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Extract from the Register of European Patents

EP About this file: EP1934198

EP1934198 - POLYMORPHS OF BENZOATE SALT OF 2-[[6-[(3R)-3-AMINO-1-PIPERIDINYL]-3,4-DIHYDRO-3-METHYL-2,4-DIOXO-1(2H)-PYRIMIDINYL]METHYL]-BENZONITRILE AND METHODS OF USE THEREFOR [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  08.06.2012
Database last updated on 19.10.2024
Most recent event   Tooltip04.10.2013Lapse of the patent in a contracting state
New state(s): HU		published on 06.11.2013  [2013/45]
Applicant(s)For all designated states
Takeda Pharmaceutical Company Limited
1-1, Doshomachi 4-chome Chuo-ku Osaka-shi
Osaka 541-0045 / JP
[2008/26]
Inventor(s)01 / ANDRES, Mark
2307 Sycamore Lane
West Lafayette, IN 47906 / US
02 / LORIMER, Keith
2109 Wake Robin Drive
West Lafayette, IN 47906 / US
 [2008/26]
Representative(s)Duncan, Garreth Andrew, et al
D Young & Co LLP
120 Holborn
London EC1N 2DY / GB
[N/P]
Former [2008/26]Duncan, Garreth Andrew, et al
D Young & Co 120 Holborn London
EC1N 2DY / GB
Application number, filing date06803516.113.09.2006
[2008/26]
WO2006US35701
Priority number, dateUS20050718133P16.09.2005         Original published format: US 718133 P
[2008/26]
Filing languageEN
Procedural languageEN
PublicationType: A2 Application without search report
No.:WO2007035372
Date:29.03.2007
Language:EN
[2007/13]
Type: A2 Application without search report 
No.:EP1934198
Date:25.06.2008
Language:EN
The application published by WIPO in one of the EPO official languages on 29.03.2007 takes the place of the publication of the European patent application.
[2008/26]
Type: B1 Patent specification 
No.:EP1934198
Date:03.08.2011
Language:EN
[2011/31]
Search report(s)International search report - published on:EP14.06.2007
ClassificationIPC:C07D401/04, A61P3/04, A61K31/513
[2008/26]
CPC:
A61K31/513 (EP,KR,US); C07D401/04 (EP,KR,US); A61P1/04 (EP);
A61P1/14 (EP); A61P15/08 (EP); A61P15/16 (EP);
A61P17/00 (EP); A61P17/06 (EP); A61P19/02 (EP);
A61P19/10 (EP); A61P25/00 (EP); A61P29/00 (EP);
A61P3/00 (EP); A61P3/04 (EP); A61P3/06 (EP);
A61P3/10 (EP); A61P31/18 (EP); A61P35/00 (EP);
A61P35/04 (EP); A61P37/04 (EP); A61P37/06 (EP);
A61P43/00 (EP) (-)
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   NL,   PL,   PT,   RO,   SE,   SI,   SK,   TR [2008/26]
Extension statesAL28.03.2008
BA28.03.2008
HR28.03.2008
MK28.03.2008
RS28.03.2008
TitleGerman:POLYMORPHE DES BENZOATSALZES VON 2-[[6-[(3R)-3-AMINO-1-PIPERIDINYL]-3,4-DIHYDRO-3-METHYL-2,4-DIOXO-1(2H)-PYRIMIDINYL]METHYL]-BENZONITRIL UND VERWENDUNGSVERFAHREN DAFÜR[2008/26]
English:POLYMORPHS OF BENZOATE SALT OF 2-[[6-[(3R)-3-AMINO-1-PIPERIDINYL]-3,4-DIHYDRO-3-METHYL-2,4-DIOXO-1(2H)-PYRIMIDINYL]METHYL]-BENZONITRILE AND METHODS OF USE THEREFOR[2008/26]
French:FORMES POLYMORPHES DE SEL BENZOATE DE 2-[[6-[(3R)-3-AMINO-1-PIPERIDINYL]-3,4-DIHYDRO-3-METHYL-2,4-DIOXO-1(2H)-PYRIMIDINYL]METHYL]-BENZONITRILE, ET LEURS PROCEDES D'UTILISATION[2008/26]
Entry into regional phase28.03.2008National basic fee paid 
28.03.2008Designation fee(s) paid 
28.03.2008Examination fee paid 
Examination procedure28.03.2008Examination requested  [2008/26]
19.08.2008Despatch of a communication from the examining division (Time limit: M04)
15.12.2008Reply to a communication from the examining division
15.01.2009Despatch of a communication from the examining division (Time limit: M04)
12.05.2009Reply to a communication from the examining division
29.06.2009Despatch of a communication from the examining division (Time limit: M04)
23.10.2009Reply to a communication from the examining division
17.02.2011Communication of intention to grant the patent
17.06.2011Fee for grant paid
17.06.2011Fee for publishing/printing paid
Divisional application(s)The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is  19.08.2008
Opposition(s)04.05.2012No opposition filed within time limit [2012/28]
Fees paidRenewal fee
25.09.2008Renewal fee patent year 03
25.09.2009Renewal fee patent year 04
27.09.2010Renewal fee patent year 05
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court		 See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipAT03.08.2011
BE03.08.2011
CY03.08.2011
CZ03.08.2011
DK03.08.2011
EE03.08.2011
FI03.08.2011
HU03.08.2011
LT03.08.2011
LV03.08.2011
NL03.08.2011
PL03.08.2011
RO03.08.2011
SE03.08.2011
SI03.08.2011
SK03.08.2011
TR03.08.2011
IE13.09.2011
LU13.09.2011
MC30.09.2011
BG03.11.2011
GR04.11.2011
ES14.11.2011
IS03.12.2011
PT05.12.2011
[2013/45]
Former [2013/44]AT03.08.2011
BE03.08.2011
CY03.08.2011
CZ03.08.2011
DK03.08.2011
EE03.08.2011
FI03.08.2011
LT03.08.2011
LV03.08.2011
NL03.08.2011
PL03.08.2011
RO03.08.2011
SE03.08.2011
SI03.08.2011
SK03.08.2011
TR03.08.2011
IE13.09.2011
LU13.09.2011
MC30.09.2011
BG03.11.2011
GR04.11.2011
ES14.11.2011
IS03.12.2011
PT05.12.2011
Former [2013/29]AT03.08.2011
BE03.08.2011
CY03.08.2011
CZ03.08.2011
DK03.08.2011
EE03.08.2011
FI03.08.2011
LT03.08.2011
LV03.08.2011
NL03.08.2011
PL03.08.2011
RO03.08.2011
SE03.08.2011
SI03.08.2011
SK03.08.2011
IE13.09.2011
LU13.09.2011
MC30.09.2011
BG03.11.2011
GR04.11.2011
ES14.11.2011
IS03.12.2011
PT05.12.2011
Former [2013/25]AT03.08.2011
BE03.08.2011
CY03.08.2011
CZ03.08.2011
DK03.08.2011
EE03.08.2011
FI03.08.2011
LT03.08.2011
LV03.08.2011
NL03.08.2011
PL03.08.2011
RO03.08.2011
SE03.08.2011
SI03.08.2011
SK03.08.2011
IE13.09.2011
LU13.09.2011
MC30.09.2011
GR04.11.2011
ES14.11.2011
IS03.12.2011
PT05.12.2011
Former [2013/22]AT03.08.2011
BE03.08.2011
CY03.08.2011
CZ03.08.2011
DK03.08.2011
EE03.08.2011
FI03.08.2011
LT03.08.2011
LV03.08.2011
NL03.08.2011
PL03.08.2011
RO03.08.2011
SE03.08.2011
SI03.08.2011
SK03.08.2011
IE13.09.2011
MC30.09.2011
GR04.11.2011
ES14.11.2011
IS03.12.2011
PT05.12.2011
Former [2012/35]AT03.08.2011
BE03.08.2011
CY03.08.2011
CZ03.08.2011
DK03.08.2011
EE03.08.2011
FI03.08.2011
LT03.08.2011
LV03.08.2011
NL03.08.2011
PL03.08.2011
RO03.08.2011
SE03.08.2011
SI03.08.2011
SK03.08.2011
IE13.09.2011
MC30.09.2011
GR04.11.2011
IS03.12.2011
PT05.12.2011
Former [2012/33]AT03.08.2011
BE03.08.2011
CY03.08.2011
CZ03.08.2011
DK03.08.2011
EE03.08.2011
FI03.08.2011
LT03.08.2011
LV03.08.2011
NL03.08.2011
PL03.08.2011
RO03.08.2011
SE03.08.2011
SI03.08.2011
SK03.08.2011
MC30.09.2011
GR04.11.2011
IS03.12.2011
PT05.12.2011
Former [2012/23]AT03.08.2011
BE03.08.2011
CY03.08.2011
CZ03.08.2011
EE03.08.2011
FI03.08.2011
LT03.08.2011
LV03.08.2011
NL03.08.2011
PL03.08.2011
RO03.08.2011
SE03.08.2011
SI03.08.2011
SK03.08.2011
MC30.09.2011
GR04.11.2011
IS03.12.2011
PT05.12.2011
Former [2012/21]AT03.08.2011
BE03.08.2011
CY03.08.2011
CZ03.08.2011
FI03.08.2011
LT03.08.2011
LV03.08.2011
NL03.08.2011
PL03.08.2011
SE03.08.2011
SI03.08.2011
MC30.09.2011
GR04.11.2011
IS03.12.2011
PT05.12.2011
Former [2012/20]AT03.08.2011
BE03.08.2011
CY03.08.2011
FI03.08.2011
LT03.08.2011
LV03.08.2011
NL03.08.2011
PL03.08.2011
SE03.08.2011
SI03.08.2011
MC30.09.2011
GR04.11.2011
IS03.12.2011
PT05.12.2011
Former [2012/17]AT03.08.2011
BE03.08.2011
CY03.08.2011
FI03.08.2011
LT03.08.2011
LV03.08.2011
NL03.08.2011
PL03.08.2011
SE03.08.2011
SI03.08.2011
GR04.11.2011
IS03.12.2011
PT05.12.2011
Former [2012/12]AT03.08.2011
CY03.08.2011
FI03.08.2011
LT03.08.2011
LV03.08.2011
NL03.08.2011
PL03.08.2011
SE03.08.2011
SI03.08.2011
GR04.11.2011
IS03.12.2011
PT05.12.2011
Former [2012/11]AT03.08.2011
FI03.08.2011
LT03.08.2011
LV03.08.2011
NL03.08.2011
PL03.08.2011
SE03.08.2011
SI03.08.2011
GR04.11.2011
IS03.12.2011
PT05.12.2011
Former [2012/09]FI03.08.2011
LT03.08.2011
NL03.08.2011
IS03.12.2011
PT05.12.2011
Former [2012/08]LT03.08.2011
NL03.08.2011
IS03.12.2011
Cited inInternational search[A]US2005070535  (FENG JUN [US], et al) [A] 1-60 * the whole document *;
 [PX]WO2005095381  (SYRRX INC [US], et al) [PX] 1-60 * page 96 *;
 [A]  - CAIRA M R, "CRYSTALLINE POLYMORPHISM OF ORGANIC COMPOUNDS", TOPICS IN CURRENT CHEMISTRY, SPRINGER, BERLIN, DE, (1998), vol. 198, ISSN 0340-1022, pages 163 - 208, XP001156954 [A] 1-60 * the whole document *

DOI:   http://dx.doi.org/10.1007/3-540-69178-2_5
ExaminationEP1586571
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.