blank Quick help
blank Maintenance news

Scheduled maintenance

Regular maintenance outages:
between 05.00 and 05.15 hrs CET (Monday to Sunday).

Other outages
Availability
Register Forum

2022.02.11

More...
blank News flashes

News flashes

New version of the European Patent Register - SPC information for Unitary Patents.

2024-03-06

More...
blank Related links

Release notes
European Patent Register Assistant
European Patent Register Resource Book
European Patent Register – pocket guide
FAQ - European Patent Register
FAQ - Register Alert
Federated Register (Flyer)
Global Dossier (Flyer)
Register events
Deep link coverage
Federated Register content
The Patent Information Tour
Fair use charter

Extract from the Register of European Patents

EP About this file: EP1494673

EP1494673 - COMPOUNDS HAVING UNIQUE CB1 RECEPTOR BINDING SELECTIVITY AND METHODS FOR THEIR PRODUCTION AND USE [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  19.06.2009
Database last updated on 15.06.2024
Most recent event   Tooltip30.09.2011Lapse of the patent in a contracting state
New state(s): CY, TR		published on 02.11.2011  [2011/44]
Applicant(s)For all designated states
RESEARCH TRIANGLE INSTITUTE
3040 Cornwallis Road, P.O. Box 12194
Research Triangle Park, NC 27709 / US
[2008/33]
Former [2005/02]For all designated states
RESEARCH TRIANGLE INSTITUTE
3040 Cornwallis Road, P.O. Box 12194
Research Triangle Park, NC 27709 / US
Inventor(s)01 / THOMAS, Brian, F.
3 Fontana Ct.
Durham, NC 27713 / US
02 / SELTZMAN, Herbert, H.
4604 Hiddenbrook Drive
Raleigh, NC 27609 / US
03 / FRANCISCO, Maria, Elena, Y.
1021 Okaland Avenue
Durham, NC 27705 / US
 [2005/02]
Representative(s)Poulin, Gérard, et al
BREVALEX
95, rue d'Amsterdam
75378 Paris Cedex 8 / FR
[N/P]
Former [2009/48]Poulin, Gérard, et al
Brevalex 3, rue du Docteur Lancereaux
75008 Paris / FR
Former [2005/02]Poulin, Gérard, et al
BREVALEX 3, rue du Docteur Lancereaux
75008 Paris / FR
Application number, filing date03719602.914.04.2003
[2005/02]
WO2003US10470
Priority number, dateUS2002012170815.04.2002         Original published format: US 121708
[2005/02]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO03088968
Date:30.10.2003
Language:EN
[2003/44]
Type: A1 Application with search report 
No.:EP1494673
Date:12.01.2005
Language:EN
The application published by WIPO in one of the EPO official languages on 30.10.2003 takes the place of the publication of the European patent application.
[2005/02]
Type: B1 Patent specification 
No.:EP1494673
Date:13.08.2008
Language:EN
[2008/33]
Search report(s)International search report - published on:US30.10.2003
(Supplementary) European search report - dispatched on:EP06.12.2005
ClassificationIPC:A61K31/4745, A61K31/415, A61K31/473, C07D471/02, C07D231/12, A61P3/04, A61P25/18
[2006/03]
CPC:
C07D471/04 (EP,US); A61P25/18 (EP); A61P3/04 (EP);
C07D231/14 (EP,US)
Former IPC [2005/02]A61K31/4745, A61K31/415, A61K31/473, C07D471/02, C07D231/12
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HU,   IE,   IT,   LI,   LU,   MC,   NL,   PT,   RO,   SE,   SI,   SK,   TR [2005/02]
Extension statesALNot yet paid
LTNot yet paid
LVNot yet paid
MKNot yet paid
TitleGerman:VERBINDUNGEN MIT EINZIGARTIGER CB1-REZEPTOR-BINDUNGSSELEKTIVITÄT UND HERSTELLUNGS- UND ANWENDUNGSVERFAHREN DAFÜR[2005/02]
English:COMPOUNDS HAVING UNIQUE CB1 RECEPTOR BINDING SELECTIVITY AND METHODS FOR THEIR PRODUCTION AND USE[2005/02]
French:COMPOSES PRESENTANT UNE SELECTIVITE DE LIAISON AU RECEPTEUR CB1 UNIQUE ET PROCEDES DE PRODUCTION ET D'UTILISATION[2005/02]
Entry into regional phase08.10.2004National basic fee paid 
08.10.2004Search fee paid 
08.10.2004Designation fee(s) paid 
08.10.2004Examination fee paid 
Examination procedure17.11.2003Request for preliminary examination filed
International Preliminary Examining Authority: US
08.10.2004Examination requested  [2005/02]
15.12.2004Amendment by applicant (claims and/or description)
09.06.2006Despatch of a communication from the examining division (Time limit: M06)
12.10.2006Reply to a communication from the examining division
25.02.2008Communication of intention to grant the patent
24.06.2008Fee for grant paid
24.06.2008Fee for publishing/printing paid
Opposition(s)14.05.2009No opposition filed within time limit [2009/30]
Fees paidRenewal fee
13.04.2005Renewal fee patent year 03
17.03.2006Renewal fee patent year 04
12.04.2007Renewal fee patent year 05
28.03.2008Renewal fee patent year 06
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court		 See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipAT13.08.2008
BE13.08.2008
CY13.08.2008
CZ13.08.2008
DK13.08.2008
EE13.08.2008
FI13.08.2008
IT13.08.2008
NL13.08.2008
RO13.08.2008
SI13.08.2008
SK13.08.2008
TR13.08.2008
BG13.11.2008
SE13.11.2008
GR14.11.2008
ES24.11.2008
PT13.01.2009
HU14.02.2009
IE14.04.2009
LU14.04.2009
CH30.04.2009
LI30.04.2009
MC30.04.2009
[2011/43]
Former [2011/31]AT13.08.2008
BE13.08.2008
CZ13.08.2008
DK13.08.2008
EE13.08.2008
FI13.08.2008
IT13.08.2008
NL13.08.2008
RO13.08.2008
SI13.08.2008
SK13.08.2008
BG13.11.2008
SE13.11.2008
GR14.11.2008
ES24.11.2008
PT13.01.2009
HU14.02.2009
IE14.04.2009
LU14.04.2009
CH30.04.2009
LI30.04.2009
MC30.04.2009
Former [2011/21]AT13.08.2008
BE13.08.2008
CZ13.08.2008
DK13.08.2008
EE13.08.2008
FI13.08.2008
IT13.08.2008
NL13.08.2008
RO13.08.2008
SI13.08.2008
SK13.08.2008
BG13.11.2008
SE13.11.2008
GR14.11.2008
ES24.11.2008
PT13.01.2009
IE14.04.2009
LU14.04.2009
CH30.04.2009
LI30.04.2009
MC30.04.2009
Former [2010/48]AT13.08.2008
BE13.08.2008
CZ13.08.2008
DK13.08.2008
EE13.08.2008
FI13.08.2008
IT13.08.2008
NL13.08.2008
RO13.08.2008
SI13.08.2008
SK13.08.2008
BG13.11.2008
SE13.11.2008
GR14.11.2008
ES24.11.2008
PT13.01.2009
IE14.04.2009
CH30.04.2009
LI30.04.2009
MC30.04.2009
Former [2010/21]AT13.08.2008
BE13.08.2008
CZ13.08.2008
DK13.08.2008
EE13.08.2008
FI13.08.2008
IT13.08.2008
NL13.08.2008
RO13.08.2008
SI13.08.2008
SK13.08.2008
BG13.11.2008
SE13.11.2008
ES24.11.2008
PT13.01.2009
IE14.04.2009
CH30.04.2009
LI30.04.2009
MC30.04.2009
Former [2010/09]AT13.08.2008
BE13.08.2008
CZ13.08.2008
DK13.08.2008
EE13.08.2008
FI13.08.2008
IT13.08.2008
NL13.08.2008
RO13.08.2008
SI13.08.2008
SK13.08.2008
BG13.11.2008
SE13.11.2008
ES24.11.2008
PT13.01.2009
CH30.04.2009
LI30.04.2009
Former [2010/08]AT13.08.2008
BE13.08.2008
CZ13.08.2008
DK13.08.2008
EE13.08.2008
FI13.08.2008
IT13.08.2008
NL13.08.2008
RO13.08.2008
SI13.08.2008
SK13.08.2008
BG13.11.2008
ES24.11.2008
PT13.01.2009
CH30.04.2009
LI30.04.2009
Former [2009/39]AT13.08.2008
BE13.08.2008
CZ13.08.2008
DK13.08.2008
EE13.08.2008
FI13.08.2008
IT13.08.2008
NL13.08.2008
RO13.08.2008
SI13.08.2008
SK13.08.2008
BG13.11.2008
ES24.11.2008
PT13.01.2009
Former [2009/36]AT13.08.2008
BE13.08.2008
CZ13.08.2008
DK13.08.2008
EE13.08.2008
FI13.08.2008
NL13.08.2008
RO13.08.2008
SI13.08.2008
SK13.08.2008
BG13.11.2008
ES24.11.2008
PT13.01.2009
Former [2009/25]AT13.08.2008
BE13.08.2008
CZ13.08.2008
DK13.08.2008
FI13.08.2008
NL13.08.2008
RO13.08.2008
SI13.08.2008
SK13.08.2008
BG13.11.2008
ES24.11.2008
PT13.01.2009
Former [2009/24]AT13.08.2008
BE13.08.2008
CZ13.08.2008
DK13.08.2008
FI13.08.2008
NL13.08.2008
SI13.08.2008
SK13.08.2008
BG13.11.2008
ES24.11.2008
Former [2009/23]AT13.08.2008
BE13.08.2008
DK13.08.2008
FI13.08.2008
NL13.08.2008
SI13.08.2008
BG13.11.2008
ES24.11.2008
Former [2009/19]AT13.08.2008
BE13.08.2008
DK13.08.2008
FI13.08.2008
NL13.08.2008
SI13.08.2008
ES24.11.2008
Former [2009/15]AT13.08.2008
FI13.08.2008
NL13.08.2008
SI13.08.2008
ES24.11.2008
Former [2009/12]FI13.08.2008
NL13.08.2008
ES24.11.2008
Former [2009/09]NL13.08.2008
ES24.11.2008
Documents cited:Search   [ ] - No further relevant documents disclosed
International search[XP]US6509367  (MARTIN BILLY R [US], et al);
 [X]  - WILEY J.L. ET AL., "Novel pyrazole cannabinoids: insights into CB1 receptor recognition and activation", J. P.E.T., (2001), vol. 296, pages 1013 - 1022, XP002968556
 [X]  - SHIM J.-Y. ET AL., "Molecular interaction of the antagonist N-(piperidin-1-yl)-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide with the CB1 cannabinoid receptor", J. MED. CHEM., (200203), vol. 45, pages 1447 - 1459, XP002968557

DOI:   http://dx.doi.org/10.1021/jm010267o
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.