EP2233467 - ALPHA-AMINO-N-SUBSTITUTED AMIDES, PHARMACEUTICAL COMPOSITION CONTAINING THEM AND USES THEREOF [Right-click to bookmark this link] | Status | No opposition filed within time limit Status updated on 26.07.2013 Database last updated on 22.05.2024 | Most recent event Tooltip | 18.07.2014 | Lapse of the patent in a contracting state New state(s): HU | published on 20.08.2014 [2014/34] | Applicant(s) | For all designated states SHANGHAI INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF SCIENCES 294 Tai-Yuan Road Shanghai 200031 / CN | [2010/39] | Inventor(s) | 01 /
NAN, Fajun 294 Taiyuan Road Shanghai 200031 / CN | 02 /
LI, Jia 294 Taiyuan Road Shanghai 200031 / CN | 03 /
DING, Jian 294 Taiyuan Road Shanghai 200031 / CN | 04 /
LIU, Gang 294 Taiyuan Road Shanghai 200031 / CN | 05 /
XIE, Chuanming 294 Taiyuan Road Shanghai 200031 / CN | 06 /
MIAO, Zehong 294 Taiyuan Road Shanghai 200031 / CN | 07 /
TAI, Wanyi 294 Taiyuan Road Shanghai 200031 / CN | [2010/39] | Representative(s) | Kador & Partner Part mbB Corneliusstraße 15 80469 München / DE | [N/P] |
Former [2012/38] | Kador & Partner Corneliusstrasse 15 80469 München / DE | ||
Former [2010/39] | Kador & Partner Corneliusstrasse 15 80469 München / DE | Application number, filing date | 08858616.9 | 11.12.2008 | [2010/39] | WO2008CN01996 | Priority number, date | CN200710172079 | 11.12.2007 Original published format: CN200710172079 | [2010/39] | Filing language | ZH | Procedural language | EN | Publication | Type: | A1 Application with search report | No.: | WO2009074020 | Date: | 18.06.2009 | Language: | ZH | [2009/25] | Type: | A1 Application with search report | No.: | EP2233467 | Date: | 29.09.2010 | Language: | EN | [2010/39] | Type: | B1 Patent specification | No.: | EP2233467 | Date: | 19.09.2012 | Language: | EN | [2012/38] | Search report(s) | International search report - published on: | CN | 18.06.2009 | (Supplementary) European search report - dispatched on: | EP | 14.06.2011 | Classification | IPC: | C07C237/16, C07C233/05, C07C233/09, C07C233/18, C07C233/20, A61K31/16, A61P35/00 | [2010/39] | CPC: |
C07C237/22 (EP,US);
A61P35/00 (EP);
C07C247/12 (EP,US);
C07C271/22 (EP,US);
C07C323/60 (EP,US);
C07D209/14 (EP,US);
C07D209/20 (EP,US);
C07D233/54 (EP,US);
C07D307/24 (EP,US);
C07D307/94 (EP,US);
C07C2601/02 (EP,US);
C07C2601/04 (EP,US);
C07C2601/08 (EP,US);
C07C2601/14 (EP,US);
C07C2601/16 (EP,US);
C07C2603/74 (EP,US)
(-)
| Designated contracting states | AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MT, NL, NO, PL, PT, RO, SE, SI, SK, TR [2010/39] | Title | German: | ALPHA-AMINO-N-SUBSTITUIERTE AMIDE, PHARMAZEUTISCHE ZUSAMMENSETZUNG, DIE DIESE ENTHÄLT, UND ANWENDUNGEN DAVON | [2010/39] | English: | ALPHA-AMINO-N-SUBSTITUTED AMIDES, PHARMACEUTICAL COMPOSITION CONTAINING THEM AND USES THEREOF | [2010/39] | French: | AMIDES N-SUBSTITUÉS PAR ALPHA-AMINO, COMPOSITION PHARMACEUTIQUE LES CONTENANT ET LEURS UTILISATIONS | [2010/39] | Entry into regional phase | 10.06.2010 | Translation filed | 10.06.2010 | National basic fee paid | 10.06.2010 | Search fee paid | 10.06.2010 | Designation fee(s) paid | 10.06.2010 | Examination fee paid | Examination procedure | 10.06.2010 | Examination requested [2010/39] | 07.07.2011 | Amendment by applicant (claims and/or description) | 03.05.2012 | Communication of intention to grant the patent | 03.08.2012 | Fee for grant paid | 03.08.2012 | Fee for publishing/printing paid | Divisional application(s) | The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is 03.05.2012 | Opposition(s) | 20.06.2013 | No opposition filed within time limit [2013/35] | Fees paid | Renewal fee | 27.12.2010 | Renewal fee patent year 03 | 29.12.2011 | Renewal fee patent year 04 |
Opt-out from the exclusive Tooltip competence of the Unified Patent Court | See the Register of the Unified Patent Court for opt-out data | ||
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Lapses during opposition Tooltip | HU | 11.12.2008 | AT | 19.09.2012 | BE | 19.09.2012 | CY | 19.09.2012 | CZ | 19.09.2012 | DK | 19.09.2012 | EE | 19.09.2012 | FI | 19.09.2012 | HR | 19.09.2012 | LT | 19.09.2012 | LV | 19.09.2012 | MT | 19.09.2012 | NL | 19.09.2012 | PL | 19.09.2012 | RO | 19.09.2012 | SE | 19.09.2012 | SI | 19.09.2012 | SK | 19.09.2012 | TR | 19.09.2012 | IE | 11.12.2012 | LU | 11.12.2012 | BG | 19.12.2012 | GB | 19.12.2012 | NO | 19.12.2012 | GR | 20.12.2012 | ES | 30.12.2012 | CH | 31.12.2012 | LI | 31.12.2012 | MC | 31.12.2012 | IS | 19.01.2013 | PT | 21.01.2013 | [2014/34] |
Former [2014/27] | AT | 19.09.2012 | |
BE | 19.09.2012 | ||
CY | 19.09.2012 | ||
CZ | 19.09.2012 | ||
DK | 19.09.2012 | ||
EE | 19.09.2012 | ||
FI | 19.09.2012 | ||
HR | 19.09.2012 | ||
LT | 19.09.2012 | ||
LV | 19.09.2012 | ||
MT | 19.09.2012 | ||
NL | 19.09.2012 | ||
PL | 19.09.2012 | ||
RO | 19.09.2012 | ||
SE | 19.09.2012 | ||
SI | 19.09.2012 | ||
SK | 19.09.2012 | ||
TR | 19.09.2012 | ||
IE | 11.12.2012 | ||
LU | 11.12.2012 | ||
BG | 19.12.2012 | ||
GB | 19.12.2012 | ||
NO | 19.12.2012 | ||
GR | 20.12.2012 | ||
ES | 30.12.2012 | ||
CH | 31.12.2012 | ||
LI | 31.12.2012 | ||
MC | 31.12.2012 | ||
IS | 19.01.2013 | ||
PT | 21.01.2013 | ||
Former [2014/21] | AT | 19.09.2012 | |
BE | 19.09.2012 | ||
CY | 19.09.2012 | ||
CZ | 19.09.2012 | ||
DK | 19.09.2012 | ||
EE | 19.09.2012 | ||
FI | 19.09.2012 | ||
HR | 19.09.2012 | ||
LT | 19.09.2012 | ||
LV | 19.09.2012 | ||
MT | 19.09.2012 | ||
NL | 19.09.2012 | ||
PL | 19.09.2012 | ||
RO | 19.09.2012 | ||
SE | 19.09.2012 | ||
SI | 19.09.2012 | ||
SK | 19.09.2012 | ||
TR | 19.09.2012 | ||
IE | 11.12.2012 | ||
BG | 19.12.2012 | ||
GB | 19.12.2012 | ||
NO | 19.12.2012 | ||
GR | 20.12.2012 | ||
ES | 30.12.2012 | ||
CH | 31.12.2012 | ||
LI | 31.12.2012 | ||
MC | 31.12.2012 | ||
IS | 19.01.2013 | ||
PT | 21.01.2013 | ||
Former [2013/52] | AT | 19.09.2012 | |
BE | 19.09.2012 | ||
CY | 19.09.2012 | ||
CZ | 19.09.2012 | ||
DK | 19.09.2012 | ||
EE | 19.09.2012 | ||
FI | 19.09.2012 | ||
HR | 19.09.2012 | ||
LT | 19.09.2012 | ||
LV | 19.09.2012 | ||
MT | 19.09.2012 | ||
NL | 19.09.2012 | ||
PL | 19.09.2012 | ||
RO | 19.09.2012 | ||
SE | 19.09.2012 | ||
SI | 19.09.2012 | ||
SK | 19.09.2012 | ||
IE | 11.12.2012 | ||
BG | 19.12.2012 | ||
GB | 19.12.2012 | ||
NO | 19.12.2012 | ||
GR | 20.12.2012 | ||
ES | 30.12.2012 | ||
CH | 31.12.2012 | ||
LI | 31.12.2012 | ||
MC | 31.12.2012 | ||
IS | 19.01.2013 | ||
PT | 21.01.2013 | ||
Former [2013/51] | AT | 19.09.2012 | |
BE | 19.09.2012 | ||
CZ | 19.09.2012 | ||
DK | 19.09.2012 | ||
EE | 19.09.2012 | ||
FI | 19.09.2012 | ||
HR | 19.09.2012 | ||
LT | 19.09.2012 | ||
LV | 19.09.2012 | ||
MT | 19.09.2012 | ||
NL | 19.09.2012 | ||
PL | 19.09.2012 | ||
RO | 19.09.2012 | ||
SE | 19.09.2012 | ||
SI | 19.09.2012 | ||
SK | 19.09.2012 | ||
IE | 11.12.2012 | ||
BG | 19.12.2012 | ||
GB | 19.12.2012 | ||
NO | 19.12.2012 | ||
GR | 20.12.2012 | ||
ES | 30.12.2012 | ||
CH | 31.12.2012 | ||
LI | 31.12.2012 | ||
MC | 31.12.2012 | ||
IS | 19.01.2013 | ||
PT | 21.01.2013 | ||
Former [2013/48] | AT | 19.09.2012 | |
BE | 19.09.2012 | ||
CZ | 19.09.2012 | ||
DK | 19.09.2012 | ||
EE | 19.09.2012 | ||
FI | 19.09.2012 | ||
HR | 19.09.2012 | ||
LT | 19.09.2012 | ||
LV | 19.09.2012 | ||
NL | 19.09.2012 | ||
PL | 19.09.2012 | ||
RO | 19.09.2012 | ||
SE | 19.09.2012 | ||
SI | 19.09.2012 | ||
SK | 19.09.2012 | ||
IE | 11.12.2012 | ||
BG | 19.12.2012 | ||
NO | 19.12.2012 | ||
GR | 20.12.2012 | ||
ES | 30.12.2012 | ||
CH | 31.12.2012 | ||
LI | 31.12.2012 | ||
MC | 31.12.2012 | ||
IS | 19.01.2013 | ||
PT | 21.01.2013 | ||
Former [2013/47] | AT | 19.09.2012 | |
BE | 19.09.2012 | ||
CZ | 19.09.2012 | ||
DK | 19.09.2012 | ||
EE | 19.09.2012 | ||
FI | 19.09.2012 | ||
HR | 19.09.2012 | ||
LT | 19.09.2012 | ||
LV | 19.09.2012 | ||
NL | 19.09.2012 | ||
PL | 19.09.2012 | ||
RO | 19.09.2012 | ||
SE | 19.09.2012 | ||
SI | 19.09.2012 | ||
SK | 19.09.2012 | ||
IE | 11.12.2012 | ||
BG | 19.12.2012 | ||
NO | 19.12.2012 | ||
GR | 20.12.2012 | ||
ES | 30.12.2012 | ||
MC | 31.12.2012 | ||
IS | 19.01.2013 | ||
PT | 21.01.2013 | ||
Former [2013/34] | AT | 19.09.2012 | |
BE | 19.09.2012 | ||
CZ | 19.09.2012 | ||
DK | 19.09.2012 | ||
EE | 19.09.2012 | ||
FI | 19.09.2012 | ||
HR | 19.09.2012 | ||
LT | 19.09.2012 | ||
LV | 19.09.2012 | ||
NL | 19.09.2012 | ||
PL | 19.09.2012 | ||
RO | 19.09.2012 | ||
SE | 19.09.2012 | ||
SI | 19.09.2012 | ||
SK | 19.09.2012 | ||
BG | 19.12.2012 | ||
NO | 19.12.2012 | ||
GR | 20.12.2012 | ||
ES | 30.12.2012 | ||
MC | 31.12.2012 | ||
IS | 19.01.2013 | ||
PT | 21.01.2013 | ||
Former [2013/33] | AT | 19.09.2012 | |
BE | 19.09.2012 | ||
CZ | 19.09.2012 | ||
EE | 19.09.2012 | ||
FI | 19.09.2012 | ||
HR | 19.09.2012 | ||
LT | 19.09.2012 | ||
LV | 19.09.2012 | ||
NL | 19.09.2012 | ||
PL | 19.09.2012 | ||
RO | 19.09.2012 | ||
SE | 19.09.2012 | ||
SI | 19.09.2012 | ||
SK | 19.09.2012 | ||
NO | 19.12.2012 | ||
GR | 20.12.2012 | ||
ES | 30.12.2012 | ||
MC | 31.12.2012 | ||
IS | 19.01.2013 | ||
PT | 21.01.2013 | ||
Former [2013/31] | AT | 19.09.2012 | |
BE | 19.09.2012 | ||
CZ | 19.09.2012 | ||
EE | 19.09.2012 | ||
FI | 19.09.2012 | ||
HR | 19.09.2012 | ||
LT | 19.09.2012 | ||
LV | 19.09.2012 | ||
NL | 19.09.2012 | ||
PL | 19.09.2012 | ||
RO | 19.09.2012 | ||
SE | 19.09.2012 | ||
SI | 19.09.2012 | ||
SK | 19.09.2012 | ||
NO | 19.12.2012 | ||
GR | 20.12.2012 | ||
ES | 30.12.2012 | ||
IS | 19.01.2013 | ||
PT | 21.01.2013 | ||
Former [2013/28] | BE | 19.09.2012 | |
CZ | 19.09.2012 | ||
EE | 19.09.2012 | ||
FI | 19.09.2012 | ||
HR | 19.09.2012 | ||
LT | 19.09.2012 | ||
LV | 19.09.2012 | ||
NL | 19.09.2012 | ||
PL | 19.09.2012 | ||
RO | 19.09.2012 | ||
SE | 19.09.2012 | ||
SI | 19.09.2012 | ||
SK | 19.09.2012 | ||
NO | 19.12.2012 | ||
GR | 20.12.2012 | ||
ES | 30.12.2012 | ||
IS | 19.01.2013 | ||
PT | 21.01.2013 | ||
Former [2013/23] | BE | 19.09.2012 | |
CZ | 19.09.2012 | ||
EE | 19.09.2012 | ||
FI | 19.09.2012 | ||
HR | 19.09.2012 | ||
LT | 19.09.2012 | ||
LV | 19.09.2012 | ||
NL | 19.09.2012 | ||
PL | 19.09.2012 | ||
RO | 19.09.2012 | ||
SE | 19.09.2012 | ||
SI | 19.09.2012 | ||
SK | 19.09.2012 | ||
NO | 19.12.2012 | ||
GR | 20.12.2012 | ||
ES | 30.12.2012 | ||
IS | 19.01.2013 | ||
Former [2013/22] | BE | 19.09.2012 | |
CZ | 19.09.2012 | ||
EE | 19.09.2012 | ||
FI | 19.09.2012 | ||
HR | 19.09.2012 | ||
LT | 19.09.2012 | ||
LV | 19.09.2012 | ||
NL | 19.09.2012 | ||
SE | 19.09.2012 | ||
SI | 19.09.2012 | ||
NO | 19.12.2012 | ||
GR | 20.12.2012 | ||
ES | 30.12.2012 | ||
IS | 19.01.2013 | ||
Former [2013/20] | BE | 19.09.2012 | |
FI | 19.09.2012 | ||
HR | 19.09.2012 | ||
LT | 19.09.2012 | ||
LV | 19.09.2012 | ||
SE | 19.09.2012 | ||
SI | 19.09.2012 | ||
NO | 19.12.2012 | ||
GR | 20.12.2012 | ||
Former [2013/12] | FI | 19.09.2012 | |
HR | 19.09.2012 | ||
LT | 19.09.2012 | ||
LV | 19.09.2012 | ||
SE | 19.09.2012 | ||
SI | 19.09.2012 | ||
NO | 19.12.2012 | ||
GR | 20.12.2012 | ||
Former [2013/11] | FI | 19.09.2012 | |
HR | 19.09.2012 | ||
LT | 19.09.2012 | ||
LV | 19.09.2012 | ||
SI | 19.09.2012 | ||
NO | 19.12.2012 | ||
GR | 20.12.2012 | ||
Former [2013/10] | FI | 19.09.2012 | |
HR | 19.09.2012 | ||
LT | 19.09.2012 | ||
NO | 19.12.2012 | ||
Former [2013/09] | FI | 19.09.2012 | |
LT | 19.09.2012 | ||
NO | 19.12.2012 | ||
Former [2013/08] | LT | 19.09.2012 | |
NO | 19.12.2012 | Documents cited: | Search | [A]US2007244087 (ZHANG JIDONG [FR], et al) [A] 1-13 * examples 1-23; claims 1-16; tables 1,2 *; | [A]US2007249584 (ZHANG JIDONG [FR], et al) [A] 1-13 * examples 1-27; claims 1-24; tables 1,2 * | International search | [XP]CN101092384 (SHANGHAI INST OF MEDICINES C A [CN]); | [A]WO2006056696 (AVENTIS PHARMA SA [FR], et al); | [A]WO2005014574 (NOVARTIS AG [CH], et al) | by applicant | - J. MED. CHEM, (2001), vol. 44, pages 3692 - 3699 | - ORG. PROCESS. RES. DEV., (2003), vol. 7, pages 856 - 865 | - J ORG. CHEM., (1982), vol. 47, pages 2027 - 2033 | - TETRAHEDRON LETTERS, (2002), vol. 43, pages 6709 - 6713 | - J MED. CHEM., (1989), vol. 32, pages 859 - 863 | - TETRAHEDRON, (2004), vol. 60, pages 8957 - 8966 | - EUR J MED. CHEM. CHIM. THER, (1978), vol. 13, page 171 | - J AM. CHEM. SOC., (2007), vol. 129, pages 2744 - 2745 |