EP2029138 - AMINOTHIAZOLE DERIVATIVES AS HUMAN STEAROYL-COA DESATURASE INHIBITORS [Right-click to bookmark this link] | Status | The application is deemed to be withdrawn Status updated on 17.04.2015 Database last updated on 15.06.2024 | Most recent event Tooltip | 17.04.2015 | Application deemed to be withdrawn | published on 20.05.2015 [2015/21] | Applicant(s) | For all designated states Xenon Pharmaceuticals Inc. 3650 Gilmore Way Burnaby, BC V5G 4W8 / CA | [N/P] |
Former [2009/10] | For all designated states Xenon Pharmaceuticals Inc. 3650 Gilmore Way Burnaby, British Columbia V5G 4W8 / CA | Inventor(s) | 01 /
FU, Jianmin 3170 Quintette Crescent Coquitlam, British Columbia V3E 3B6 / CA | 02 /
HOU, Duanjie 46-7088 17th Avenue Burnaby, BC V3N 1K5 / CA | 03 /
KAMBOJ, Rajender 5809 Sperling Avenue Burnaby, British Columbia V5E 2T6 / CA | 04 /
KODUMURU, Vishnumurthy 7480 Vista Cres. Burnaby, British Columbia V5E 2E1 / CA | 05 /
POKROVSKAIA, Natalia 100-845 Mcbride Blvd New Westminster, BC V3L 2C2 / CA | 06 /
RAINA, Vandna 6654 Linden Avenue Burnaby, British Columbia V5E 3G4 / CA | 07 /
SUN, Shaoyi 5-1200 Brunette Avenue Coquitlam, British Columbia V3K 1G3 / CA | 08 /
SVIRIDOV, Serguei 1904-5885 Olive Avenue Burnaby, British Columbia V5H 4N8 / CA | 09 /
ZHANG, Zaihui 4038 MacDonald Street Vancouver, British Columbia V6L 2N9 / CA | [2009/10] | Representative(s) | Grünecker Patent- und Rechtsanwälte PartG mbB Leopoldstraße 4 80802 München / DE | [N/P] |
Former [2009/10] | Grünecker, Kinkeldey, Stockmair & Schwanhäusser Anwaltssozietät Leopoldstrasse 4 80802 München / DE | Application number, filing date | 06784578.4 | 05.06.2006 | [2009/10] | WO2006US21660 | Priority number, date | US20050687133P | 03.06.2005 Original published format: US 687133 P | [2012/42] |
Former [2009/10] | US20060687133P | 03.06.2006 | Filing language | EN | Procedural language | EN | Publication | Type: | A1 Application with search report | No.: | WO2007130075 | Date: | 15.11.2007 | Language: | EN | [2007/46] | Type: | A1 Application with search report | No.: | EP2029138 | Date: | 04.03.2009 | Language: | EN | The application published by WIPO in one of the EPO official languages on 15.11.2007 takes the place of the publication of the European patent application. | [2009/10] | Search report(s) | International search report - published on: | EP | 15.11.2007 | Classification | IPC: | A61K31/426, A61K31/427, A61K31/4439, A61P3/00, A61P9/12, A61P17/06, A61P17/10, A61P19/06, C07D277/82, C07D417/12 | [2009/10] | CPC: |
A61K31/426 (EP,US);
C07D277/587 (US);
A61K31/427 (EP,US);
A61K31/4439 (EP,US);
A61K31/5377 (US);
A61K31/616 (US);
A61K38/26 (US);
A61K38/28 (US);
A61K45/06 (US);
A61P1/16 (EP);
A61P17/00 (EP);
A61P17/02 (EP);
A61P17/06 (EP);
A61P17/08 (EP);
A61P17/10 (EP);
A61P19/06 (EP);
A61P3/00 (EP);
A61P3/04 (EP);
A61P3/06 (EP);
A61P3/10 (EP);
A61P35/00 (EP);
A61P43/00 (EP);
A61P7/02 (EP);
A61P9/10 (EP);
A61P9/12 (EP);
C07D277/56 (EP,US);
C07D417/06 (US);
C07D417/12 (EP,US)
(-)
| Designated contracting states | AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LI, LT, LU, LV, MC, NL, PL, PT, RO, SE, SI, SK, TR [2009/10] | Title | German: | AMINOTHIAZOLDERIVATE ALS HUMANE STEAROYL-COA DESATURASEHEMMER | [2009/10] | English: | AMINOTHIAZOLE DERIVATIVES AS HUMAN STEAROYL-COA DESATURASE INHIBITORS | [2009/10] | French: | DERIVES AMINOTHIAZOLE UTILISES EN TANT QU'INHIBITEURS DE LA STEAROYLE-COA DESATURASE HUMAINE | [2009/10] | Entry into regional phase | 28.12.2007 | National basic fee paid | 28.12.2007 | Designation fee(s) paid | 28.12.2007 | Examination fee paid | Examination procedure | 28.12.2007 | Examination requested [2009/10] | 13.08.2010 | Despatch of a communication from the examining division (Time limit: M06) | 31.01.2011 | Reply to a communication from the examining division | 21.07.2014 | Despatch of a communication from the examining division (Time limit: M04) | 02.12.2014 | Application deemed to be withdrawn, date of legal effect [2015/21] | 14.01.2015 | Despatch of communication that the application is deemed to be withdrawn, reason: reply to the communication from the examining division not received in time [2015/21] | Divisional application(s) | EP12005821.9 / EP2540296 | The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is 13.08.2010 | Fees paid | Renewal fee | 25.06.2008 | Renewal fee patent year 03 | 26.06.2009 | Renewal fee patent year 04 | 25.06.2010 | Renewal fee patent year 05 | 27.06.2011 | Renewal fee patent year 06 | 26.06.2012 | Renewal fee patent year 07 | 27.06.2013 | Renewal fee patent year 08 | Penalty fee | Additional fee for renewal fee | 30.06.2014 | 09   M06   Not yet paid |
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Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Cited in | International search | [DA]WO2005011655 (XENON PHARMACEUTICALS INC [CA], et al) [DA] 1-24* Page 144, lines 16-17,; page 1, line 3 - line 8 *; | [X] - WITYAK, JOHN ET AL, "Discovery and initial SAR of 2-amino-5-carboxamidothiazoles as inhibitors of the Src-family kinase p56Lck", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS , 13(22), 4007-4010 CODEN: BMCLE8; ISSN: 0960-894X, (2003), XP002402709 [X] 11,21,23 * the whole document * DOI: http://dx.doi.org/10.1016/j.bmcl.2003.08.054 | [X] - OHKUBO, MITSURU ET AL, "Studies on cerebral protective agents. VIII. Synthesis of 2-aminothiazoles and 2-thiazolecarboxamides with anti-anoxic activity", CAPLUS, CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US, Database accession no. 1995:902192, URL: STN, XP002402712 [X] 11,21,23 * the whole document * | [X] - SINGH, S. N. ET AL, "New local anesthetics", CA, CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US, Database accession no. 1972:564589, URL: STN, XP002402713 [X] 11,21,23 * the whole document * | Examination | EP0518731 | US6114365 | WO0250071 | WO2004112782 | EP1244641 | - HELAL C J ET AL, "Discovery and SAR of 2-aminothiazole inhibitors of cyclin-dependent kinase 5/p25 as a potential treatment for Alzheimer's disease", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, PERGAMON, AMSTERDAM, NL, (20041115), vol. 14, no. 22, doi:10.1016/J.BMCL.2004.09.006, ISSN 0960-894X, pages 5521 - 5525, XP004598586 DOI: http://dx.doi.org/10.1016/j.bmcl.2004.09.006 | - MISRA RAJ N ET AL, "N-(cycloalkylamino)acyl-2-aminothiazole inhibitors of cyclin-dependent kinase 2. N-[5-[[[5-(1,1-dimethylethyl)-2-oxazolyl]methyl]thio]-2-thi azolyl]-4- piperidinecarboxamide (BMS-387032), a highly efficacious and selective antitumor agent", JOURNAL OF MEDICINAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY, US, (20040325), vol. 47, no. 7, doi:10.1021/JM0305568, ISSN 0022-2623, pages 1719 - 1728, XP002302339 DOI: http://dx.doi.org/10.1021/jm0305568 | - KIM KYOUNG SOON ET AL, "DISCOVERY OF AMINOTHIAZOLE INHIBITORS OF CYCLIN-DEPENDENT KINASE 2: SYNTHESIS, X-RAY CRYSTALLOGRAPHIC ANALYSIS, AND BIOLOGICAL ACTIVITIES", JOURNAL OF MEDICINAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY, US, (20020101), vol. 45, no. 18, doi:10.1021/JM0201520, ISSN 0022-2623, pages 3905 - 3927, XP009073889 DOI: http://dx.doi.org/10.1021/jm0201520 |