EP2635577 - SUBSTITUTED 6-FLUORO-1H-PYRAZOLO[4,3-B]PYRIDINES AND USE THEREOF [Right-click to bookmark this link] | Status | No opposition filed within time limit Status updated on 07.08.2015 Database last updated on 20.07.2024 | Most recent event Tooltip | 12.10.2018 | Lapse of the patent in a contracting state New state(s): AL | published on 14.11.2018 [2018/46] | Applicant(s) | For all designated states Bayer Intellectual Property GmbH Alfred-Nobel-Strasse 10 40789 Monheim / DE | [2013/37] | Inventor(s) | 01 /
FOLLMANN, Markus Rosmarinweg 28 50859 Köln / DE | 02 /
STASCH, Johannes-Peter Alfred-Nobel-Str. 109 42651 Solingen / DE | 03 /
REDLICH, Gorden Schadowstr. 50 44799 Bochum / DE | 04 /
ACKERSTAFF, Jens Schliemannstr. 15 10437 Berlin / DE | 05 /
GRIEBENOW, Nils Kurfürstenstr. 39 41541 Dormagen (Zons) / DE | 06 /
KNORR, Andreas Trillser Graben 10 40699 Erkrath / DE | 07 /
WUNDER, Frank Schwarzer Weg 251 42117 Wuppertal / DE | 08 /
LI, Volkhart, Min-Jian Im Wiesengrund 40 42553 Velbert / DE | 09 /
MITTENDORF, Joachim Wildsteig 30a 42113 Wuppertal / DE | 10 /
SCHLEMMER, Karl-Heinz Wildsteig 22 a 42113 Wuppertal / DE | 11 /
JAUTELAT, Rolf Zur Pumpstation 35 42781 Haan / DE | [2013/37] | Representative(s) | BIP Patents c/o Bayer Intellectual Property GmbH Alfred-Nobel-Straße 50 40789 Monheim am Rhein / DE | [N/P] |
Former [2013/37] | BIP Patents c/o Bayer Intellectual Property GmbH Creative Campus Monheim Alfred-Nobel-Straße 10 40789 Monheim / DE | Application number, filing date | 11788085.6 | 03.11.2011 | WO2011EP69346 | Priority number, date | DE20101043379 | 04.11.2010 Original published format: DE102010043379 | [2013/37] | Filing language | DE | Procedural language | DE | Publication | Type: | A1 Application with search report | No.: | WO2012059549 | Date: | 10.05.2012 | Language: | DE | [2012/19] | Type: | A1 Application with search report | No.: | EP2635577 | Date: | 11.09.2013 | Language: | DE | The application published by WIPO in one of the EPO official languages on 10.05.2012 takes the place of the publication of the European patent application. | [2013/37] | Type: | B1 Patent specification | No.: | EP2635577 | Date: | 01.10.2014 | Language: | DE | [2014/40] | Search report(s) | International search report - published on: | EP | 10.05.2012 | Classification | IPC: | C07D471/04, A61K31/437, A61P9/00 | [2013/37] | CPC: |
C07D471/04 (EP,US);
A61K31/506 (EP,US);
A61K45/06 (US);
A61P7/02 (EP);
A61P9/00 (EP);
A61P9/04 (EP);
| Designated contracting states | AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR [2013/37] | Extension states | BA | Not yet paid | ME | Not yet paid | Title | German: | SUBSTITUIERTE 6-FLUOR-1H-PYRAZOLO[4,3-B]PYRIDINE UND IHRE VERWENDUNG | [2013/37] | English: | SUBSTITUTED 6-FLUORO-1H-PYRAZOLO[4,3-B]PYRIDINES AND USE THEREOF | [2013/37] | French: | 6-FLUORO-1H-PYRAZOLO[4,3-B]PYRIDINES SUBSTITUÉES ET LEUR UTILISATION | [2013/37] | Entry into regional phase | 04.06.2013 | National basic fee paid | 04.06.2013 | Designation fee(s) paid | 04.06.2013 | Examination fee paid | Examination procedure | 04.06.2013 | Examination requested [2013/37] | 19.12.2013 | Amendment by applicant (claims and/or description) | 15.05.2014 | Communication of intention to grant the patent | 20.08.2014 | Fee for grant paid | 20.08.2014 | Fee for publishing/printing paid | 20.08.2014 | Receipt of the translation of the claim(s) | Divisional application(s) | The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is 15.05.2014 | Opposition(s) | 02.07.2015 | No opposition filed within time limit [2015/37] | Fees paid | Renewal fee | 18.11.2013 | Renewal fee patent year 03 |
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Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Lapses during opposition Tooltip | HU | 03.11.2011 | AL | 01.10.2014 | BG | 01.10.2014 | CY | 01.10.2014 | CZ | 01.10.2014 | DK | 01.10.2014 | EE | 01.10.2014 | FI | 01.10.2014 | HR | 01.10.2014 | LT | 01.10.2014 | LV | 01.10.2014 | MC | 01.10.2014 | MK | 01.10.2014 | MT | 01.10.2014 | NL | 01.10.2014 | PL | 01.10.2014 | RO | 01.10.2014 | RS | 01.10.2014 | SE | 01.10.2014 | SI | 01.10.2014 | SK | 01.10.2014 | SM | 01.10.2014 | TR | 01.10.2014 | IE | 03.11.2014 | LU | 03.11.2014 | BE | 30.11.2014 | CH | 30.11.2014 | LI | 30.11.2014 | NO | 01.01.2015 | GR | 02.01.2015 | IS | 01.02.2015 | PT | 02.02.2015 | [2018/46] |
Former [2018/31] | HU | 03.11.2011 | |
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CZ | 01.10.2014 | ||
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EE | 01.10.2014 | ||
FI | 01.10.2014 | ||
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LT | 01.10.2014 | ||
LV | 01.10.2014 | ||
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MK | 01.10.2014 | ||
MT | 01.10.2014 | ||
NL | 01.10.2014 | ||
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TR | 01.10.2014 | ||
IE | 03.11.2014 | ||
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CH | 30.11.2014 | ||
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NO | 01.01.2015 | ||
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PT | 02.02.2015 | ||
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TR | 01.10.2014 | ||
IE | 03.11.2014 | ||
LU | 03.11.2014 | ||
BE | 30.11.2014 | ||
CH | 30.11.2014 | ||
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GR | 02.01.2015 | ||
IS | 01.02.2015 | ||
PT | 02.02.2015 | ||
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IE | 03.11.2014 | ||
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PT | 02.02.2015 | ||
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BE | 30.11.2014 | ||
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LI | 30.11.2014 | ||
NO | 01.01.2015 | ||
GR | 02.01.2015 | ||
IS | 01.02.2015 | ||
PT | 02.02.2015 | ||
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BE | 30.11.2014 | ||
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LI | 30.11.2014 | ||
NO | 01.01.2015 | ||
GR | 02.01.2015 | ||
IS | 01.02.2015 | ||
PT | 02.02.2015 | ||
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Former [2015/16] | NL | 01.10.2014 | Cited in | International search | [AD]WO2008031513 (BAYER HEALTHCARE AG [DE], et al) [AD] 1-11 * page 2, line 2 - page 2, line 4; example 9 *; | [A]WO2010079120 (BAYER SCHERING PHARMA AG [DE], et al) [A] 1-11 * page 2, line 25 - page 2, line 28; examples 8,9 * | by applicant | WO9816223 | WO2008031513 | WO2005030121 | WO2011119518 | WO2011115804 | - WU ET AL., BLOOD, (1994), vol. 84, page 4226 | - MÜLSCH ET AL., BRIT. J PHARMACOL., (1997), vol. 120, page 681 | - GOLDBERG ET AL., J BIOL. CHEM., (1977), vol. 252, page 1279 | - PETTIBONE ET AL., EUR. J PHARMACOL., (1985), vol. 116, page 307 | - YU ET AL., BRIT. J PHARMACOL., (1995), vol. 114, page 1587 | - L.F.CAVALIERI, J.F.TANKER, A.BENDICH, J.AM.CHEM.SOC., (1949), vol. 71, page 533 | - HELVETICA CHIMICA ACTA, (1951), vol. 34, pages 835 - 40 | - F. WUNDER ET AL., ANAL. BIOCHEM., (2005), vol. 339, pages 104 - 112 | - KLAUS WITTE, KAI HU, JOHANNA SWIATEK, CLAUDIA MÜSSIG, GEORG ERTL, BJÖRN LEMMER, "Experimental heart failure in rats: effects on cardiovascular circadian rhythms and on myocardial ßadrenergic signaling", CARDIOVASC RES, (2000), vol. 47, no. 2, pages 203 - 405 | - KOZO OKAMOTO, "Spontaneous hypertension in rats", INT REV EXP PATHOL, (1969), vol. 7, pages 227 - 270 | - MAARTEN VAN DEN BUUSE, "Circadian Rhythms of Blood Pressure, Heart Rate, and Locomotor Activity in Spontaneously Hypertensive Rats as Measured With Radio-Telemetry", PHYSIOLOGY & BEHAVIOR, (1994), vol. 55, no. 4, pages 783 - 787 |