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EP1881981
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EP About this file: EP1881981
| EP1881981 - 4, 6-DIAMINO-[1,7] NAPHTHYRIDINE-3-CARBONITRILE INHIBITORS OF TPL2 KINASE AND METHODS OF MAKING AND USING THE SAME [Right-click to bookmark this link] | Status | The application is deemed to be withdrawn Status updated on 27.04.2012 Database last updated on 17.08.2024 | Most recent event Tooltip | 27.04.2012 | Application deemed to be withdrawn | published on 30.05.2012 [2012/22] | Applicant(s) | For all designated states Wyeth LLC Five Giralda Farms Madison, NJ 07940 / US | [2010/16] |
| Former [2008/05] | For all designated states Wyeth Five Giralda Farms Madison, New Jersey 07940 / US | Inventor(s) | 01 /
GREEN, Neal, Jeffrey 51 Cotton Street Newton, Massachusetts 02458 / US | 02 /
GAVRIN, Lori, Krim 11 Knollwood Avenue Woburn, Massachusetts 01801 / US | 03 /
KAILA, Neelu 17 Augustus Road Lexington, Massachusetts 02421 / US | 04 /
HU, Yonghan 502 Tumbling Hawk Road Acton, Massachusetts 01718 / US | 05 /
JANZ, Kristin, Marie 35 Everett Street, Apt. 1 Arlington, Massachusetts 02474 / US | 06 /
THOMASON, Jennifer, R. 51 Broadway 2 Chelsea, Massachusetts 02150 / US | 07 /
GOPALSAMY, Ariamala 21 Whispering Pines Drive Mahwah, New Jersey 07430 / US | 08 /
TAM, Steve, Y. 88 Woodside Avenue Wellesley, Massachusetts 02482 / US | 09 /
LIN, Lih-Ling 107 College Road Concord, Massachusetts 01742 / US | 10 /
CUOZZO, John, William 106 Bacon Street Natick, Massachusetts 01760 / US | 11 /
POWELL, Dennis, William 50 Maple Moor Lane Cortlandt Manor, New York 10567 / US | [2008/05] | Representative(s) | Motion, Keith Robert, et al Pfizer ATTENTION: ADDRESS INACTIVE - USE ASS-NR - CDR / FR | [N/P] |
| Former [2010/32] | Motion, Keith Robert, et al Pfizer Limited European Patent Department Ramsgate Road Sandwich, Kent CT13 9NJ / GB | ||
| Former [2009/29] | Mannion, Sally Kim Wyeth Laboratories Huntercombe Lane South Taplow Maidenhead Berkshire SL6 0PH / GB | ||
| Former [2008/05] | Mannion, Sally Kim Wyeth Laboratories Patent & Trademarks Department Huntercombe Lane South Taplow, Maidenhead SL6 0PH / GB | Application number, filing date | 06759971.2 | 17.05.2006 | [2008/05] | WO2006US18996 | Priority number, date | US20050682044P | 18.05.2005 Original published format: US 682044 P | [2008/05] | Filing language | EN | Procedural language | EN | Publication | Type: | A1 Application with search report | No.: | WO2006124944 | Date: | 23.11.2006 | Language: | EN | [2006/47] | Type: | A1 Application with search report | No.: | EP1881981 | Date: | 30.01.2008 | Language: | EN | The application published by WIPO in one of the EPO official languages on 23.11.2006 takes the place of the publication of the European patent application. | [2008/05] | Search report(s) | International search report - published on: | EP | 23.11.2006 | Classification | IPC: | C07D471/04, A61K31/4375 | [2008/05] | CPC: |
C07D471/04 (EP,US);
A61P19/02 (EP);
A61P29/00 (EP);
A61P43/00 (EP);
Y02P20/582 (EP,US)
| Designated contracting states | AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LI, LT, LU, LV, MC, NL, PL, PT, RO, SE, SI, SK, TR [2008/05] | Extension states | AL | Not yet paid | BA | Not yet paid | HR | Not yet paid | MK | Not yet paid | YU | Not yet paid | Title | German: | 4,6-DIAMINO-[1,7] NAPHTHYRIDIN-3-CARBONITRIL-HEMMER DER TPL2-KINASE SOWIE HERSTELLUNGS- UND VERWENDUNGSVERFAHREN DAFÜR | [2008/05] | English: | 4, 6-DIAMINO-[1,7] NAPHTHYRIDINE-3-CARBONITRILE INHIBITORS OF TPL2 KINASE AND METHODS OF MAKING AND USING THE SAME | [2008/05] | French: | INHIBITEURS DE 4, 6-DIAMINO-[1,7] NAPHTHYRIDINE-3-CARBONITRILE DE LA TPL2 KINASE ET PROCEDES DE FABRICATION ET D'UTILISATION DE CEUX-CI | [2008/05] | Entry into regional phase | 05.11.2007 | National basic fee paid | 05.11.2007 | Designation fee(s) paid | 05.11.2007 | Examination fee paid | Examination procedure | 05.11.2007 | Examination requested [2008/05] | 01.12.2011 | Application deemed to be withdrawn, date of legal effect [2012/22] | 09.01.2012 | Despatch of communication that the application is deemed to be withdrawn, reason: renewal fee not paid in time [2012/22] | Fees paid | Renewal fee | 18.03.2008 | Renewal fee patent year 03 | 07.05.2009 | Renewal fee patent year 04 | 31.03.2010 | Renewal fee patent year 05 | Penalty fee | Additional fee for renewal fee | 31.05.2011 | 06 M06 Not yet paid |
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| Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Cited in | International search | [AX]WO0066583 (AMERICAN CYANAMID CO [US]) [A] 1-30,36 * examples 58,63; claims 1,16 * * examples 57,59,60,64,66-71,73-78,83 * [X] 37; | [AX] - A. WISSNER ET AL, "Synthesis and EGFR kinase inhibitory activity of 6-substituted -4-anilino [1,7] and [1,8] naphthyridine-3-carbonitriles", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, (2004), vol. 14, no. 6, pages 1411 - 1416, XP002399928 [A] 1-30 * page 1412, scheme 2, compound 26 * * page 1421, scheme 1, compounds 9a, 9b; scheme 2, compounds 23a, 23b, 24, 25, 27 * [X] 37 DOI: http://dx.doi.org/10.1016/j.bmcl.2004.01.034 | [PX] - GAVRIN ET AL, "Inhibition of Tpl2 kinase and TNF-alpha production with 1,7-naphthyridine-3-carbonitriles: Synthesis and structure-activity relationships", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, OXFORD, GB, (20051201), vol. 15, no. 23, ISSN 0960-894X, pages 5288 - 5292, XP005116293 [PX] 1,2,4-6,8,9,13-16,19,20,26-28,31-37 * scheme 1;;; tables 1,2 * DOI: http://dx.doi.org/10.1016/j.bmcl.2005.08.029 |