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Extract from the Register of European Patents

EP About this file: EP1513520

EP1513520 - SUBSTITUTED PYRROLINES AS KINASE INHIBITORS [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  31.07.2009
Database last updated on 05.07.2024
Most recent event   Tooltip30.09.2011Lapse of the patent in a contracting state
New state(s): CY, TR		published on 02.11.2011  [2011/44]
Applicant(s)For all designated states
Janssen Pharmaceutica NV
Turnhoutseweg 30
2340 Beerse / BE
[2008/39]
Former [2005/11]For all designated states
JANSSEN PHARMACEUTICA N.V.
Turnhoutseweg 30
2340 Beerse / BE
Inventor(s)01 / ZHANG, Han-Cheng
109 Bryan Way
Lansdale, PA 19446 / US
02 / MARYANOFF, Bruce E.
P.O. Box 239
New Hope, PA 18938 / US
03 / MCCOMSEY, David F.
1125 Victoria Road
Warminster, PA 18974 / US
04 / WHITE, Kimberly
120 Blue Ribbon Drive
North Wales, PA 19454 / US
05 / YE, Hong
124 Canterbury Lane
Lansdale, PA 19446 / US
06 / HECKER, Leonard
212 Tanglewood Way
Harleysville, PA 19438 / US
07 / CONWAY, Bruce R.
3302 Ephross Circle
Doylestown, PA 18901 / US
08 / DEMAREST, Keith
1 Newell Road
Flemington, NJ 08822 / US
 [2006/18]
Former [2005/11]01 / ZHANG, Han-Cheng
109 Bryan Way
Lansdale, PA 19446 / US
02 / MARYANOFF, Bruce E.
4029 Devonshire Drive
Forest Grove, PA 18922 / US
03 / MCCOMSEY, David F.
1125 Victoria Road
Warminster, PA 18974 / US
04 / WHITE, Kimberly
120 Blue Ribbon Drive
North Wales, PA 19454 / US
05 / YE, Hong
124 Canterbury Lane
Lansdale, PA 19446 / US
06 / HECKER, Leonard
212 Tanglewood Way
Harleysville, PA 19438 / US
07 / CONWAY, Bruce R.
3302 Ephross Circle
Doylestown, PA 18901 / US
08 / DEMAREST, Keith
1 Newell Road
Flemington, NJ 08822 / US
Representative(s)Mercer, Christopher Paul, et al
Carpmaels & Ransford LLP
One Southampton Row
London
WC1B 5HA / GB
[N/P]
Former [2009/51]Mercer, Christopher Paul, et al
Carpmaels & Ransford 43-45 Bloomsbury Square
London WC1A 2RA / GB
Former [2005/11]Mercer, Christopher Paul, et al
Carpmaels & Ransford, 43-45 Bloomsbury Square
London WC1A 2RA / GB
Application number, filing date03731528.004.06.2003
[2005/11]
WO2003US17518
Priority number, dateUS20020386002P05.06.2002         Original published format: US 386002 P
[2005/11]
Filing languageEN
Procedural languageEN
PublicationType: A2 Application without search report
No.:WO03103663
Date:18.12.2003
Language:EN
[2003/51]
Type: A2 Application without search report 
No.:EP1513520
Date:16.03.2005
Language:EN
The application published by WIPO in one of the EPO official languages on 18.12.2003 takes the place of the publication of the European patent application.
[2005/11]
Type: B1 Patent specification 
No.:EP1513520
Date:24.09.2008
Language:EN
[2008/39]
Search report(s)International search report - published on:EP08.07.2004
ClassificationIPC:A61K31/404, A61K31/416, A61P29/00, A61P37/02, C07D403/04
[2005/11]
CPC:
C07D409/14 (EP,US); A61P11/06 (EP); A61P13/12 (EP);
A61P17/00 (EP); A61P17/06 (EP); A61P17/14 (EP);
A61P25/00 (EP); A61P25/02 (EP); A61P25/04 (EP);
A61P25/18 (EP); A61P25/24 (EP); A61P25/28 (EP);
A61P27/02 (EP); A61P29/00 (EP); A61P3/10 (EP);
A61P35/00 (EP); A61P37/00 (EP); A61P37/02 (EP);
A61P37/06 (EP); A61P43/00 (EP); A61P7/02 (EP);
A61P9/00 (EP); A61P9/04 (EP); A61P9/10 (EP);
A61P9/12 (EP); C07D401/14 (EP,US); C07D403/04 (EP,US);
C07D403/14 (EP,US); C07D405/14 (EP,US); C07D417/14 (EP,US) (-)
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HU,   IE,   IT,   LI,   LU,   MC,   NL,   PT,   RO,   SE,   SI,   SK,   TR [2005/11]
Extension statesALNot yet paid
LTNot yet paid
LVNot yet paid
MKNot yet paid
TitleGerman:SUBSTITUIERTE PYRROLINE ALS KINASE INHIBITOREN[2005/11]
English:SUBSTITUTED PYRROLINES AS KINASE INHIBITORS[2005/11]
French:PYRROLINES SUBSTITUEES EN TANT QU'INHIBITEURS DE KINASE[2005/11]
Entry into regional phase04.01.2005National basic fee paid 
04.01.2005Designation fee(s) paid 
04.01.2005Examination fee paid 
Examination procedure12.12.2003Request for preliminary examination filed
International Preliminary Examining Authority: EP
04.01.2005Amendment by applicant (claims and/or description)
04.01.2005Examination requested  [2005/11]
24.06.2005Despatch of a communication from the examining division (Time limit: M06)
04.01.2006Reply to a communication from the examining division
16.11.2006Despatch of a communication from the examining division (Time limit: M04)
19.03.2007Reply to a communication from the examining division
11.10.2007Despatch of a communication from the examining division (Time limit: M04)
20.02.2008Reply to a communication from the examining division
31.03.2008Communication of intention to grant the patent
04.08.2008Fee for grant paid
04.08.2008Fee for publishing/printing paid
Opposition(s)25.06.2009No opposition filed within time limit [2009/36]
Fees paidRenewal fee
04.01.2005Renewal fee patent year 03
14.06.2006Renewal fee patent year 04
14.06.2007Renewal fee patent year 05
28.03.2008Renewal fee patent year 06
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court		 See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipAT24.09.2008
BE24.09.2008
CY24.09.2008
CZ24.09.2008
DK24.09.2008
EE24.09.2008
FI24.09.2008
NL24.09.2008
RO24.09.2008
SI24.09.2008
SK24.09.2008
TR24.09.2008
BG24.12.2008
SE24.12.2008
GR25.12.2008
PT24.02.2009
HU25.03.2009
IE04.06.2009
IT04.06.2009
LU04.06.2009
ES05.06.2009
[2011/43]
Former [2011/31]AT24.09.2008
BE24.09.2008
CZ24.09.2008
DK24.09.2008
EE24.09.2008
FI24.09.2008
NL24.09.2008
RO24.09.2008
SI24.09.2008
SK24.09.2008
BG24.12.2008
SE24.12.2008
GR25.12.2008
PT24.02.2009
HU25.03.2009
IE04.06.2009
IT04.06.2009
LU04.06.2009
ES05.06.2009
Former [2011/21]AT24.09.2008
BE24.09.2008
CZ24.09.2008
DK24.09.2008
EE24.09.2008
FI24.09.2008
NL24.09.2008
RO24.09.2008
SI24.09.2008
SK24.09.2008
BG24.12.2008
SE24.12.2008
GR25.12.2008
PT24.02.2009
IE04.06.2009
IT04.06.2009
LU04.06.2009
ES05.06.2009
Former [2011/14]AT24.09.2008
BE24.09.2008
CZ24.09.2008
DK24.09.2008
EE24.09.2008
FI24.09.2008
NL24.09.2008
RO24.09.2008
SI24.09.2008
SK24.09.2008
BG24.12.2008
SE24.12.2008
GR25.12.2008
PT24.02.2009
IE04.06.2009
IT04.06.2009
ES05.06.2009
Former [2010/46]AT24.09.2008
BE24.09.2008
CZ24.09.2008
DK24.09.2008
EE24.09.2008
FI24.09.2008
NL24.09.2008
RO24.09.2008
SI24.09.2008
SK24.09.2008
BG24.12.2008
SE24.12.2008
GR25.12.2008
PT24.02.2009
IE04.06.2009
ES05.06.2009
Former [2010/21]AT24.09.2008
BE24.09.2008
CZ24.09.2008
DK24.09.2008
EE24.09.2008
FI24.09.2008
NL24.09.2008
RO24.09.2008
SI24.09.2008
SK24.09.2008
BG24.12.2008
SE24.12.2008
PT24.02.2009
IE04.06.2009
Former [2010/09]AT24.09.2008
BE24.09.2008
CZ24.09.2008
DK24.09.2008
EE24.09.2008
FI24.09.2008
NL24.09.2008
RO24.09.2008
SI24.09.2008
SK24.09.2008
BG24.12.2008
SE24.12.2008
PT24.02.2009
Former [2009/36]AT24.09.2008
BE24.09.2008
CZ24.09.2008
DK24.09.2008
EE24.09.2008
FI24.09.2008
NL24.09.2008
RO24.09.2008
SI24.09.2008
SK24.09.2008
BG24.12.2008
PT24.02.2009
Former [2009/34]AT24.09.2008
BE24.09.2008
CZ24.09.2008
DK24.09.2008
FI24.09.2008
NL24.09.2008
RO24.09.2008
SI24.09.2008
SK24.09.2008
BG24.12.2008
PT24.02.2009
Former [2009/26]AT24.09.2008
BE24.09.2008
CZ24.09.2008
FI24.09.2008
NL24.09.2008
RO24.09.2008
SI24.09.2008
SK24.09.2008
BG24.12.2008
PT24.02.2009
Former [2009/24]AT24.09.2008
BE24.09.2008
CZ24.09.2008
FI24.09.2008
SI24.09.2008
SK24.09.2008
BG24.12.2008
Former [2009/23]AT24.09.2008
BE24.09.2008
FI24.09.2008
SI24.09.2008
BG24.12.2008
Former [2009/19]AT24.09.2008
BE24.09.2008
FI24.09.2008
SI24.09.2008
Former [2009/15]AT24.09.2008
FI24.09.2008
SI24.09.2008
Cited inInternational search[A]WO9113071  (BOEHRINGER MANNHEIM GMBH [DE]) [A] 1-58 * examples 69,70; claim 1 *;
 [DX]US5057614  (DAVIS PETER D [GB], et al) [DX] 1-58 * column 4, line 10 - column 5, line 65; examples 4,5,40,86,87; claims 1,10 *;
 [X]WO0238561  (NOVARTIS AG [CH], et al) [X] 1-58 * claim -; table 7 *;
 [PA]WO0246183  (ORTHO MCNEIL PHARM INC [US]) [PA] 1-58* example -; claim - *;
 [X]  - DAVIS P D ET AL, "INHIBITORS OF PROTEIN KINASE C 1. 2,3-BISARYLMALEIMIDES", JOURNAL OF MEDICINAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY. WASHINGTON, US, (1992), vol. 35, no. 1, ISSN 0022-2623, pages 177 - 184, XP000910195 [X] 1-58 * page 179, column R - page 181, column L; examples 19-26; table 3 *

DOI:   http://dx.doi.org/10.1021/jm00079a024
 [X]  - ZHU G ET AL, "Synthesis of Quinolinly/Isoquinolinyl(a)pyrrolo(3,4-c) Carbazoles as Cyclin D1/CDK4 Inhibitors", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, OXFORD, GB, (20030401), vol. 13, ISSN 0960-894X, pages 1231 - 1235, XP002255246 [X] 1-58 * examples 2A,-,2R *

DOI:   http://dx.doi.org/10.1016/S0960-894X(03)00133-1
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.