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Extract from the Register of European Patents

EP About this file: EP2097405

EP2097405 - ANTI-VIRAL COMPOUNDS [Right-click to bookmark this link]
StatusThe application is deemed to be withdrawn
Status updated on  21.10.2011
Database last updated on 11.09.2024
Most recent event   Tooltip21.10.2011Application deemed to be withdrawnpublished on 23.11.2011  [2011/47]
Applicant(s)For all designated states
GlaxoSmithKline LLC
One Franklin Plaza
200 North 16th Street
Philadelphia, PA 19102 / US
[N/P]
Former [2010/09]For all designated states
GlaxoSmithKline LLC
One Franklin Plaza 200 North 16th Street
Philadelphia, PA 19102 / US
Former [2009/37]For all designated states
Smithkline Beecham Corporation
One Franklin Plaza PO Box 7929
Philadelphia, PA 19101 / US
Inventor(s)01 / LEIVERS, Martin Robert
91 Central Ave. 103
San Francisco, CA 94117 / US
02 / SCHMITZ, Franz Ulrich
544 Marin Avenue
Mill Valley, CA 94941 / US
03 / ROBERTS, Christopher Don
1160 Granada St.
Belmont, CA 94002 / US
04 / DEHGHANI MOHAMMAD ABADI, Ali
4971 Ponderosa Terrace
Campbell, CA 95008 / US
 [2009/37]
Representative(s)Crawley, Karen Anne, et al
GlaxoSmithKline
Global Patents (CN925.1)
980 Great West Road
Brentford, Middlesex TW8 9GS / GB
[N/P]
Former [2009/37]Crawley, Karen Anne, et al
GlaxoSmithKline Corporate Intellectual Property (CN9.25.1) 980 Great West Road
Brentford, Middlesex TW8 9GS / GB
Application number, filing date07871535.620.11.2007
[2009/37]
WO2007US85218
Priority number, dateUS20060860614P21.11.2006         Original published format: US 860614 P
[2009/37]
Filing languageEN
Procedural languageEN
PublicationType: A2 Application without search report
No.:WO2008070447
Date:12.06.2008
Language:EN
[2008/24]
Type: A2 Application without search report 
No.:EP2097405
Date:09.09.2009
Language:EN
The application published by WIPO in one of the EPO official languages on 12.06.2008 takes the place of the publication of the European patent application.
[2009/37]
Search report(s)International search report - published on:EP05.03.2009
ClassificationIPC:C07D403/04, C07D207/09, C07D417/14, C07D401/14, C07D403/14, C07D405/14, C07D409/14, C07D413/04
[2009/37]
CPC:
C07D403/04 (EP,US); A61P1/16 (EP); A61P31/12 (EP);
A61P31/14 (EP); A61P43/00 (EP); C07D207/08 (EP,US);
C07D207/09 (EP,US); C07D401/14 (EP,US); C07D403/14 (EP,US);
C07D405/14 (EP,US); C07D409/14 (EP,US); C07D413/04 (EP,US);
C07D413/14 (EP,US); C07D417/04 (EP,US); C07D417/12 (EP,US);
C07D417/14 (EP,US); C07D471/04 (EP,US) (-)
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MT,   NL,   PL,   PT,   RO,   SE,   SI,   SK,   TR [2009/37]
Extension statesHR05.06.2009
TitleGerman:ANTIVIRALE VERBINDUNGEN[2009/37]
English:ANTI-VIRAL COMPOUNDS[2009/37]
French:COMPOSÉS ANTI-VIRAUX[2009/37]
Entry into regional phase05.06.2009National basic fee paid 
05.06.2009Designation fee(s) paid 
05.06.2009Examination fee paid 
Examination procedure05.06.2009Amendment by applicant (claims and/or description)
05.06.2009Examination requested  [2009/37]
01.06.2011Application deemed to be withdrawn, date of legal effect  [2011/47]
05.07.2011Despatch of communication that the application is deemed to be withdrawn, reason: renewal fee not paid in time  [2011/47]
Fees paidRenewal fee
06.11.2009Renewal fee patent year 03
Penalty fee
Additional fee for renewal fee
30.11.201004   M06   Not yet paid
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Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Cited inInternational search[X]EP1604989  (SANTHERA PHARMACEUTICALS DEUTS [DE]) [X] 1-33 * scheme H; example 17, step 1 *;
 [X]US5977101  (ALI FADIA EL-FEHAIL [US], et al) [X] 1-33 * examples 43a,44a *;
 [X]JP2001247569  (JAPAN TOBACCO INC) [X] 1-33 * page 42, compound 135; pages 47-48, compounds 163, 164, 167 *;
 [X]WO03057667  (UNIV OHIO STATE RES FOUND [US], et al) [X] 1-33 * figure 5, compound 38; example 6 *;
 [X]US2006074071  (MELIKIAN ANITA [US], et al) [X] 1-33 * example 25 *;
 [PX]WO2007077186  (NOVARTIS AG [CH], et al) [PX] 1-33 * compounds E-4, F-4, K-3; page 39, line 2 from bottom; page 40, 3 last lines; examples 6, 14-26, 39, 45-48, 55, 72, 75-79, 96 *;
 [PX]WO2007106192  (GENENTECH INC [US], et al) [PX] 1-33 * scheme 3, compounds e; scheme 5, compounds d; scheme 7, compounds e; examples 9d, 10c, 11c, 12c *;
 [PX]WO2007070600  (GENELABS TECH INC [US], et al) [PX] 1-33 * the whole document *;
 [E]WO2008021936  (SQUIBB BRISTOL MYERS CO [US], et al) [E] 1 * example -; claims 1,19,20,26 *;
 [X]US5948793  (ABREO MELWYN A [US], et al) [X] 1 * reaction scheme I, compounds 3; examples 2a, 14a, 15b, 17a, 18a, 74a, 74b, ... *;
 [X]WO0200631  (FUJISAWA PHARMACEUTICAL CO [JP], et al) [X] 1 * preparation 42 *;
 [X]WO9741119  (REDDY RESEARCH FOUNDATION [IN], et al) [X] 1 * preparation 10; example 6;; claims 1,9,17,18 *;
 [X]US6660759  (HATTORI KOUJI [JP], et al) [X] 1 * preparations 5, 10 *;
 [X]US2006116515  (GAHMAN TIMOTHY C [US], et al) [X] 1 * examples 3e,89g,89h,89i,137a,140a,140b,140c,...; claims 1,51 *;
 [X]US4801604  (VONVOIGTLANDER PHILIP F [US], et al) [X] 1 * example 9A *;
 [X]WO2006117669  (PFIZER [US], et al) [X] 1 * general procedures G7, G8, G14a-c;;; examples 4-8,44,57,62,73,84,92,...; claims 1,4,7,9 *;
 [X]US5707987  (NAKAGAWA SUSUMU [JP], et al) [X] 1 * reference examples 100(7), 101(2),103(5), 104(8), 109(5), ... *
 [X]  - KAZUYUKI MAEKAWA AND JIRO OHTANI, "Synthese von 2-(1'-Amino-1'-substituiertem alkyl)-benzimidazol aus Aminosäuren und ihre biologische Aktivität", AGRICULTURAL AND BIOLOGICAL CHEMISTRY, (1976), vol. 40, no. 4, ISSN 0002-1369, pages 791 - 799, XP008069983 [X] 1-33 * table 1, entry 6; table 3, entry 16 (Z-Pro*-) *
 [X]  - GHOTAS EVINDAR AND ROBERT A. BATEY, "Parallel synthesis of a library of benzoxazoles and benzothiazoles using ligand-accelerated copper-catalyzed cyclizations of ortho-halobenzanilides", JOURNAL OF ORGANIC CHEMISTRY, (2006), vol. 71, no. 5, pages 1802 - 1808, XP002508116 [X] 1-33 * table 3, entries 23, 24 *

DOI:   http://dx.doi.org/10.1021/JO051927Q
 [X]  - ROGER JOYEAU ET AL, "Synthesis and activity of pyrrolidinyl- and thiazolidinyl-dipeptide derivatives as inhibitors of the Tc80 prolyl oligopeptidase from Trypanosoma cruzi", EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, (2000), vol. 35, no. 2, ISSN 0223-5234, pages 257 - 266, XP004330419 [X] 1-33 * compound 17 *

DOI:   http://dx.doi.org/10.1016/S0223-5234(00)00118-5
 [X]  - BRIAN K. ALBRECHT AND ROBERT M. WILLIAMS, "A concise formal total synthesis of TMC-95A/B proteasome inhibitors", ORGANIC LETTERS, (2003), vol. 5, no. 2, pages 197 - 200, XP002508117 [X] 1-33 * scheme 1, 13 -> 14; *

DOI:   http://dx.doi.org/10.1021/OL0272545
 [DA]  - ZHI-JIE NI AND ALLAN S. WAGMAN, "Progress and development of small molecule HCV antivirals", CURRENT OPINION IN DRUG DISCOVERY & DEVELOPMENT, (2004), vol. 7, no. 4, ISSN 1367-6733, pages 446 - 459, XP009037092 [DA] 1-33 * the whole document *
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.