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Extract from the Register of European Patents

EP About this file: EP2595994

EP2595994 - PROCESS FOR PREPARING PYRANO - [2,3-C]PYRIDINE DERIVATIVES [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  24.02.2017
Database last updated on 02.09.2024
Most recent event   Tooltip12.10.2018Lapse of the patent in a contracting state
New state(s): AL		published on 14.11.2018  [2018/46]
Applicant(s)For all designated states
Glaxo Group Limited
980 Great West Road
Brentford, Middlesex TW8 9GS / GB
[2013/22]
Inventor(s)01 / SISKO, Joseph
GlaxoSmithKline
c/o Global Patents
709 Swedeland Road
King of Prussia, PA 19406 / US
02 / MANS, Douglas
GlaxoSmithKline
c/o Global Patents
709 Swedeland Road
King of Prussia, PA 19406 / US
03 / YIN, Hao
GlaxoSmithKline
c/o Global Patents
709 Swedeland Road
King of Prussia, PA 19406 / US
 [2016/16]
Former [2013/22]01 / SISKO, Joseph
GlaxoSmithKline
c/o Global Patents
709 Swedeland Road
King of Prussia
PA 19406 / US
02 / MANS, Douglas
GlaxoSmithKline
c/o Global Patents
709 Swedeland Road
King or Prussia
PA 19406 / US
03 / YIN, Hao
GlaxoSmithKline
c/o Global Patents
709 Swedeland Road
King of Prussia
PA 19406 / US
Representative(s)Quillin, Helen Kaye, et al
GlaxoSmithKline
Global Patents (CN925.1)
980 Great West Road
Brentford, Middlesex TW8 9GS / GB
[N/P]
Former [2016/16]Valentine, Jill Barbara
GlaxoSmithKline
Global Patents (CN925.1)
980 Great West Road
Brentford, Middlesex TW8 9GS / GB
Former [2013/22]Valentine, Jill Barbara
GlaxoSmithKline Corporate Intellectual Property (CN9.25.1) 980 Great West Road
Brentford, Middlesex TW8 9GS / GB
Application number, filing date11810260.719.07.2011
[2016/16]
WO2011US44489
Priority number, dateUS20100365880P20.07.2010         Original published format: US 365880 P
[2013/22]
Filing languageEN
Procedural languageEN
PublicationType: A2 Application without search report
No.:WO2012012391
Date:26.01.2012
Language:EN
[2012/04]
Type: A2 Application without search report 
No.:EP2595994
Date:29.05.2013
Language:EN
The application published by WIPO in one of the EPO official languages on 26.01.2012 takes the place of the publication of the European patent application.
[2013/22]
Type: B1 Patent specification 
No.:EP2595994
Date:20.04.2016
Language:EN
[2016/16]
Search report(s)International search report - published on:US08.08.2013
(Supplementary) European search report - dispatched on:EP06.11.2014
ClassificationIPC:C07D491/052, C07D491/044
[2014/50]
CPC:
C07D491/052 (EP,CN,US); C07D491/04 (KR); A61K31/436 (KR);
A61P31/00 (EP); C07D491/044 (EP,US)
Former IPC [2013/22]C07D498/02
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   RS,   SE,   SI,   SK,   SM,   TR [2013/22]
Extension statesBA11.02.2013
ME11.02.2013
TitleGerman:VERFAHREN ZUR HERSTELLUNG VON PYRANO-[2,3-C-] PYRIDIN-DERIVATEN[2013/22]
English:PROCESS FOR PREPARING PYRANO - [2,3-C]PYRIDINE DERIVATIVES[2013/22]
French:PROCÉDÉ DE PRÉPARATION DE DÉRIVÉS PYRANO-[2,3-C]PYRIDINE[2013/22]
Entry into regional phase11.02.2013National basic fee paid 
11.02.2013Search fee paid 
11.02.2013Designation fee(s) paid 
11.02.2013Examination fee paid 
Examination procedure11.02.2013Amendment by applicant (claims and/or description)
11.02.2013Examination requested  [2013/22]
07.07.2015Communication of intention to grant the patent
18.12.2015Communication of intention to grant the patent
23.02.2016Fee for grant paid
23.02.2016Fee for publishing/printing paid
23.02.2016Receipt of the translation of the claim(s)
Divisional application(s)The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is  07.07.2015
Opposition(s)23.01.2017No opposition filed within time limit [2017/13]
Fees paidRenewal fee
08.07.2013Renewal fee patent year 03
08.07.2014Renewal fee patent year 04
09.07.2015Renewal fee patent year 05
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court		 See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipHU19.07.2011
AL20.04.2016
AT20.04.2016
BE20.04.2016
BG20.04.2016
CY20.04.2016
CZ20.04.2016
DK20.04.2016
EE20.04.2016
FI20.04.2016
HR20.04.2016
IS20.04.2016
LT20.04.2016
LV20.04.2016
MC20.04.2016
MK20.04.2016
NL20.04.2016
PL20.04.2016
RO20.04.2016
RS20.04.2016
SE20.04.2016
SI20.04.2016
SK20.04.2016
SM20.04.2016
TR20.04.2016
IE19.07.2016
LU19.07.2016
NO20.07.2016
GR21.07.2016
CH31.07.2016
LI31.07.2016
MT31.07.2016
PT22.08.2016
[2018/46]
Former [2018/38]HU19.07.2011
AT20.04.2016
BE20.04.2016
BG20.04.2016
CY20.04.2016
CZ20.04.2016
DK20.04.2016
EE20.04.2016
FI20.04.2016
HR20.04.2016
IS20.04.2016
LT20.04.2016
LV20.04.2016
MC20.04.2016
MK20.04.2016
NL20.04.2016
PL20.04.2016
RO20.04.2016
RS20.04.2016
SE20.04.2016
SI20.04.2016
SK20.04.2016
SM20.04.2016
TR20.04.2016
IE19.07.2016
LU19.07.2016
NO20.07.2016
GR21.07.2016
CH31.07.2016
LI31.07.2016
MT31.07.2016
PT22.08.2016
Former [2018/31]HU19.07.2011
AT20.04.2016
BE20.04.2016
CY20.04.2016
CZ20.04.2016
DK20.04.2016
EE20.04.2016
FI20.04.2016
HR20.04.2016
IS20.04.2016
LT20.04.2016
LV20.04.2016
MC20.04.2016
MK20.04.2016
NL20.04.2016
PL20.04.2016
RO20.04.2016
RS20.04.2016
SE20.04.2016
SI20.04.2016
SK20.04.2016
SM20.04.2016
TR20.04.2016
IE19.07.2016
LU19.07.2016
NO20.07.2016
GR21.07.2016
CH31.07.2016
LI31.07.2016
MT31.07.2016
PT22.08.2016
Former [2018/29]HU19.07.2011
AT20.04.2016
BE20.04.2016
CY20.04.2016
CZ20.04.2016
DK20.04.2016
EE20.04.2016
FI20.04.2016
HR20.04.2016
LT20.04.2016
LV20.04.2016
MC20.04.2016
MK20.04.2016
NL20.04.2016
PL20.04.2016
RO20.04.2016
RS20.04.2016
SE20.04.2016
SI20.04.2016
SK20.04.2016
SM20.04.2016
TR20.04.2016
IE19.07.2016
LU19.07.2016
NO20.07.2016
GR21.07.2016
CH31.07.2016
LI31.07.2016
PT22.08.2016
Former [2018/28]HU19.07.2011
AT20.04.2016
BE20.04.2016
CY20.04.2016
CZ20.04.2016
DK20.04.2016
EE20.04.2016
FI20.04.2016
HR20.04.2016
LT20.04.2016
LV20.04.2016
MC20.04.2016
MK20.04.2016
NL20.04.2016
PL20.04.2016
RO20.04.2016
RS20.04.2016
SE20.04.2016
SI20.04.2016
SK20.04.2016
SM20.04.2016
IE19.07.2016
LU19.07.2016
NO20.07.2016
GR21.07.2016
CH31.07.2016
LI31.07.2016
PT22.08.2016
Former [2017/37]AT20.04.2016
BE20.04.2016
CZ20.04.2016
DK20.04.2016
EE20.04.2016
FI20.04.2016
HR20.04.2016
LT20.04.2016
LV20.04.2016
MC20.04.2016
NL20.04.2016
PL20.04.2016
RO20.04.2016
RS20.04.2016
SE20.04.2016
SI20.04.2016
SK20.04.2016
SM20.04.2016
IE19.07.2016
LU19.07.2016
NO20.07.2016
GR21.07.2016
CH31.07.2016
LI31.07.2016
PT22.08.2016
Former [2017/25]AT20.04.2016
BE20.04.2016
CZ20.04.2016
DK20.04.2016
EE20.04.2016
FI20.04.2016
HR20.04.2016
LT20.04.2016
LV20.04.2016
MC20.04.2016
NL20.04.2016
PL20.04.2016
RO20.04.2016
RS20.04.2016
SE20.04.2016
SI20.04.2016
SK20.04.2016
SM20.04.2016
NO20.07.2016
GR21.07.2016
CH31.07.2016
LI31.07.2016
PT22.08.2016
Former [2017/22]AT20.04.2016
BE20.04.2016
CZ20.04.2016
DK20.04.2016
EE20.04.2016
FI20.04.2016
HR20.04.2016
LT20.04.2016
LV20.04.2016
MC20.04.2016
NL20.04.2016
PL20.04.2016
RO20.04.2016
RS20.04.2016
SE20.04.2016
SK20.04.2016
SM20.04.2016
NO20.07.2016
GR21.07.2016
CH31.07.2016
LI31.07.2016
PT22.08.2016
Former [2017/11]AT20.04.2016
BE20.04.2016
CZ20.04.2016
DK20.04.2016
EE20.04.2016
FI20.04.2016
HR20.04.2016
LT20.04.2016
LV20.04.2016
NL20.04.2016
PL20.04.2016
RO20.04.2016
RS20.04.2016
SE20.04.2016
SK20.04.2016
SM20.04.2016
NO20.07.2016
GR21.07.2016
PT22.08.2016
Former [2017/10]AT20.04.2016
BE20.04.2016
CZ20.04.2016
DK20.04.2016
EE20.04.2016
FI20.04.2016
HR20.04.2016
LT20.04.2016
LV20.04.2016
NL20.04.2016
PL20.04.2016
RO20.04.2016
RS20.04.2016
SE20.04.2016
SK20.04.2016
NO20.07.2016
GR21.07.2016
PT22.08.2016
Former [2017/09]AT20.04.2016
BE20.04.2016
CZ20.04.2016
DK20.04.2016
EE20.04.2016
FI20.04.2016
HR20.04.2016
LT20.04.2016
LV20.04.2016
NL20.04.2016
PL20.04.2016
RO20.04.2016
RS20.04.2016
SE20.04.2016
NO20.07.2016
GR21.07.2016
PT22.08.2016
Former [2017/07]AT20.04.2016
BE20.04.2016
DK20.04.2016
FI20.04.2016
HR20.04.2016
LT20.04.2016
LV20.04.2016
NL20.04.2016
PL20.04.2016
RS20.04.2016
SE20.04.2016
NO20.07.2016
GR21.07.2016
PT22.08.2016
Former [2017/03]AT20.04.2016
BE20.04.2016
FI20.04.2016
HR20.04.2016
LT20.04.2016
LV20.04.2016
NL20.04.2016
PL20.04.2016
RS20.04.2016
SE20.04.2016
NO20.07.2016
GR21.07.2016
PT22.08.2016
Former [2016/52]AT20.04.2016
FI20.04.2016
HR20.04.2016
LT20.04.2016
LV20.04.2016
NL20.04.2016
PL20.04.2016
RS20.04.2016
SE20.04.2016
NO20.07.2016
GR21.07.2016
PT22.08.2016
Former [2016/51]AT20.04.2016
FI20.04.2016
HR20.04.2016
LT20.04.2016
LV20.04.2016
NL20.04.2016
PL20.04.2016
RS20.04.2016
NO20.07.2016
GR21.07.2016
PT22.08.2016
Former [2016/50]AT20.04.2016
FI20.04.2016
HR20.04.2016
LT20.04.2016
LV20.04.2016
NL20.04.2016
PL20.04.2016
RS20.04.2016
NO20.07.2016
Former [2016/49]FI20.04.2016
LT20.04.2016
NL20.04.2016
PL20.04.2016
NO20.07.2016
Former [2016/46]LT20.04.2016
NO20.07.2016
Documents cited:Search[A]US2003130305  (WALKER DANIEL PATRICK [US], et al) [A] 1-13 * example 18; claim - *;
 [T]  - S.N. GOODMAN ET. AL., "Synthesis of Fused Dihydropyrano(furano)pyridines via [4+2] Cycloaddition of 5-Alkenoxy Substitued Oxazoles.", ORGANIC LETTERS, (20120307), vol. 14, no. 6, pages 1604 - 1607, XP002723731 [T] 1-13 * page 1606; figure 2 *

DOI:   http://dx.doi.org/10.1021/ol300351v
International search[A]  - MOVASSAGHI ET AL., "A Versatile Cyclodehydration Reaction for the Synthesis of lsoquinoline and beta-Carboline Derivatives", ORG LETT., vol. 10, no. 16, (2008), pages 3485 - 3488, URL: http:/lwww.ncbi.nlm.nih.govlpmdarticIesIPMC26928361pdfinihms-108650.pdf, XP055079588

DOI:   http://dx.doi.org/10.1021/ol801264u
 [A]  - WILLIAMS ET AL., "Studies of stereocontrolled allylation reactions for the total synthesis of phorboxazole A", PNAS, vol. 101, no. 33, (2004), pages 12058 - 12063, URL: http://www.pnas.orglcontenU101/33/12058.fufl.pdf+html, XP055079589

DOI:   http://dx.doi.org/10.1073/pnas.0402477101
 [A]  - MARTIN ET AL., "A Convenient, One Step Synthesis of Pyrano(2,3-b)Pyridines", TETRAHEDRON, (1988), vol. 44, no. 18, pages 5861 - 5868, XP055079591

DOI:   http://dx.doi.org/10.1016/S0040-4020(01)81443-5
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