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EP2454250
European procedure
Extract from the Register of European Patents
EP About this file: EP2454250
| EP2454250 - APOPTOSIS SIGNAL-REGULATING KINASE INHIBITORS [Right-click to bookmark this link] | Status | No opposition filed within time limit Status updated on 20.11.2015 Database last updated on 11.04.2026 | Most recent event Tooltip | 20.11.2015 | No opposition filed within time limit | published on 23.12.2015 [2015/52] | Applicant(s) | For all designated states Gilead Sciences, Inc. 333 Lakeside Drive Foster City, CA 94404 / US | [2012/21] | Inventor(s) | 01 /
CORKEY, Britton 355 Buena Vista Ave East Apt 415 San Francisco CA 94117 / US | 02 /
GRAUPE, Michael 1131 Banyan Way Pacifica CA 94044 / US | 03 /
KOCH, Keith 384 Baker Lane Erie CO 80516 / US | 04 /
MELVIN, Lawrence S. 7623 Crestview Drive Longmont CO 80504 / US | 05 /
NOTTE, Gregory 707 Highland Ave Apt 2 San Mateo CA 94401 / US | [2012/21] | Representative(s) | Wallace, Sheila Jane, et al Marks & Clerk LLP 15 Fetter Lane London EC4A 1BW / GB | [N/P] |
| Former [2015/03] | Wallace, Sheila Jane, et al Marks & Clerk LLP 90 Long Acre London WC2E 9RA / GB | ||
| Former [2014/27] | Wallace, Sheila Jane, et al Marks & Clerk LLP 90 Long Acre London WC2E 9RA / GB | ||
| Former [2012/21] | Schnappauf, Georg, et al Dr. Volker Vossius Patent- und Rechtsanwaltskanzlei Geibelstrasse 6 81679 München / DE | Application number, filing date | 10733116.7 | 12.07.2010 | WO2010US41739 | Priority number, date | US20090289263P | 22.12.2009 Original published format: US 289263 P | US20090225076P | 13.07.2009 Original published format: US 225076 P | US20090225079P | 13.07.2009 Original published format: US 225079 P | [2012/21] | Filing language | EN | Procedural language | EN | Publication | Type: | A1 Application with search report | No.: | WO2011008709 | Date: | 20.01.2011 | Language: | EN | [2011/03] | Type: | A1 Application with search report | No.: | EP2454250 | Date: | 23.05.2012 | Language: | EN | The application published by WIPO in one of the EPO official languages on 20.01.2011 takes the place of the publication of the European patent application. | [2012/21] | Type: | B1 Patent specification | No.: | EP2454250 | Date: | 14.01.2015 | Language: | EN | [2015/03] | Search report(s) | International search report - published on: | EP | 20.01.2011 | Classification | IPC: | C07D401/12, C07D401/14, C07D407/14, C07D413/14, C07D471/04, C07D491/048, A61K31/437, A61K31/4439, A61K31/444, A61K31/497, A61K31/506, A61P9/00, A61P25/28, A61P29/00, A61P37/00 | [2012/21] | CPC: |
A61K31/444 (EP,US);
C07D401/12 (EP,KR,US);
A61K31/4196 (EP);
A61K31/4439 (EP,KR,US);
A61K31/4709 (US);
A61K31/496 (US);
A61K31/497 (US);
A61K31/506 (EP,US);
A61K31/5377 (US);
A61K31/585 (US);
A61K45/06 (US);
A61P25/28 (EP);
A61P29/00 (EP);
A61P37/00 (EP);
A61P9/00 (EP);
C07D401/14 (EP,US);
C07D405/14 (US);
C07D413/12 (US);
C07D413/14 (US);
C07D417/14 (US);
C07D471/04 (KR,US);
C07D491/048 (KR,US)
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| Designated contracting states | AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, SM, TR [2012/21] | Extension states | BA | 10.02.2012 | ME | 10.02.2012 | RS | 10.02.2012 | Title | German: | APOPTOSESIGNALREGULIERENDE KINASEHEMMER | [2012/21] | English: | APOPTOSIS SIGNAL-REGULATING KINASE INHIBITORS | [2012/21] | French: | INHIBITEURS DE LA KINASE RÉGULANT LES SIGNAUX DE L'APOPTOSE | [2012/21] | Entry into regional phase | 23.01.2012 | National basic fee paid | 23.01.2012 | Designation fee(s) paid | 23.01.2012 | Examination fee paid | Examination procedure | 23.01.2012 | Amendment by applicant (claims and/or description) | 23.01.2012 | Examination requested [2012/21] | 16.10.2012 | Despatch of a communication from the examining division (Time limit: M06) | 02.04.2013 | Reply to a communication from the examining division | 04.08.2014 | Communication of intention to grant the patent | 03.12.2014 | Fee for grant paid | 03.12.2014 | Fee for publishing/printing paid | 03.12.2014 | Receipt of the translation of the claim(s) | Divisional application(s) | EP15151030.2 / EP2933252 | EP17208659.7 / EP3363797 | EP20210819.7 | The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is 16.10.2012 | Opposition(s) | 15.10.2015 | No opposition filed within time limit [2015/52] | Fees paid | Renewal fee | 25.07.2012 | Renewal fee patent year 03 | 29.07.2013 | Renewal fee patent year 04 | 28.07.2014 | Renewal fee patent year 05 |
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| Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Cited in | International search | [I] EP2058309 (TAKEDA PHARMACEUTICAL et al.) [I] 1-36 * claims 1, 14-18 * * page 98 - page 99; examples 88, 89 * * page 1, paragraph [0001] * * ASK1 inhibitory activity; page 220 - page 221 * | by applicant | US2007276050 | US2007167386 | WO2009027283 | US3845770 | US4326525 | US4902514 | US5616345 | US5023252 | US4992445 | US5001139 | KUMAR, S.; BOEHM, J.; LEE., J.C., NAT. REV. DRUG DIS., vol. 2, 2003, pages 717 - 726 | PIMIENTA, G.; PASCUAL, J., CELL CYCLE, vol. 6, 2007, pages 2826 - 2632 | ICHIJO, H.; NISHIDA, E.; IRIE, K.; DIJKE, P. T.; SAITOH, M.; MORIGUCHI, T.; MATSUMOTO, K.; MIYAZONO, K.; GOTOH, Y., SCIENCE, vol. 275, 1997, pages 90 - 94 | HATTORI, K; NAGURO, I; RUNCHEL, C; ICHIJO, H, CELL COMM. SIGNA, vol. 7, 2009, pages 1 - 10 | TAKEDA, K.; NOGUCHI, T.; NAGURO, I.; ICHIJO, H., ANNU. REV. PHARMACOL. TOXICOL., vol. 48, 2007, pages 1 - 8.27 | NAGAI, H.; NOGUCHI, T.; TAKCDA, K.; ICHIJO, 1., J. BIOCHCM. MOL. BIOL., vol. 40, 2007, pages 1 - 6 | WANG, X. S.; DIENER, K.; TAN, T-H.; YAO, Z., BIOCHEM. BIOPHYS. RES. COMMUN., vol. 253, 1998, pages 33 - 37 | TAKEDA, K.; SHIMOZONO, R.; NOGUCHI, T.; UMEDA, T.; MORIMOTO, Y.; NAGURO, I.; TOBIUME, K.; SAITOH, M.; MATSUZAWA, A.; ICHIJO, H., J. BIOL. CHEM., vol. 282, 2007, pages 7522 - 7531 | IRIYAMA, T. ET AL., EMBO J., vol. 28, 2009, pages 843 - 853 | SAITOH, M.; NISHITOH, H.; FUJI, M.; TAKEDA, K.; TOBIUME, K.; SAWADA, Y.; KAWABATA, M.; MIYAZONO, K.; LCHIJO, H., EMBO J., vol. 17, 1998, pages 2596 - 2606 | ZHANG, L.; CHEN, J.; FU, H., PROC. NATL. ACAD. SCI. U.S.A, vol. 96, 1999, pages 8511 - 8515 | WATANABE ET AL., BBRC, vol. 33, no. 3, 2005, pages 562 - 567 | ZHANG ET AL., LIFE SCI, 2003, pages 7443 - 37 | TERADA ET AL., BBRC, vol. 364, 2007, pages 1043 - 49 | FOSTER: "Deuterium Isotope Effects in Studies of Drug Metabolism", TRENDS PHARMACOL. SCI., vol. 5, no. 12, 1984, pages 524 - 527 |