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Extract from the Register of European Patents

EP About this file: EP1638969

EP1638969 - CGRP RECEPTOR ANTAGONISTS [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  11.09.2009
Database last updated on 31.08.2024
Most recent event   Tooltip23.04.2010Lapse of the patent in a contracting statepublished on 26.05.2010  [2010/21]
Applicant(s)For all designated states
Merck & Co., Inc.
126 East Lincoln Avenue
Rahway, New Jersey 07065-0907 / US
[2008/45]
Former [2006/13]For all designated states
Merck & Co., Inc.
126 East Lincoln Avenue Rahway
New Jersey 07065-0907 / US
Inventor(s)01 / BURGEY, Christopher, S.
126 East Lincoln Avenue
Rahway, NJ 07065-0907 / US
02 / DENG, Zhengwu, J.
126 East Lincoln Avenue
Rahway, NJ 07065-0907 / US
03 / NGUYEN, Diem, N.
126 East Lincoln Avenue
Rahway, NJ 07065-0907 / US
04 / PAONE, Daniel, V.
126 East Lincoln Avenue
Rahway, NJ 07065-0907 / US
05 / SHAW, Anthony, W.
126 East Lincoln Avenue
Rahway, NJ 07065-0907 / US
06 / WILLIAMS, Theresa, M.
126 East Lincoln Avenue
Rahway, NJ 07065-0907 / US
 [2006/13]
Representative(s)Man, Jocelyn, et al
Merck & Co., Inc.
European Patent Department
Merck Sharp & Dohme Limited
Hertford Road, Hoddesdon
Hertfordshire, EN11 9BU / GB
[N/P]
Former [2006/48]Man, Jocelyn, et al
Merck & Co., Inc. European Patent Department Merck Sharp & Dohme Limited, Hertford Road, Hoddesdon
Hertfordshire, EN11 9BU / GB
Former [2006/13]Man, Jocelyn
Merck & Co.,Inc. European Patent Department Terlings Park Eastwick Road
Harlow, Essex CM20 2QR / GB
Application number, filing date04749887.809.04.2004
[2006/13]
WO2004US10851
Priority number, dateUS20030463089P15.04.2003         Original published format: US 463089 P
US20030510352P10.10.2003         Original published format: US 510352 P
[2006/13]
Filing languageEN
Procedural languageEN
PublicationType: A2 Application without search report
No.:WO2004092166
Date:28.10.2004
Language:EN
[2004/44]
Type: A2 Application without search report 
No.:EP1638969
Date:29.03.2006
Language:EN
The application published by WIPO in one of the EPO official languages on 28.10.2004 takes the place of the publication of the European patent application.
[2006/13]
Type: B1 Patent specification 
No.:EP1638969
Date:05.11.2008
Language:EN
[2008/45]
Search report(s)International search report - published on:EP20.01.2005
ClassificationIPC:C07D471/04, A61K31/4188, A61P25/06
[2006/13]
CPC:
C07D487/04 (EP,US); C07D471/04 (EP,KR,US); A61P1/02 (EP);
A61P1/04 (EP); A61P11/00 (EP); A61P11/06 (EP);
A61P13/10 (EP); A61P17/00 (EP); A61P19/02 (EP);
A61P25/00 (EP); A61P25/04 (EP); A61P25/06 (EP);
A61P25/08 (EP); A61P25/30 (EP); A61P27/02 (EP);
A61P27/16 (EP); A61P29/00 (EP); A61P3/10 (EP);
A61P31/04 (EP); A61P37/08 (EP); A61P43/00 (EP);
A61P7/08 (EP); A61P9/00 (EP) (-)
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HU,   IE,   IT,   LI,   LU,   MC,   NL,   PL,   PT,   RO,   SE,   SI,   SK,   TR [2006/13]
Extension statesALNot yet paid
HR15.11.2005
LT15.11.2005
LV15.11.2005
MKNot yet paid
TitleGerman:CGRP-REZEPTORANTAGONISTEN[2006/13]
English:CGRP RECEPTOR ANTAGONISTS[2006/13]
French:ANTAGONISTES DES RECEPTEURS CGRP[2006/13]
Entry into regional phase15.11.2005National basic fee paid 
15.11.2005Designation fee(s) paid 
15.11.2005Examination fee paid 
Examination procedure18.10.2005Amendment by applicant (claims and/or description)
15.11.2005Examination requested  [2006/13]
31.03.2008Communication of intention to grant the patent
07.08.2008Fee for grant paid
07.08.2008Fee for publishing/printing paid
Divisional application(s)EP08105721.8  / EP2039694
Opposition(s)06.08.2009No opposition filed within time limit [2009/42]
Fees paidRenewal fee
27.03.2006Renewal fee patent year 03
10.04.2007Renewal fee patent year 04
18.03.2008Renewal fee patent year 05
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court
See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipMC30.04.2009
[2010/21]
Cited inInternational search[A]WO0018764  (MERCK SHARP & DOHME [GB], et al) [A] 1-29 * claim 1 *;
 [PA]WO03104236  (BRISTOL MYERS SQUIBB CO [US], et al) [PA] 1-29 * claim 1 *;
 [A]  - MALLEE J J ET AL, "Receptor Activity-modifying Protein 1 Determines the Species Selectivity of Non-peptide CGRP Receptor Antagonists", JOURNAL OF BIOLOGICAL CHEMISTRY, AMERICAN SOCIETY OF BIOLOGICAL CHEMISTS, BALTIMORE, MD, US, (20020419), vol. 277, no. 16, ISSN 0021-9258, pages 14294 - 14298, XP002271313 [A] 1-29 * the whole document *

DOI:   http://dx.doi.org/10.1074/jbc.M109661200
 [A]  - VAN ROSSUM, D., HANISCH, U.K. QUIRION, R., "Neuroanatomical Localization, Pharmcological Characterization and Functions of CGRP, related peptides and Their Receptors", NEUROSCIENCE AND BEHAVIORAL REVIEWS, (1997), vol. 21, no. 5, pages 649 - 678, XP002299339 [A] 1-29 * the whole document *

DOI:   http://dx.doi.org/10.1016/S0149-7634(96)00023-1
by applicantUS4166452
 US4256108
 US4265874
 WO9635713
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The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.