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EP About this file: EP2311455

EP2311455 - Compounds for nonsense suppression, and methods for their use [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  20.05.2016
Database last updated on 14.09.2024
Most recent event   Tooltip13.10.2017Lapse of the patent in a contracting state
New state(s): BG, CY, HU, NL, TR
published on 15.11.2017  [2017/46]
Applicant(s)For all designated states
PTC Therapeutics, Inc.
100 Corporate Court
South Plainfield, NJ 07080 / US
[2011/16]
Inventor(s)01 / Almstead, Neil
179 Longview Drive
Princeton, NJ 08540 / US
02 / Chen, Guangming
1402 Stech Drive
Bridgewater, NJ 08807 / US
03 / Karp, Gary Mitchell
37 Cartwright Drive
Princeton Junction, NJ 08550 / US
04 / Welch, Ellen
33 Hollow Brook Road
Califon, NJ 07830 / US
05 / Wilde, Richard Gerald
13 Cascades Terrace
Sommerville, NJ 08876 / US
06 / Campbell, Jeffrey Allen
328 Adams Street
Apt. 103
Bethlehem, PA 18015 / US
 [2015/29]
Former [2011/34]01 / Almstead, Neil
179 Longview Drive
Princeton, NJ 08540 / US
02 / Chen, Guangming
1402 Stech Drive
Bridgewater, NJ 08807 / US
03 / Karp, Gary Mitchell
37 Cartwright Drive
Princeton Junction, NJ 08550 / US
04 / Welch, Ellen
33 Hollow Brook Road
Califon, NJ 07830 / US
05 / Wilde, Richard Gerald
13 Cascades Terrace
Sommerville, NJ 08876 / US
06 / Campbell, Jeffrey Allen
328 Adams Street Apt. 103
Bethlehem, PA 18015 / US
Former [2011/16]01 / Almstead, Neil
179 Longview Drive
Princeton, NJ 08540 / US
02 / Chen, Guangming
1402 Stech Drive
Bridgewater, NJ 08807 / US
03 / Karp, Gary Mitchell
37 Cartwright Drive
Princeton Junction, NJ 08550 / US
04 / Welch, Ellen
33 Hollow Brook Road
Califon, NJ 07830 / US
05 / Wilde, Richard Gerald
13 Cascades Terrace
Sommerville, NJ 08876 / US
06 / Campbell, Jeffrey Allen
31 Bell Avenue
Glen Gardner, NJ 08826 / US
Representative(s)Uexküll & Stolberg
Partnerschaft von
Patent- und Rechtsanwälten mbB
Beselerstraße 4
22607 Hamburg / DE
[N/P]
Former [2015/29]UEXKÜLL & STOLBERG
Patentanwälte
Beselerstrasse 4
22607 Hamburg / DE
Former [2011/16]UEXKÜLL & STOLBERG
Patentanwälte Beselerstrasse 4
22607 Hamburg / DE
Application number, filing date10185130.113.10.2005
[2011/16]
Priority number, dateUS20040617653P13.10.2004         Original published format: US 617653 P
US20040617670P13.10.2004         Original published format: US 617670 P
US20040617633P13.10.2004         Original published format: US 617633 P
US20040617634P13.10.2004         Original published format: US 617634 P
US20040617655P13.10.2004         Original published format: US 617655 P
US20040624170P03.11.2004         Original published format: US 624170 P
[2011/16]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report 
No.:EP2311455
Date:20.04.2011
Language:EN
[2011/16]
Type: B1 Patent specification 
No.:EP2311455
Date:15.07.2015
Language:EN
[2015/29]
Search report(s)(Supplementary) European search report - dispatched on:EP17.02.2011
ClassificationIPC:A61K31/4245, A61K31/433, A61P35/00, C07D417/10, C07D277/30
[2011/16]
CPC:
C07D271/06 (EP,US); A61K31/4155 (KR); A61K31/53 (KR);
A61P1/16 (EP); A61P11/00 (EP); A61P13/12 (EP);
A61P19/00 (EP); A61P19/02 (EP); A61P19/08 (EP);
A61P21/00 (EP); A61P25/00 (EP); A61P25/16 (EP);
A61P25/28 (EP); A61P27/02 (EP); A61P29/00 (EP);
A61P3/04 (EP); A61P3/06 (EP); A61P3/10 (EP);
A61P35/00 (EP); A61P35/02 (EP); A61P37/00 (EP);
A61P37/02 (EP); A61P37/06 (EP); A61P43/00 (EP);
A61P5/14 (EP); A61P7/00 (EP); A61P7/04 (EP);
A61P9/00 (EP); A61P9/10 (EP); C07D231/12 (EP,US);
C07D233/64 (EP,US); C07D249/08 (EP,US); C07D251/24 (EP,US);
C07D261/08 (EP,US); C07D263/32 (EP,US); C07D271/10 (EP,US);
C07D271/107 (EP,US); C07D277/30 (EP,US); C07D285/12 (EP,US);
C07D307/68 (EP,US); C07D333/24 (EP,US); C07D401/04 (EP,US);
C07D403/04 (EP,US); C07D405/04 (EP,US); C07D409/04 (EP,US);
C07D413/04 (EP,US); C07D413/06 (EP,US); C07D413/12 (EP,KR,US);
C07D417/04 (EP,US); C07F9/65306 (US) (-)
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   NL,   PL,   PT,   RO,   SE,   SI,   SK,   TR [2015/29]
Former [2011/16]AT,  BE,  BG,  CH,  CY,  CZ,  DE,  DK,  EE,  ES,  FI,  FR,  GB,  GR,  HU,  IE,  IS,  IT,  LI,  LT,  LU,  LV,  MC,  NL,  PL,  PT,  RO,  SE,  SI,  SK,  TR 
TitleGerman:Verbindungen zur Nonsense-Unterdrückung und Verfahren zu deren Verwendung[2011/16]
English:Compounds for nonsense suppression, and methods for their use[2011/16]
French:Composes de suppression de non-sens et procedes de leur utilisation[2011/16]
Examination procedure20.10.2011Amendment by applicant (claims and/or description)
20.10.2011Examination requested  [2011/48]
06.02.2013Despatch of a communication from the examining division (Time limit: M04)
17.06.2013Reply to a communication from the examining division
14.11.2013Communication of intention to grant the patent
12.03.2014Receipt of the translation of the claim(s)
14.03.2014Disapproval of the communication of intention to grant the patent by the applicant or resumption of examination proceedings by the EPO
10.04.2014Communication of intention to grant the patent
19.08.2014Disapproval of the communication of intention to grant the patent by the applicant or resumption of examination proceedings by the EPO
08.01.2015Communication of intention to grant the patent
15.05.2015Fee for grant paid
15.05.2015Fee for publishing/printing paid
15.05.2015Receipt of the translation of the claim(s)
Parent application(s)   TooltipEP05815159.8  / EP1815206
Divisional application(s)The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued (EP20050815159) is  27.05.2008
Opposition(s)18.04.2016No opposition filed within time limit [2016/25]
Fees paidRenewal fee
06.12.2010Renewal fee patent year 03
06.12.2010Renewal fee patent year 04
06.12.2010Renewal fee patent year 05
06.12.2010Renewal fee patent year 06
25.10.2011Renewal fee patent year 07
26.10.2012Renewal fee patent year 08
30.10.2013Renewal fee patent year 09
14.10.2014Renewal fee patent year 10
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court
See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipHU13.10.2005
AT15.07.2015
BE15.07.2015
BG15.07.2015
CY15.07.2015
CZ15.07.2015
DK15.07.2015
EE15.07.2015
ES15.07.2015
FI15.07.2015
IS15.07.2015
IT15.07.2015
LT15.07.2015
LV15.07.2015
MC15.07.2015
NL15.07.2015
PL15.07.2015
RO15.07.2015
SE15.07.2015
SI15.07.2015
SK15.07.2015
TR15.07.2015
IE13.10.2015
LU13.10.2015
GR16.10.2015
CH31.10.2015
LI31.10.2015
PT16.11.2015
[2017/39]
Former [2017/03]AT15.07.2015
BE15.07.2015
CZ15.07.2015
DK15.07.2015
EE15.07.2015
ES15.07.2015
FI15.07.2015
IS15.07.2015
IT15.07.2015
LT15.07.2015
LV15.07.2015
MC15.07.2015
PL15.07.2015
RO15.07.2015
SE15.07.2015
SI15.07.2015
SK15.07.2015
IE13.10.2015
LU13.10.2015
GR16.10.2015
CH31.10.2015
LI31.10.2015
PT16.11.2015
Former [2016/45]AT15.07.2015
CZ15.07.2015
DK15.07.2015
EE15.07.2015
ES15.07.2015
FI15.07.2015
IS15.07.2015
IT15.07.2015
LT15.07.2015
LV15.07.2015
MC15.07.2015
PL15.07.2015
RO15.07.2015
SE15.07.2015
SI15.07.2015
SK15.07.2015
IE13.10.2015
LU13.10.2015
GR16.10.2015
CH31.10.2015
LI31.10.2015
PT16.11.2015
Former [2016/36]AT15.07.2015
CZ15.07.2015
DK15.07.2015
EE15.07.2015
ES15.07.2015
FI15.07.2015
IS15.07.2015
IT15.07.2015
LT15.07.2015
LV15.07.2015
MC15.07.2015
PL15.07.2015
RO15.07.2015
SE15.07.2015
SI15.07.2015
SK15.07.2015
LU13.10.2015
GR16.10.2015
CH31.10.2015
LI31.10.2015
PT16.11.2015
Former [2016/34]AT15.07.2015
CZ15.07.2015
DK15.07.2015
EE15.07.2015
ES15.07.2015
FI15.07.2015
IS15.07.2015
IT15.07.2015
LT15.07.2015
LV15.07.2015
MC15.07.2015
PL15.07.2015
RO15.07.2015
SE15.07.2015
SK15.07.2015
LU13.10.2015
GR16.10.2015
CH31.10.2015
LI31.10.2015
PT16.11.2015
Former [2016/31]AT15.07.2015
CZ15.07.2015
DK15.07.2015
EE15.07.2015
ES15.07.2015
FI15.07.2015
IS15.07.2015
IT15.07.2015
LT15.07.2015
LV15.07.2015
MC15.07.2015
PL15.07.2015
RO15.07.2015
SE15.07.2015
SK15.07.2015
LU13.10.2015
GR16.10.2015
PT16.11.2015
Former [2016/28]AT15.07.2015
CZ15.07.2015
DK15.07.2015
EE15.07.2015
ES15.07.2015
FI15.07.2015
IT15.07.2015
LT15.07.2015
LV15.07.2015
MC15.07.2015
PL15.07.2015
RO15.07.2015
SE15.07.2015
SK15.07.2015
LU13.10.2015
GR16.10.2015
PT16.11.2015
Former [2016/26]AT15.07.2015
CZ15.07.2015
DK15.07.2015
EE15.07.2015
ES15.07.2015
FI15.07.2015
IT15.07.2015
LT15.07.2015
LV15.07.2015
PL15.07.2015
RO15.07.2015
SE15.07.2015
SK15.07.2015
LU13.10.2015
GR16.10.2015
PT16.11.2015
Former [2016/23]AT15.07.2015
CZ15.07.2015
DK15.07.2015
EE15.07.2015
ES15.07.2015
FI15.07.2015
IT15.07.2015
LT15.07.2015
LV15.07.2015
PL15.07.2015
RO15.07.2015
SE15.07.2015
SK15.07.2015
GR16.10.2015
PT16.11.2015
Former [2016/22]AT15.07.2015
CZ15.07.2015
DK15.07.2015
EE15.07.2015
ES15.07.2015
FI15.07.2015
IT15.07.2015
LT15.07.2015
LV15.07.2015
PL15.07.2015
SE15.07.2015
GR16.10.2015
PT16.11.2015
Former [2016/21]AT15.07.2015
DK15.07.2015
ES15.07.2015
FI15.07.2015
IT15.07.2015
LT15.07.2015
LV15.07.2015
PL15.07.2015
SE15.07.2015
GR16.10.2015
PT16.11.2015
Former [2016/20]AT15.07.2015
DK15.07.2015
ES15.07.2015
FI15.07.2015
LT15.07.2015
LV15.07.2015
PL15.07.2015
SE15.07.2015
GR16.10.2015
PT16.11.2015
Former [2016/11]AT15.07.2015
ES15.07.2015
FI15.07.2015
LT15.07.2015
LV15.07.2015
PL15.07.2015
SE15.07.2015
GR16.10.2015
PT16.11.2015
Former [2016/10]ES15.07.2015
FI15.07.2015
LT15.07.2015
LV15.07.2015
PL15.07.2015
SE15.07.2015
GR16.10.2015
PT16.11.2015
Former [2016/09]FI15.07.2015
LT15.07.2015
LV15.07.2015
GR16.10.2015
Former [2016/07]LT15.07.2015
Documents cited:Search[X]US3947263  (BROUWER WALTER G, et al) [X] 1 * column 6; compounds G,O *;
 [X]US3964896  (BROUWER WALTER G, et al) [X] 1 * column 9 - column 10; examples 29-31 *;
 [X]US4210762  (HOWE ROBERT K [US]) [X] 1 * examples 5,6,8 *;
 [X]DE3819037  (HOECHST AG [DE]) [X] 1-3 * example 43; claim - *;
 [X]EP0838453  (EISAI CO LTD [JP]) [X] 1-14 * page 2, line 10 - line 27; examples 18,19,22,23; claims 1,8-10 *;
 [X]EP0889032  (EISAI CO LTD [JP]) [X] 1-14 * page 3, line 13 - line 30; examples 1,62,63; claims 1,14-19 *;
 [X]WO02068417  (NPS PHARMA INC [US], et al) [X] 1-14 * page 46; examples 10,B147,B265; claims 1,7,8,10,14 *;
 [X]WO2004072050  (NOVARTIS AG [CH], et al) [X] 1-14 * examples 13-16; claim - *;
 [X]  - MACDONALD G J ET AL, "Design and Synthesis of trans-3(2-(4-((3-(3-(5-Methyl-1,2,4-oxadiozol yl))-phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-te trahydro1H-3-benzazepine (SB-414796): A Potent and Selective Dopamine D.sub.3 Receptor Antagonist", JOURNAL OF MEDICINAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY, WASHINGTON, US, (20031106), vol. 46, no. 23, doi:10.1021/JM030817D, ISSN 0022-2623, pages 4952 - 4964, XP002994764 [X] 1 * Schemes 1 and 2 *; page 4954, column r, line 25, paragraph 2 - line 28; compounds 31,33,56 *

DOI:   http://dx.doi.org/10.1021/jm030817d
by applicantUS4892538
 WO9325673
 US5283187
 US5681746
 US2003023185
 US6800604
 US6800731
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