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Extract from the Register of European Patents

EP About this file: EP2597086

EP2597086 - CYCLIC N,N'-DIARYLTHIOUREAS AND N,N'-DIARYLUREAS AS ANDROGEN RECEPTOR ANTAGONISTS, ANTI-CANCER AGENT, METHOD FOR PRODUCING AND USING SAME [Right-click to bookmark this link]
StatusThe application is deemed to be withdrawn
Status updated on  12.12.2014
Database last updated on 19.10.2024
Most recent event   Tooltip12.12.2014Application deemed to be withdrawnpublished on 14.01.2015  [2015/03]
Applicant(s)For all designated states
Ivachtchenko, Alexandre Vasilievich
2874 Calle Rancho Vista
Encinitas, CA 92024 / RU
For all designated states
Ivashchenko, Andrey Alexandrovich
ul. Abramtsevskaya, 4/2-27
Moscow 127576 / RU
For all designated states
Savchuk, Nikolay Filippovich
ul. Nametkina 9-35
Moscow 117420 / RU
[2013/22]
Inventor(s)01 / MITKIN, Oleg Dmitrievich
Kurkinskoe shosse 20-62
Khimki
Moskovskaya obl. 141400 / RU
 [2013/22]
Representative(s)Zellentin & Partner mbB Patentanwälte
Rubensstraße 30
67061 Ludwigshafen / DE
[N/P]
Former [2013/22]Patentanwälte Zellentin & Partner
Rubensstrasse 30
67061 Ludwigshafen / DE
Application number, filing date11809933.201.07.2011
WO2011RU00476
Priority number, dateRU2010013061822.07.2010         Original published format: RU 2010130618
[2013/22]
Filing languageRU
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2012011840
Date:26.01.2012
Language:RU
[2012/04]
Type: A1 Application with search report 
No.:EP2597086
Date:29.05.2013
Language:EN
[2013/22]
Search report(s)International search report - published on:RU26.01.2012
(Supplementary) European search report - dispatched on:EP09.10.2013
ClassificationIPC:C07D239/10, C07D239/22, C07D233/86, C07D233/72, C07D471/10, C07D491/107, C07D249/12, A61K31/4196, A61K31/513, A61K31/4166, A61K31/4188, A61K31/527, A61K9/20, A61K9/48, A61K9/08, A61P35/00
[2013/22]
CPC:
C07D233/86 (EP,KR,US); A61K9/0019 (EP,KR,US); A61K9/2018 (EP,US);
A61K9/2059 (EP,KR,US); A61K9/2095 (EP,US); A61K9/4858 (EP,US);
A61P13/08 (EP); A61P35/00 (EP); A61P43/00 (EP);
C07D233/72 (EP,US); C07D233/74 (KR); C07D239/10 (EP,US);
C07D239/22 (EP,US); C07D249/12 (EP,US); C07D471/10 (EP,US);
C07D491/107 (EP,US) (-)
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   RS,   SE,   SI,   SK,   SM,   TR [2013/22]
TitleGerman:ZYKLISCHE N,N'-DIARYLTHIOHARNSTOFFE UND N,N'-DIARYLHARNSTOFFE AS ANDROGENREZEPTORANTAGONISTEN, ANTI-KREBSMITTEL DAMIT SOWIE VERFAHREN ZU IHRER HERSTELLUNG UND VERWENDUNG[2013/22]
English:CYCLIC N,N'-DIARYLTHIOUREAS AND N,N'-DIARYLUREAS AS ANDROGEN RECEPTOR ANTAGONISTS, ANTI-CANCER AGENT, METHOD FOR PRODUCING AND USING SAME[2013/22]
French:N,N'-DIARYLURÉES ET N,N'-DIARYLTHIOURÉES CYCLIQUES, ANTAGONISTES DE RÉCEPTEURS D'ANDROGÈNES, AGENT ANTI-CANCER ET PROCÉDÉ DE PRODUCTION ET D'APPLICATION[2013/22]
Entry into regional phase22.02.2013Translation filed 
22.02.2013National basic fee paid 
22.02.2013Search fee paid 
22.02.2013Designation fee(s) paid 
22.02.2013Examination fee paid 
Examination procedure25.01.2012Request for preliminary examination filed
International Preliminary Examining Authority: RU
22.02.2013Amendment by applicant (claims and/or description)
22.02.2013Examination requested  [2013/22]
07.05.2014Application deemed to be withdrawn, date of legal effect  [2015/03]
09.07.2014Despatch of communication that the application is deemed to be withdrawn, reason: reply to the communication from the examining division not received in time  [2015/03]
Divisional application(s)EP14001526.4  / EP2767531
Fees paidRenewal fee
31.07.2013Renewal fee patent year 03
Penalty fee
Additional fee for renewal fee
31.07.201404   M06   Not yet paid
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Documents cited:Search   [ ] - No further relevant documents disclosed
International search[X]WO2006124118  (UNIV CALIFORNIA [US], et al);
 [X]WO2007127010  (UNIV CALIFORNIA [US], et al);
 [A]RU2152934  (ROUSSEL UCLAF [FR])
 [X]  - PRAKASH VISHNU ET AL., "Update on options for treatment of metastatic castration-resistant prostate cancer", ONCO TARGETS AND THERAPY, (2010), vol. 3, pages 39 - 51
 [X]  - CA, ACS, Database accession no. 151: 115902
    [ ] - TRAN CHRIS ET AL., "Development of a Second-Generation Antiandrogen for Treatment of Advanced Prostate Cancer", SCIENCE, (2009), vol. 324, no. 5298, doi:doi:10.1126/science.1168175, pages 787 - 790, XP002696684

DOI:   http://dx.doi.org/10.1126/science.1168175
by applicantWO2006124118
 WO2007127010
    - DRUG DATA REP., (2009), vol. 31, no. 6, page 609
    - BERGE S.M. ET AL., "Pharmaceutical Salts", J.PHARM.SCI., (1977), vol. 66, doi:doi:10.1002/jps.2600660104, pages 1 - 19, XP002675560

DOI:   http://dx.doi.org/10.1002/jps.2600660104
    - CHENG, Y.; PRUSOFF, W. H., "Relationship between the inhibition constant (K;) and the concentration of inhibitor which causes 50 per cent inhibition (IC5o) of an enzymatic reaction", BIOCHEM PHARMACOL., (1973), vol. 22, doi:doi:10.1016/0006-2952(73)90196-2, pages 3099 - 3108, XP001106687

DOI:   http://dx.doi.org/10.1016/0006-2952(73)90196-2
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.