EP2609100 - FUROPYRIDINE DERIVATIVES [Right-click to bookmark this link] | Status | No opposition filed within time limit Status updated on 29.04.2016 Database last updated on 04.06.2024 | Most recent event Tooltip | 19.10.2018 | Lapse of the patent in a contracting state New state(s): AL | published on 21.11.2018 [2018/47] | Applicant(s) | For all designated states Merck Patent GmbH Frankfurter Strasse 250 64293 Darmstadt / DE | [2013/27] | Inventor(s) | 01 /
BURGDORF, Lars Gabelsbergerstrasse 21 60389 Frankfurt am Main / DE | 02 /
SCHULTZ, Melanie Wienerstrasse 63 64287 Darmstadt / DE | 03 /
ROSS, Tatjana Taunusblick 13 65760 Eschborn / DE | 04 /
HODOUS, Brian 250 Chestnut Street Cambridge MA 02139 / US | 05 /
POTNICK, Justin 53 Conant Street Acton, MA 01720 / US | 06 /
SUTTON, Amanda E. 4 Triphammer Road Hingham Massachusetts 02043 / US | 07 /
HUCK, Bayard R. 50 Woodmere Drive Sudbury Massachusetts 01776 / US | [2013/32] |
Former [2013/28] | 01 /
BURGDORF, Lars Gabelsbergerstrasse 21 60389 Frankfurt am Main / DE | ||
02 /
SCHULTZ, Melanie Wienerstrasse 63 64287 Darmstadt / DE | |||
03 /
HOFMANN, Tatjana Josef-Traxel-Weg 4 55128 Mainz / DE | |||
04 /
HODOUS, Brian 250 Chestnut Street Cambridge MA 02139 / US | |||
05 /
POTNICK, Justin 53 Conant Street Acton, MA 01720 / US | |||
06 /
SUTTON, Amanda E. 4 Triphammer Road Hingham Massachusetts 02043 / US | |||
07 /
HUCK, Bayard R. 50 Woodmere Drive Sudbury Massachusetts 01776 / US | |||
Former [2013/27] | 01 /
BURGDORF, Lars Gabelsbergerstrasse 21 60389 Frankfurt am Main / DE | ||
02 /
SCHULTZ, Melanie Wienerstrasse 63 64287 Darmstadt / DE | |||
03 /
HOFMANN, Tatjana Josef-Traxel-Weg 4 55128 Mainz / DE | |||
04 /
HODOUS, Brian 250 Chestnut Street Cambridge MA 02139 / US | |||
05 /
POTNICK, Justin 499 Boston Rd. Unit 1220 Billerica Massachusetts 01821 / US | |||
06 /
SUTTON, Amanda E. 4 Triphammer Road Hingham Massachusetts 02043 / US | |||
07 /
HUCK, Bayard R. 50 Woodmere Drive Sudbury Massachusetts 01776 / US | Application number, filing date | 11738631.8 | 29.07.2011 | WO2011EP03831 | Priority number, date | EP20100008928 | 27.08.2010 Original published format: EP 10008928 | [2013/27] | Filing language | EN | Procedural language | EN | Publication | Type: | A2 Application without search report | No.: | WO2012025187 | Date: | 01.03.2012 | Language: | EN | [2012/09] | Type: | A2 Application without search report | No.: | EP2609100 | Date: | 03.07.2013 | Language: | EN | The application published by WIPO in one of the EPO official languages on 01.03.2012 takes the place of the publication of the European patent application. | [2013/27] | Type: | B1 Patent specification | No.: | EP2609100 | Date: | 24.06.2015 | Language: | EN | [2015/26] | Search report(s) | International search report - published on: | EP | 21.06.2012 | Classification | IPC: | A61K45/06, A61K31/4709, A61K31/496, A61K31/506, A61K31/5377, A61K31/5383, C07D491/048, C07D519/00, C07D491/04, A61K31/4355 | [2015/08] | CPC: |
C07D491/048 (EP,US);
C07D491/04 (EP,KR,US);
A61K31/4355 (EP,KR,US);
A61K31/4709 (EP,US);
A61K31/496 (EP,US);
A61K31/506 (EP,US);
A61K31/5377 (EP,US);
A61K31/5383 (EP,US);
A61K45/06 (US);
A61P11/00 (EP);
A61P11/02 (EP);
A61P11/06 (EP);
A61P15/08 (EP);
A61P19/02 (EP);
A61P25/00 (EP);
A61P29/00 (EP);
A61P3/00 (EP);
A61P31/00 (EP);
A61P35/00 (EP);
A61P35/02 (EP);
A61P37/02 (EP);
A61P37/06 (EP);
A61P37/08 (EP);
A61P7/02 (EP);
|
Former IPC [2013/27] | C07D491/04, A61K31/4355 | Designated contracting states | AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR [2013/27] | Extension states | BA | Not yet paid | ME | Not yet paid | Title | German: | FUROPYRIDINDERIVATE | [2013/27] | English: | FUROPYRIDINE DERIVATIVES | [2013/27] | French: | DÉRIVÉS DE FUROPYRIDINE | [2013/27] | Entry into regional phase | 09.01.2013 | National basic fee paid | 09.01.2013 | Designation fee(s) paid | 09.01.2013 | Examination fee paid | Examination procedure | 09.01.2013 | Examination requested [2013/27] | 08.10.2013 | Amendment by applicant (claims and/or description) | 30.09.2014 | Despatch of a communication from the examining division (Time limit: M02) | 10.10.2014 | Reply to a communication from the examining division | 06.03.2015 | Communication of intention to grant the patent | 12.05.2015 | Fee for grant paid | 12.05.2015 | Fee for publishing/printing paid | 12.05.2015 | Receipt of the translation of the claim(s) | Divisional application(s) | The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is 30.09.2014 | Opposition(s) | 29.03.2016 | No opposition filed within time limit [2016/22] | Fees paid | Renewal fee | 10.07.2013 | Renewal fee patent year 03 | 14.07.2014 | Renewal fee patent year 04 |
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Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Lapses during opposition Tooltip | HU | 29.07.2011 | AL | 24.06.2015 | AT | 24.06.2015 | BE | 24.06.2015 | CY | 24.06.2015 | CZ | 24.06.2015 | DK | 24.06.2015 | EE | 24.06.2015 | FI | 24.06.2015 | HR | 24.06.2015 | LT | 24.06.2015 | LV | 24.06.2015 | MC | 24.06.2015 | MK | 24.06.2015 | MT | 24.06.2015 | NL | 24.06.2015 | PL | 24.06.2015 | RO | 24.06.2015 | RS | 24.06.2015 | SE | 24.06.2015 | SI | 24.06.2015 | SK | 24.06.2015 | SM | 24.06.2015 | TR | 24.06.2015 | IE | 29.07.2015 | LU | 29.07.2015 | BG | 24.09.2015 | NO | 24.09.2015 | GR | 25.09.2015 | IS | 24.10.2015 | PT | 26.10.2015 | [2018/47] |
Former [2018/31] | HU | 29.07.2011 | |
AT | 24.06.2015 | ||
BE | 24.06.2015 | ||
CY | 24.06.2015 | ||
CZ | 24.06.2015 | ||
DK | 24.06.2015 | ||
EE | 24.06.2015 | ||
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LT | 24.06.2015 | ||
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TR | 24.06.2015 | ||
IE | 29.07.2015 | ||
LU | 29.07.2015 | ||
BG | 24.09.2015 | ||
NO | 24.09.2015 | ||
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IS | 24.10.2015 | ||
PT | 26.10.2015 | ||
Former [2018/02] | HU | 29.07.2011 | |
AT | 24.06.2015 | ||
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CY | 24.06.2015 | ||
CZ | 24.06.2015 | ||
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SM | 24.06.2015 | ||
IE | 29.07.2015 | ||
LU | 29.07.2015 | ||
BG | 24.09.2015 | ||
NO | 24.09.2015 | ||
GR | 25.09.2015 | ||
IS | 24.10.2015 | ||
PT | 26.10.2015 | ||
Former [2017/39] | HU | 29.07.2011 | |
AT | 24.06.2015 | ||
BE | 24.06.2015 | ||
CY | 24.06.2015 | ||
CZ | 24.06.2015 | ||
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EE | 24.06.2015 | ||
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RO | 24.06.2015 | ||
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SI | 24.06.2015 | ||
SK | 24.06.2015 | ||
SM | 24.06.2015 | ||
IE | 29.07.2015 | ||
BG | 24.09.2015 | ||
NO | 24.09.2015 | ||
GR | 25.09.2015 | ||
IS | 24.10.2015 | ||
PT | 26.10.2015 | ||
Former [2017/22] | AT | 24.06.2015 | |
BE | 24.06.2015 | ||
CZ | 24.06.2015 | ||
DK | 24.06.2015 | ||
EE | 24.06.2015 | ||
FI | 24.06.2015 | ||
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LT | 24.06.2015 | ||
LV | 24.06.2015 | ||
MC | 24.06.2015 | ||
MT | 24.06.2015 | ||
PL | 24.06.2015 | ||
RO | 24.06.2015 | ||
RS | 24.06.2015 | ||
SI | 24.06.2015 | ||
SK | 24.06.2015 | ||
IE | 29.07.2015 | ||
BG | 24.09.2015 | ||
NO | 24.09.2015 | ||
GR | 25.09.2015 | ||
IS | 24.10.2015 | ||
PT | 26.10.2015 | ||
Former [2017/03] | AT | 24.06.2015 | |
BE | 24.06.2015 | ||
CZ | 24.06.2015 | ||
DK | 24.06.2015 | ||
EE | 24.06.2015 | ||
FI | 24.06.2015 | ||
HR | 24.06.2015 | ||
LT | 24.06.2015 | ||
LV | 24.06.2015 | ||
MC | 24.06.2015 | ||
PL | 24.06.2015 | ||
RO | 24.06.2015 | ||
RS | 24.06.2015 | ||
SI | 24.06.2015 | ||
SK | 24.06.2015 | ||
IE | 29.07.2015 | ||
BG | 24.09.2015 | ||
NO | 24.09.2015 | ||
GR | 25.09.2015 | ||
IS | 24.10.2015 | ||
PT | 26.10.2015 | ||
Former [2016/36] | AT | 24.06.2015 | |
CZ | 24.06.2015 | ||
DK | 24.06.2015 | ||
EE | 24.06.2015 | ||
FI | 24.06.2015 | ||
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LT | 24.06.2015 | ||
LV | 24.06.2015 | ||
MC | 24.06.2015 | ||
PL | 24.06.2015 | ||
RO | 24.06.2015 | ||
RS | 24.06.2015 | ||
SI | 24.06.2015 | ||
SK | 24.06.2015 | ||
IE | 29.07.2015 | ||
BG | 24.09.2015 | ||
NO | 24.09.2015 | ||
GR | 25.09.2015 | ||
IS | 24.10.2015 | ||
PT | 26.10.2015 | ||
Former [2016/33] | AT | 24.06.2015 | |
CZ | 24.06.2015 | ||
DK | 24.06.2015 | ||
EE | 24.06.2015 | ||
FI | 24.06.2015 | ||
HR | 24.06.2015 | ||
LT | 24.06.2015 | ||
LV | 24.06.2015 | ||
MC | 24.06.2015 | ||
PL | 24.06.2015 | ||
RO | 24.06.2015 | ||
RS | 24.06.2015 | ||
SK | 24.06.2015 | ||
IE | 29.07.2015 | ||
BG | 24.09.2015 | ||
NO | 24.09.2015 | ||
GR | 25.09.2015 | ||
IS | 24.10.2015 | ||
PT | 26.10.2015 | ||
Former [2016/20] | AT | 24.06.2015 | |
CZ | 24.06.2015 | ||
DK | 24.06.2015 | ||
EE | 24.06.2015 | ||
FI | 24.06.2015 | ||
HR | 24.06.2015 | ||
LT | 24.06.2015 | ||
LV | 24.06.2015 | ||
MC | 24.06.2015 | ||
PL | 24.06.2015 | ||
RO | 24.06.2015 | ||
RS | 24.06.2015 | ||
SK | 24.06.2015 | ||
BG | 24.09.2015 | ||
NO | 24.09.2015 | ||
GR | 25.09.2015 | ||
IS | 24.10.2015 | ||
PT | 26.10.2015 | ||
Former [2016/18] | AT | 24.06.2015 | |
CZ | 24.06.2015 | ||
EE | 24.06.2015 | ||
FI | 24.06.2015 | ||
HR | 24.06.2015 | ||
LT | 24.06.2015 | ||
LV | 24.06.2015 | ||
MC | 24.06.2015 | ||
PL | 24.06.2015 | ||
RO | 24.06.2015 | ||
RS | 24.06.2015 | ||
SK | 24.06.2015 | ||
BG | 24.09.2015 | ||
NO | 24.09.2015 | ||
GR | 25.09.2015 | ||
IS | 24.10.2015 | ||
PT | 26.10.2015 | ||
Former [2016/11] | AT | 24.06.2015 | |
CZ | 24.06.2015 | ||
EE | 24.06.2015 | ||
FI | 24.06.2015 | ||
HR | 24.06.2015 | ||
LT | 24.06.2015 | ||
LV | 24.06.2015 | ||
PL | 24.06.2015 | ||
RO | 24.06.2015 | ||
RS | 24.06.2015 | ||
SK | 24.06.2015 | ||
BG | 24.09.2015 | ||
NO | 24.09.2015 | ||
GR | 25.09.2015 | ||
IS | 24.10.2015 | ||
PT | 26.10.2015 | ||
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EE | 24.06.2015 | ||
FI | 24.06.2015 | ||
HR | 24.06.2015 | ||
LT | 24.06.2015 | ||
LV | 24.06.2015 | ||
PL | 24.06.2015 | ||
RO | 24.06.2015 | ||
RS | 24.06.2015 | ||
SK | 24.06.2015 | ||
BG | 24.09.2015 | ||
NO | 24.09.2015 | ||
GR | 25.09.2015 | ||
IS | 24.10.2015 | ||
PT | 26.10.2015 | ||
Former [2016/09] | EE | 24.06.2015 | |
FI | 24.06.2015 | ||
HR | 24.06.2015 | ||
LT | 24.06.2015 | ||
LV | 24.06.2015 | ||
RS | 24.06.2015 | ||
BG | 24.09.2015 | ||
NO | 24.09.2015 | ||
GR | 25.09.2015 | ||
Former [2015/50] | FI | 24.06.2015 | |
HR | 24.06.2015 | ||
LT | 24.06.2015 | ||
LV | 24.06.2015 | ||
RS | 24.06.2015 | ||
BG | 24.09.2015 | ||
NO | 24.09.2015 | ||
GR | 25.09.2015 | ||
Former [2015/49] | FI | 24.06.2015 | |
HR | 24.06.2015 | ||
LT | 24.06.2015 | ||
LV | 24.06.2015 | ||
RS | 24.06.2015 | ||
NO | 24.09.2015 | ||
GR | 25.09.2015 | Cited in | International search | [I]WO9940091 (AMGEN INC [US]) [I] 1-17 * page 13, line 5 - page 29, line 28; page 30, line 4 - page 34, line 9; examples 228, 230, 231; figure 1B *; | [A]US2002004511 (LUZZIO MICHAEL JOSEPH [US], et al) [A] 1-17 * [0008]-[0018]; [0180]-[0189]; examples * | by applicant | WO2008118823 | WO2009136995 | WO2010027500 | - J. A.TAYLOR ET AL., MOLEC. 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ET AL., "Inhibition of Syk with fostamatinib disodium has significant clinical activity in non-Hodgkin lymphoma and chronic lymphocytic leukemia", BLOOD, vol. 115, doi:doi:10.1182/blood-2009-08-236471, pages 2578 - 2585, XP055213215 DOI: http://dx.doi.org/10.1182/blood-2009-08-236471 | - GAO, C. ET AL., "Eptifibatide-induced thrombocytopenia and thrombosis in humans require FcgammaRlla and the integrin beta3 cytoplasmic domain", J CLIN INVEST, (2009), vol. 119, pages 504 - 511 | - MARJON, K.D., MARNELL, L.L., MOLD, C., DU CLOS, T.W., "Macrophages activated by C-reactive protein through Fc gamma RI transfer suppression of immune thrombocytopenia", J IMMUNOL, (2009), vol. 182, pages 1397 - 1403 | - CHEN, L. ET AL., "SYK-dependent tonic B-cell receptor signaling is a rational treatment target in diffuse large B-cell lymphoma", BLOOD, (2008), vol. 111, pages 2230 - 2237 | - PECHLOFF, K. 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