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Extract from the Register of European Patents

EP About this file: EP1756080

EP1756080 - CHROMONE DERIVATIVES USEFUL AS VANILLOID ANTAGONISTS [Right-click to bookmark this link]
Status	The application is deemed to be withdrawn Status updated on 25.05.2012 Database last updated on 19.07.2024
Most recent event Tooltip	25.05.2012	Application deemed to be withdrawn	published on 27.06.2012 [2012/26]
Applicant(s)	For:BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU MC Novartis AG Lichtstrasse 35 4056 Basel / CH
	For:AT Novartis Pharma GmbH Brunner Strasse 59 1230 Wien / AT
	[N/P]
Former [2009/43]	For:BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU MC Novartis AG Lichtstrasse 35 4056 Basel / CH
	For:AT Novartis Pharma GmbH Brunner Strasse 59 1230 Wien / AT
Former [2007/09]	For:BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU MC Novartis AG Lichtstrasse 35 4056 Basel / CH
	For:AT NOVARTIS-PHARMA GMBH Brunner Strasse 59 1230 Vienna / AT
Inventor(s)	01 / RITCHIE, Timothy J., Novartis Pharmaceuticals UK Patents and Trademarks, Wimblehurst Road Horsham, West Sussex RH12 5AB / GB
	02 / CULSHAW, Andrew J., Novartis Pharmaceuticals UK Patents and Trademarks, Wimblehurst Road Horsham, WestSussex RH12 5AB / GB
	03 / BRAIN, Christopher T, Novartis Pharmaceutical UK Patents and Trademarks, Wimblehurst Road Horsham, West Sussex RH12 5AB / GB
	04 / DZIADULEWICZ, Edward, Novartis Pharmaceuticals UK Patents and Trademarks, Wimblehurst Road Horsham, West Sussex RH12 5AB / GB
	05 / Hart, Terance.W. Peakdale Molecular Ltd. Peakdale Science Park, Sheffield Road. Chapel en le Frith, High Peak. SK23 0PG / GB
	[2007/09]
Representative(s)	Vögeli-Lange, Regina Novartis AG Corporate Intellectual Property 4002 Basel / CH
	[N/P]
Former [2007/09]	Vögeli-Lange, Regina Novartis AG Corporate Intellectual Property Basel, 4002 / CH
Application number, filing date	05748025.3	08.06.2005
	[2007/09]
	WO2005EP06252
Priority number, date	GB20040012768	08.06.2004 Original published format: GB 0412768
	[2007/09]
Filing language	EN
Procedural language	EN
Publication	Type:	A1 Application with search report
	No.:	WO2005121116
	Date:	22.12.2005
	Language:	EN
	[2005/51]
	Type:	A1 Application with search report
	No.:	EP1756080
	Date:	28.02.2007
	Language:	EN
	The application published by WIPO in one of the EPO official languages on 22.12.2005 takes the place of the publication of the European patent application.
	[2007/09]
Search report(s)	International search report - published on:	EP	22.12.2005
Classification	IPC:	C07D311/36, C07D407/04, A61K31/352	[2007/09]
	CPC:	C07D407/04 (EP,KR,US); C07D311/36 (EP,KR,US); A61P1/04 (EP); A61P1/18 (EP); A61P11/00 (EP); A61P11/02 (EP); (+) A61P11/06 (EP); A61P11/14 (EP); A61P13/10 (EP); A61P17/00 (EP); A61P17/06 (EP); A61P19/02 (EP); A61P21/02 (EP); A61P25/00 (EP); A61P25/04 (EP); A61P25/06 (EP); A61P29/00 (EP); A61P37/08 (EP); A61P43/00 (EP); A61P7/10 (EP); A61P7/12 (EP); C07D405/12 (EP,KR,US) (-)
Designated contracting states	AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LI, LT, LU, MC, NL, PL, PT, RO, SE, SI, SK, TR [2007/09]
Extension states	AL	Not yet paid
	BA	Not yet paid
	HR	Not yet paid
	LV	Not yet paid
	MK	Not yet paid
	YU	Not yet paid
Title	German:	ALS VANILLOIDANTAGONISTEN GEEIGNETE CHROMONDERIVATE	[2007/09]
	English:	CHROMONE DERIVATIVES USEFUL AS VANILLOID ANTAGONISTS	[2007/09]
	French:	DERIVES DE CHROMONE UTILES EN TANT QU'ANTAGONISTES DE VANILLOIDE	[2007/09]
Entry into regional phase	08.01.2007	National basic fee paid
	08.01.2007	Designation fee(s) paid
	08.01.2007	Examination fee paid
Examination procedure	08.01.2007	Examination requested [2007/09]
	03.04.2009	Despatch of a communication from the examining division (Time limit: M06)
	10.10.2009	Reply to a communication from the examining division
	01.01.2012	Application deemed to be withdrawn, date of legal effect [2012/26]
	09.02.2012	Despatch of communication that the application is deemed to be withdrawn, reason: renewal fee not paid in time [2012/26]
Divisional application(s)	The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is 03.04.2009
Fees paid	Renewal fee
	02.07.2007	Renewal fee patent year 03
	28.03.2008	Renewal fee patent year 04
	16.06.2009	Renewal fee patent year 05
	11.06.2010	Renewal fee patent year 06
	Penalty fee
	Additional fee for renewal fee
	30.06.2011	07 M06 Not yet paid
Opt-out from the exclusive Tooltip competence of the Unified Patent Court	See the Register of the Unified Patent Court for opt-out data
	Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Cited in	International search	[X]WO9503293 (CHINOIN GYOGYSZER ES VEGYESZET [HU], et al) [X] 1,3-5 * claim 1 *;
		[X]US4841076 (KITAGAWA MASAYUKI [JP], et al) [X] 1,3-5 * column 18; compound 23 * * column 23; compound 52 * * claim 1 *;
		[X]GB1495305 (PFIZER LTD) [X] 1,3-5 * page 2, lines 20-25 * * Table, second and fourth compounds * * claim 1 *;
		[X]WO0117985 (INDENA SPA [IT], et al) [X] 1,3-5 * page 26; compound VIB 105 *;
		[X]US3864362 (FEUER LASZLO, et al) [X] 4 * column 6; compound VI *;
		[X]US4841077 (ITO NORIKI [JP], et al) [X] 4 * column 11, lines 10-23,44-58 * * column 12, lines 20-25 *;
		[A]WO9829403 (CHIESI FARMA SPA [IT], et al) [A] 1-6 * page 10, lines 4-11 * * claim 1 *;
		[A]US4501755 (WU EDWIN S [US]) [A] 1-6 * column 1, lines 10-14 * * claim 1 *;
		[A]WO0228851 (NEGMA LERADS [FR], et al) [A] 1-6 * claims 1,4 *
		[X] - MOERSCH, GEORGE W. ET AL, "Antifertility activity of isoflavones related to genistein", JOURNAL OF MEDICINAL CHEMISTRY ( 1967 ), 10(2), 154-8 CODEN: JMCMAR; ISSN: 0022-2623, (1967), XP002339302 [X] 1,3-5 * page 158; table IV; compounds XVI,XVII * DOI: http://dx.doi.org/10.1021/jm00314a005
		[X] - EDWARDS J M ET AL, "ANTINEOPLASTIC ACTIVITY AND CYTOTOXICITY OF FLAVONES, ISOFLAVONES, AND FLAVANONES", JOURNAL OF NATURAL PRODUCTS, (1979), vol. 42, no. 1, ISSN 0163-3864, pages 85 - 91, XP009035912 [X] 1,3-5 * page 90; table 3; compounds 93361,93362 * DOI: http://dx.doi.org/10.1021/np50001a002
		[X] - SHAO, GUO-XIAN ET AL, "Studies on the synthesis and structure-antihypoxia activity relations of daidzein, an active principle of Pueraria pseudohiruta, and its derivatives", CA, CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US, (19810101), Database accession no. 1981:174809, URL: STN, XP002339319 [X] 1,3-5 * abstract * * page 1; compound I *
		[X] - VILAIN, C., "Ichthyocidal properties of rotenoids and isoflavones", CA, CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US, (1979), Database accession no. 1979:469937, URL: STN, XP002339320 [X] 1,3-5 * abstract * * compounds: RN = 5093-58-3; RN = 70894-40-5 *
		[X] - BRADY, WILLIAM T. ET AL, "Intramolecular [2 + 2] ketene cycloadditions. Synthesis of isoflavones and 3-aroylbenzofurans", JOURNAL OF ORGANIC CHEMISTRY ( 1988 ), 53(7), 1353-6 CODEN: JOCEAH; ISSN: 0022-3263, (1988), XP002339303 [X] 4 * page 1353; compounds 8E,8F * DOI: http://dx.doi.org/10.1021/jo00242a002
		[X] - AL-MAHARIK, NAWAF I. ET AL, "Synthesis of C-C-Bridged Bis-Isoflavones", JOURNAL OF ORGANIC CHEMISTRY ( 2000 ), 65(8), 2305-2308 CODEN: JOCEAH; ISSN: 0022-3263, (2000), XP002339304 [X] 4 * page 2306; compound 4 * DOI: http://dx.doi.org/10.1021/jo991404g
		[X] - LEVAI, ALBERT ET AL, "A comparative study of the epoxidation of 2-substituted isoflavones by dimethyldioxirane, sodium hypochlorite, and alkaline hydrogen peroxide (Weitz-Scheffer reaction)", JOURNAL OF HETEROCYCLIC CHEMISTRY ( 2000 ), 37(5), 1065-1069 CODEN: JHTCAD; ISSN: 0022-152X, (2000), XP002339305 [X] 4 * page 1066; compounds 4-10,6-12,10-18,12-20 * DOI: http://dx.doi.org/10.1002/jhet.5570370507
		[X] - BONDARENKO, S. P. ET AL, "Synthesis of 3',4'-Dimethoxyisoflavone Derivatives", CHEMISTRY OF NATURAL COMPOUNDS (TRANSLATION OF KHIMIYA PRIRODNYKH SOEDINENII) ( 2003 ), 39(4), 340-343 CODEN: CHNCA8; ISSN: 0009-3130, (2003), XP002339306 [X] 4 * page 340; compounds 3-9,11-15 * DOI: http://dx.doi.org/10.1023/B:CONC.0000003412.37888.78
		[X] - BONDARENKO, S. P. ET AL, "Synthesis of Formononetin Analogs", CHEMISTRY OF NATURAL COMPOUNDS (TRANSLATION OF KHIMIYA PRIRODNYKH SOEDINENII) ( 2003 ), 39(4), 344-348 CODEN: CHNCA8; ISSN: 0009-3130, (2003), XP002339307 [X] 4 * page 345; compounds 2,3,4,6-12,14,16,17,19,20 * DOI: http://dx.doi.org/10.1023/B:CONC.0000003413.23808.2b
		[X] - PARMAR, VIRINDER S. ET AL, "Fragmentation pathways in the mass spectra of 2-methylisoflavone derivatives. Useful in their diagnosis", JOURNAL OF THE INDIAN CHEMICAL SOCIETY ( 1987 ), 64(1), 64-6 CODEN: JICSAH; ISSN: 0019-4522, (1987), XP009051764 [X] 4 * page 65; compounds 2-7 *
		[X] - KUROSAWA, KAZU ET AL, "Reactions of 2'-hydroxyisoflavone and 2'-hydroxy-2-methylisoflavones with metal salts", CA, CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US, (1979), Database accession no. 1979:420255, URL: STN, XP002339321 [X] 4 * abstract * * compounds: RN = 70387-00-7; RN = 70387-01-8; RN = 70387-03-0 *
		[X] - ANIRUDHAN, C. A. ET AL, "The chemistry of the "insoluble red" woods. X. Syntheses of isoflavans, isoflav-3-enes, and isoflavylium salts", CA, CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US, (1966), Database accession no. 1966:67663, URL: STN, XP002339322 [X] 4 * abstract * * compounds: RN = 5093-58-3; RN = 5093-58-3; RN = 5093-60-7 *
		[X] - KUKLA, A. S. ET AL, "Insecticidal properties and chemical constitution. VII. Allylated isoflavone derivatives", CA, CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US, (1963), Database accession no. 1964:3073, URL: STN, XP002339323 [X] 4 * abstract * * compounds: RN = 54528-39-1; RN = 100211-03-8 *
		[X] - FUKUI, KENJI ET AL, "Synthesis of 7-hydroxy-2',4',5'-trimethoxyisoflavone and related compounds", CA, CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US, (1963), Database accession no. 1963:448229, URL: STN, XP002339324 [X] 4 * abstract * * compound: RN = 99886-39-2 *

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