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Extract from the Register of European Patents

EP About this file: EP1539741

EP1539741 - 2-THIO-SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR USE IN PHARMACEUTICS [Right-click to bookmark this link]
StatusThe application is deemed to be withdrawn
Status updated on  22.06.2012
Database last updated on 29.07.2024
Most recent event   Tooltip22.06.2012Application deemed to be withdrawnpublished on 25.07.2012  [2012/30]
Applicant(s)For all designated states
MERCKLE GMBH
Chem.-pharm. Fabrik, Graf-Arco-Strasse 3
D-89079 Ulm / DE
[N/P]
Former [2005/24]For all designated states
MERCKLE GMBH
Chem.-pharm. Fabrik, Graf-Arco-Strasse 3
D-89079 Ulm / DE
Inventor(s)01 / LAUFER, Stefan
Karlstrasse 65/2
89143 Blaubeuren / DE
02 / STRIEGEL, Hans-Günter
Reiherweg 6
89143 Blaubeuren / DE
03 / TOLLMANN, Karola
Limburger Strasse 18
65611 Brechen / DE
04 / ALBRECHT, Wolfgang
Alfred-Mendler-Weg 25/1
89075 Ulm / DE
 [2006/16]
Former [2005/24]01 / LAUFER, Stefan
Karlstrasse 65/2
89143 Blaubeuren / DE
02 / STRIEGEL, Hans-Günter
Ulmer-Strasse 6-7
89134 Blaustein / DE
03 / TOLLMANN, Karola
Limburger Strasse 18
65611 Brechen / DE
04 / ALBRECHT, Wolfgang
Alfred-Mendler-Weg 25/1
89075 Ulm / DE
Representative(s)Reitstötter Kinzebach
Patentanwälte
Sternwartstraße 4
81679 München / DE
[N/P]
Former [2005/24]Reitstötter - Kinzebach
Patentanwälte, Sternwartstrasse 4
81679 München / DE
Application number, filing date03747916.920.08.2003
[2005/24]
WO2003EP09219
Priority number, dateDE2002103804520.08.2002         Original published format: DE 10238045
[2005/24]
Filing languageDE
Procedural languageDE
PublicationType: A1 Application with search report
No.:WO2004018458
Date:04.03.2004
Language:DE
[2004/10]
Type: A1 Application with search report 
No.:EP1539741
Date:15.06.2005
Language:DE
The application published by WIPO in one of the EPO official languages on 04.03.2004 takes the place of the publication of the European patent application.
[2005/24]
Search report(s)International search report - published on:EP04.03.2004
ClassificationIPC:C07D401/14, C07D401/04
[2005/24]
CPC:
C07D401/04 (EP,KR,US); C07D401/14 (KR); A61P1/02 (EP);
A61P1/04 (EP); A61P1/16 (EP); A61P11/00 (EP);
A61P17/06 (EP); A61P17/14 (EP); A61P19/02 (EP);
A61P19/06 (EP); A61P19/10 (EP); A61P25/00 (EP);
A61P25/04 (EP); A61P25/08 (EP); A61P25/28 (EP);
A61P29/00 (EP); A61P3/10 (EP); A61P31/18 (EP);
A61P35/00 (EP); A61P37/00 (EP); A61P37/02 (EP);
A61P37/06 (EP); A61P37/08 (EP); A61P9/00 (EP);
A61P9/04 (EP); A61P9/10 (EP) (-)
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HU,   IE,   IT,   LI,   LU,   MC,   NL,   PT,   RO,   SE,   SI,   SK,   TR [2005/24]
Extension statesALNot yet paid
LT18.02.2005
LV18.02.2005
MKNot yet paid
TitleGerman:2-THIO-SUBSTITUIERTE IMIDAZOLDERIVATE UND IHRE VERWENDUNG IN DER PHARMAZIE[2005/24]
English:2-THIO-SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR USE IN PHARMACEUTICS[2005/24]
French:DERIVES D'IMIDAZOL 2-THIO-SUBSTITUES ET LEUR UTILISATION DANS LE DOMAINE PHARMACEUTIQUE[2005/24]
Entry into regional phase18.02.2005National basic fee paid 
18.02.2005Designation fee(s) paid 
18.02.2005Examination fee paid 
Examination procedure16.03.2004Request for preliminary examination filed
International Preliminary Examining Authority: EP
18.02.2005Amendment by applicant (claims and/or description)
18.02.2005Examination requested  [2005/24]
27.04.2009Despatch of a communication from the examining division (Time limit: M04)
28.07.2009Reply to a communication from the examining division
18.02.2010Despatch of a communication from the examining division (Time limit: M06)
15.12.2010Reply to a communication from the examining division
10.01.2011Despatch of a communication from the examining division (Time limit: M06)
18.07.2011Reply to a communication from the examining division
21.09.2011Communication of intention to grant the patent
02.02.2012Application deemed to be withdrawn, date of legal effect  [2012/30]
09.03.2012Despatch of communication that the application is deemed to be withdrawn, reason: fee for grant / fee for printing not paid in time  [2012/30]
Divisional application(s)The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is  27.04.2009
Request for further processing for:The application is deemed to be withdrawn due to failure to reply to the examination report
15.12.2010Request for further processing filed
15.12.2010Full payment received (date of receipt of payment)
Request granted
04.01.2011Decision despatched
Fees paidRenewal fee
12.08.2005Renewal fee patent year 03
14.08.2006Renewal fee patent year 04
14.08.2007Renewal fee patent year 05
14.08.2008Renewal fee patent year 06
31.08.2009Renewal fee patent year 07
31.08.2010Renewal fee patent year 08
Penalty fee
Additional fee for renewal fee
31.08.201109   M06   Not yet paid
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Patent Court		 See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Cited inInternational search[DX]EP0004648  (CIBA GEIGY AG [CH]) [DX] 1-14 * page 1 - page 2, paragraph 2 * * page 5, paragraph 2 *;
 [DY]WO9314081  (SMITHKLINE BEECHAM CORP [US]) [DY] 1-14 * page 9, line 32 - line 34 * * page 10, line 13 - line 14 *;
 [X]US6040320  (BEERS SCOTT A [US], et al) [X] 1-14 * column 2, line 36 - column 4, line 30; example 1 * * example 78; table A *;
 [DX]WO0017192  (MERCKLE GMBH [DE], et al) [DX] 1-14 * page 5, paragraphs 2-4 *;
 [PY]WO02066458  (MERCKLE GMBH [DE], et al) [PY] 1-14 * page 26; table 2 *;
 [PY]DE10114775  (DANNHARDT GERHARD [DE]) [PY] 1-14* the whole document *;
 [Y]  - LAUFER, STEFAN ET AL, "Ones, thiones, and N-oxides: An exercise in imidazole chemistry", ANGEWANDTE CHEMIE, INTERNATIONAL EDITION (2002), 41(13), 2290-2293, XP002261426 [Y] 1-14 * page 2291, column 1, line 2 - line 3; figure 1 *

DOI:   http://dx.doi.org/10.1002/1521-3773(20020703)41:13<2290::AID-ANIE2290>3.0.CO;2-R
 [DY]  - LIVERTON, N.J.; ET AL., J. MED. CHEM., (1999), vol. 42, pages 2180 - 2190, XP002261427 [DY] 1-14 * page 2180, column 2, paragraph 2 * * page 2181; example 48; table 1 * * page 2183; figure 6; examples 45,46 *

DOI:   http://dx.doi.org/10.1021/jm9805236
 [DY]  - BOEHM, J.C.; ET AL., J. MED. CGEM., (1996), vol. 39, pages 3929 - 3937, XP002261428 [DY] 1-14 * page 3932; examples 44,45; table 2 *

DOI:   http://dx.doi.org/10.1021/jm960415o
Examination   - WAGNER, G. K. ET AL., "Indentification of regioisomers in a series of N-substituted pyridin-4-yl imidazole derivatives by regiospecific synthesis, GC/MS, and 1H NMR.", J. ORG. CHEM., (2003), vol. 68, doi:doi:10.1021/jo026619w, pages 4527 - 4530, XP002382672

DOI:   http://dx.doi.org/10.1021/jo026619w
by applicantRU1415725
 JPS6440467
 WO9110662
 WO9113876
 WO9314081
 WO9500501
 WO9903837
 DE10114775
    - J. MED. CHEM., (1996), vol. 39, pages 3927 - 37
    - ACTA CHIM., (1969), vol. 61, pages 69 - 77
    - J. PRAKT. CHEM., (1972), vol. 314, pages 785 - 792
    - INDIAN J. CHEM., SECT. B, (1983), vol. 22B, no. 3, pages 268 - 269
    - BIOORGANIC & MEDICINAL CHEM. LETT., (1995), vol. 5, no. 2, pages 177 - 180
    - PHOSPHORUS SULFUR, (1988), vol. 35, no. 1-2, pages 83 - 88
    - ARCH. BIOCHEM. BIOPHYS., (1992), vol. 297, pages 258 - 264
    - J. MED. CHEM., (1995), vol. 38, pages 1067 - 1083
    - HELV. CHIM. ACTA, (1999), vol. 82, pages 290 - 296
    - HELV. CHIM. ACTA, (1998), vol. 81, pages 1585 - 1595
    - LAUFER ET AL., ANGEW. CHEM. INT. ED., (2002), vol. 41, no. 13
    - LIVERTON ET AL., J. MED. CHEM., (1999), vol. 42, pages 2180 - 2190
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.