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Extract from the Register of European Patents

EP About this file: EP2018379

EP2018379 - SCOPINE SALTS AND THEIR USE IN PROCESSES FOR THE PREPARATION OF N-DEMETHYL-TIOTROPIUM AND TIOTROPIUM BROMIDE [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  22.02.2013
Database last updated on 30.09.2024
Most recent event   Tooltip18.07.2014Lapse of the patent in a contracting state
New state(s): HU		published on 20.08.2014  [2014/34]
Applicant(s)For all designated states
Sicor, Inc.
19 Hughes
Irvine, CA 92618 / US
[2012/16]
Former [2009/05]For all designated states
Sicor, Inc.
19 Hughes
Irvine, CA 92618 / US
Inventor(s)01 / BUSOLLI, Jonathan
Via Buronzo N. 65
I-13040 Carisio (vc) / IT
02 / DIULGHEROFF, Nicola
C. So Tassoni, 34
Torino / IT
03 / VOLONTÈ Roberta
Via de Amicis N. 4
I-22069 Rovellasca (co) / IT
04 / PONTIROLI, Alessandro
Via Begoglio 40
S. Maria Della Versa (pv) / IT
 [2012/14]
Former [2009/05]01 / BUSOLLI, Jonathan
Via Buronzo N. 65
I-13040 Carisio (vc) / IT
02 / DIULGHEROFF, Nicola
C. So Tassoni, 34
Torino / IT
03 / VOLONTÈ Roberta
Via de Amicis N. 4
I-22069 Rovellasca (co) / IT
04 / PONTIROLI, Alessandro
Via Begoglio 40
S. Maria Della Versa (pv) / IT
05 / PONTIROLI, Alessandro
Via Begoglio 40
S. Maria Della Versa (pv) / IT
Representative(s)Gallagher, Kirk James, et al
D Young & Co LLP
120 Holborn
London EC1N 2DY / GB
[N/P]
Former [2011/50]Gallagher, Kirk James, et al
D Young & Co LLP 120 Holborn
London EC1N 2DY / GB
Former [2009/05]Russell, Tim, et al
D Young & Co 120 Holborn
London EC1N 2DY / GB
Application number, filing date07810332.210.07.2007
[2009/05]
WO2007US15787
Priority number, dateUS20060830231P10.07.2006         Original published format: US 830231 P
US20060835200P03.08.2006         Original published format: US 835200 P
US20060835201P03.08.2006         Original published format: US 835201 P
US20060836037P07.08.2006         Original published format: US 836037 P
US2006064301319.12.2006         Original published format: US 643013
[2009/05]
Filing languageEN
Procedural languageEN
PublicationType: A2 Application without search report
No.:WO2008008376
Date:17.01.2008
Language:EN
[2008/03]
Type: A2 Application without search report 
No.:EP2018379
Date:28.01.2009
Language:EN
The application published by WIPO in one of the EPO official languages on 17.01.2008 takes the place of the publication of the European patent application.
[2009/05]
Type: B1 Patent specification 
No.:EP2018379
Date:18.04.2012
Language:EN
[2012/16]
Search report(s)International search report - published on:EP13.11.2008
ClassificationIPC:C07D451/06, C07D451/10
[2009/05]
CPC:
C07D451/06 (EP,US); A61P11/00 (EP); A61P11/06 (EP);
A61P11/08 (EP); A61P43/00 (EP); C07D451/10 (EP,US)
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MT,   NL,   PL,   PT,   RO,   SE,   SI,   SK,   TR [2009/05]
TitleGerman:SCOPIN-SALZE UND DEREN VERWENDUNG IN VERFAHREN ZUR HERSTELLUNG VON N-DEMETHYL-TIOTROPIUM UND TIOTROPIUMBROMID[2011/42]
English:SCOPINE SALTS AND THEIR USE IN PROCESSES FOR THE PREPARATION OF N-DEMETHYL-TIOTROPIUM AND TIOTROPIUM BROMIDE[2009/05]
French:SELS DE SCOPINE ET LEUR UTILISATION DANS DES PROCÉDÉS POUR LA PRÉPARATION DE N-DÉMÉTHYL-TIOTROPIUM ET DE BROMURE DE TIOTROPIUM[2011/42]
Former [2009/05]VERFAHREN ZUR HERSTELLUNG VON TIOTROPIUMBROMID
Former [2009/05]PROCÉDÉ POUR LA PRÉPARATION DE BROMURE DE TIOTROPIUM
Entry into regional phase03.03.2008National basic fee paid 
03.03.2008Designation fee(s) paid 
03.03.2008Examination fee paid 
Examination procedure29.02.2008Amendment by applicant (claims and/or description)
03.03.2008Examination requested  [2009/05]
12.08.2009Despatch of a communication from the examining division (Time limit: M04)
21.12.2009Reply to a communication from the examining division
03.03.2011Despatch of a communication from the examining division (Time limit: M04)
21.06.2011Reply to a communication from the examining division
24.10.2011Communication of intention to grant the patent
21.02.2012Fee for grant paid
21.02.2012Fee for publishing/printing paid
Divisional application(s)The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is  12.08.2009
Opposition(s)21.01.2013No opposition filed within time limit [2013/13]
Fees paidRenewal fee
20.07.2009Renewal fee patent year 03
27.07.2010Renewal fee patent year 04
25.07.2011Renewal fee patent year 05
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court		 See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipHU10.07.2007
CY18.04.2012
CZ18.04.2012
DK18.04.2012
EE18.04.2012
FI18.04.2012
LT18.04.2012
LV18.04.2012
MT18.04.2012
RO18.04.2012
SI18.04.2012
SK18.04.2012
IE10.07.2012
LU10.07.2012
BG18.07.2012
CH31.07.2012
LI31.07.2012
MC31.07.2012
IS18.08.2012
PT20.08.2012
[2014/34]
Former [2014/27]CY18.04.2012
CZ18.04.2012
DK18.04.2012
EE18.04.2012
FI18.04.2012
LT18.04.2012
LV18.04.2012
MT18.04.2012
RO18.04.2012
SI18.04.2012
SK18.04.2012
IE10.07.2012
LU10.07.2012
BG18.07.2012
CH31.07.2012
LI31.07.2012
MC31.07.2012
IS18.08.2012
PT20.08.2012
Former [2013/34]CY18.04.2012
CZ18.04.2012
DK18.04.2012
EE18.04.2012
FI18.04.2012
LT18.04.2012
LV18.04.2012
MT18.04.2012
RO18.04.2012
SI18.04.2012
SK18.04.2012
IE10.07.2012
BG18.07.2012
CH31.07.2012
LI31.07.2012
MC31.07.2012
IS18.08.2012
PT20.08.2012
Former [2013/33]CY18.04.2012
CZ18.04.2012
DK18.04.2012
EE18.04.2012
FI18.04.2012
LT18.04.2012
LV18.04.2012
RO18.04.2012
SI18.04.2012
SK18.04.2012
IE10.07.2012
CH31.07.2012
LI31.07.2012
MC31.07.2012
IS18.08.2012
PT20.08.2012
Former [2013/20]CY18.04.2012
CZ18.04.2012
DK18.04.2012
EE18.04.2012
FI18.04.2012
LT18.04.2012
LV18.04.2012
RO18.04.2012
SI18.04.2012
SK18.04.2012
CH31.07.2012
LI31.07.2012
MC31.07.2012
IS18.08.2012
PT20.08.2012
Former [2013/11]CY18.04.2012
CZ18.04.2012
DK18.04.2012
EE18.04.2012
FI18.04.2012
LT18.04.2012
LV18.04.2012
RO18.04.2012
SI18.04.2012
SK18.04.2012
MC31.07.2012
IS18.08.2012
PT20.08.2012
Former [2013/10]CY18.04.2012
CZ18.04.2012
DK18.04.2012
EE18.04.2012
FI18.04.2012
LT18.04.2012
LV18.04.2012
RO18.04.2012
SI18.04.2012
SK18.04.2012
IS18.08.2012
PT20.08.2012
Former [2013/09]CY18.04.2012
DK18.04.2012
EE18.04.2012
FI18.04.2012
LT18.04.2012
LV18.04.2012
SI18.04.2012
IS18.08.2012
PT20.08.2012
Former [2013/08]CY18.04.2012
DK18.04.2012
FI18.04.2012
LT18.04.2012
LV18.04.2012
SI18.04.2012
IS18.08.2012
PT20.08.2012
Former [2013/01]CY18.04.2012
FI18.04.2012
LT18.04.2012
LV18.04.2012
SI18.04.2012
IS18.08.2012
PT20.08.2012
Former [2012/51]CY18.04.2012
FI18.04.2012
LT18.04.2012
LV18.04.2012
SI18.04.2012
IS18.08.2012
Former [2012/50]CY18.04.2012
FI18.04.2012
LT18.04.2012
LV18.04.2012
IS18.08.2012
Former [2012/49]CY18.04.2012
FI18.04.2012
LT18.04.2012
IS18.08.2012
Former [2012/48]FI18.04.2012
LT18.04.2012
Former [2012/47]LT18.04.2012
Cited inInternational search[DX]GB1469781  (BOEHRINGER SOHN INGELHEIM) [DX] 1,3,4 * example 1 *;
 [DAX]US5610163  (BANHOLZER ROLF [DE], et al) [DA] 1-26,29-33 * column 7, lines 1-53; examples 1-4 * [X] 27-32;
 [A]WO0232898  (BOEHRINGER INGELHEIM PHARMA [DE], et al) [A] 27-32* page 7, line 12 - page 8, line 5; claim 12 *;
 [X]US2004242622  (MAMMEN MATHAI [US], et al) [X] 27-32 * page 29, paragraphs 504,505 *;
 [X]  - JINGXI XIE ET AL, "Improvement of studies on total synthesis of anisodine", CAPLUS, CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US, XP002482293 [X] 1-4 * compounds RN 83350-03-2 *
 [X]  - YAPING ZHUANG AND LIQIN ZHAO, "Systemic analysis of 150 kinds of tablet", CAPLUS, CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US, XP002482294 [X] 1-4 * compounds RN 83350-03-2 *
 [X]  - HANS E SCHINK, HELENA PETTERSSON AND JAN-E BÄCKVALL, "Stereocontrolled epoxidations of cycloheptene derivatives in the palladium-catalysed route to tropane alkaloids", JOURNAL OF ORGANIC CHEMISTRY, (1991), vol. 56, no. 8, pages 2769 - 2774, XP002482292 [X] 1,3,4 * Scheme II p.2770; 2nd full par. p.2771; Scopine Hydrochloride (1.HCl) p.2773 *

DOI:   http://dx.doi.org/10.1021/jo00008a037
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.