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Extract from the Register of European Patents

EP About this file: EP1773768

EP1773768 - PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  28.06.2019
Database last updated on 19.10.2024
FormerThe patent has been granted
Status updated on  20.07.2018
FormerGrant of patent is intended
Status updated on  15.01.2018
FormerExamination is in progress
Status updated on  07.11.2016
Most recent event   Tooltip28.06.2019No opposition filed within time limitpublished on 31.07.2019  [2019/31]
Applicant(s)For all designated states
Exelixis, Inc.
1851 Harbor Bay Parkway
Alameda, CA 94502-3010 / US
[2018/38]
Former [2018/27]For all designated states
Exelixis, Inc.
210 East Grand Avenue
South San Francisco, CA 94080 / US
Former [2007/16]For all designated states
Exelixis, Inc.
170 Harbor Way, P.O. Box 511
South San Francisco, CA 94083-0511 / US
Inventor(s)01 / CANNE BANNEN, Lynne
1086 Rio Vista Drive
Pacifica, California 94044 / US
02 / CHEN, Jeff
140 South Van Ness Avenue, Apartment 407
San Francisco, California 94103 / US
03 / DALRYMPLE, Lisa, Esther
650 Anderson Street
San Francisco, California 94110 / US
04 / FLATT, Brenton, T.
12721 Pedriza Drive
Poway, California 92064 / US
05 / FORSYTH, Timothy, Patrick
1928 Wingate Way
Hayward, California 94541 / US
06 / GU, Xiao-Hui
7699 Palmilla Drive, 3408
San Diego, California 92122 / US
07 / MAC, Morrison, B.
2567 30th Avenue
San Francisco, California 94116 / US
08 / MANN, Larry, W.
6450 Whitney Woods
Richland, Michigan 49083 / US
09 / MANN, Grace
231 Callippe Court
Brisbane, California 94005 / US
10 / MARTIN, Richard
4293 Cordobes Cove
San Diego, California 92130 / US
11 / MOHAN, Raju
3125 Caminito Ricardo
Encinitas, California 92024 / US
12 / MURPHY, Brett
487 E. Montana Drive
Sandy, UT 84070 / US
13 / NYMAN, Michael, Charles
4511 Rhode Island Street
San Diego, California 92116 / US
14 / STEVENS, William, C., Jr.
11632 Candy Rose Way
San Diego, CA 92131 / US
15 / WANG, Tie-Lin
7746 Roan Road
San Diego, California 92129 / US
16 / WANG, Yong
667 Catamaran Street, Apartment 3
Foster City, California 94404 / US
17 / WU, Jason, H.
8310 Regents Road, B
San Diego, California 92122 / US
 [2007/42]
Former [2007/30]01 / CANNE BANNEN, Lynne
1086 Rio Vista Drive
Pacifica, California 94044 / US
02 / CHEN, Jeff
140 South Van Ness Avenue, Apartment 407
San Francisco, California 94103 / US
03 / DALRYMPLE, Lisa, Esther
650 Anderson Street
San Francisco, California 94110 / US
04 / FLATT, Brenton, T.
12721 Pedriza Drive
Poway, California 92064 / US
05 / FORSYTH, Timothy, Patrick
1928 Wingate Way
Hayward, California 94541 / US
06 / GU, Xiao-Hu
7699 Palmilla Drive, 3408
San Diego, California 92122 / US
07 / MAC, Morrison, B.
2567 30th Avenue
San Francisco, California 94116 / US
08 / MANN, Larry, W.
6450 Whitney Woods
Richland, Michigan 49083 / US
09 / MANN, Grace
231 Callippe Court
Brisbane, California 94005 / US
10 / MARTIN, Richard
4293 Cordobes Cove
San Diego, California 92130 / US
11 / MOHAN, Raju
3125 Caminito Ricardo
Encinitas, California 92024 / US
12 / MURPHY, Brett
487 E. Montana Drive
Sandy, UT 84070 / US
13 / NYMAN, Michael, Charles
4511 Rhode Island Street
San Diego, California 92116 / US
14 / STEVENS, William, C., Jr.
11632 Candy Rose Way
San Diego, CA 92131 / US
15 / WANG, Tie-Lin
7746 Roan Road
San Diego, California 92129 / US
16 / WANG, Yong
667 Catamaran Street, Apartment 3
Foster City, California 94404 / US
17 / WU, Jason, H.
8310 Regents Road, B
San Diego, California 92122 / US
Former [2007/27]01 / CANNE BANNEN, Lynne
801 Saint Lawrence Drive
Pacifica, California 94044 / US
02 / CHEN, Jeff
140 South Van Ness Avenue, Apartment 407
San Francisco, California 94103 / US
03 / DALRYMPLE, Lisa, Esther
650 Anderson Street
San Francisco, California 94110 / US
04 / FLATT, Brenton, T.
12721 Pedriza Drive
Poway, California 92064 / US
05 / FORSYTH, Timothy, Patrick
1928 Wingate Way
Hayward, California 94541 / US
06 / GU, Xiao-Hu
7699 Palmilla Drive, 3408
San Diego, California 92122 / US
07 / MAC, Morrison, B.
2567 30th Avenue
San Francisco, California 94116 / US
08 / MANN, Larry, W.
6450 Whitney Woods
Richland, Michigan 49083 / US
09 / MANN, Grace
231 Callippe Court
Brisbane, California 94005 / US
10 / MARTIN, Richard
4293 Cordobes Cove
San Diego, California 92130 / US
11 / MOHAN, Raju
3125 Caminito Ricardo
Encinitas, California 92024 / US
12 / MURPHY, Brett
487 E. Montana Drive
Sandy, UT 84070 / US
13 / NYMAN, Michael, Charles
4511 Rhode Island Street
San Diego, California 92116 / US
14 / STEVENS, William, C., Jr.
11632 Candy Rose Way
San Diego, CA 92131 / US
15 / WANG, Tie-Lin
7746 Roan Road
San Diego, California 92129 / US
16 / WANG, Yong
667 Catamaran Street, Apartment 4
Foster City, California 94404 / US
17 / WU, Jason, H.
8310 Regents Road, B
San Diego, California 92122 / US
Former [2007/16]01 / CANNE BANNEN, Lynne
801 Saint Lawrence Drive
Pacifica, California 94044 / US
02 / CHEN, Jeff
140 South Van Ness Avenue, Apartment 407
San Francisco, California 94103 / US
03 / DALRYMPLE, Lisa, Esther
650 Anderson Street
San Francisco, California 94110 / US
04 / FLATT, Brenton, T.
12721 Pedriza Drive
Poway, California 92064 / US
05 / FORSYTH, Timothy, Patrick
1928 Wingate Way
Hayward, California 94541 / US
06 / GU, Xiao-Hu
7699 Palmilla Drive, 3408
San Diego, California 92122 / US
07 / MAC, Morrison, B.
2567 30th Avenue
San Francisco, California 94116 / US
08 / MANN, Larry, W.
6450 Whitney Woods
Richland, Michigan 49083 / US
09 / MANN, Grace
231 Callippe Court
Brisbane, California 94005 / US
10 / MARTIN, Richard
4293 Cordobes Cove
San Diego, California 92130 / US
11 / MOHAN, Raju
3125 Caminito Ricardo
Encinitas, California 92024 / US
12 / MURPHY, Brett
32485 Skylark Drive
Lake Elsinore, California 92530 / US
13 / NYMAN, Michael, Charles
4511 Rhode Island Street
San Diego, California 92116 / US
14 / STEVENS, William, C., Jr.
8850 West Lilac Road
Escondido, California 92026 / US
15 / WANG, Tie-Lin
7746 Roan Road
San Diego, California 92129 / US
16 / WANG, Yong
667 Catamaran Street, Apartment 4
Foster City, California 94404 / US
17 / WU, Jason, H.
8310 Regents Road, B
San Diego, California 92122 / US
Representative(s)Murgitroyd & Company
165-169 Scotland Street
Glasgow G5 8PL / GB
[N/P]
Former [2018/34]Murgitroyd & Company
Scotland House
165-169 Scotland Street
Glasgow G5 8PL / GB
Former [2007/16]Main, Malcolm Charles
Murgitroyd & Company Scotland House 165-169 Scotland Street
Glasgow G5 8PL / GB
Application number, filing date05803281.430.07.2005
[2007/16]
WO2005US26916
Priority number, dateUS20040592469P30.07.2004         Original published format: US 592469 P
US20040592439P30.07.2004         Original published format: US 592439 P
[2007/16]
Filing languageEN
Procedural languageEN
PublicationType: A2 Application without search report
No.:WO2006012642
Date:02.02.2006
Language:EN
[2006/05]
Type: A2 Application without search report 
No.:EP1773768
Date:18.04.2007
Language:EN
The application published by WIPO in one of the EPO official languages on 02.02.2006 takes the place of the publication of the European patent application.
[2007/16]
Type: B1 Patent specification 
No.:EP1773768
Date:22.08.2018
Language:EN
[2018/34]
Type: B8 Corrected title page of specification 
No.:EP1773768
Date:26.12.2018
[2018/52]
Search report(s)International search report - published on:US27.07.2006
(Supplementary) European search report - dispatched on:EP04.07.2008
ClassificationIPC:C07D207/416, C07D401/12, C07D403/12, C07D405/12, C07D409/12, C07D417/12, A61K31/40, A61K31/4025, A61K31/415, A61K31/426, A61K31/428, A61K31/433, A61K31/4439, A61P3/00, A61P15/08, A61P19/00, A61P35/00
[2008/32]
CPC:
C07D207/416 (EP,NO,US); C07D207/34 (KR); A61K31/40 (KR,NO);
A61K31/4025 (NO); A61K31/405 (NO); A61K31/415 (NO);
A61K31/426 (NO); A61K31/428 (NO); A61K31/433 (NO);
A61K31/4439 (NO); A61P13/12 (EP); A61P15/00 (EP);
A61P15/08 (EP,NO); A61P15/18 (EP); A61P17/00 (EP);
A61P19/00 (EP,NO); A61P19/08 (EP); A61P21/00 (EP);
A61P25/00 (EP); A61P25/28 (EP); A61P3/00 (EP,NO);
A61P3/10 (EP); A61P35/00 (EP,NO); A61P37/00 (EP);
A61P37/02 (EP); A61P37/04 (EP); A61P43/00 (EP);
A61P5/00 (EP); A61P5/42 (EP); A61P5/44 (EP);
A61P9/00 (EP); A61P9/12 (EP); C07D401/12 (EP,NO,US);
C07D403/12 (EP,NO,US); C07D405/12 (EP,NO,US); C07D409/12 (EP,NO,US);
C07D417/12 (EP,NO,US) (-)
Former IPC [2007/16]C07D207/325, A61K31/40
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   NL,   PL,   PT,   RO,   SE,   SI,   SK,   TR [2018/34]
Former [2007/16]AT,  BE,  BG,  CH,  CY,  CZ,  DE,  DK,  EE,  ES,  FI,  FR,  GB,  GR,  HU,  IE,  IS,  IT,  LI,  LT,  LU,  LV,  MC,  NL,  PL,  PT,  RO,  SE,  SI,  SK,  TR 
Extension statesAL18.01.2007
BA18.01.2007
HR18.01.2007
MK18.01.2007
YU18.01.2007
TitleGerman:PYRROLDERIVATE ALS PHARMAZEUTISCHE WIRKSTOFFE[2007/16]
English:PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS[2007/16]
French:DERIVES DE PYRROLE EN TANT QU'AGENTS PHARMACEUTIQUES[2007/16]
Entry into regional phase18.01.2007National basic fee paid 
18.01.2007Search fee paid 
18.01.2007Designation fee(s) paid 
18.01.2007Examination fee paid 
Examination procedure18.01.2007Examination requested  [2007/16]
15.01.2009Despatch of a communication from the examining division (Time limit: M06)
18.09.2009Despatch of communication that the application is deemed to be withdrawn, reason: reply to the communication from the examining division not received in time
30.11.2009Reply to a communication from the examining division
12.11.2013Despatch of a communication from the examining division (Time limit: M06)
19.05.2014Reply to a communication from the examining division
28.04.2016Despatch of a communication from the examining division (Time limit: M06)
03.11.2016Reply to a communication from the examining division
16.01.2018Communication of intention to grant the patent
24.05.2018Fee for grant paid
24.05.2018Fee for publishing/printing paid
24.05.2018Receipt of the translation of the claim(s)
Divisional application(s)The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is  15.01.2009
Opposition(s)23.05.2019No opposition filed within time limit [2019/31]
Request for further processing for:The application is deemed to be withdrawn due to failure to reply to the examination report
30.11.2009Request for further processing filed
30.11.2009Full payment received (date of receipt of payment)
Fees paidRenewal fee
13.07.2007Renewal fee patent year 03
14.07.2008Renewal fee patent year 04
10.07.2009Renewal fee patent year 05
14.07.2010Renewal fee patent year 06
12.07.2011Renewal fee patent year 07
13.07.2012Renewal fee patent year 08
10.07.2013Renewal fee patent year 09
14.07.2014Renewal fee patent year 10
10.07.2015Renewal fee patent year 11
11.07.2016Renewal fee patent year 12
12.07.2017Renewal fee patent year 13
11.07.2018Renewal fee patent year 14
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Documents cited:Search[X]WO03016280  (LION BIOSCIENCE AG [DE], et al) [X] 1-124 * page 5; examples; claim 1 *;
 [A]WO03016288  (LION BIOSCIENCE AG [DE], et al) [A] 1-124 * examples; claims *; paragraph [0001] *;
 [A]WO03015777  (LION BIOSCIENCE AG [DE], et al) [A] 1-124* examples; claims *; paragraph [0001] *;
 [A]EP1398029  (LION BIOSCIENCE AG [DE]) [A] 1-124 * examples; claims *; paragraphs [0013] , [0014] *
International search[A]WO2004058249  (ASTRAZENECA AB [SE], et al);
 [AP]US2004267028  (SMITH ROGER A [US], et al)
ExaminationEP0022087
 WO9841527
 WO0009482
 EP1176140
    - H. Kamogawa ET AL, "Vinyl polymers bearing pyrrole ring: I. Syntheses of pyrroles having 3-substituent bearing vinyl group", Bulletin of the chemical society of Japan, (19910101), vol. 64, no. 3, pages 1066 - 1068, XP055086620

DOI:   http://dx.doi.org/10.1246/bcsj.64.1066
    - H. Jendralla ET AL, "Synthesis and biological activity of new HMG-CoA reductase inhibitors. 2. Derivatives of 7-(1H-pyrrol-3-yl)-substituted-3,5-dihydroxyhept-6(E)-enoic (-heptanoic) acids", Journal of Medicinal Chemistry, (19900101), vol. 33, no. 1, doi:10.1021/jm00163a011, ISSN 0022-2623, pages 61 - 70, XP055086421

DOI:   http://dx.doi.org/10.1021/jm00163a011
    - Paul A. Keifer ET AL, "Bioactive bromopyrrole metabolites from the Caribbean sponge Agelas conifera", The Journal of Organic Chemistry, (19910401), vol. 56, no. 9, doi:10.1021/jo00009a008, ISSN 0022-3263, pages 2965 - 2975, XP055086428

DOI:   http://dx.doi.org/10.1021/jo00009a008
    - Robert Moffett, "Central Nervous System Depressants. VIII. Pyroles.", Journal of Medicinal Chemistry, (19681101), vol. 11, no. 6, doi:10.1021/jm00312a604, ISSN 0022-2623, pages 1251 - 1252, XP055086598

DOI:   http://dx.doi.org/10.1021/jm00312a604
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.