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Extract from the Register of European Patents

EP About this file: EP1446402

EP1446402 - 2-AMINO-4-HETEROARYLETHYL THIAZOLINE DERIVATIVES AND THEIR USE AN INHIBITORS OF INDUCIBLE NO-SYNTHASE [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  08.09.2006
Database last updated on 26.06.2024
Most recent event   Tooltip13.04.2007Lapse of the patent in a contracting state
New state(s): CY
published on 16.05.2007  [2007/20]
Applicant(s)For all designated states
Aventis Pharma S.A.
20, avenue Raymond Aron
92160 Antony / FR
[2004/34]
Inventor(s)01 / BACQUE, Eric
123 Allée de la Clairière
F-91190 Gif sur Yvette / FR
02 / BIGOT, Antony
8 rue Jean Rostand
F-91300 Massy / FR
03 / CARRY, Jean-Christophe
41 rue du Dauphiné
F-94100 Saint Maur des Fosses / FR
04 / MIGNANI, Serge
14 Avenue de Robinson
F-92290 Chatenay Malabry / FR
 [2004/34]
Representative(s)Rousseau, Pierick Edouard, et al
Aventis Pharma S.A.
Direction des Brevets
Tri LEO/144
20, avenue Raymond Aron
92165 Antony Cedex / FR
[N/P]
Former [2004/34]Rousseau, Pierrick Edouard, et al
Aventis Pharma S.A. Direction des Brevets, Tri LEO/144 20, avenue Raymond Aron
92165 Antony Cedex / FR
Application number, filing date02793211.007.11.2002
[2004/34]
WO2002FR03809
Priority number, dateFR2001001450909.11.2001         Original published format: FR 0114509
US20020352977P30.01.2002         Original published format: US 352977 P
[2004/34]
Filing languageFR
Procedural languageFR
PublicationType: A1 Application with search report
No.:WO03040142
Date:15.05.2003
Language:FR
[2003/20]
Type: A1 Application with search report 
No.:EP1446402
Date:18.08.2004
Language:FR
The application published by WIPO in one of the EPO official languages on 15.05.2003 takes the place of the publication of the European patent application.
[2004/34]
Type: B1 Patent specification 
No.:EP1446402
Date:02.11.2005
Language:FR
[2005/44]
Search report(s)International search report - published on:EP15.05.2003
ClassificationIPC:C07D417/06, C07D277/28, A61K31/427, A61K31/426, A61K31/4439, A61K31/506, A61P25/16, C07D333/20, C07D413/06
[2004/34]
CPC data not yet available
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   IE,   IT,   LI,   LU,   MC,   NL,   PT,   SE,   SK,   TR [2004/34]
Extension statesAL09.06.2004
LT09.06.2004
LV09.06.2004
MK09.06.2004
RO09.06.2004
SI09.06.2004
TitleGerman:2-AMINO-4-HETEROARYLETHYL-THIAZOLINDERIVATE UND IHRE VERWENDUNG ALS HEMMSTOFFE DER INDUZIERBAREN NO-SYNTHASE[2004/34]
English:2-AMINO-4-HETEROARYLETHYL THIAZOLINE DERIVATIVES AND THEIR USE AN INHIBITORS OF INDUCIBLE NO-SYNTHASE[2004/34]
French:DERIVES DE 2-AMINO-4-HETEROARYLETHYL THIAZOLINE ET LEUR UTILISATION COMME INHIBITEURS DE NO-SYNTHASE INDUCTIBLE[2004/34]
Entry into regional phase09.06.2004National basic fee paid 
09.06.2004Designation fee(s) paid 
09.06.2004Examination fee paid 
Examination procedure26.06.2003Request for preliminary examination filed
International Preliminary Examining Authority: EP
09.06.2004Examination requested  [2004/34]
15.04.2005Communication of intention to grant the patent
25.08.2005Fee for grant paid
25.08.2005Fee for publishing/printing paid
Opposition(s)03.08.2006No opposition filed within time limit [2006/41]
Fees paidRenewal fee
30.11.2004Renewal fee patent year 03
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Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipCZ02.11.2005
EE02.11.2005
SK02.11.2005
CY07.11.2005
MC30.11.2005
LU02.01.2006
BG02.02.2006
[2007/20]
Former [2007/11]CZ02.11.2005
EE02.11.2005
SK02.11.2005
MC30.11.2005
LU02.01.2006
BG02.02.2006
Former [2006/41]CZ02.11.2005
SK02.11.2005
MC30.11.2005
BG02.02.2006
Former [2006/35]CZ02.11.2005
SK02.11.2005
MC30.11.2005
Former [2006/30]MC30.11.2005
Cited inInternational search[DA]WO9412165  (WELLCOME FOUND [GB], et al) [DA] 1,6 * the whole document *;
 [DA]WO9511231  (SEARLE & CO [US], et al) [DA] 1,6 * the whole document *;
 [DA]WO9614842  (MERCK & CO INC [US], et al) [DA] 1,6 * the whole document *;
 [PX]WO0194325  (AVENTIS PHARMA SA [FR]) [PX] 1-12* the whole document *;
 [X]  - NOIKE Y, "Syntheses of quinolizine derivatives. VI. Syntheses of 3-aminoquinolizines. 1. Syntheses of dl-3-amino, dl-3-epiamino-, and dl-3-epidimethylaminoquinolizidines", CHEMICAL ABSTRACTS, (19600610), vol. 54, no. 11, Database accession no. 11021h, XP002110770 [X] 12 * abrégé, en particulier composé X *
    [ ] - YAKUGAKU ZASSHI, (1959), vol. 79, pages 1514 - 1518
 [X]  - SABAT M ET AL, "Synthesis of unnatural amino acids via Suzuki cross-coupling of enantiopure vinyloxazolidine derivatives", ORGANIC LETTERS, (20000420), vol. 2, no. 8, pages 1089 - 1092, XP002205081 [X] 12 * the whole document *

DOI:   http://dx.doi.org/10.1021/ol005645i
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.