. 6, no. 17, ISSN 0960-894X, pages 2121 - 2126, XP004135669 [YD] 1-7,9-17 * the whole document, in particular page 2124, last paragraph *

DOI:   http://dx.doi.org/10.1016/0960-894X(96)00383-6
International search[X]WO9920275  (RHONE POULENC RORER PHARMA [US], et al);
 [X]WO9919300  (PFIZER [US], et al);
 [X]EP0763524  (SANKYO CO [JP]);
 [X]EP0516069  (SUMITOMO PHARMA [JP]);
 [X]GB1436502  (GALLARDO ANTONIO SA);
 [X]WO9631492  (TEXAS BIOTECHNOLOGY CORP [US], et al);
 [X]EP0911025  (SSP CO LTD [JP]);
 [X]WO9736862  (SEARLE & CO [US], et al)
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.