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Extract from the Register of European Patents

EP About this file: EP2254415

EP2254415 - ARYL-HYDROXYETHYLAMINO-PYRIMIDINES AND TRIAZINES AS MODULATORS OF FATTY ACID AMIDE HYDROLASE [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  29.11.2013
Database last updated on 24.07.2024
Most recent event   Tooltip17.07.2015Lapse of the patent in a contracting state
New state(s): HU, LU		published on 19.08.2015  [2015/34]
Applicant(s)For all designated states
Janssen Pharmaceutica, N.V.
Turnhoutseweg 30
2340 Beerse / BE
[2010/48]
Inventor(s)01 / APODACA, Richard
8448 Via Sonoma, 98
La Jolla CA 92037 / US
02 / BREITENBUCHER, J., Guy
2433 North Summit Circle Glen
Escondido CA 92026 / US
03 / CHAMBERS, Alison, L.
5235 Fiore Terrace, C312
San Diego CA 92122 / US
04 / DENG, Xiaohu
8219 Bryn Glen Way
San Diego CA 92129 / US
05 / HAWRYLUK, Natalie, A.
4379 Mistral Place
San Diego CA 92130 / US
06 / KEITH, John, M.
16724 Alondra Drive
San Diego CA 92128 / US
07 / MANI, Neelakandha, S.
13109 Russet Leaf Lane
San Diego CA 92128 / US
08 / MERIT, Jeffrey, E.
344 Olmsted Road, 431
Stanford CA 94305 / US
09 / PIERCE, Joan, M.
3167 Via Alicante
Unit 244
La Jolla CA 92037 / US
10 / SEIERSTAD, Mark
2230 Shadyridge Avenue
Escondido CA 92029 / US
11 / XIAO, Wei
4043 Carmel Springs Way
San Diego CA 92130 / US
 [2013/04]
Former [2010/48]01 / APODACA, Richard
8448 Via Sonoma, 98
La Jolla CA 92037 / US
02 / BREITENBUCHER, J., Guy
2433 North Summit Circle Glen
Escondido CA 92026 / US
03 / CHAMBERS, Alison, L.
5235 Fiore Terrace, C312
San Diego CA 92122 / US
04 / DENG, Xiaohu
8219 Bryn Glen Way
San Diego CA 92129 / US
05 / HAWRYLUK, Natalie, A.
4379 Mistral Place
San Diego CA 92130 / US
06 / KEITH, John, M.
16724 Alondra Drive
San Diego CA 92128 / US
07 / MANI, Neelakandha, S.
13109 Russet Leaf Lane
San Diego CA 92128 / US
08 / MERIT, Jeffrey, E.
344 Olmsted Road, 431
Stanford CA 94305 / US
09 / PIERCE, Joan, M.
3167 Via Alicante Unit 244
La Jolla CA 92037 / US
10 / SEIERSTAD, Mark
2230 Shadyridge Avenue
Escondido CA 92029 / US
11 / XIAO, Wei
4043 Carmel Springs Way
San Diego CA 92130 / US
Representative(s)Warner, James Alexander, et al
Carpmaels & Ransford LLP
One Southampton Row
London WC1B 5HA / GB
[N/P]
Former [2010/48]Warner, James Alexander, et al
Carpmaels & Ransford One Southampton Row London
WC1B 5HA / GB
Application number, filing date09712375.618.02.2009
[2010/48]
WO2009US01043
Priority number, dateUS20080029619P19.02.2008         Original published format: US 29619 P
US20080086353P05.08.2008         Original published format: US 86353 P
[2010/48]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2009105220
Date:27.08.2009
Language:EN
[2009/35]
Type: A1 Application with search report 
No.:EP2254415
Date:01.12.2010
Language:EN
The application published by WIPO in one of the EPO official languages on 27.08.2009 takes the place of the publication of the European patent application.
[2010/48]
Type: B1 Patent specification 
No.:EP2254415
Date:23.01.2013
Language:EN
[2013/04]
Search report(s)International search report - published on:US27.08.2009
(Supplementary) European search report - dispatched on:EP12.12.2011
ClassificationIPC:A61K31/53, C07D239/42, C07D239/47, C07D239/48, C07D251/22, C07D401/04, C07D401/12, C07D403/04, C07D405/04, C07D405/12, A61P25/00
[2012/35]
CPC:
C07D239/42 (EP,US); A61P1/00 (EP); A61P11/00 (EP);
A61P25/00 (EP); A61P3/00 (EP); C07D239/47 (EP,US);
C07D239/48 (EP,US); C07D251/22 (EP,US); C07D401/04 (EP,US);
C07D401/12 (EP,US); C07D403/04 (EP,US); C07D403/12 (EP,US);
C07D405/04 (EP,US); C07D405/12 (EP,US); C07D409/04 (EP,US);
C07D409/12 (EP,US); C07D409/14 (EP,US); C07D413/04 (EP,US);
C07D413/14 (EP,US); C07D417/12 (EP,US) (-)
Former IPC [2010/48]A01N43/66, A61K31/53
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   SE,   SI,   SK,   TR [2010/48]
TitleGerman:ARYLHYDROXYETHYLAMINOPYRIMIDINE UND TRIAZINE ALS MODULATOREN DER FETTSÄUREAMIDHYDROLASE[2010/48]
English:ARYL-HYDROXYETHYLAMINO-PYRIMIDINES AND TRIAZINES AS MODULATORS OF FATTY ACID AMIDE HYDROLASE[2010/48]
French:ARYL-HYDROXYÉTHYLAMINO-PYRIMIDINES ET TRIAZINES EN TANT QUE MODULATEURS D'AMIDE D'ACIDE GRAS HYDROLASE[2010/48]
Entry into regional phase20.09.2010National basic fee paid 
20.09.2010Search fee paid 
20.09.2010Designation fee(s) paid 
20.09.2010Examination fee paid 
Examination procedure20.09.2010Examination requested  [2010/48]
06.07.2012Amendment by applicant (claims and/or description)
09.08.2012Communication of intention to grant the patent
07.12.2012Fee for grant paid
07.12.2012Fee for publishing/printing paid
Divisional application(s)The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is  09.08.2012
Opposition(s)24.10.2013No opposition filed within time limit [2014/01]
Fees paidRenewal fee
15.02.2011Renewal fee patent year 03
15.02.2012Renewal fee patent year 04
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court		 See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipHU18.02.2009
AT23.01.2013
BE23.01.2013
CY23.01.2013
CZ23.01.2013
DK23.01.2013
EE23.01.2013
FI23.01.2013
HR23.01.2013
IT23.01.2013
LT23.01.2013
LV23.01.2013
MK23.01.2013
MT23.01.2013
NL23.01.2013
PL23.01.2013
RO23.01.2013
SE23.01.2013
SI23.01.2013
SK23.01.2013
TR23.01.2013
LU18.02.2013
CH28.02.2013
LI28.02.2013
MC28.02.2013
BG23.04.2013
NO23.04.2013
GR24.04.2013
ES04.05.2013
IS23.05.2013
PT23.05.2013
[2015/34]
Former [2015/32]AT23.01.2013
BE23.01.2013
CY23.01.2013
CZ23.01.2013
DK23.01.2013
EE23.01.2013
FI23.01.2013
HR23.01.2013
IT23.01.2013
LT23.01.2013
LV23.01.2013
MK23.01.2013
MT23.01.2013
NL23.01.2013
PL23.01.2013
RO23.01.2013
SE23.01.2013
SI23.01.2013
SK23.01.2013
TR23.01.2013
CH28.02.2013
LI28.02.2013
MC28.02.2013
BG23.04.2013
NO23.04.2013
GR24.04.2013
ES04.05.2013
IS23.05.2013
PT23.05.2013
Former [2014/32]AT23.01.2013
BE23.01.2013
CY23.01.2013
CZ23.01.2013
DK23.01.2013
EE23.01.2013
FI23.01.2013
HR23.01.2013
IT23.01.2013
LT23.01.2013
LV23.01.2013
MT23.01.2013
NL23.01.2013
PL23.01.2013
RO23.01.2013
SE23.01.2013
SI23.01.2013
SK23.01.2013
CH28.02.2013
LI28.02.2013
MC28.02.2013
BG23.04.2013
NO23.04.2013
GR24.04.2013
ES04.05.2013
IS23.05.2013
PT23.05.2013
Former [2014/03]AT23.01.2013
BE23.01.2013
CY23.01.2013
CZ23.01.2013
DK23.01.2013
EE23.01.2013
FI23.01.2013
HR23.01.2013
IT23.01.2013
LT23.01.2013
LV23.01.2013
NL23.01.2013
PL23.01.2013
RO23.01.2013
SE23.01.2013
SI23.01.2013
SK23.01.2013
CH28.02.2013
LI28.02.2013
MC28.02.2013
BG23.04.2013
NO23.04.2013
GR24.04.2013
ES04.05.2013
IS23.05.2013
PT23.05.2013
Former [2013/52]AT23.01.2013
BE23.01.2013
CY23.01.2013
CZ23.01.2013
DK23.01.2013
EE23.01.2013
FI23.01.2013
HR23.01.2013
LT23.01.2013
LV23.01.2013
NL23.01.2013
PL23.01.2013
RO23.01.2013
SE23.01.2013
SI23.01.2013
SK23.01.2013
CH28.02.2013
LI28.02.2013
MC28.02.2013
BG23.04.2013
NO23.04.2013
GR24.04.2013
ES04.05.2013
IS23.05.2013
PT23.05.2013
Former [2013/49]AT23.01.2013
BE23.01.2013
CZ23.01.2013
DK23.01.2013
EE23.01.2013
FI23.01.2013
HR23.01.2013
LT23.01.2013
LV23.01.2013
NL23.01.2013
PL23.01.2013
RO23.01.2013
SE23.01.2013
SI23.01.2013
SK23.01.2013
CH28.02.2013
LI28.02.2013
MC28.02.2013
BG23.04.2013
NO23.04.2013
GR24.04.2013
ES04.05.2013
IS23.05.2013
PT23.05.2013
Former [2013/48]AT23.01.2013
BE23.01.2013
DK23.01.2013
EE23.01.2013
FI23.01.2013
HR23.01.2013
LT23.01.2013
LV23.01.2013
NL23.01.2013
PL23.01.2013
SE23.01.2013
SI23.01.2013
CH28.02.2013
LI28.02.2013
MC28.02.2013
BG23.04.2013
NO23.04.2013
GR24.04.2013
ES04.05.2013
IS23.05.2013
PT23.05.2013
Former [2013/42]AT23.01.2013
BE23.01.2013
FI23.01.2013
HR23.01.2013
LT23.01.2013
LV23.01.2013
NL23.01.2013
PL23.01.2013
SE23.01.2013
SI23.01.2013
MC28.02.2013
BG23.04.2013
NO23.04.2013
GR24.04.2013
ES04.05.2013
IS23.05.2013
PT23.05.2013
Former [2013/41]AT23.01.2013
BE23.01.2013
FI23.01.2013
HR23.01.2013
LT23.01.2013
LV23.01.2013
NL23.01.2013
PL23.01.2013
SE23.01.2013
SI23.01.2013
BG23.04.2013
NO23.04.2013
GR24.04.2013
ES04.05.2013
IS23.05.2013
PT23.05.2013
Former [2013/40]AT23.01.2013
BE23.01.2013
FI23.01.2013
LT23.01.2013
LV23.01.2013
NL23.01.2013
PL23.01.2013
SE23.01.2013
SI23.01.2013
BG23.04.2013
NO23.04.2013
GR24.04.2013
ES04.05.2013
IS23.05.2013
PT23.05.2013
Former [2013/38]AT23.01.2013
BE23.01.2013
FI23.01.2013
LT23.01.2013
LV23.01.2013
NL23.01.2013
PL23.01.2013
SE23.01.2013
SI23.01.2013
BG23.04.2013
NO23.04.2013
GR24.04.2013
ES04.05.2013
IS23.05.2013
Former [2013/37]AT23.01.2013
BE23.01.2013
FI23.01.2013
LT23.01.2013
NL23.01.2013
PL23.01.2013
SE23.01.2013
SI23.01.2013
BG23.04.2013
NO23.04.2013
GR24.04.2013
ES04.05.2013
IS23.05.2013
Former [2013/36]AT23.01.2013
BE23.01.2013
LT23.01.2013
PL23.01.2013
SE23.01.2013
BG23.04.2013
NO23.04.2013
ES04.05.2013
IS23.05.2013
Former [2013/35]BE23.01.2013
LT23.01.2013
SE23.01.2013
BG23.04.2013
NO23.04.2013
IS23.05.2013
Former [2013/34]LT23.01.2013
SE23.01.2013
BG23.04.2013
NO23.04.2013
IS23.05.2013
Former [2013/33]LT23.01.2013
NO23.04.2013
Documents cited:Search[A]WO2006074025  (JANSSEN PHARMACEUTICA NV [BE], et al) [A] 1-16 * the whole document *;
 [A]US2007004741  (APODACA RICHARD [US], et al) [A] 1-16 * the whole document *
International search[Y]US2006025433  (BARBOSA ANTONIO J JR [US], et al);
 [Y]US5594141  (YUAN JUN [US], et al);
 [Y]US3624084  (MATHIEU JACQUES);
 [Y]US2005234030  (BARTOLINI WILMIN [US], et al);
 [Y]  - WESTHUYZEN ET AL., "Effect of substituent structure on pyrimidine electrophilic substitution.", TETRAHEDRON, (2007), vol. 63, pages 5394 - 5405
 [Y]  - BORK ET AL., "The Combinatorial Synthesis of Purine, Pyrimidine and Triazinebased Libraries.", QSAR COMB. SCI., (2004), vol. 23, pages 245 - 260, XP008140827

DOI:   http://dx.doi.org/10.1002/qsar.200420016
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