Deutsch English Français

Contact

EP2588441

European procedure

Quick help

Maintenance news

Scheduled maintenance

Regular maintenance outages:
between 05.00 and 05.15 hrs CET (Monday to Sunday).

Other outages
Availability

2022.02.11

More...

News flashes

News Flashes

New version of the European Patent Register – SPC proceedings information in the Unitary Patent Register.

2024-07-24

More...

Extract from the Register of European Patents

EP About this file: EP2588441

EP2588441 - NOVEL PROCESSES FOR THE PREPARATION OF PHENYLCYCLOPROPYLAMINE DERIVATIVES AND USE THEREOF FOR PREPARING TICAGRELOR [Right-click to bookmark this link]
Status	The application is deemed to be withdrawn Status updated on 13.05.2016 Database last updated on 19.10.2024
Most recent event Tooltip	13.05.2016	Application deemed to be withdrawn	published on 15.06.2016 [2016/24]
Applicant(s)	For all designated states Actavis Group Ptc Ehf Reykjavikurvegi 76-78 220 Hafnarfjörour / IS
	[2013/19]
Inventor(s)	01 / KHILE, Anil, Shahaji Flat No.502, Shree Gayatri Chs Ltd. Plot No.7, Sector 11, 5th Floor Khanda Colony New Panvel (W), Navi Mumbai Raigad 410206 / IN
	02 / NAIR, Vignesh Thadavillayil Vadakkathil P.O- Vallikunnam Dist-Alapuzha Kerala 590601 / IN
	03 / TRIVEDI, Nikhil 601 Parimal Apartments Plot No. C-1, Sector-23 Nerul Navimumbai Maharashtra PIN - 400 706 / IN
	04 / PRADHAN, Nitin, Sharadchandra C-602 Runwal Estate Ghoad Bunder Road Opposite Lawkim Company Manpada, Thane (West) Maharashtra 400601 / IN
	[2013/19]
Representative(s)	Wichmann, Hendrik, et al Wuesthoff & Wuesthoff Patentanwälte und Rechtsanwalt PartG mbB Schweigerstraße 2 81541 München / DE
	[N/P]
Former [2013/19]	Wichmann, Hendrik, et al Wuesthoff & Wuesthoff Patent- und Rechtsanwälte Schweigerstraße 2 DE-81541 München / DE
Application number, filing date	11776239.3	28.06.2011
	WO2011IB02246
Priority number, date	IN2010MUM1841	30.06.2010 Original published format: IN MU18412010
	IN2010MUM2043	19.07.2010 Original published format: IN MU20432010
	[2013/19]
Filing language	EN
Procedural language	EN
Publication	Type:	A2 Application without search report
	No.:	WO2012001531
	Date:	05.01.2012
	Language:	EN
	[2012/01]
	Type:	A2 Application without search report
	No.:	EP2588441
	Date:	08.05.2013
	Language:	EN
	The application published by WIPO in one of the EPO official languages on 05.01.2012 takes the place of the publication of the European patent application.
	[2013/19]
Search report(s)	International search report - published on:	EP	16.08.2012
Classification	IPC:	C07C209/56	[2013/19]
	CPC:	C07C209/62 (EP,US); C07C209/56 (EP,US); C07C211/35 (EP,US); C07C211/40 (US); C07B2200/13 (EP,US); C07C2601/02 (EP,US); (+) C07C2601/16 (EP,US) (-)
Designated contracting states	AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR [2013/19]
Title	German:	NEUE VERFAHREN ZUR HERSTELLUNG VON PHENYLCYCLOPROPYLAMINDERIVATEN UND VERWENDUNG DAVON ZUR HERSTELLUNG VON TICAGRELOR	[2013/19]
	English:	NOVEL PROCESSES FOR THE PREPARATION OF PHENYLCYCLOPROPYLAMINE DERIVATIVES AND USE THEREOF FOR PREPARING TICAGRELOR	[2013/19]
	French:	NOUVEAUX PROCÉDÉS POUR LA PRÉPARATION DE DÉRIVÉS DE PHÉNYLCYCLOPROPYLAMINE ET LEUR UTILISATION POUR LA PRÉPARATION DE TICAGRELOR	[2013/19]
Entry into regional phase	19.12.2012	National basic fee paid
	19.12.2012	Designation fee(s) paid
	19.12.2012	Examination fee paid
Examination procedure	19.12.2012	Examination requested [2013/19]
	08.08.2013	Amendment by applicant (claims and/or description)
	01.01.2016	Application deemed to be withdrawn, date of legal effect [2016/24]
	01.02.2016	Despatch of communication that the application is deemed to be withdrawn, reason: renewal fee not paid in time [2016/24]
Fees paid	Renewal fee
	20.06.2013	Renewal fee patent year 03
	25.06.2014	Renewal fee patent year 04
	Penalty fee
	Additional fee for renewal fee
	30.06.2015	05 M06 Not yet paid
Opt-out from the exclusive Tooltip competence of the Unified Patent Court	See the Register of the Unified Patent Court for opt-out data
	Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Cited in	International search	[AD]US2003120105 (CLARK ADRIAN [SE], et al) [AD] 1-9* the whole document *;
		[AD]WO2008018823 (ASTRAZENECA AB [SE], et al) [AD] 1-9 * example 5 * * page 28, paragraph l - page 29, paragraph 1 *;
		[Y] - FILLER R AND WHITE W, "New Reactions of polyfluoroaromatic compounds. II. Polyfluoroaralkyl amines", JOURNAL OF THE CHEMICAL SOCIETY, SECTION C: ORGANIC CHEMISTRY, CHEMICAL SOCIETY. LETCHWORTH, GB, (19710101), ISSN 0022-4952, pages 2062 - 2068, XP009102773 [Y] 1-9 * page 2063, column l, paragraph l * scheme 3 * page 2067, column r, paragraph 3 *
		[Y] - Shinya Mimasu ET AL, "Structurally Designed Trans-2-phenylcyclopropylamine Derivatives Potently Inhibit Histone Demethylase LSD1/KDM1-Supporting Information", (20100622), pages 1 - 15, URL: http://pubs.acs.org/doi/suppl/10.1021/bi100299r/suppl_file/bi100299r_si_001.pdf, (20120402), XP055023540 [Y] 1-9 * page 3 *
		[Y] - TENG P-F ET AL, "Asymmetric inter- and intramolecular cyclopropanations of alkenes catalyzed by rhodium D4-porphyrin: a comparison of rhodium- and ruthenium-centred catalysts", TETRAHEDRON ASYMMETRY, PERGAMON PRESS LTD, OXFORD, GB, (20030404), vol. 14, no. 7, doi:10.1016/S0957-4166(03)00047-8, ISSN 0957-4166, pages 837 - 844, XP004417215 [Y] 1-9 * table 1 * DOI: http://dx.doi.org/10.1016/S0957-4166(03)00047-8
		[Y] - Takayuki Shioiri, "Diphenyl Phosphorazidate (DPPA) - More Than Three Decades Later", TCIMAIL number 134, (20071001), pages 2 - 19, URL: http://www.tciamerica.com/tcimail/backnumber/article/134drE.pdf, (20120402), XP055023593 [Y] 1-9 * page 6 *
		[Y] - MA B ET AL, "A modified Curtius reaction: an efficient and simple method for direct isolation of free amine", TETRAHEDRON LETTERS, ELSEVIER, AMSTERDAM, NL, vol. 51, no. 2, ISSN 0040-4039, (20100113), pages 385 - 386, (20091113), XP027259063 [Y] 1-9 * the whole document *
		[AD] - TSAI T Y ET AL, "Novel trans-2-aryl-cyclopropylamine analogues as potent and selective dipeptidyl peptidase IV inhibitors", BIOORGANIC & MEDICINAL CHEMISTRY, PERGAMON, GB, vol. 17, no. 6, doi:10.1016/J.BMC.2009.02.020, ISSN 0968-0896, (20090315), pages 2388 - 2399, (20090220), XP025981936 [AD] 1-9 scheme 1; page 2389 * * page 2395, column r, paragraph 3 * DOI: http://dx.doi.org/10.1016/j.bmc.2009.02.020
		[A] - PRYDE ET AL, "Novel selective inhibitors of neutral endopeptidase for the treatment of female sexual arousal disorder", BIOORGANIC & MEDICINAL CHEMISTRY, PERGAMON, GB, (20061115), vol. 15, no. 1, doi:10.1016/J.BMC.2006.10.002, ISSN 0968-0896, pages 142 - 159, XP005764596 [A] 1-9 * page 156, column r, paragraph l * items 5.11.7.1 to 5.11.10; page 157, column r * DOI: http://dx.doi.org/10.1016/j.bmc.2006.10.002
		[A] - VALLGARDA J ET AL, "trans-2-Aryl-N,N-diyclopropylamines: synthesis and interactions with 5-HT1a receptors", JOURNAL OF MEDICINAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY, US, (19960101), vol. 39, no. 7, doi:10.1021/JM9507136, ISSN 0022-2623, pages 1485 - 1493, XP002262871 [A] 1-9 scheme 1; page 1486 * DOI: http://dx.doi.org/10.1021/jm9507136
	by applicant	EP0996621
		US6251910
		EP1135391
		US6525060
		US6974868
		US7067663
		US7122695
		US7250419
		US2007265282
		WO2008018823
		US2008132719
		US2008214812
		WO2010030224
		- BIOORGANIC & MEDICINAL CHEMISTRY, (2009), vol. 17, no. 6, pages 2388 - 2399
		- J. MED. CHEM., (1977), vol. 20, no. 7, pages 934 - 939
		- J. ORG. CHEM., (1992), vol. 57, pages 3757 - 3759

The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.

Legal notice
Terms of use
24.2.25; 35p