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Extract from the Register of European Patents

EP About this file: EP2418201

EP2418201 - Polymorph forms of (2S)-(4E)-N-methyl-5-[3-(5-isopropoxypyridin) yl]-4-penten-2-amine p-hydroxybenzoate for the treatment of central nervous system disorders [Right-click to bookmark this link]
Former [2012/07]Polymorph forms of (2S) - (4E) -N-methyl-5- (3-isopropoxypyridin) yl]-4-penten-2-amine for the treatment of central nervous system disorders
[2013/40]
StatusNo opposition filed within time limit
Status updated on  19.12.2014
Database last updated on 24.04.2024
Most recent event   Tooltip19.12.2014No opposition filed within time limitpublished on 21.01.2015  [2015/04]
Applicant(s)For all designated states
Targacept, Inc.
100 North Main Street
Suite 1510
Winston-Salem, NC 27101 / US
[2014/24]
Former [2012/07]For all designated states
Targacept, Inc.
200 East First Street, Suite 300
Winston-Salem, NC 27101-4165 / US
Inventor(s)01 / Munoz, Julio A.
214 Lakeside Drive
Walnut Grove, NC 27052 / US
02 / Dull, Gary Maurice
6025 Shallowford Road
Lewisville, NC 27003 / US
 [2012/07]
Representative(s)Crooks, Elizabeth Caroline, et al
Kilburn & Strode LLP
Lacon London
84 Theobalds Road
London WC1X 8NL / GB
[N/P]
Former [2013/25]Crooks, Elizabeth Caroline, et al
Kilburn & Strode LLP 20 Red Lion Street
London WC1R 4PJ / GB
Former [2012/07]Harris, Jennifer Lucy, et al
Kilburn & Strode LLP 20 Red Lion Street
London WC1R 4PJ / GB
Application number, filing date11167528.608.05.2007
[2012/07]
Priority number, dateUS20060746821P09.05.2006         Original published format: US 746821 P
[2012/07]
Previously filed application, dateWO2007US6844608.05.2007
[2012/07]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report 
No.:EP2418201
Date:15.02.2012
Language:EN
[2012/07]
Type: B1 Patent specification 
No.:EP2418201
Date:12.02.2014
Language:EN
[2014/07]
Search report(s)(Supplementary) European search report - dispatched on:EP16.01.2012
ClassificationIPC:C07D213/63, A61K31/44, A61P25/28
[2012/07]
CPC:
C07D213/65 (EP,US); C07D213/63 (KR); A61K31/44 (KR);
A61P25/00 (EP); A61P25/02 (EP); A61P25/18 (EP);
A61P25/28 (EP); A61P43/00 (EP) (-)
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MT,   NL,   PL,   PT,   RO,   SE,   SI,   SK,   TR [2012/07]
Extension statesAL09.08.2012
BA09.08.2012
HR09.08.2012
MK09.08.2012
RS09.08.2012
TitleGerman:Polymorphe Formen von (2S)-(4E)-N-Methyl-5-[(3-(5-Isopropoxypyridin)yl]-4-Penten-2-Amin p-Hydroxybenzoate zur Behandlung von Erkrankungen des zentralen Nervensystems[2013/40]
English:Polymorph forms of (2S)-(4E)-N-methyl-5-[3-(5-isopropoxypyridin) yl]-4-penten-2-amine p-hydroxybenzoate for the treatment of central nervous system disorders[2013/40]
French:Formes polymorphes de (2S)-(4E)-N-méthyl-5- [3-(5-isopropoxypyridine)yl]-4-penten-2-amine p-hydroxybenzoate destinées au traitement de troubles du système nerveux central[2013/40]
Former [2012/07]Polymorphe Formen von (2S)-(4E)-N-Methyl-5-(3-Isopropoxypyridin)-[l]-4-penten-2-amin zur Behandlung von Erkrankungen des zentralen Nervensystems
Former [2012/07]Polymorph forms of (2S) - (4E) -N-methyl-5- (3-isopropoxypyridin) yl]-4-penten-2-amine for the treatment of central nervous system disorders
Former [2012/07]Formes polymorphes de (2S) - (4E) -N-méthyl-5- (3-isopropoxypyridine) yl ̈-4-penten-2-amine destinées au traitement de troubles du système nerveux central
Examination procedure09.08.2012Amendment by applicant (claims and/or description)
09.08.2012Examination requested  [2012/38]
29.10.2012Despatch of a communication from the examining division (Time limit: M06)
12.06.2013Despatch of communication that the application is deemed to be withdrawn, reason: reply to the communication from the examining division not received in time
14.08.2013Reply to a communication from the examining division
19.09.2013Communication of intention to grant the patent
17.12.2013Fee for grant paid
17.12.2013Fee for publishing/printing paid
Parent application(s)   TooltipEP07783431.5  / EP2021326
Divisional application(s)The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued (EP20070783431) is  18.11.2009
Opposition(s)13.11.2014No opposition filed within time limit [2015/04]
Request for further processing for:The application is deemed to be withdrawn due to failure to reply to the examination report
14.08.2013Request for further processing filed
14.08.2013Full payment received (date of receipt of payment)
Request granted
26.08.2013Decision despatched
Fees paidRenewal fee
25.05.2011Renewal fee patent year 03
25.05.2011Renewal fee patent year 04
25.05.2011Renewal fee patent year 05
25.05.2012Renewal fee patent year 06
10.05.2013Renewal fee patent year 07
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Documents cited:Search[AD]WO9965876  (REYNOLDS TOBACCO CO R [US], et al) [AD] 1-14 * example 12 *;
 [XP]WO2006053039  (TARGACEPT INC [US], et al) [XP] 1-14* example 2 *
by applicantUS4922901
 WO9408992
 WO9631475
 US5583140
 US5597919
 US5604231
 US5853696
 US5969144
 WO9965876
 US6953855
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