EP2041119 - PYRAZOLYLBENZIMIDAZOLE DERIVATIVES, COMPOSITIONS CONTAINING THEM AND USE THEREOF [Right-click to bookmark this link] | Status | No opposition filed within time limit Status updated on 16.03.2018 Database last updated on 26.06.2024 | |
Former | The patent has been granted Status updated on 07.04.2017 | ||
Former | Grant of patent is intended Status updated on 03.04.2017 | ||
Former | Examination is in progress Status updated on 22.03.2017 | ||
Former | Grant of patent is intended Status updated on 27.11.2016 | Most recent event Tooltip | 29.05.2020 | Lapse of the patent in a contracting state New state(s): PT | published on 01.07.2020 [2020/27] | Applicant(s) | For all designated states Aventis Pharma S.A. 20, avenue Raymond Aron 92160 Antony / FR | [2009/14] | Inventor(s) | 01 /
CHERRIER, Marie-Pierre Sanofi-Aventis Département Brevets tri E2/300 20 avenue Raymond Aron 92160 Antony / FR | 02 /
PARMANTIER, Eric Sanofi-Aventis Département Brevets tri E2/300 20 avenue Raymond Aron 92160 Antony / FR | 03 /
MINOUX, Hervé Sanofi-Aventis Département Brevets tri E2/300 20 avenue Raymond Aron 92160 Antony / FR | 04 /
CLERC, François Sanofi-Aventis Département Brevets tri E2/300 20 avenue Raymond Aron 92160 Antony / FR | 05 /
ANGOUILLANT-BONIFACE, Odile Sanofi-Aventis Département Brevets tri E2/300 20 avenue Raymond Aron 92160 Antony / FR | 06 /
BROLLO, Maurice Sanofi-Aventis Département Brevets tri E2/300 20 avenue Raymond Aron 92160 Antony / FR | 07 /
SCHIO, Laurent Sanofi-Aventis Département Brevets tri E2/300 20 avenue Raymond Aron 92160 Antony / FR | [2017/19] |
Former [2009/14] | 01 /
CHERRIER, Marie-Pierre Sanofi-Aventis Département Brevets tri E2/300 20 avenue Raymond Aron 92160 Antony / FR | ||
02 /
PARMANTIER, Eric Sanofi-Aventis Département Brevets tri E2/300 20 avenue Raymond Aron 92160 Antony / FR | |||
03 /
MINOUX, Hervé Sanofi-Aventis Département Brevets tri E2/300 20 avenue Raymond Aron 92160 Antony / FR | |||
04 /
CLERC, François Sanofi-Aventis Département Brevets tri E2/300 20 avenue Raymond Aron 92160 Antony / FR | |||
05 /
ANGOUILLANT-BONIFACE, Odile Sanofi-Aventis Département Brevets tri E2/300 20 avenue Raymond Aron 92160 Antony / FR | |||
06 /
BROLLO, Maurice Sanofi-Aventis Département Brevets tri E2/300 20 avenue Raymond Aron 92160 Antony / FR | |||
07 /
SCHIO, Laurent Sanofi-Aventis Département Brevets tri E2/300 20 avenue Raymond Aron 92160 Antony / FR | Representative(s) | Lavoix 2, place d'Estienne d'Orves 75441 Paris Cedex 09 / FR | [2017/19] |
Former [2011/15] | Lavé, Stéphanie, et al Cabinet Lavoix 2, Place d'Estienne d'Orves 75441 Paris Cedex 09 / FR | ||
Former [2009/14] | Le Pennec, Magali, et al Sanofi-Aventis 20 Avenue Raymond Aron 92165 Antony Cedex / FR | Application number, filing date | 07803834.6 | 03.07.2007 | [2009/14] | WO2007FR01126 | Priority number, date | FR20060006064 | 04.07.2006 Original published format: FR 0606064 | [2009/14] | Filing language | FR | Procedural language | FR | Publication | Type: | A1 Application with search report | No.: | WO2008003857 | Date: | 10.01.2008 | Language: | FR | [2008/02] | Type: | A1 Application with search report | No.: | EP2041119 | Date: | 01.04.2009 | Language: | FR | The application published by WIPO in one of the EPO official languages on 10.01.2008 takes the place of the publication of the European patent application. | [2009/14] | Type: | B1 Patent specification | No.: | EP2041119 | Date: | 10.05.2017 | Language: | FR | [2017/19] | Search report(s) | International search report - published on: | EP | 10.01.2008 | Classification | IPC: | C07D403/04, C07D413/14, C07D403/14, C07D405/14, A61K31/551, A61K31/4184, A61K31/5377, A61K31/496, A61P35/00 | [2009/14] | CPC: |
C07D403/04 (EP,US);
A61P1/04 (EP);
A61P1/16 (EP);
A61P1/18 (EP);
A61P11/00 (EP);
A61P11/04 (EP);
A61P13/02 (EP);
A61P13/08 (EP);
A61P13/10 (EP);
A61P13/12 (EP);
A61P15/00 (EP);
A61P15/08 (EP);
A61P15/14 (EP);
A61P17/00 (EP);
A61P17/06 (EP);
A61P19/00 (EP);
A61P25/00 (EP);
A61P27/02 (EP);
A61P27/06 (EP);
A61P29/00 (EP);
A61P35/00 (EP);
A61P35/02 (EP);
A61P43/00 (EP);
A61P5/00 (EP);
A61P5/10 (EP);
A61P5/14 (EP);
A61P5/38 (EP);
A61P9/00 (EP);
C07D235/04 (EP,US);
C07D401/14 (EP,US);
| Designated contracting states | AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MT, NL, PL, PT, RO, SE, SI, SK, TR [2017/19] |
Former [2009/14] | AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MT, NL, PL, PT, RO, SE, SI, SK, TR | Extension states | AL | 04.02.2009 | BA | 04.02.2009 | HR | 04.02.2009 | MK | 04.02.2009 | RS | 04.02.2009 | Title | German: | PYRAZOLYLBENZIMIDAZOLDERIVATE, DIESE ENTHALTENDE ZUSAMMENSETZUNGEN UND IHRE VERWENDUNG | [2009/14] | English: | PYRAZOLYLBENZIMIDAZOLE DERIVATIVES, COMPOSITIONS CONTAINING THEM AND USE THEREOF | [2009/14] | French: | DERIVES DE PYRAZOLYLBENZIMIDAZOLE, COMPOSITIONS LES CONTENANT ET LEUR UTILISATION | [2009/14] | Entry into regional phase | 04.02.2009 | National basic fee paid | 04.02.2009 | Designation fee(s) paid | 04.02.2009 | Examination fee paid | Examination procedure | 05.05.2008 | Request for preliminary examination filed International Preliminary Examining Authority: EP | 04.02.2009 | Examination requested [2009/14] | 12.07.2010 | Despatch of a communication from the examining division (Time limit: M06) | 14.01.2011 | Reply to a communication from the examining division | 13.03.2012 | Despatch of a communication from the examining division (Time limit: M04) | 10.07.2012 | Reply to a communication from the examining division | 24.02.2014 | Despatch of a communication from the examining division (Time limit: M04) | 23.06.2014 | Reply to a communication from the examining division | 24.06.2015 | Despatch of a communication from the examining division (Time limit: M04) | 04.09.2015 | Reply to a communication from the examining division | 04.03.2016 | Despatch of a communication from the examining division (Time limit: M04) | 15.04.2016 | Reply to a communication from the examining division | 28.11.2016 | Communication of intention to grant the patent | 16.03.2017 | Disapproval of the communication of intention to grant the patent by the applicant or resumption of examination proceedings by the EPO | 16.03.2017 | Fee for grant paid | 16.03.2017 | Fee for publishing/printing paid | 03.04.2017 | Information about intention to grant a patent | 03.04.2017 | Receipt of the translation of the claim(s) | Divisional application(s) | The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is 12.07.2010 | Opposition(s) | 13.02.2018 | No opposition filed within time limit [2018/16] | Fees paid | Renewal fee | 10.07.2009 | Renewal fee patent year 03 | 14.07.2010 | Renewal fee patent year 04 | 12.07.2011 | Renewal fee patent year 05 | 13.07.2012 | Renewal fee patent year 06 | 10.07.2013 | Renewal fee patent year 07 | 14.07.2014 | Renewal fee patent year 08 | 10.07.2015 | Renewal fee patent year 09 | 11.07.2016 | Renewal fee patent year 10 |
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Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Lapses during opposition Tooltip | HU | 03.07.2007 | AT | 10.05.2017 | CY | 10.05.2017 | CZ | 10.05.2017 | DK | 10.05.2017 | EE | 10.05.2017 | ES | 10.05.2017 | FI | 10.05.2017 | IT | 10.05.2017 | LT | 10.05.2017 | LV | 10.05.2017 | MC | 10.05.2017 | MT | 10.05.2017 | NL | 10.05.2017 | PL | 10.05.2017 | PT | 10.05.2017 | RO | 10.05.2017 | SE | 10.05.2017 | SI | 10.05.2017 | SK | 10.05.2017 | TR | 10.05.2017 | IE | 03.07.2017 | LU | 03.07.2017 | BE | 31.07.2017 | CH | 31.07.2017 | LI | 31.07.2017 | BG | 10.08.2017 | GR | 11.08.2017 | IS | 10.09.2017 | [2020/27] |
Former [2020/15] | HU | 03.07.2007 | |
AT | 10.05.2017 | ||
CY | 10.05.2017 | ||
CZ | 10.05.2017 | ||
DK | 10.05.2017 | ||
EE | 10.05.2017 | ||
ES | 10.05.2017 | ||
FI | 10.05.2017 | ||
IT | 10.05.2017 | ||
LT | 10.05.2017 | ||
LV | 10.05.2017 | ||
MC | 10.05.2017 | ||
MT | 10.05.2017 | ||
NL | 10.05.2017 | ||
PL | 10.05.2017 | ||
RO | 10.05.2017 | ||
SE | 10.05.2017 | ||
SI | 10.05.2017 | ||
SK | 10.05.2017 | ||
TR | 10.05.2017 | ||
IE | 03.07.2017 | ||
LU | 03.07.2017 | ||
BE | 31.07.2017 | ||
CH | 31.07.2017 | ||
LI | 31.07.2017 | ||
BG | 10.08.2017 | ||
GR | 11.08.2017 | ||
IS | 10.09.2017 | ||
Former [2019/46] | HU | 03.07.2007 | |
AT | 10.05.2017 | ||
CY | 10.05.2017 | ||
CZ | 10.05.2017 | ||
DK | 10.05.2017 | ||
EE | 10.05.2017 | ||
ES | 10.05.2017 | ||
FI | 10.05.2017 | ||
IT | 10.05.2017 | ||
LT | 10.05.2017 | ||
LV | 10.05.2017 | ||
MC | 10.05.2017 | ||
MT | 10.05.2017 | ||
NL | 10.05.2017 | ||
PL | 10.05.2017 | ||
RO | 10.05.2017 | ||
SE | 10.05.2017 | ||
SI | 10.05.2017 | ||
SK | 10.05.2017 | ||
IE | 03.07.2017 | ||
LU | 03.07.2017 | ||
BE | 31.07.2017 | ||
CH | 31.07.2017 | ||
LI | 31.07.2017 | ||
BG | 10.08.2017 | ||
GR | 11.08.2017 | ||
IS | 10.09.2017 | ||
Former [2019/31] | HU | 03.07.2007 | |
AT | 10.05.2017 | ||
CZ | 10.05.2017 | ||
DK | 10.05.2017 | ||
EE | 10.05.2017 | ||
ES | 10.05.2017 | ||
FI | 10.05.2017 | ||
IT | 10.05.2017 | ||
LT | 10.05.2017 | ||
LV | 10.05.2017 | ||
MC | 10.05.2017 | ||
MT | 10.05.2017 | ||
NL | 10.05.2017 | ||
PL | 10.05.2017 | ||
RO | 10.05.2017 | ||
SE | 10.05.2017 | ||
SI | 10.05.2017 | ||
SK | 10.05.2017 | ||
IE | 03.07.2017 | ||
LU | 03.07.2017 | ||
BE | 31.07.2017 | ||
CH | 31.07.2017 | ||
LI | 31.07.2017 | ||
BG | 10.08.2017 | ||
GR | 11.08.2017 | ||
IS | 10.09.2017 | ||
Former [2019/30] | AT | 10.05.2017 | |
CZ | 10.05.2017 | ||
DK | 10.05.2017 | ||
EE | 10.05.2017 | ||
ES | 10.05.2017 | ||
FI | 10.05.2017 | ||
IT | 10.05.2017 | ||
LT | 10.05.2017 | ||
LV | 10.05.2017 | ||
MC | 10.05.2017 | ||
MT | 10.05.2017 | ||
NL | 10.05.2017 | ||
PL | 10.05.2017 | ||
RO | 10.05.2017 | ||
SE | 10.05.2017 | ||
SI | 10.05.2017 | ||
SK | 10.05.2017 | ||
IE | 03.07.2017 | ||
LU | 03.07.2017 | ||
BE | 31.07.2017 | ||
CH | 31.07.2017 | ||
LI | 31.07.2017 | ||
BG | 10.08.2017 | ||
GR | 11.08.2017 | ||
IS | 10.09.2017 | ||
Former [2018/43] | AT | 10.05.2017 | |
CZ | 10.05.2017 | ||
DK | 10.05.2017 | ||
EE | 10.05.2017 | ||
ES | 10.05.2017 | ||
FI | 10.05.2017 | ||
IT | 10.05.2017 | ||
LT | 10.05.2017 | ||
LV | 10.05.2017 | ||
MT | 10.05.2017 | ||
NL | 10.05.2017 | ||
PL | 10.05.2017 | ||
RO | 10.05.2017 | ||
SE | 10.05.2017 | ||
SI | 10.05.2017 | ||
SK | 10.05.2017 | ||
IE | 03.07.2017 | ||
LU | 03.07.2017 | ||
BE | 31.07.2017 | ||
CH | 31.07.2017 | ||
LI | 31.07.2017 | ||
BG | 10.08.2017 | ||
GR | 11.08.2017 | ||
IS | 10.09.2017 | ||
Former [2018/39] | AT | 10.05.2017 | |
CZ | 10.05.2017 | ||
DK | 10.05.2017 | ||
EE | 10.05.2017 | ||
ES | 10.05.2017 | ||
FI | 10.05.2017 | ||
IT | 10.05.2017 | ||
LT | 10.05.2017 | ||
LV | 10.05.2017 | ||
NL | 10.05.2017 | ||
PL | 10.05.2017 | ||
RO | 10.05.2017 | ||
SE | 10.05.2017 | ||
SI | 10.05.2017 | ||
SK | 10.05.2017 | ||
IE | 03.07.2017 | ||
LU | 03.07.2017 | ||
BE | 31.07.2017 | ||
CH | 31.07.2017 | ||
LI | 31.07.2017 | ||
BG | 10.08.2017 | ||
GR | 11.08.2017 | ||
IS | 10.09.2017 | ||
Former [2018/34] | AT | 10.05.2017 | |
CZ | 10.05.2017 | ||
DK | 10.05.2017 | ||
EE | 10.05.2017 | ||
ES | 10.05.2017 | ||
FI | 10.05.2017 | ||
IT | 10.05.2017 | ||
LT | 10.05.2017 | ||
LV | 10.05.2017 | ||
NL | 10.05.2017 | ||
PL | 10.05.2017 | ||
RO | 10.05.2017 | ||
SE | 10.05.2017 | ||
SI | 10.05.2017 | ||
SK | 10.05.2017 | ||
IE | 03.07.2017 | ||
LU | 03.07.2017 | ||
CH | 31.07.2017 | ||
LI | 31.07.2017 | ||
BG | 10.08.2017 | ||
GR | 11.08.2017 | ||
IS | 10.09.2017 | ||
Former [2018/23] | AT | 10.05.2017 | |
CZ | 10.05.2017 | ||
DK | 10.05.2017 | ||
EE | 10.05.2017 | ||
ES | 10.05.2017 | ||
FI | 10.05.2017 | ||
IT | 10.05.2017 | ||
LT | 10.05.2017 | ||
LV | 10.05.2017 | ||
NL | 10.05.2017 | ||
PL | 10.05.2017 | ||
RO | 10.05.2017 | ||
SE | 10.05.2017 | ||
SI | 10.05.2017 | ||
SK | 10.05.2017 | ||
IE | 03.07.2017 | ||
CH | 31.07.2017 | ||
LI | 31.07.2017 | ||
BG | 10.08.2017 | ||
GR | 11.08.2017 | ||
IS | 10.09.2017 | ||
Former [2018/21] | AT | 10.05.2017 | |
CZ | 10.05.2017 | ||
DK | 10.05.2017 | ||
EE | 10.05.2017 | ||
ES | 10.05.2017 | ||
FI | 10.05.2017 | ||
IT | 10.05.2017 | ||
LT | 10.05.2017 | ||
LV | 10.05.2017 | ||
NL | 10.05.2017 | ||
PL | 10.05.2017 | ||
RO | 10.05.2017 | ||
SE | 10.05.2017 | ||
SK | 10.05.2017 | ||
CH | 31.07.2017 | ||
LI | 31.07.2017 | ||
BG | 10.08.2017 | ||
GR | 11.08.2017 | ||
IS | 10.09.2017 | ||
Former [2018/11] | AT | 10.05.2017 | |
CZ | 10.05.2017 | ||
DK | 10.05.2017 | ||
EE | 10.05.2017 | ||
ES | 10.05.2017 | ||
FI | 10.05.2017 | ||
IT | 10.05.2017 | ||
LT | 10.05.2017 | ||
LV | 10.05.2017 | ||
NL | 10.05.2017 | ||
PL | 10.05.2017 | ||
RO | 10.05.2017 | ||
SE | 10.05.2017 | ||
SK | 10.05.2017 | ||
BG | 10.08.2017 | ||
GR | 11.08.2017 | ||
IS | 10.09.2017 | ||
Former [2018/10] | AT | 10.05.2017 | |
CZ | 10.05.2017 | ||
DK | 10.05.2017 | ||
EE | 10.05.2017 | ||
ES | 10.05.2017 | ||
FI | 10.05.2017 | ||
LT | 10.05.2017 | ||
LV | 10.05.2017 | ||
NL | 10.05.2017 | ||
PL | 10.05.2017 | ||
RO | 10.05.2017 | ||
SE | 10.05.2017 | ||
SK | 10.05.2017 | ||
BG | 10.08.2017 | ||
GR | 11.08.2017 | ||
IS | 10.09.2017 | ||
Former [2018/09] | AT | 10.05.2017 | |
DK | 10.05.2017 | ||
EE | 10.05.2017 | ||
ES | 10.05.2017 | ||
FI | 10.05.2017 | ||
LT | 10.05.2017 | ||
LV | 10.05.2017 | ||
NL | 10.05.2017 | ||
PL | 10.05.2017 | ||
SE | 10.05.2017 | ||
BG | 10.08.2017 | ||
GR | 11.08.2017 | ||
IS | 10.09.2017 | ||
Former [2017/52] | AT | 10.05.2017 | |
ES | 10.05.2017 | ||
FI | 10.05.2017 | ||
LT | 10.05.2017 | ||
LV | 10.05.2017 | ||
NL | 10.05.2017 | ||
PL | 10.05.2017 | ||
SE | 10.05.2017 | ||
BG | 10.08.2017 | ||
GR | 11.08.2017 | ||
IS | 10.09.2017 | ||
Former [2017/50] | AT | 10.05.2017 | |
ES | 10.05.2017 | ||
FI | 10.05.2017 | ||
LT | 10.05.2017 | ||
LV | 10.05.2017 | ||
PL | 10.05.2017 | ||
SE | 10.05.2017 | ||
BG | 10.08.2017 | ||
GR | 11.08.2017 | ||
IS | 10.09.2017 | ||
Former [2017/49] | AT | 10.05.2017 | |
ES | 10.05.2017 | ||
FI | 10.05.2017 | ||
LT | 10.05.2017 | ||
GR | 11.08.2017 | ||
IS | 10.09.2017 | Cited in | International search | [DX]WO2005002552 (ASTEX TECHNOLOGY LTD [GB], et al) [DX] 1-30 * claim 1 * * page 158; examples 87,88 *; | [DX]WO03035065 (AVENTIS PHARMA INC [US], et al) [DX] 1-30 * claim 1 * * page 446 - page 448; examples 257-c,257-d,257-e,257-h,257-i * * page 450 - page 452; examples 258-d,258-e,258-h * * page 459 - page 460; examples 260-d,260-f,260-g * | Examination | - G.A. PATANI ET AL., "Bioisosterism: A Rational Approach in Drug Design", CHEM. REV., (1996), vol. 96, doi:doi:10.1021/cr950066q, pages 3147 - 3176, XP000652176 DOI: http://dx.doi.org/10.1021/cr950066q |