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Extract from the Register of European Patents

EP About this file: EP2641590

EP2641590 - Pharmaceutical compositions comprising imidazoquinolin(amines) and derivatives thereof suitable for local administration [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  09.02.2018
Database last updated on 21.05.2024
FormerThe patent has been granted
Status updated on  03.03.2017
FormerGrant of patent is intended
Status updated on  13.01.2017
FormerExamination is in progress
Status updated on  21.12.2016
FormerGrant of patent is intended
Status updated on  16.12.2016
Most recent event   Tooltip26.06.2020Lapse of the patent in a contracting state
New state(s): CY, MK
published on 29.07.2020  [2020/31]
Applicant(s)For all designated states
Urogen Pharma Ltd.
9 Ha`Tassiya Street
4365007 Ra`anana / IL
[2016/42]
Former [2013/39]For all designated states
Telormedix SA
Via della Posta 10
6934 Bioggio / CH
Inventor(s)01 / Leoni, Lorenzo
Via Perdaglie 32
6527 Lodrino / CH
02 / Maj, Roberto
Via Favia 7
21047 Saronno / IT
03 / Pattarino, Franco
Via Genova 77
10126 Torino / IT
04 / Vecchio, Carlo
Via Comignago 2B Revislate
28010 Veruno / IT
 [2013/39]
Representative(s)Graf von Stosch, Andreas, et al
Graf von Stosch
Patentanwaltsgesellschaft mbH
Prinzregentenstraße 22
80538 München / DE
[2017/14]
Former [2013/39]Graf von Stosch, Andreas, et al
Graf von Stosch Patentanwaltsgesellschaft mbH Prinzregentenstrasse 22
80538 München / DE
Application number, filing date13001958.105.02.2010
[2013/39]
Priority number, dateWO2009EP0083406.02.2009         Original published format: PCT/EP2009/000834
[2013/39]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report 
No.:EP2641590
Date:25.09.2013
Language:EN
[2013/39]
Type: B1 Patent specification 
No.:EP2641590
Date:05.04.2017
Language:EN
[2017/14]
Search report(s)(Supplementary) European search report - dispatched on:EP23.08.2013
ClassificationIPC:A61K9/00, A61K47/12, A61K31/4745, A61P13/10, A61P35/00, // A61K47/10, A61K47/34, A61K47/40
[2016/34]
CPC:
A61K47/40 (EP,IL,KR,US); A61K31/4745 (EP,IL,KR,US); A61K47/10 (EP,KR,US);
A61K47/12 (EP,IL,KR,US); A61K47/34 (EP,IL,KR,US); A61K9/00 (IL);
A61K9/0014 (EP,KR,US); A61K9/0034 (EP,KR,US); A61P13/00 (EP);
A61P13/10 (EP); A61P17/00 (EP); A61P17/12 (EP);
A61P35/00 (EP); Y02A50/30 (EP) (-)
Former IPC [2013/39]A61K9/00, A61K47/12, A61K31/4745, A61P13/10, A61P35/00, // A61K47/10, A61K47/40
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   SE,   SI,   SK,   SM,   TR [2013/39]
Extension statesAL15.04.2013
BA15.04.2013
RS15.04.2013
TitleGerman:Pharmazeutische Zusammensetzungen mit Imidazochinolin(aminen) und Derivativen daraus zur lokalen Verabreichung[2013/39]
English:Pharmaceutical compositions comprising imidazoquinolin(amines) and derivatives thereof suitable for local administration[2013/39]
French:Compositions pharmaceutiques comprenant des imidazoquinolines (amines) et ses dérivés appropriés pour une administration locale[2013/39]
Examination procedure15.04.2013Examination requested  [2013/39]
25.03.2014Amendment by applicant (claims and/or description)
16.02.2016Despatch of a communication from the examining division (Time limit: M04)
24.06.2016Reply to a communication from the examining division
10.08.2016Communication of intention to grant the patent
12.12.2016Disapproval of the communication of intention to grant the patent by the applicant or resumption of examination proceedings by the EPO
12.12.2016Fee for grant paid
12.12.2016Fee for publishing/printing paid
12.01.2017Information about intention to grant a patent
12.01.2017Receipt of the translation of the claim(s)
Parent application(s)   TooltipEP10703023.1  / EP2393474
Divisional application(s)The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued (EP20100703023) is  18.07.2012
Opposition(s)08.01.2018No opposition filed within time limit [2018/11]
Fees paidRenewal fee
15.04.2013Renewal fee patent year 03
15.04.2013Renewal fee patent year 04
30.12.2013Renewal fee patent year 05
16.12.2014Renewal fee patent year 06
26.02.2016Renewal fee patent year 07
20.02.2017Renewal fee patent year 08
Opt-out from the exclusive  Tooltip
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Patent Court
See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipHU05.02.2010
AT05.04.2017
CY05.04.2017
CZ05.04.2017
DK05.04.2017
EE05.04.2017
ES05.04.2017
FI05.04.2017
HR05.04.2017
IT05.04.2017
LT05.04.2017
LV05.04.2017
MC05.04.2017
MK05.04.2017
NL05.04.2017
PL05.04.2017
PT05.04.2017
RO05.04.2017
SE05.04.2017
SI05.04.2017
SK05.04.2017
SM05.04.2017
TR05.04.2017
BG05.07.2017
NO05.07.2017
GR06.07.2017
IS05.08.2017
[2020/31]
Former [2020/27]HU05.02.2010
AT05.04.2017
CZ05.04.2017
DK05.04.2017
EE05.04.2017
ES05.04.2017
FI05.04.2017
HR05.04.2017
IT05.04.2017
LT05.04.2017
LV05.04.2017
MC05.04.2017
NL05.04.2017
PL05.04.2017
PT05.04.2017
RO05.04.2017
SE05.04.2017
SI05.04.2017
SK05.04.2017
SM05.04.2017
TR05.04.2017
BG05.07.2017
NO05.07.2017
GR06.07.2017
IS05.08.2017
Former [2020/15]AT05.04.2017
CZ05.04.2017
DK05.04.2017
EE05.04.2017
ES05.04.2017
FI05.04.2017
HR05.04.2017
IT05.04.2017
LT05.04.2017
LV05.04.2017
MC05.04.2017
NL05.04.2017
PL05.04.2017
RO05.04.2017
SE05.04.2017
SI05.04.2017
SK05.04.2017
SM05.04.2017
TR05.04.2017
BG05.07.2017
NO05.07.2017
GR06.07.2017
IS05.08.2017
Former [2018/44]AT05.04.2017
CZ05.04.2017
DK05.04.2017
EE05.04.2017
ES05.04.2017
FI05.04.2017
HR05.04.2017
IT05.04.2017
LT05.04.2017
LV05.04.2017
MC05.04.2017
NL05.04.2017
PL05.04.2017
RO05.04.2017
SE05.04.2017
SI05.04.2017
SK05.04.2017
SM05.04.2017
BG05.07.2017
NO05.07.2017
GR06.07.2017
IS05.08.2017
Former [2018/25]AT05.04.2017
CZ05.04.2017
DK05.04.2017
EE05.04.2017
ES05.04.2017
FI05.04.2017
HR05.04.2017
IT05.04.2017
LT05.04.2017
LV05.04.2017
NL05.04.2017
PL05.04.2017
RO05.04.2017
SE05.04.2017
SI05.04.2017
SK05.04.2017
SM05.04.2017
BG05.07.2017
NO05.07.2017
GR06.07.2017
IS05.08.2017
Former [2018/11]AT05.04.2017
CZ05.04.2017
DK05.04.2017
EE05.04.2017
ES05.04.2017
FI05.04.2017
HR05.04.2017
IT05.04.2017
LT05.04.2017
LV05.04.2017
NL05.04.2017
PL05.04.2017
RO05.04.2017
SE05.04.2017
SK05.04.2017
SM05.04.2017
BG05.07.2017
NO05.07.2017
GR06.07.2017
IS05.08.2017
Former [2018/10]AT05.04.2017
CZ05.04.2017
DK05.04.2017
EE05.04.2017
ES05.04.2017
FI05.04.2017
HR05.04.2017
LT05.04.2017
LV05.04.2017
NL05.04.2017
PL05.04.2017
RO05.04.2017
SE05.04.2017
SK05.04.2017
BG05.07.2017
NO05.07.2017
GR06.07.2017
IS05.08.2017
Former [2018/09]AT05.04.2017
DK05.04.2017
EE05.04.2017
ES05.04.2017
FI05.04.2017
HR05.04.2017
LT05.04.2017
LV05.04.2017
NL05.04.2017
PL05.04.2017
SE05.04.2017
BG05.07.2017
NO05.07.2017
GR06.07.2017
IS05.08.2017
Former [2017/50]AT05.04.2017
ES05.04.2017
FI05.04.2017
HR05.04.2017
LT05.04.2017
LV05.04.2017
NL05.04.2017
PL05.04.2017
SE05.04.2017
BG05.07.2017
NO05.07.2017
GR06.07.2017
IS05.08.2017
Former [2017/49]AT05.04.2017
ES05.04.2017
FI05.04.2017
HR05.04.2017
LT05.04.2017
NL05.04.2017
NO05.07.2017
GR06.07.2017
IS05.08.2017
Former [2017/48]NL05.04.2017
Documents cited:Search[XI]EP0394026  (RIKER LABORATORIES INC [US]) [X] 1,5,7,11,13,15 * page 2, line 34 - line 37 * * page 2, line 54 - page 3, line 3 * * examples 1,2,16 * [I] 2-4,6,8-10,12,14,16-19;
 [XI]US2007264317  (YOSHA IDO [IL], et al) [X] 1,5,7,11,13,15 * paragraph [0029]; example 6; table 6 * [I] 2-4,6,8-10,12,14,16-19;
 [XI]US2008207674  (STOESZ JAMES D [US], et al) [X] 1,4,5,7,11,13,15 * page 3 - page 4; tables 3-4 * * examples 13-18 * * paragraph [0041] * [I] 2,3,6,8-10,12,14,16-19;
 [XI]WO2008118763  (GRACEWAY PHARMACEUTICALS LLC [US], et al) [X] 1,5,7,11,13,15 * page 1, paragraph 1 * * page 26; example 16 * [I] 2-4,6,8-10,12,14,16-19;
 [XP]WO2009091541  (DOW PHARMACEUTICAL SCIENCES [US], et al) [XP] 1,3,5,6,11,13,15,17,18 * page 1, paragraph 2 - paragraph 3 * * examples 1,5-9; tables 1,12,14-17 * * page 12, paragraph L - page 13, paragraph 1 *;
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DOI:   http://dx.doi.org/10.1097/01.SMJ.0000176712.01491.98
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DOI:   http://dx.doi.org/10.1016/S1473-3099(01)00095-0
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DOI:   http://dx.doi.org/10.1007/s11095-006-9104-4
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DOI:   http://dx.doi.org/10.2165/00003495-200767150-00006
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DOI:   http://dx.doi.org/10.2165/00003495-200767150-00006
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DOI:   http://dx.doi.org/10.1016/j.juro.2007.01.112
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DOI:   http://dx.doi.org/10.1016/j.juro.2007.01.112
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DOI:   http://dx.doi.org/10.1016/j.juro.2007.01.112
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DOI:   http://dx.doi.org/10.1007/s00262-004-0621-x
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DOI:   http://dx.doi.org/10.1016/S0140-6736(98)07422-4
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DOI:   http://dx.doi.org/10.1016/0090-4295(91)80166-5
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DOI:   http://dx.doi.org/10.1097/01.ju.0000091826.83705.79
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DOI:   http://dx.doi.org/10.1016/j.urolonc.2007.11.031
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DOI:   http://dx.doi.org/10.1097/01.ju.0000073852.24341.4a
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DOI:   http://dx.doi.org/10.1016/S0168-3659(02)00273-0
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DOI:   http://dx.doi.org/10.1016/S0140-6736(98)07422-4
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    - SMITH EB; SCHWARTZ M; KAWAMOTO H ET AL., "Antitumor effects of imidazoquinolines in urothelial cell carcinoma of the bladder", THE JOURNAL OF UROLOGY, (2007), vol. 177, pages 347 - 51
    - MANGSBO SM; NINALGA C; ESSAND M; LOSKOG A; TOTTERMAN TH, "CpG therapy is superior to BCG in an orthotopic bladder cancer model and generates CD4+ T-ell immunity", J IMMUNOTHER, (2008), vol. 31, pages 34 - 42
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    - SMITH EB; SCHWARTZ M; KAWAMOTO H ET AL., "Antitumor effects of imidazoquinolines in urothelial cell carcinoma of the bladder", THEJOURNALOF UROLOGY, (2007), vol. 177, doi:doi:10.1016/j.juro.2007.01.112, pages 2347 - 51, XP022078754

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