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Extract from the Register of European Patents

EP About this file: EP1812003

EP1812003 - ORTHO- CONDENSED PYRIDINE AND PYRIMIDINE DERIVATIVES (E. G. PURINES) AS PROTEIN KINASES INHIBITORS [Right-click to bookmark this link]
StatusThe application has been withdrawn
Status updated on  06.05.2011
Database last updated on 26.06.2024
Most recent event   Tooltip06.05.2011Withdrawal of applicationpublished on 08.06.2011  [2011/23]
Applicant(s)For all designated states
Astex Therapeutics Limited
436 Cambridge Science Park Milton Road, Cambridge
CB4 0QA / GB
For all designated states
The Institute of Cancer Research: Royal Cancer Hospital
123 Old Brompton Road
London SW7 3RP / GB
For all designated states
Cancer Research Technology Limited
Sardinia House, Sardinia Street
London WC2A 3NL / GB
[N/P]
Former [2007/31]For all designated states
Astex Therapeutics Limited
436 Cambridge Science Park Milton Road, Cambridge
CB4 0QA / GB
For all designated states
THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL
123 Old Brompton Road
London SW7 3RP / GB
For all designated states
Cancer Research Technology Limited
Sardinia House, Sardinia Street
London WC2A 3NL / GB
Inventor(s)01 / BERDINI, Valerio
436 Cambridge Science Park Milton Road
Cambridge CB4 0QA / GB
02 / BOYLE, Robert, George
436 Cambridge Science Park Milton Road
Cambridge CB4 0QA / GB
03 / SAXTY, Gordon
436 Cambridge Science Park Milton Road
Cambridge CB4 0QA / GB
04 / VERDONK, Marinus, Leendert
436 Cambridge Science Park Milton Road
Cambridge CB4 0QA / GB
05 / WOODHEAD, Steven, John
436 Cambridge Science Park Milton Road
Cambridge CB4 0QA / GB
06 / WYATT, Paul, Graham
436 Cambridge Science Park Milton Road
Cambridge CB4 0QA / GB
07 / SORE, Hannah, Fiona
436 Cambridge Science Park Milton Road
Cambridge CB4 0QA / GB
08 / CALDWELL, John
Cancer Research UK 15 Cotswold Road
Sutton SM2 5NG / GB
09 / COLLINS, Ian
Cancer Research UK 15 Cotswold Road
Sutton SM2 5NG / GB
10 / DA FONSECA, Tatiana, Faria
Cancer Research UK 15 Cotswold Road
Sutton SM2 5NG / GB
11 / DONALD, Alastair
Cancer Research UK 15 Cotswold Road
Sutton SM2 5NG / GB
 [2007/31]
Representative(s)Hutchins, Michael Richard
Elkington and Fife LLP
Prospect House
8 Pembroke Road
Sevenoaks
Kent TN13 1XR / GB
[N/P]
Former [2008/13]Hutchins, Michael Richard
Elkington and Fife LLP Prospect House 8 Pembroke Road Sevenoaks
Kent TN13 1XR / GB
Former [2007/31]Hutchins, Michael Richard
M.R. Hutchins & Co, 23 Mount Sion Tunbridge Wells
Kent TN1 1TZ / GB
Application number, filing date05796842.225.10.2005
[2007/31]
WO2005GB04115
Priority number, dateGB2004002368425.10.2004         Original published format: GB 0423684
US20040621719P25.10.2004         Original published format: US 621719 P
US20050683980P24.05.2005         Original published format: US 683980 P
[2007/31]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2006046023
Date:04.05.2006
Language:EN
[2006/18]
Type: A1 Application with search report 
No.:EP1812003
Date:01.08.2007
Language:EN
The application published by WIPO in one of the EPO official languages on 04.05.2006 takes the place of the publication of the European patent application.
[2007/31]
Search report(s)International search report - published on:EP04.05.2006
ClassificationIPC:A61K31/52, A61K31/519, C07D473/34, A61K31/437, C07D471/04, C07D487/04, C07D473/00
[2007/31]
CPC:
C07D471/04 (EP,US); A61P25/00 (EP); A61P3/04 (EP);
A61P3/10 (EP); A61P35/00 (EP); A61P37/02 (EP);
A61P43/00 (EP); A61P9/10 (EP); C07D473/00 (EP,US);
C07D473/34 (EP,US); C07D487/04 (EP,US) (-)
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   NL,   PL,   PT,   RO,   SE,   SI,   SK,   TR [2007/31]
Extension statesALNot yet paid
BANot yet paid
HRNot yet paid
MKNot yet paid
YUNot yet paid
TitleGerman:ORTHOKONDENSIERTE PYRIDIN- UND PYRIMIDIN-DERIVATE (Z.B. PURINE) ALS PROTEINKINASE-HEMMER[2007/31]
English:ORTHO- CONDENSED PYRIDINE AND PYRIMIDINE DERIVATIVES (E. G. PURINES) AS PROTEIN KINASES INHIBITORS[2007/31]
French:DERIVES ORTHO-CONDENSES DE PYRIDINE ET PYRIMIDINE (PAR EXEMPLE PURINES) EN TANT QU'INHIBITEURS DE PROTEINES KINASES[2007/31]
Entry into regional phase25.05.2007National basic fee paid 
25.05.2007Designation fee(s) paid 
25.05.2007Examination fee paid 
Examination procedure25.05.2007Examination requested  [2007/31]
14.06.2007Amendment by applicant (claims and/or description)
03.09.2008Despatch of a communication from the examining division (Time limit: M06)
12.03.2009Reply to a communication from the examining division
21.09.2010Despatch of a communication from the examining division (Time limit: M06)
30.03.2011Reply to a communication from the examining division
28.04.2011Application withdrawn by applicant  [2011/23]
Divisional application(s)The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is  03.09.2008
Fees paidRenewal fee
29.10.2007Renewal fee patent year 03
26.03.2008Renewal fee patent year 04
13.10.2009Renewal fee patent year 05
12.10.2010Renewal fee patent year 06
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Cited inInternational search[X]GB1047935  (AMERICAN CYANAMID CO) [X] 1,3 * example 5 * * page 2, line 74 - line 88 *;
 [X]US6432947  (ARNAIZ DAMIAN O [US], et al) [X] 3 * column 55, line 31 - line 39 *;
 [A]EP1444982  (MERCKLE GMBH [DE]) [A] 1,3 * page 3, line 24 - page 4, line 51 ** claim 1, definition of R1 *
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 US2003139427
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