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Extract from the Register of European Patents

EP About this file: EP2258400

EP2258400 - Multivalent VLA-4 antagonists comprising polymer moieties [Right-click to bookmark this link]
StatusThe application is deemed to be withdrawn
Status updated on  10.07.2015
Database last updated on 14.06.2024
Most recent event   Tooltip10.07.2015Application deemed to be withdrawnpublished on 12.08.2015  [2015/33]
Applicant(s)For all designated states
ELAN PHARMACEUTICALS, INC.
800 Gateway Boulevard
South San Francisco, CA 94080 / US
[2010/49]
Inventor(s)01 / Konradi, Andrei, W.
30 Victoria Road
Burlingame, CA 94010 / US
02 / Pleiss, Michael, A.
848 Stella Court
Sunnyvale, CA 94087 / US
03 / Semko, Christopher, M.
4993 Norris Road
Fremont, CA 94536 / US
04 / Yednock, Theodore
184 Arroyo Road
Forest Knolls, CA 94933 / US
05 / Smith, Jenifer, L.
1770 W 13th Avenue
Eugene, Oregon 97402 / US
 [2011/14]
Former [2011/08]01 / Konradi, Andrei, W.
30 Victoria Road
Burlingame, CA 94010 / US
02 / Pleiss, Michael, A.
848 Stella Court
Sunnyvale, CA 94087 / US
03 / Semko, Christopher, M.
4993 Norris Road
Fremont, CA 94536 / US
04 / Yednock, Theodore
184 Arroyo Road
Forest Knolls, CA 94933 / US
05 / Smith, Jenifer, L.
1770 W 13th Avenue
Eugene, Oregon 97402 / US
Former [2010/49]01 / Konradi, Andrei, W.
30 Victoria Road
Burlingame, CA 94010 / US
02 / Pleiss, Michael, A.
848 Stella Court
Sunnyvale, CA 94087 / US
03 / Semko, Christopher, M.
4993 Norris Road
Fremont, CA 94536 / US
04 / Yednock, Theodore
184 Arroyo Road
Forest Knolls, CA 94933 / US
05 / Smith, Jenifer, L.
512 Cortesti Avenue
San Francisco, CA 94080 / US
Representative(s)Smaggasgale, Gillian Helen, et al
WP Thompson
138 Fetter Lane
London EC4A 1BT / GB
[N/P]
Former [2011/08]Smaggasgale, Gillian Helen, et al
W.P. Thompson & Co 55 Drury Lane
London WC2B 5SQ / GB
Former [2010/49]Smaggasgale, Gillian Helen
W.P. Thompson & Co 55 Drury Lane
London WC2B 5SQ / GB
Application number, filing date10180274.208.07.2005
[2010/49]
Priority number, dateUS20040586975P08.07.2004         Original published format: US 586975 P
[2010/49]
Filing languageEN
Procedural languageEN
PublicationType: A2 Application without search report 
No.:EP2258400
Date:08.12.2010
Language:EN
[2010/49]
Type: A3 Search report 
No.:EP2258400
Date:10.08.2011
[2011/32]
Search report(s)(Supplementary) European search report - dispatched on:EP13.07.2011
ClassificationIPC:A61K47/48, A61P37/00
[2010/49]
CPC:
A61K31/785 (EP,KR,US); C07D417/12 (KR); A61K45/06 (US);
A61K47/50 (KR); A61K47/60 (EP,US); A61P1/00 (EP);
A61P1/02 (EP); A61P1/04 (EP); A61P1/16 (EP);
A61P11/00 (EP); A61P11/02 (EP); A61P11/06 (EP);
A61P13/02 (EP); A61P13/10 (EP); A61P17/00 (EP);
A61P17/04 (EP); A61P17/06 (EP); A61P19/02 (EP);
A61P21/00 (EP); A61P25/00 (EP); A61P25/28 (EP);
A61P27/02 (EP); A61P29/00 (EP); A61P3/10 (EP);
A61P31/12 (EP); A61P31/18 (EP); A61P35/00 (EP);
A61P35/04 (EP); A61P37/00 (EP); A61P37/02 (EP);
A61P37/04 (EP); A61P37/06 (EP); A61P37/08 (EP);
A61P5/00 (EP); A61P5/14 (EP); A61P7/06 (EP);
A61P9/00 (EP); A61P9/04 (EP); A61P9/10 (EP);
A61P9/14 (EP); A61Q5/00 (EP,US) (-)
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   NL,   PL,   PT,   RO,   SE,   SI,   SK,   TR [2010/49]
Extension statesALNot yet paid
BANot yet paid
HRNot yet paid
MKNot yet paid
YUNot yet paid
TitleGerman:Multivalente VLA-4-Antagonisten enthaltend Polymeren[2010/49]
English:Multivalent VLA-4 antagonists comprising polymer moieties[2010/49]
French:Antagonistes multivalents de l'antigène VLA-4 comprénant des polymères[2010/49]
Examination procedure10.02.2012Examination requested  [2012/12]
01.06.2012Amendment by applicant (claims and/or description)
04.03.2013Despatch of a communication from the examining division (Time limit: M06)
03.09.2013Reply to a communication from the examining division
03.02.2015Application deemed to be withdrawn, date of legal effect  [2015/33]
24.03.2015Despatch of communication that the application is deemed to be withdrawn, reason: renewal fee not paid in time  [2015/33]
Parent application(s)   TooltipEP05770402.5  / EP1765412
Divisional application(s)The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued (EP20050770402) is  22.01.2008
Request for further processing for:The application is deemed to be withdrawn due to failure to reply to the Extended European Search Report/Written Opinion of the International Searching Authority/International Preliminary Examination Report/Supplementary international search report/Supplementary European search report
01.06.2012Request for further processing filed
01.06.2012Full payment received (date of receipt of payment)
Request granted
28.06.2012Decision despatched
Fees paidRenewal fee
27.09.2010Renewal fee patent year 03
27.09.2010Renewal fee patent year 04
27.09.2010Renewal fee patent year 05
27.09.2010Renewal fee patent year 06
12.07.2011Renewal fee patent year 07
13.07.2012Renewal fee patent year 08
10.07.2013Renewal fee patent year 09
Penalty fee
Additional fee for renewal fee
31.07.201410   M06   Not yet paid
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Patent Court
See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Documents cited:Search[A]WO0154690  (BIOGEN INC [US], et al) [A] 1-22 * Claims *;
 [AP]WO2005000244  (ELAN PHARM INC [US], et al) [AP] 1-22 * page 268 line 9-page 279; page 613-618 *;
 [A]  - HURYN D M ET AL, Synthesis, characterization and evaluation of pro-drugs of VLA-4 antagonists, BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, OXFORD, GB, PAGE(S) 1651-1654, (200404), ISSN 0960-894X, XP002327663 [A] 1-22 * abstract * * page 1653, column 1, paragraph 2; figure 1 *

DOI:   http://dx.doi.org/10.1016/j.bmcl.2004.01.062
 [AP]  - PEPINSKY R. B. ET AL, "Design, synthesis and analysis of a polyethylene glycol-modified (PEGylated) small molecule inhibitor of integrin a4b1 with improved pharmaceutical properties", JOURNAL OF PHARMOCOLOGY AND EXPERIMENTAL THERAPEUTICS, (20050201), vol. 312, no. 2, pages 742 - 750, XP008067961 [AP] 1-22 * see discussion; page 744, column 1; figures 1,2; tables 1,2 *

DOI:   http://dx.doi.org/10.1124/jpet.104.075648
by applicantUS4235871
 US4501728
 US4837028
 US5011472
 US5023252
 WO9216555
 US5177059
 US5824701
 WO9853817
 US5880131
 WO0154690
 US6436904
 US6489300
 US6664331
 US2004043030
 US6716821
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The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.