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Extract from the Register of European Patents

EP About this file: EP1572113

EP1572113 - CALCIUM RECEPTOR MODULATING COMPOUND AND USE THEREOF [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  23.03.2018
Database last updated on 28.05.2024
FormerThe patent has been granted
Status updated on  14.04.2017
FormerGrant of patent is intended
Status updated on  11.04.2017
FormerExamination is in progress
Status updated on  24.03.2017
FormerGrant of patent is intended
Status updated on  09.11.2016
Most recent event   Tooltip29.05.2020Lapse of the patent in a contracting state
New state(s): PT		published on 01.07.2020  [2020/27]
Applicant(s)For all designated states
Takeda Pharmaceutical Company Limited
1-1, Doshomachi 4-chome Chuo-ku
Osaka- shi, Osaka 541-0045 / JP
[2017/17]
Former [2005/37]For all designated states
Takeda Pharmaceutical Company Limited
1-1, Doshomachi 4-chome Chuo-ku
Osaka 541-0045 / JP
Inventor(s)01 / YASUMA, Tsuneo
20-5, Takada-cho
Ibaraki-shi, Osaka 567-0011 / JP
02 / MORI, Akira
358, Kashira-cho
Nijo-sagaru
Shinainomachi
Sakyo-ku
Kyoto-shi, Kyoto 606-8354 / JP
03 / KAWASE, Masahiro
14-5, Wakaba 2-chome
Inagawa-cho
Kawabe-gun, Hyogo 666-0251 / JP
04 / KIMURA, Hiroyuki
2-20-808, Ohamanakamachi 1-cho
Sakai-shi, Osaka 590-0975 / JP
05 / YOSHIDA, Masato
228-2, Hirono, Sanda-shi
Hyogo 669-1331 / JP
06 / GYORKOS, Albert, Charles
11795 Decatur Drive
Westminster, CO 80234 / US
07 / PRATT, Scott, Alan
13099 Alcott Place
Broomfield, CO 80020 / US
08 / CORRETTE, Christopher, Peter
13839 W. 66th Way
Arvada, CO 80004 / US
 [2017/20]
Former [2005/37]01 / YASUMA, Tsuneo
20-5, Takada-cho
Ibaraki-shi, Osaka 567-0011 / JP
02 / MORI, Akira
358 Kashiracho, Nijosagaru, Shinainomachi, Sakyoku
Kyoto-shi, Kyoto 606-8354 / JP
03 / KAWASE, Masahiro
14-5, Wakaba 2-chome, Inagawa-cho
Kawabe-gun Hyogo 666-0251 / JP
04 / KIMURA, Hiroyuki
2-20-808, Ohamanakamachi 1-cho
Sakai-shi, Osaka 590-0975 / JP
05 / YOSHIDA, Masato
228-2, Hirono, Sanda-shi
Hyogo 669-1331 / JP
06 / GYORKOS, Albert, Charles
11795 Decatur Drive
Westminster, CO 80234 / US
07 / PRATT, Scott, Alan
13099 Alcott Place
Broomfield, CO 80020 / US
08 / CORRETTE, Christopher, Peter
13839 W. 66th Way Arvada
Longmont, CO 80004 / US
Representative(s)Dossmann, Gérard, et al
Casalonga & Partners
Bayerstrasse 71-73
80335 München / DE
[2017/20]
Former [2009/31]Dossmann, Gérard, et al
Bureau CASALONGA & JOSSE Bayerstrasse 71/73
80335 München / DE
Former [2005/37]Rickard, Timothy Mark Adrian
Takeda Euro IP Department, 11-12 Charles II Street
London SW1Y 4QU / GB
Application number, filing date03793273.821.08.2003
[2005/37]
WO2003US26317
Priority number, dateUS20020406012P26.08.2002         Original published format: US 406012 P
US20030466129P28.04.2003         Original published format: US 466129 P
[2005/37]
Filing languageEN
Procedural languageEN
PublicationType: A2 Application without search report
No.:WO2004017908
Date:04.03.2004
Language:EN
[2004/10]
Type: A2 Application without search report 
No.:EP1572113
Date:14.09.2005
Language:EN
The application published by WIPO in one of the EPO official languages on 04.03.2004 takes the place of the publication of the European patent application.
[2005/37]
Type: B1 Patent specification 
No.:EP1572113
Date:17.05.2017
Language:EN
[2017/20]
Search report(s)International search report - published on:US05.01.2006
(Supplementary) European search report - dispatched on:EP19.10.2006
ClassificationIPC:C07D487/04, C07D221/04, C07D471/04, A61K31/519, A61K31/473, A61K31/551, A61K31/53, A61P19/10
[2006/47]
CPC:
C07D487/04 (EP,KR,US); A61P13/12 (EP); A61P19/00 (EP);
A61P19/02 (EP); A61P19/08 (EP); A61P19/10 (EP);
A61P25/28 (EP); A61P29/00 (EP); A61P3/10 (EP);
A61P3/14 (EP); A61P35/00 (EP); A61P43/00 (EP);
A61P5/14 (EP); A61P9/12 (EP); C07D403/04 (KR) (-)
Former IPC [2006/28]C07D221/04, C07D487/04, C07D471/04, A61K31/519, A61K31/473, A61K31/551, A61K31/53
Former IPC [2005/37]A61K6/00
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HU,   IE,   IT,   LI,   LU,   MC,   NL,   PT,   RO,   SE,   SI,   SK,   TR [2017/20]
Former [2005/37]AT,  BE,  BG,  CH,  CY,  CZ,  DE,  DK,  EE,  ES,  FI,  FR,  GB,  GR,  HU,  IE,  IT,  LI,  LU,  MC,  NL,  PT,  RO,  SE,  SI,  SK,  TR 
Extension statesAL14.02.2005
LT14.02.2005
LV14.02.2005
MK14.02.2005
TitleGerman:CALCIUM-REZEPTOR-MODULIERENDE VERBINDUNG UND IHRE VERWENDUNG[2005/37]
English:CALCIUM RECEPTOR MODULATING COMPOUND AND USE THEREOF[2005/37]
French:COMPOSE MODULATEUR DE RECEPTEUR DE CALCIUM ET UTILISATION ASSOCIEE[2005/37]
Entry into regional phase14.02.2005National basic fee paid 
14.02.2005Search fee paid 
14.02.2005Designation fee(s) paid 
14.02.2005Examination fee paid 
Examination procedure30.01.2004Request for preliminary examination filed
International Preliminary Examining Authority: US
14.02.2005Examination requested  [2005/37]
28.12.2007Despatch of a communication from the examining division (Time limit: M04)
04.03.2008Reply to a communication from the examining division
02.04.2008Despatch of a communication from the examining division (Time limit: M04)
11.08.2008Reply to a communication from the examining division
30.06.2011Despatch of a communication from the examining division (Time limit: M02)
24.08.2011Reply to a communication from the examining division
12.03.2015Despatch of a communication from the examining division (Time limit: M06)
01.09.2015Reply to a communication from the examining division
15.01.2016Despatch of a communication from the examining division (Time limit: M02)
15.03.2016Reply to a communication from the examining division
11.11.2016Communication of intention to grant the patent
21.03.2017Disapproval of the communication of intention to grant the patent by the applicant or resumption of examination proceedings by the EPO
21.03.2017Fee for grant paid
21.03.2017Fee for publishing/printing paid
11.04.2017Information about intention to grant a patent
11.04.2017Receipt of the translation of the claim(s)
Divisional application(s)The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is  28.12.2007
Opposition(s)20.02.2018No opposition filed within time limit [2018/17]
Fees paidRenewal fee
14.02.2005Renewal fee patent year 03
14.08.2006Renewal fee patent year 04
14.08.2007Renewal fee patent year 05
31.03.2008Renewal fee patent year 06
12.08.2009Renewal fee patent year 07
17.08.2010Renewal fee patent year 08
11.08.2011Renewal fee patent year 09
10.08.2012Renewal fee patent year 10
19.08.2013Renewal fee patent year 11
13.08.2014Renewal fee patent year 12
10.08.2015Renewal fee patent year 13
11.08.2016Renewal fee patent year 14
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court		 See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipHU21.08.2003
AT17.05.2017
CY17.05.2017
CZ17.05.2017
DK17.05.2017
EE17.05.2017
FI17.05.2017
MC17.05.2017
NL17.05.2017
PT17.05.2017
RO17.05.2017
SE17.05.2017
SI17.05.2017
SK17.05.2017
TR17.05.2017
BG17.08.2017
GR18.08.2017
IE21.08.2017
LU21.08.2017
BE31.08.2017
[2020/27]
Former [2020/15]HU21.08.2003
AT17.05.2017
CY17.05.2017
CZ17.05.2017
DK17.05.2017
EE17.05.2017
FI17.05.2017
MC17.05.2017
NL17.05.2017
RO17.05.2017
SE17.05.2017
SI17.05.2017
SK17.05.2017
TR17.05.2017
BG17.08.2017
GR18.08.2017
IE21.08.2017
LU21.08.2017
BE31.08.2017
Former [2019/46]HU21.08.2003
AT17.05.2017
CY17.05.2017
CZ17.05.2017
DK17.05.2017
EE17.05.2017
FI17.05.2017
MC17.05.2017
NL17.05.2017
RO17.05.2017
SE17.05.2017
SI17.05.2017
SK17.05.2017
BG17.08.2017
GR18.08.2017
IE21.08.2017
LU21.08.2017
BE31.08.2017
Former [2019/31]HU21.08.2003
AT17.05.2017
CZ17.05.2017
DK17.05.2017
EE17.05.2017
FI17.05.2017
MC17.05.2017
NL17.05.2017
RO17.05.2017
SE17.05.2017
SI17.05.2017
SK17.05.2017
BG17.08.2017
GR18.08.2017
IE21.08.2017
LU21.08.2017
BE31.08.2017
Former [2018/39]AT17.05.2017
CZ17.05.2017
DK17.05.2017
EE17.05.2017
FI17.05.2017
MC17.05.2017
NL17.05.2017
RO17.05.2017
SE17.05.2017
SI17.05.2017
SK17.05.2017
BG17.08.2017
GR18.08.2017
IE21.08.2017
LU21.08.2017
BE31.08.2017
Former [2018/34]AT17.05.2017
CZ17.05.2017
DK17.05.2017
EE17.05.2017
FI17.05.2017
MC17.05.2017
NL17.05.2017
RO17.05.2017
SE17.05.2017
SI17.05.2017
SK17.05.2017
BG17.08.2017
GR18.08.2017
IE21.08.2017
LU21.08.2017
Former [2018/25]AT17.05.2017
CZ17.05.2017
DK17.05.2017
EE17.05.2017
FI17.05.2017
MC17.05.2017
NL17.05.2017
RO17.05.2017
SE17.05.2017
SI17.05.2017
SK17.05.2017
BG17.08.2017
GR18.08.2017
Former [2018/18]AT17.05.2017
CZ17.05.2017
DK17.05.2017
EE17.05.2017
FI17.05.2017
MC17.05.2017
NL17.05.2017
RO17.05.2017
SE17.05.2017
SK17.05.2017
BG17.08.2017
GR18.08.2017
Former [2018/10]AT17.05.2017
CZ17.05.2017
DK17.05.2017
EE17.05.2017
FI17.05.2017
NL17.05.2017
RO17.05.2017
SE17.05.2017
SK17.05.2017
BG17.08.2017
GR18.08.2017
Former [2018/09]AT17.05.2017
DK17.05.2017
EE17.05.2017
FI17.05.2017
NL17.05.2017
SE17.05.2017
BG17.08.2017
GR18.08.2017
Former [2017/52]AT17.05.2017
FI17.05.2017
NL17.05.2017
SE17.05.2017
BG17.08.2017
GR18.08.2017
Former [2017/50]AT17.05.2017
FI17.05.2017
SE17.05.2017
BG17.08.2017
GR18.08.2017
Former [2017/49]AT17.05.2017
FI17.05.2017
GR18.08.2017
Documents cited:Search[PX]WO02072585  (GRUENENTHAL GMBH [DE], et al) [PX] 1-11,22* figure 1A; claim - *;
 [DX]  - K. REDDY ET AL., "synthesis of alkyl/aryl substituted pyrazolo[1,5-a]pyrimidines.", INDIAN JOURNAL OF CHEMISTRY SECTION B, india, (1993), vol. 32b, no. 5, pages 586 - 589, XP008069928 [DX] 1,2,11,22 * page 586 - page 587; table 1; compound 2 *
International search[X]  - BRANOWSKA ET AL., "Tandem vicarious nucleophilic subsitution of hydrogen/intramolecular Diels-Alder reaction of 1,24-triazines into functionalized cacloalkenopyradines.", CHEM PHARM BULL, (200204), vol. 50, no. 4, pages 463 - 466, XP008073107

DOI:   http://dx.doi.org/10.1248/cpb.50.463
ExaminationEP0217142
 US4746656
    - MUTSCHLERE ET AL, MUTSCHLER ARZNEIMITTELWIRKUNGEN : LEHRBUCH DER PHARMAKOLOGIE UND TOXIKOLOGIE, MUTSCHLER ARZNEIMITTELWIRKUNGEN : LEHRBUCH DER PHARMAKOLOGIE UND TOXIKOLOGIE, STUTTGART : WISSENSCHAFTL. VERL.-GES, DE, PAGE(S) 396 - 397, (20010101), ISBN 978-3-8047-1763-3, XP007904326
by applicantUS4746656
 JPS6333380
 EP0217142
    - NATURE, (1993), vol. 366, pages 575 - 580
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.