EP2350060 - MELANOCORTIN RECEPTOR AGONISTS [Right-click to bookmark this link] | Status | No opposition filed within time limit Status updated on 25.07.2014 Database last updated on 15.06.2024 | Most recent event Tooltip | 04.09.2015 | Lapse of the patent in a contracting state New state(s): MT | published on 07.10.2015 [2015/41] | Applicant(s) | For all designated states LG Life Sciences Ltd LG Twin Tower, East Tower 20, Yoido-dong Youngdungpo-ku Seoul 150-010 / KR | [2011/31] | Inventor(s) | 01 /
LEE, Koo R&D Park LG Life Sciences Ltd. 104-1 Moongi-dong Yuseong-gu Daejeon 305-380 / KR | 02 /
LEE, Sang Dae R&D Park LG Life Sciences Ltd. 104-1 Moongi-dong Yuseong-gu Daejeon 305-380 / KR | 03 /
MOON, Sang Pil R&D Park LG Life Sciences Ltd. 104-1 Moongi-dong Yuseong-gu Daejeon 305-380 / KR | 04 /
AHN, In Ae R&D Park LG Life Sciences Ltd. 104-1 Moongi-dong Yuseong-gu Daejeon 305-380 / KR | 05 /
CHOI, Sung Pil R&D Park LG Life Sciences Ltd. 104-1 Moongi-dong Yuseong-gu Daejeon 305-380 / KR | 06 /
LEE, Hyun Ho R&D Park LG Life Sciences Ltd. 104-1 Moongi-dong Yuseong-gu Daejeon 305-380 / KR | 07 /
SHIM, Dong Sup R&D Park LG Life Sciences Ltd. 104-1 Moongi-dong Yuseong-gu Daejeon 305-380 / KR | 08 /
CHUNG, Soo Yong R&D Park LG Life Sciences Ltd. 104-1 Moongi-dong Yuseong-gu Daejeon 305-380 / KR | 09 /
LEE, Hyun Min R&D Park LG Life Sciences Ltd. 104-1 Moongi-dong Yuseong-gu Daejeon 305-380 / KR | [2013/38] |
Former [2011/31] | 01 /
LEE, Koo R&D Park LG Life Sciences Ltd. 104-1 Moongi-dong Yuseong-gu Daejeon 305-380 / KR | ||
02 /
LEE, Sang Dae R&D Park LG Life Sciences Ltd. 104-1 Moongi-dong Yuseong-gu Daejeon 305-380 / KR | |||
03 /
MOON, Sang Pil R&D Park LG Life Sciences Ltd. 104-1 Moongi-dong Yuseong-gu Daejeon 305-380 / KR | |||
04 /
AHN, In Ae R&D Park LG Life Sciences Ltd. 104-1 Moongi-dong Yuseong-gu Daejeon 305-380 / KR | |||
05 /
CHOI, Sung Pil R&D Park LG Life Sciences Ltd. 104-1 Moongi-dong Yuseong-gu Daejeon 305-380 / KR | |||
06 /
LEE, Hyun Ho R&D Park LG Life Sciences Ltd. 104-1 Moongi-dong Yuseong-gu Daejeon 305-380 / KR | |||
07 /
SHIM, Dong Sup R&D Park LG Life Sciences Ltd. 104-1 Moongi-dong Yuseong-gu Daejeon 305-380 / KR | |||
08 /
CHUNG, Soo Yong R&D Park LG Life Sciences Ltd. 104-1 Moongi-dong Yuseong-gu Daejeon 305-380 / KR | |||
09 /
LEE, Hyun Min R&D Park LG Life Sciences Ltd. 104-1 Moongi-dong Yuseong-gu Daejeon 305-380 / KR | Representative(s) | Busher, Samantha Jane, et al Elkington and Fife LLP 3-4 Holborn Circus London, EC1N 2HA / GB | [2014/27] |
Former [2013/38] | Gillard, Richard Edward Elkington and Fife LLP Thavies Inn House 3-4 Holborn Circus London EC1N 2HA / GB | ||
Former [2011/31] | Gillard, Richard Edward Elkington and Fife LLP Thavies Inn House 3-4 Holborn Circus London EC1N 2HA / GB | Application number, filing date | 09826254.6 | 10.11.2009 | [2011/31] | WO2009KR06568 | Priority number, date | KR20080112403 | 12.11.2008 Original published format: KR 20080112403 | [2011/31] | Filing language | EN | Procedural language | EN | Publication | Type: | A2 Application without search report | No.: | WO2010056022 | Date: | 20.05.2010 | Language: | EN | [2010/20] | Type: | A2 Application without search report | No.: | EP2350060 | Date: | 03.08.2011 | Language: | EN | The application published by WIPO in one of the EPO official languages on 20.05.2010 takes the place of the publication of the European patent application. | [2011/31] | Type: | B1 Patent specification | No.: | EP2350060 | Date: | 18.09.2013 | Language: | EN | [2013/38] | Search report(s) | International search report - published on: | KR | 10.09.2010 | (Supplementary) European search report - dispatched on: | EP | 22.06.2012 | Classification | IPC: | C07D403/14, C07D401/14, C07D403/06, C07D405/14, C07D409/14, A61K31/4025, A61P3/04, A61P3/10, A61P15/10, A61P29/00 | [2012/30] | CPC: |
C07D417/14 (EP,US);
C07D403/14 (KR);
A61K31/4025 (EP,KR,US);
A61K31/496 (EP,US);
A61P15/00 (EP);
A61P15/10 (EP);
A61P27/06 (EP);
A61P29/00 (EP);
A61P3/04 (EP);
A61P3/10 (EP);
A61P37/00 (EP);
A61P43/00 (EP);
C07D207/16 (EP,US);
C07D401/14 (EP,KR,US);
C07D403/06 (EP,US);
|
Former IPC [2011/31] | C07D403/14 | Designated contracting states | AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, SM, TR [2011/31] | Extension states | AL | Not yet paid | BA | Not yet paid | RS | Not yet paid | Title | German: | MELANOCORTIN-REZEPTOR-AGONISTEN | [2011/31] | English: | MELANOCORTIN RECEPTOR AGONISTS | [2011/31] | French: | ANTAGONISTES DE RÉCEPTEUR DE MÉLANOCORTINE | [2011/31] | Entry into regional phase | 06.05.2011 | National basic fee paid | 06.05.2011 | Search fee paid | 06.05.2011 | Designation fee(s) paid | 06.05.2011 | Examination fee paid | Examination procedure | 01.06.2010 | Request for preliminary examination filed International Preliminary Examining Authority: KR | 06.05.2011 | Examination requested [2011/31] | 21.01.2013 | Amendment by applicant (claims and/or description) | 27.03.2013 | Communication of intention to grant the patent | 06.08.2013 | Fee for grant paid | 06.08.2013 | Fee for publishing/printing paid | Divisional application(s) | The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is 27.03.2013 | Opposition(s) | 19.06.2014 | No opposition filed within time limit [2014/35] | Fees paid | Renewal fee | 14.11.2011 | Renewal fee patent year 03 | 13.11.2012 | Renewal fee patent year 04 |
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Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Lapses during opposition Tooltip | HU | 10.11.2009 | AT | 18.09.2013 | BE | 18.09.2013 | BG | 18.09.2013 | CY | 18.09.2013 | CZ | 18.09.2013 | DK | 18.09.2013 | EE | 18.09.2013 | ES | 18.09.2013 | FI | 18.09.2013 | HR | 18.09.2013 | IT | 18.09.2013 | LT | 18.09.2013 | LV | 18.09.2013 | MC | 18.09.2013 | MK | 18.09.2013 | MT | 18.09.2013 | NL | 18.09.2013 | PL | 18.09.2013 | RO | 18.09.2013 | SE | 18.09.2013 | SI | 18.09.2013 | SK | 18.09.2013 | SM | 18.09.2013 | IE | 10.11.2013 | LU | 10.11.2013 | CH | 30.11.2013 | LI | 30.11.2013 | NO | 18.12.2013 | GR | 19.12.2013 | IS | 18.01.2014 | PT | 20.01.2014 | [2015/41] |
Former [2015/34] | HU | 10.11.2009 | |
AT | 18.09.2013 | ||
BE | 18.09.2013 | ||
BG | 18.09.2013 | ||
CY | 18.09.2013 | ||
CZ | 18.09.2013 | ||
DK | 18.09.2013 | ||
EE | 18.09.2013 | ||
ES | 18.09.2013 | ||
FI | 18.09.2013 | ||
HR | 18.09.2013 | ||
IT | 18.09.2013 | ||
LT | 18.09.2013 | ||
LV | 18.09.2013 | ||
MC | 18.09.2013 | ||
MK | 18.09.2013 | ||
NL | 18.09.2013 | ||
PL | 18.09.2013 | ||
RO | 18.09.2013 | ||
SE | 18.09.2013 | ||
SI | 18.09.2013 | ||
SK | 18.09.2013 | ||
SM | 18.09.2013 | ||
IE | 10.11.2013 | ||
LU | 10.11.2013 | ||
CH | 30.11.2013 | ||
LI | 30.11.2013 | ||
NO | 18.12.2013 | ||
GR | 19.12.2013 | ||
IS | 18.01.2014 | ||
PT | 20.01.2014 | ||
Former [2015/32] | AT | 18.09.2013 | |
BE | 18.09.2013 | ||
CY | 18.09.2013 | ||
CZ | 18.09.2013 | ||
DK | 18.09.2013 | ||
EE | 18.09.2013 | ||
ES | 18.09.2013 | ||
FI | 18.09.2013 | ||
HR | 18.09.2013 | ||
IT | 18.09.2013 | ||
LT | 18.09.2013 | ||
LV | 18.09.2013 | ||
MC | 18.09.2013 | ||
MK | 18.09.2013 | ||
NL | 18.09.2013 | ||
PL | 18.09.2013 | ||
RO | 18.09.2013 | ||
SE | 18.09.2013 | ||
SI | 18.09.2013 | ||
SK | 18.09.2013 | ||
SM | 18.09.2013 | ||
IE | 10.11.2013 | ||
CH | 30.11.2013 | ||
LI | 30.11.2013 | ||
NO | 18.12.2013 | ||
GR | 19.12.2013 | ||
IS | 18.01.2014 | ||
PT | 20.01.2014 | ||
Former [2015/24] | AT | 18.09.2013 | |
BE | 18.09.2013 | ||
CY | 18.09.2013 | ||
CZ | 18.09.2013 | ||
DK | 18.09.2013 | ||
EE | 18.09.2013 | ||
ES | 18.09.2013 | ||
FI | 18.09.2013 | ||
HR | 18.09.2013 | ||
IT | 18.09.2013 | ||
LT | 18.09.2013 | ||
LV | 18.09.2013 | ||
MC | 18.09.2013 | ||
NL | 18.09.2013 | ||
PL | 18.09.2013 | ||
RO | 18.09.2013 | ||
SE | 18.09.2013 | ||
SI | 18.09.2013 | ||
SK | 18.09.2013 | ||
SM | 18.09.2013 | ||
IE | 10.11.2013 | ||
CH | 30.11.2013 | ||
LI | 30.11.2013 | ||
NO | 18.12.2013 | ||
GR | 19.12.2013 | ||
IS | 18.01.2014 | ||
PT | 20.01.2014 | ||
Former [2015/23] | AT | 18.09.2013 | |
BE | 18.09.2013 | ||
CY | 18.09.2013 | ||
CZ | 18.09.2013 | ||
DK | 18.09.2013 | ||
EE | 18.09.2013 | ||
ES | 18.09.2013 | ||
FI | 18.09.2013 | ||
HR | 18.09.2013 | ||
IT | 18.09.2013 | ||
LT | 18.09.2013 | ||
LV | 18.09.2013 | ||
MC | 18.09.2013 | ||
NL | 18.09.2013 | ||
PL | 18.09.2013 | ||
RO | 18.09.2013 | ||
SE | 18.09.2013 | ||
SI | 18.09.2013 | ||
SK | 18.09.2013 | ||
IE | 10.11.2013 | ||
CH | 30.11.2013 | ||
LI | 30.11.2013 | ||
NO | 18.12.2013 | ||
GR | 19.12.2013 | ||
IS | 18.01.2014 | ||
PT | 20.01.2014 | ||
Former [2014/48] | AT | 18.09.2013 | |
BE | 18.09.2013 | ||
CY | 18.09.2013 | ||
CZ | 18.09.2013 | ||
DK | 18.09.2013 | ||
EE | 18.09.2013 | ||
ES | 18.09.2013 | ||
FI | 18.09.2013 | ||
HR | 18.09.2013 | ||
IT | 18.09.2013 | ||
LT | 18.09.2013 | ||
LV | 18.09.2013 | ||
MC | 18.09.2013 | ||
NL | 18.09.2013 | ||
PL | 18.09.2013 | ||
SE | 18.09.2013 | ||
SI | 18.09.2013 | ||
SK | 18.09.2013 | ||
IE | 10.11.2013 | ||
CH | 30.11.2013 | ||
LI | 30.11.2013 | ||
NO | 18.12.2013 | ||
GR | 19.12.2013 | ||
IS | 18.01.2014 | ||
PT | 20.01.2014 | ||
Former [2014/41] | AT | 18.09.2013 | |
BE | 18.09.2013 | ||
CY | 18.09.2013 | ||
CZ | 18.09.2013 | ||
DK | 18.09.2013 | ||
EE | 18.09.2013 | ||
ES | 18.09.2013 | ||
FI | 18.09.2013 | ||
HR | 18.09.2013 | ||
IT | 18.09.2013 | ||
LT | 18.09.2013 | ||
LV | 18.09.2013 | ||
MC | 18.09.2013 | ||
NL | 18.09.2013 | ||
PL | 18.09.2013 | ||
SE | 18.09.2013 | ||
SI | 18.09.2013 | ||
SK | 18.09.2013 | ||
CH | 30.11.2013 | ||
LI | 30.11.2013 | ||
NO | 18.12.2013 | ||
GR | 19.12.2013 | ||
IS | 18.01.2014 | ||
PT | 20.01.2014 | ||
Former [2014/38] | AT | 18.09.2013 | |
BE | 18.09.2013 | ||
CY | 18.09.2013 | ||
CZ | 18.09.2013 | ||
EE | 18.09.2013 | ||
ES | 18.09.2013 | ||
FI | 18.09.2013 | ||
HR | 18.09.2013 | ||
IT | 18.09.2013 | ||
LT | 18.09.2013 | ||
LV | 18.09.2013 | ||
MC | 18.09.2013 | ||
NL | 18.09.2013 | ||
PL | 18.09.2013 | ||
SE | 18.09.2013 | ||
SI | 18.09.2013 | ||
SK | 18.09.2013 | ||
CH | 30.11.2013 | ||
LI | 30.11.2013 | ||
NO | 18.12.2013 | ||
GR | 19.12.2013 | ||
IS | 18.01.2014 | ||
PT | 20.01.2014 | ||
Former [2014/34] | AT | 18.09.2013 | |
BE | 18.09.2013 | ||
CY | 18.09.2013 | ||
CZ | 18.09.2013 | ||
EE | 18.09.2013 | ||
ES | 18.09.2013 | ||
FI | 18.09.2013 | ||
HR | 18.09.2013 | ||
LT | 18.09.2013 | ||
LV | 18.09.2013 | ||
MC | 18.09.2013 | ||
NL | 18.09.2013 | ||
PL | 18.09.2013 | ||
SE | 18.09.2013 | ||
SI | 18.09.2013 | ||
SK | 18.09.2013 | ||
CH | 30.11.2013 | ||
LI | 30.11.2013 | ||
NO | 18.12.2013 | ||
GR | 19.12.2013 | ||
IS | 18.01.2014 | ||
PT | 20.01.2014 | ||
Former [2014/33] | AT | 18.09.2013 | |
BE | 18.09.2013 | ||
CY | 18.09.2013 | ||
CZ | 18.09.2013 | ||
EE | 18.09.2013 | ||
ES | 18.09.2013 | ||
FI | 18.09.2013 | ||
HR | 18.09.2013 | ||
LT | 18.09.2013 | ||
LV | 18.09.2013 | ||
MC | 18.09.2013 | ||
NL | 18.09.2013 | ||
PL | 18.09.2013 | ||
SE | 18.09.2013 | ||
SI | 18.09.2013 | ||
SK | 18.09.2013 | ||
NO | 18.12.2013 | ||
GR | 19.12.2013 | ||
IS | 18.01.2014 | ||
PT | 20.01.2014 | ||
Former [2014/28] | AT | 18.09.2013 | |
BE | 18.09.2013 | ||
CY | 18.09.2013 | ||
CZ | 18.09.2013 | ||
EE | 18.09.2013 | ||
ES | 18.09.2013 | ||
FI | 18.09.2013 | ||
HR | 18.09.2013 | ||
LT | 18.09.2013 | ||
LV | 18.09.2013 | ||
NL | 18.09.2013 | ||
PL | 18.09.2013 | ||
SE | 18.09.2013 | ||
SI | 18.09.2013 | ||
SK | 18.09.2013 | ||
NO | 18.12.2013 | ||
GR | 19.12.2013 | ||
IS | 18.01.2014 | ||
PT | 20.01.2014 | ||
Former [2014/24] | AT | 18.09.2013 | |
BE | 18.09.2013 | ||
CY | 18.09.2013 | ||
CZ | 18.09.2013 | ||
EE | 18.09.2013 | ||
ES | 18.09.2013 | ||
FI | 18.09.2013 | ||
HR | 18.09.2013 | ||
LT | 18.09.2013 | ||
LV | 18.09.2013 | ||
NL | 18.09.2013 | ||
PL | 18.09.2013 | ||
SE | 18.09.2013 | ||
SI | 18.09.2013 | ||
SK | 18.09.2013 | ||
NO | 18.12.2013 | ||
GR | 19.12.2013 | ||
IS | 18.01.2014 | ||
Former [2014/23] | BE | 18.09.2013 | |
CY | 18.09.2013 | ||
CZ | 18.09.2013 | ||
EE | 18.09.2013 | ||
FI | 18.09.2013 | ||
HR | 18.09.2013 | ||
LT | 18.09.2013 | ||
LV | 18.09.2013 | ||
NL | 18.09.2013 | ||
SE | 18.09.2013 | ||
SI | 18.09.2013 | ||
SK | 18.09.2013 | ||
NO | 18.12.2013 | ||
GR | 19.12.2013 | ||
IS | 18.01.2014 | ||
Former [2014/22] | BE | 18.09.2013 | |
CY | 18.09.2013 | ||
FI | 18.09.2013 | ||
HR | 18.09.2013 | ||
LT | 18.09.2013 | ||
LV | 18.09.2013 | ||
NL | 18.09.2013 | ||
SE | 18.09.2013 | ||
SI | 18.09.2013 | ||
NO | 18.12.2013 | ||
GR | 19.12.2013 | ||
Former [2014/18] | BE | 18.09.2013 | |
CY | 18.09.2013 | ||
FI | 18.09.2013 | ||
HR | 18.09.2013 | ||
LT | 18.09.2013 | ||
LV | 18.09.2013 | ||
SE | 18.09.2013 | ||
SI | 18.09.2013 | ||
NO | 18.12.2013 | ||
GR | 19.12.2013 | ||
Former [2014/12] | CY | 26.06.2013 | |
FI | 18.09.2013 | ||
HR | 18.09.2013 | ||
LT | 18.09.2013 | ||
LV | 18.09.2013 | ||
SE | 18.09.2013 | ||
SI | 18.09.2013 | ||
NO | 18.12.2013 | ||
GR | 19.12.2013 | ||
Former [2014/10] | CY | 26.06.2013 | |
HR | 18.09.2013 | ||
LT | 18.09.2013 | ||
SE | 18.09.2013 | ||
NO | 18.12.2013 | ||
Former [2014/09] | HR | 18.09.2013 | |
LT | 18.09.2013 | ||
SE | 18.09.2013 | ||
NO | 18.12.2013 | ||
Former [2014/08] | LT | 18.09.2013 | |
NO | 18.12.2013 | ||
Former [2014/07] | NO | 18.12.2013 | Documents cited: | Search | [YD]WO2005047251 (LG LIFE SCIENCES LTD [KR], et al) [YD] 1-15* examples 7-186,190-293; claim - *; | [YD]WO2008007930 (LG LIFE SCIENCES LTD [KR], et al) [YD] 1-15 * examples A8,A55,A86,A93-A96; table 18 * | International search | [A]US6534503 (DINES KEVIN C [US], et al); | [A]US2003236262 (BAKSHI RAMAN K [US], et al); | [A]US2004019094 (LUNDSTEDT TORBJORN [SE], et al); | [A]US2007129346 (LEE KOO [KR], et al); | [A] - HERPIN, TIMOTHY F. ET AL., "Discovery of Tyrosine-Based Potent and Selective Melanocortin-1 Receptor Small-Molecule Agonists with Anti-inflammatory Properties", J. MED. CHEM., (2003), vol. 46, pages 1123 - 1126, XP001182772 DOI: http://dx.doi.org/10.1021/jm025600i | by applicant | WO0155109 | WO0170337 | WO0170708 | WO0215909 | WO0218327 | WO02059095 | WO02059107 | WO02059117 | WO02059108 | WO02067869 | WO02068387 | WO02068388 | WO02081443 | WO02085925 | WO03009847 | WO03009850 | WO2004078716 | WO2004078717 | WO2004087159 | WO2005040109 | WO2005047251 | WO2005077935 | WO2006019787 | WO2006020277 | WO2006072393 | WO2007015157 | WO2007015162 | WO2007041052 | WO2007041061 | WO2007047496 | JP2007131570 | WO2007096186 | WO2007096763 | WO2007141343 | WO2008007930 | WO2008039418 | - J. MED. CHEM., (2002), vol. 45, page 4589 | - BIOORG. MED. CHEM. LETT., (2005), vol. 15, page 171 | - BIOORG. MED. CHEM. LETT., (2005), vol. 15, page 3430 | - BIOORG. MED. CHEM. LETT., (2005), vol. 15, page 350 1 | - J MED CHEM, (2003), vol. 46, page 1123 |