blank Quick help
blank Maintenance news

Scheduled maintenance

Regular maintenance outages:
between 05.00 and 05.15 hrs CET (Monday to Sunday).

Other outages
Availability
Register Forum

2022.02.11

More...
blank News flashes

News flashes

New version of the European Patent Register - SPC information for Unitary Patents.

2024-03-06

More...
blank Related links

Extract from the Register of European Patents

EP About this file: EP2702042

EP2702042 - NOVEL BICYCLIC NITROGEN CONTAINING HETEROARYL TGR5 RECEPTOR MODULATORS [Right-click to bookmark this link]
StatusThe application is deemed to be withdrawn
Status updated on  14.11.2014
Database last updated on 06.07.2024
Most recent event   Tooltip14.11.2014Application deemed to be withdrawnpublished on 17.12.2014  [2014/51]
Applicant(s)For all designated states
Bristol-Myers Squibb Company
Route 206 and Province Line Road
Princeton, NJ 08543 / US
[N/P]
Former [2014/10]For all designated states
Bristol-Myers Squibb Company
Route 206 and Province Line Road
Princeton, NJ 05843-4000 / US
Inventor(s)01 / ROBL, Jeffrey A.
c/o Bristol-Myers Squibb Company
311 Pennington-Rocky Hill Road
Pennington, New Jersey 08534 / US
02 / LI, Jun
c/o Bristol-Myers Squibb Company
311 Pennington-Rocky Hill Road
Pennington, New Jersey 08534 / US
03 / KENNEDY, Lawrence J.
c/o Bristol-Myers Squibb Company
311 Pennington-Rocky Hill Road
Pennington, New Jersey 08534 / US
04 / WALKER, Steven J.
c/o Bristol-Myers Squibb Company
311 Pennington-Rocky Hill Road
Pennington, New Jersey 08534 / US
05 / WANG, Haixia
c/o Bristol-Myers Squibb Company
311 Pennington-Rocky Hill Road
Pennington, New Jersey 08534 / US
06 / WASHBURN, William N.
c/o Bristol-Myers Squibb Company
311 Pennington-Rocky Hill Road
Pennington, New Jersey 08534 / US
07 / AHMAD, Saleem
c/o Bristol-Myers Squibb Company
Route 206 and Province Line Road
Princeton, New Jersey 08543-4000 / US
08 / NGU, Khehyong
c/o Bristol-Myers Squibb Company
Route 206 and Province Line Road
Princeton, New Jersey 08543-4000 / US
 [2014/10]
Representative(s)Reitstötter Kinzebach
Patentanwälte
Sternwartstraße 4
81679 München / DE
[N/P]
Former [2014/10]Reitstötter - Kinzebach
Patentanwälte
Sternwartstrasse 4
81679 München / DE
Application number, filing date12723982.027.04.2012
WO2012US35327
Priority number, dateUS201161479917P28.04.2011         Original published format: US 201161479917 P
[2014/10]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2012149236
Date:01.11.2012
Language:EN
[2012/44]
Type: A1 Application with search report 
No.:EP2702042
Date:05.03.2014
Language:EN
The application published by WIPO in one of the EPO official languages on 01.11.2012 takes the place of the publication of the European patent application.
[2014/10]
Search report(s)International search report - published on:EP01.11.2012
ClassificationIPC:C07D215/08, C07D401/04, C07D403/04, C07D413/04, C07D417/04, A61K31/4709, A61K31/553, A61K31/554, A61P3/00, A61P9/00, C07D401/14, C07D413/14
[2014/10]
CPC:
C07D401/04 (EP,CN,US); A61K31/47 (EP,US); A61K31/4709 (EP,US);
A61K31/473 (EP,US); A61K31/4747 (EP,US); A61K31/496 (EP,US);
A61K31/506 (EP,US); A61K31/5377 (EP,US); A61K31/5415 (EP,US);
A61K31/55 (EP,US); A61K31/553 (EP,US); A61K31/554 (EP,US);
A61K31/675 (EP,US); A61K45/06 (US); A61P1/18 (EP);
A61P13/12 (EP); A61P17/02 (EP); A61P25/00 (EP);
A61P27/02 (EP); A61P3/00 (EP); A61P3/04 (EP);
A61P3/06 (EP); A61P3/10 (EP); A61P43/00 (EP);
A61P5/50 (EP); A61P9/00 (EP); A61P9/10 (EP);
A61P9/12 (EP); C07D215/08 (EP,CN,US); C07D215/12 (CN);
C07D215/14 (CN); C07D221/16 (EP,US); C07D401/12 (EP,CN,US);
C07D401/14 (EP,CN,US); C07D403/04 (EP,CN,US); C07D405/14 (EP,US);
C07D409/14 (EP,US); C07D413/04 (EP,CN,US); C07D413/14 (EP,CN,US);
C07D417/04 (EP,CN,US); C07F9/60 (US) (-)
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   RS,   SE,   SI,   SK,   SM,   TR [2014/10]
TitleGerman:NEUE BICYCLISCHE STICKSTOFFHALTIGE HETEROARYL-TGR5-REZEPTORMODULATOREN[2014/10]
English:NOVEL BICYCLIC NITROGEN CONTAINING HETEROARYL TGR5 RECEPTOR MODULATORS[2014/10]
French:NOUVEAUX MODULATEURS DU RÉCEPTEUR TGR5 SOUS FORME D'HÉTÉROARYLES BICYCLIQUES CONTENANT DE L'AZOTE[2014/10]
Entry into regional phase26.11.2013National basic fee paid 
26.11.2013Designation fee(s) paid 
26.11.2013Examination fee paid 
Examination procedure26.11.2013Examination requested  [2014/10]
24.06.2014Application deemed to be withdrawn, date of legal effect  [2014/51]
30.07.2014Despatch of communication that the application is deemed to be withdrawn, reason: reply to the Extended European Search Report/Written Opinion of the International Searching Authority/International Preliminary Examination Report/Supplementary international search report not received in time  [2014/51]
Fees paidRenewal fee
25.03.2014Renewal fee patent year 03
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court
See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Cited inInternational search[A]JPH07242663  (YOSHITOMI PHARMACEUTICAL) [A] 1-15 * compounds 6, 8-11 *;
 [A]US2010105906  (BISSANTZ CATERINA [FR], et al) [A] 1-15 * paragraph [0455] - paragraph [0463]; examples 74, 130 *;
 [I]WO2010107768  (SCHERING CORP [US], et al) [I] 1-15 * examples C-7; claims 7, 11 *;
 [A]  - ZHAO ET AL, "3,4-Dihydro-2H-benzo[1,4]oxazine derivatives as 5-HT6 receptor antagonists", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, PERGAMON, ELSEVIER SCIENCE, GB, (20070615), vol. 17, no. 12, doi:10.1016/J.BMCL.2006.12.093, ISSN 0960-894X, pages 3504 - 3507, XP022097811 [A] 1-15 * compound 13 *

DOI:   http://dx.doi.org/10.1016/j.bmcl.2006.12.093
by applicantWO2008067222
 WO2008067219
 WO2008097976
 WO2009026241
 WO2010016846
 WO2010059859
 WO2010093845
 WO2011071565
    - Remington's Pharmaceutical Sciences, MACK PUBLISHING COMPANY, (1985), page 1418
    - "Design and Application of Prodrugs", BUNDGAARD, H. ET AL., A Textbook of Drug Design and Development, HARWOOD ACADEMIC PUBLISHERS, (1991), pages 113 - 191
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.