Extract from the Register of European Patents

EP About this file: EP2201018

EP2201018 - SOLID FORMS COMPRISING N-(5-TERT-BUTYL-ISOXAZOL-3-YL)-N'-{4-Ý7-(2-MORPHOLIN-4-YL-ETHOXY)IMIDAZOÝ2,1-B ̈Ý1,3 ̈BENZOTHIAZOL-2-YL ̈PHENYL}UREA, COMPOSITIONS THEREOF, AND USES THEREWITH [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  20.01.2017
Database last updated on 14.03.2026
Most recent event   Tooltip20.01.2017No opposition filed within time limitpublished on 22.02.2017  [2017/08]
Applicant(s)For all designated states
Ambit Biosciences Corporation
11080 Roselle Street
San Diego, CA 92121 / US
[2013/16]
Former [2010/26]For all designated states
Ambit Biosciences Corporation
4215 Sorrento Valley Boulevard
San Diego, CA 92121 / US
Inventor(s)01 / BHAGWAT, Shripad
5015 Ashley Falls Court
San Diego CA 92130 / US
02 / LAI, Wei
2107 Longspur Drive
West Lafayette IN 47906 / US
03 / PARENT, Stephan, D.
2120 Cumulus Court
West Lafayette IN 47906 / US
04 / ROE, Melanie, J.
3701 Nicholas Drive Apt. A2
Lafayette IN 47909 / US
05 / SCHWARTZ, Alan
2874 Corte Morera
Carlsbad CA 92009 / US
06 / SMOLENSKAYA, Valeriya, N.
c/o SSCI - a Division of Aptuit, Inc.
3065 Kent Avenue
West Lafayette, IN 47906 / US
 [2016/11]
Former [2010/31]01 / BHAGWAT, Shripad
5015 Ashley Falls Court
San Diego CA 92130 / US
02 / LAI, Wei
2107 Longspur Drive
West Lafayette IN 47906 / US
03 / PARENT, Stephan, D.
2120 Cumulus Court
West Lafayette IN 47906 / US
04 / ROE, Melanie, J.
3701 Nicholas Drive Apt. A2
Lafayette IN 47909 / US
05 / SCHWARTZ, Alan
2874 Corte Morera
Carlsbad CA 92009 / US
06 / SMOLENSKAYA, Valeriya, N.
c/o SSCI - a Division of Aptuit, Inc. 3065 Kent Avenue
West Lafayette, IN 47906 / US
Former [2010/26]01 / BHAGWAT, Shripad
5015 Ashley Falls Court
San Diego CA 92130 / US
02 / LAI, Wei
2107 Longspur Drive
West Lafayette IN 47906 / US
03 / PARENT, Stephan, D.
2120 Cumulus Court
West Lafayette IN 47906 / US
04 / ROE, Melanie, J.
3701 Nicholas Drive Apt. A2
Lafayette IN 47909 / US
05 / SCHWARTZ, Alan
2874 Corte Morera
Carlsbad CA 92009 / US
06 / SMOLENSKAYA, Valeriya, N.
1302 Elizabeth Street Apt. 4
Lafayette IN 47904 / US
Representative(s)Savic, Bojan, et al
Jones Day
Rechtsanwälte Attorneys-at-Law Patentanwälte
Prinzregentenstraße 11
80538 München / DE
[2013/52]
Former [2010/26]Ritter, Thomas Kurt, et al
Jones Day Prinzregentenstraße 11
80538 München / DE
Application number, filing date08832577.419.09.2008
[2010/26]
WO2008US10884
Priority number, dateUS20070994635P19.09.2007         Original published format: US 994635 P
[2010/26]
Filing languageEN
Procedural languageEN
PublicationType: A2 Application without search report
No.:WO2009038757
Date:26.03.2009
Language:EN
[2009/13]
Type: A2 Application without search report 
No.:EP2201018
Date:30.06.2010
Language:EN
The application published by WIPO in one of the EPO official languages on 26.03.2009 takes the place of the publication of the European patent application.
[2010/26]
Type: B1 Patent specification 
No.:EP2201018
Date:16.03.2016
Language:EN
[2016/11]
Search report(s)International search report - published on:EP28.05.2009
ClassificationIPC:C07D513/04, A61K31/5377, A61P35/00
[2010/26]
CPC:
A61K31/5377 (EP,KR,US); C07D513/04 (EP,KR,US); A61K31/185 (EP,US);
A61P1/04 (EP); A61P11/00 (EP); A61P11/02 (EP);
A61P11/06 (EP); A61P13/12 (EP); A61P17/02 (EP);
A61P19/02 (EP); A61P19/10 (EP); A61P25/00 (EP);
A61P29/00 (EP); A61P3/10 (EP); A61P31/04 (EP);
A61P31/12 (EP); A61P35/00 (EP); A61P35/02 (EP);
A61P37/02 (EP); A61P37/06 (EP); A61P37/08 (EP);
A61P43/00 (EP); A61P9/10 (EP); C07D413/04 (KR) (-)
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MT,   NL,   NO,   PL,   PT,   RO,   SE,   SI,   SK,   TR [2016/11]
Former [2010/26]AT,  BE,  BG,  CH,  CY,  CZ,  DE,  DK,  EE,  ES,  FI,  FR,  GB,  GR,  HR,  HU,  IE,  IS,  IT,  LI,  LT,  LU,  LV,  MC,  MT,  NL,  NO,  PL,  PT,  RO,  SE,  SI,  SK,  TR 
Extension statesALNot yet paid
BANot yet paid
MKNot yet paid
RSNot yet paid
TitleGerman:FESTE FORMEN, DIE N-(5-TERT.-BUTYLISOXAZOL-3-YL)-N'-{4-[7-(2-MORPHOLIN-4-YLETHOXY)IMIDAZO[2,1-B][1,3]BENZOTHIAZOL-2-YL]PHENYL}HARNSTOFF UMFASSEN ZUSAMMENSETZUNGEN DAVON UND ANWENDUNGEN DAMIT[2010/26]
English:SOLID FORMS COMPRISING N-(5-TERT-BUTYL-ISOXAZOL-3-YL)-N'-{4-Ý7-(2-MORPHOLIN-4-YL-ETHOXY)IMIDAZOÝ2,1-B ̈Ý1,3 ̈BENZOTHIAZOL-2-YL ̈PHENYL}UREA, COMPOSITIONS THEREOF, AND USES THEREWITH[2010/26]
French:FORMES SOLIDES COMPRENANT DE LA N-(5-TERT-BUTYL-ISOXAZOL-3-YL)-N'-{4-Ý7-(2-MORPHOLIN-4-YL-ÉTHOXY)IMIDAZOÝ2,L-B ̈ÝL,3 ̈BENZOTHIAZOL-2-YL ̈PHÉNYL}URÉE, COMPOSITIONS EN CONTENANT ET LEURS UTILISATIONS[2010/26]
Entry into regional phase14.04.2010National basic fee paid 
14.04.2010Designation fee(s) paid 
14.04.2010Examination fee paid 
Examination procedure14.04.2010Examination requested  [2010/26]
28.05.2010Amendment by applicant (claims and/or description)
04.12.2014Despatch of a communication from the examining division (Time limit: M04)
02.04.2015Reply to a communication from the examining division
29.09.2015Communication of intention to grant the patent
14.01.2016Fee for grant paid
14.01.2016Fee for publishing/printing paid
14.01.2016Receipt of the translation of the claim(s)
Divisional application(s)The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is  04.12.2014
Opposition(s)19.12.2016No opposition filed within time limit [2017/08]
Fees paidRenewal fee
14.09.2010Renewal fee patent year 03
29.09.2011Renewal fee patent year 04
12.09.2012Renewal fee patent year 05
12.09.2013Renewal fee patent year 06
12.09.2014Renewal fee patent year 07
11.09.2015Renewal fee patent year 08
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Cited inInternational search[A]   SAWHNEY S N ET AL: "SYNTHESIS AND ANTIINFLAMMATORY ACTIVITY OF SOME ARYLIMIDAZO(2,1-B)THIAZOLYL- AND ARYLIMIDAZO(2,1-B) BENZOTHIAZOLYLACETIC ACIDS", INDIAN JOURNAL OF CHEMISTRY. SECTION B: ORGANIC AND MEDICINAL CHEMISTRY, SCIENTIFIC PUBLISHERS, JODHPUR, IN, vol. 21B, no. 2, 1 February 1982 (1982-02-01), pages 134 - 138, XP009080136, ISSN: 0376-4699
 [A]   TOSHIYASU MASE ET AL: "Imidazo[2,1-b]benzothiazoles. 2. New immunosuppressive agents", JOURNAL OF MEDICINAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY, WASHINGTON., US, vol. 29, no. 3, 1 January 1986 (1986-01-01), pages 386 - 394, XP002414254, ISSN: 0022-2623 [A] 1,4,22-27 * the whole document *

DOI:   http://dx.doi.org/10.1021/jm00153a014
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