EP2480557 - PROCESS FOR THE PREPARATION OF RAPAMYCIN DERIVATIVES [Right-click to bookmark this link] | Status | The application is deemed to be withdrawn Status updated on 20.03.2015 Database last updated on 26.07.2024 | Most recent event Tooltip | 17.03.2017 | Change - priority | published on 19.04.2017 [2017/16] | Applicant(s) | For all designated states Cadila Healthcare Limited Zydus Tower Satellite Cross Roads Ahmedabad 380 015, Gujarat / IN | [2012/31] | Inventor(s) | 01 /
DAVE, Mayank, Ghanshyambhai Cadila Healthcare Limited Zydus Tower Satellite Cross Roads Ahmedabad 380015 Gujarat / IN | 02 /
PANDEY, Bipin Cadila Healthcare Limited Zydus Tower Satellite Cross Roads Ahmedabad 380015 Gujarat / IN | [2012/31] | Representative(s) | Harris, Jennifer Lucy, et al Kilburn & Strode LLP Lacon London 84 Theobalds Road London WC1X 8NL / GB | [N/P] |
Former [2013/22] | Harris, Jennifer Lucy, et al Kilburn & Strode LLP 20 Red Lion Street London WC1R 4PJ / GB | ||
Former [2012/31] | Jennings, Nigel Robin, et al Kilburn & Strode LLP 20 Red Lion Street London WC1R 4PJ / GB | Application number, filing date | 10810987.7 | 24.09.2010 | WO2010IN00646 | Priority number, date | IN2009MUM2234 | 25.09.2009 Original published format: IN 2234MU2009 | [2017/16] |
Former [2012/31] | IN2009MUM2234 | 25.09.2009 | Filing language | EN | Procedural language | EN | Publication | Type: | A2 Application without search report | No.: | WO2011051960 | Date: | 05.05.2011 | Language: | EN | [2011/18] | Type: | A2 Application without search report | No.: | EP2480557 | Date: | 01.08.2012 | Language: | EN | The application published by WIPO in one of the EPO official languages on 05.05.2011 takes the place of the publication of the European patent application. | [2012/31] | Search report(s) | International search report - published on: | EP | 23.06.2011 | Classification | IPC: | C07D498/18, A61K31/435, A61P37/06, C07D319/06, C07D319/08 | [2012/31] | CPC: |
C07D498/18 (EP,US);
A61P37/06 (EP);
C07D319/06 (EP,US);
C07D319/08 (EP,US)
| Designated contracting states | AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, SM, TR [2012/31] | Title | German: | VERFAHREN ZUR HERSTELLUNG VON RAPAMYCINDERIVATEN | [2012/31] | English: | PROCESS FOR THE PREPARATION OF RAPAMYCIN DERIVATIVES | [2012/31] | French: | PROCÉDÉ DE PRÉPARATION DE DÉRIVÉS DE RAPAMYCINE | [2012/31] | Entry into regional phase | 19.04.2012 | National basic fee paid | 19.04.2012 | Designation fee(s) paid | 19.04.2012 | Examination fee paid | Examination procedure | 07.04.2011 | Request for preliminary examination filed International Preliminary Examining Authority: EP | 19.04.2012 | Amendment by applicant (claims and/or description) | 19.04.2012 | Examination requested [2012/31] | 04.04.2013 | Despatch of a communication from the examining division (Time limit: M04) | 28.04.2013 | Observations by third parties | 13.08.2013 | Reply to a communication from the examining division | 26.09.2013 | Despatch of a communication from the examining division (Time limit: M04) | 24.01.2014 | Reply to a communication from the examining division | 17.02.2014 | Despatch of a communication from the examining division (Time limit: M04) | 17.06.2014 | Reply to a communication from the examining division | 03.07.2014 | Despatch of a communication from the examining division (Time limit: M04) | 14.11.2014 | Application deemed to be withdrawn, date of legal effect [2015/17] | 15.12.2014 | Despatch of communication that the application is deemed to be withdrawn, reason: reply to the communication from the examining division not received in time [2015/17] | Divisional application(s) | EP14182880.6 Application refused : 02.02.2015 | The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is 04.04.2013 | Fees paid | Renewal fee | 11.07.2012 | Renewal fee patent year 03 | 12.07.2013 | Renewal fee patent year 04 | 25.07.2014 | Renewal fee patent year 05 |
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Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Cited in | International search | [XDYI]US5362718 (SKOTNICKI JERAULD S [US], et al) [XD] 8,10,12 * examples 13,14; claims 1,17 * [Y] 1-7 [I] 9,11,13; | [Y]WO2005016935 (WYETH CORP [US], et al) [Y] 14-22,24-27 * page 11 *; | [A]WO2005035528 (REDDYS LAB LTD DR [IN], et al) [A] 9* page 40; compound B *; | [Y]WO2006095185 (BIOTICA TECH LTD [GB], et al) [Y] 1-7 * pages 34,35 *; | [XYI] - SORBERA L A ET AL, "CCI-779: Oncolytic mTOR inhibitor", DRUGS OF THE FUTURE 2002 ES LNKD- DOI:10.1358/DOF.2002.027.01.654066, (2002), vol. 27, no. 1, ISSN 0377-8282, pages 7 - 13, XP002631962 [X] 8,10,12 * Scheme 1, 2 * [Y] 1-7,14 [I] 9,11,13 DOI: http://dx.doi.org/10.1358/DOF.2002.027.01.654066 | [XI] - GU JIANXIN ET AL, "lipase-catalyzed regioselective esterification of rapamycin: synthesis of temsirolimus (CCI-779).", ORGANIC LETTERS 1 SEP 2005 LNKD- PUBMED:16119938, (20050901), vol. 7, no. 18, ISSN 1523-7060, pages 3945 - 3948, XP002631963 [X] 8 * compounds 8,9 * [I] 9,12 DOI: http://dx.doi.org/10.1021/OL0514395 | [XY] - CHEN YANQIU ET AL, "Conformational changes of rapamycin and analogs upon complexing with FKBP associated with activity: An application of second derivative CD spectroscopy", JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, (1994), vol. 116, no. 6, ISSN 0002-7863, pages 2683 - 2684, XP002631964 [X] 23 * compounds 4-6 * [Y] 14-22,24-27 | by applicant | US5362718 | US6277983 | WO2005016935 | US2005234086 | US2007129395 | - T. W. GREENE; PETER G. M WUTS, Protective Groups in Organic Synthesis, JOHN WILEY AND SONS | other | US5362718 | WO03099787 | WO2006095185 | - BRUICE T.C. ET AL, "A search for carboxyl-group catalysis in ketal hydrolysis", JOURNAL OF THE AMERICAL CHEMICAL SOCIETY, (19670705), vol. 89, no. 14, pages 3568 - 3576, XP003031122 DOI: http://dx.doi.org/10.1021/ja00990a039 |