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EP About this file: EP2722051

EP2722051 - Monomethylvaline compounds having phenylalanine side-chain modifications at the C-terminus [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  13.09.2019
Database last updated on 11.09.2024
FormerThe patent has been granted
Status updated on  05.10.2018
FormerGrant of patent is intended
Status updated on  23.05.2018
FormerExamination is in progress
Status updated on  12.05.2017
Most recent event   Tooltip09.07.2021Lapse of the patent in a contracting state
New state(s): HU
published on 11.08.2021  [2021/32]
Applicant(s)For all designated states
Seattle Genetics, Inc.
21823 30th Drive, S.E.
Bothell, WA 98021 / US
[2014/17]
Inventor(s)01 / Doronina, Svetlana O.
10910 198th Place SE
Snohomish, WA 98296 / US
02 / Kline, Toni Beth
767 Bryant Street, No. 406
San Francisco, CA 94107 / US
 [2014/24]
Former [2014/17]01 / Doronina, Svetlana O.
10910 198th Place SE
Snohomish, Washington 98296 / US
02 / Kline, Toni Beth
2034B NW 60th Street
Seattle, Washington 981017 / US
Representative(s)Mewburn Ellis LLP
Aurora Building
Counterslip
Bristol BS1 6BX / GB
[N/P]
Former [2018/45]Andrews, Robert, et al
Mewburn Ellis LLP
City Tower
40 Basinghall Street
London EC2V 5DE / GB
Former [2014/17]Andrews, Robert, et al
Mewburn Ellis LLP
33 Gutter Lane
London Greater London EC2V 8AS / GB
Application number, filing date13190752.907.07.2006
[2014/17]
Priority number, dateUS20050697767P07.07.2005         Original published format: US 697767 P
[2014/17]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report 
No.:EP2722051
Date:23.04.2014
Language:EN
[2014/17]
Type: B1 Patent specification 
No.:EP2722051
Date:07.11.2018
Language:EN
[2018/45]
Search report(s)(Supplementary) European search report - dispatched on:EP21.03.2014
ClassificationIPC:A61K38/00, C07K7/02
[2018/22]
CPC:
A61K47/65 (EP,US); C07K16/00 (US); A61K47/6811 (EP,US);
A61K47/6849 (EP,US); A61P1/00 (EP); A61P11/00 (EP);
A61P13/12 (EP); A61P17/00 (EP); A61P19/00 (EP);
A61P21/00 (EP); A61P25/00 (EP); A61P27/02 (EP);
A61P3/10 (EP); A61P31/00 (EP); A61P35/00 (EP);
A61P35/02 (EP); A61P37/00 (EP); A61P37/02 (EP);
A61P37/06 (EP); A61P37/08 (EP); A61P43/00 (EP);
A61P5/14 (EP); A61P7/00 (EP); A61P9/00 (EP);
A61P9/10 (EP); C07K16/2878 (EP,US); C07K5/0205 (EP,US);
C07K5/10 (US); C07K7/02 (EP,US); C07K7/06 (US);
A61K38/00 (EP,US); Y02A50/30 (EP,US) (-)
Former IPC [2014/17]A61K38/00, C07K7/02, A61K47/48
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   NL,   PL,   PT,   RO,   SE,   SI,   SK,   TR [2014/17]
TitleGerman:Monomethylvalinverbindungen mit Phenylalaninseitenkettenmodifikationen am C-Terminus[2014/17]
English:Monomethylvaline compounds having phenylalanine side-chain modifications at the C-terminus[2014/17]
French:Composés de monométhylvaline présentant des modifications de la chaîne latérale de phénylalanine au niveau de la terminaison C[2014/17]
Examination procedure12.11.2013Examination requested  [2014/17]
13.02.2015Amendment by applicant (claims and/or description)
13.11.2015Despatch of a communication from the examining division (Time limit: M06)
17.06.2016Despatch of communication that the application is deemed to be withdrawn, reason: reply to the communication from the examining division not received in time
25.08.2016Reply to a communication from the examining division
03.05.2017Despatch of a communication from the examining division (Time limit: M04)
11.09.2017Reply to a communication from the examining division
24.05.2018Communication of intention to grant the patent
28.09.2018Fee for grant paid
28.09.2018Fee for publishing/printing paid
28.09.2018Receipt of the translation of the claim(s)
Parent application(s)   TooltipEP06786489.2  / EP1917020
Divisional application(s)EP18200998.5  / EP3498289
The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued (EP20060786489) is  25.10.2011
Opposition(s)08.08.2019No opposition filed within time limit [2019/42]
Request for further processing for:The application is deemed to be withdrawn due to failure to reply to the examination report
25.08.2016Request for further processing filed
25.08.2016Full payment received (date of receipt of payment)
Request granted
05.09.2016Decision despatched
The application is deemed to be withdrawn due to failure to reply to the Extended European Search Report/Written Opinion of the International Searching Authority/International Preliminary Examination Report/Supplementary international search report/Supplementary European search report
13.02.2015Request for further processing filed
13.02.2015Full payment received (date of receipt of payment)
Request granted
27.02.2015Decision despatched
Fees paidRenewal fee
12.11.2013Renewal fee patent year 03
12.11.2013Renewal fee patent year 04
12.11.2013Renewal fee patent year 05
12.11.2013Renewal fee patent year 06
12.11.2013Renewal fee patent year 07
12.11.2013Renewal fee patent year 08
28.07.2014Renewal fee patent year 09
27.07.2015Renewal fee patent year 10
27.07.2016Renewal fee patent year 11
27.07.2017Renewal fee patent year 12
27.07.2018Renewal fee patent year 13
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court
See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipHU07.07.2006
AT07.11.2018
CY07.11.2018
CZ07.11.2018
DK07.11.2018
EE07.11.2018
FI07.11.2018
LT07.11.2018
LV07.11.2018
MC07.11.2018
PL07.11.2018
RO07.11.2018
SE07.11.2018
SI07.11.2018
SK07.11.2018
TR07.11.2018
BG07.02.2019
GR08.02.2019
IS07.03.2019
PT07.03.2019
LU07.07.2019
[2021/32]
Former [2021/26]AT07.11.2018
CY07.11.2018
CZ07.11.2018
DK07.11.2018
EE07.11.2018
FI07.11.2018
LT07.11.2018
LV07.11.2018
MC07.11.2018
PL07.11.2018
RO07.11.2018
SE07.11.2018
SI07.11.2018
SK07.11.2018
TR07.11.2018
BG07.02.2019
GR08.02.2019
IS07.03.2019
PT07.03.2019
LU07.07.2019
Former [2020/27]AT07.11.2018
CZ07.11.2018
DK07.11.2018
EE07.11.2018
FI07.11.2018
LT07.11.2018
LV07.11.2018
MC07.11.2018
PL07.11.2018
RO07.11.2018
SE07.11.2018
SI07.11.2018
SK07.11.2018
TR07.11.2018
BG07.02.2019
GR08.02.2019
IS07.03.2019
PT07.03.2019
LU07.07.2019
Former [2020/17]AT07.11.2018
CZ07.11.2018
DK07.11.2018
EE07.11.2018
FI07.11.2018
LT07.11.2018
LV07.11.2018
MC07.11.2018
PL07.11.2018
RO07.11.2018
SE07.11.2018
SI07.11.2018
SK07.11.2018
TR07.11.2018
BG07.02.2019
GR08.02.2019
IS07.03.2019
PT07.03.2019
Former [2020/14]AT07.11.2018
CZ07.11.2018
DK07.11.2018
EE07.11.2018
FI07.11.2018
LT07.11.2018
LV07.11.2018
MC07.11.2018
PL07.11.2018
RO07.11.2018
SE07.11.2018
SI07.11.2018
SK07.11.2018
BG07.02.2019
GR08.02.2019
IS07.03.2019
PT07.03.2019
Former [2019/50]AT07.11.2018
CZ07.11.2018
DK07.11.2018
EE07.11.2018
FI07.11.2018
LT07.11.2018
LV07.11.2018
PL07.11.2018
RO07.11.2018
SE07.11.2018
SI07.11.2018
SK07.11.2018
BG07.02.2019
GR08.02.2019
IS07.03.2019
PT07.03.2019
Former [2019/40]AT07.11.2018
CZ07.11.2018
DK07.11.2018
EE07.11.2018
FI07.11.2018
LT07.11.2018
LV07.11.2018
PL07.11.2018
RO07.11.2018
SE07.11.2018
SK07.11.2018
BG07.02.2019
GR08.02.2019
IS07.03.2019
PT07.03.2019
Former [2019/37]AT07.11.2018
CZ07.11.2018
DK07.11.2018
EE07.11.2018
FI07.11.2018
LT07.11.2018
LV07.11.2018
PL07.11.2018
RO07.11.2018
SE07.11.2018
BG07.02.2019
GR08.02.2019
IS07.03.2019
PT07.03.2019
Former [2019/35]AT07.11.2018
CZ07.11.2018
DK07.11.2018
FI07.11.2018
LT07.11.2018
LV07.11.2018
PL07.11.2018
SE07.11.2018
BG07.02.2019
GR08.02.2019
IS07.03.2019
PT07.03.2019
Former [2019/34]AT07.11.2018
DK07.11.2018
FI07.11.2018
LT07.11.2018
LV07.11.2018
SE07.11.2018
BG07.02.2019
GR08.02.2019
IS07.03.2019
PT07.03.2019
Former [2019/26]AT07.11.2018
FI07.11.2018
LT07.11.2018
LV07.11.2018
SE07.11.2018
BG07.02.2019
GR08.02.2019
IS07.03.2019
PT07.03.2019
Former [2019/24]AT07.11.2018
FI07.11.2018
LT07.11.2018
LV07.11.2018
SE07.11.2018
BG07.02.2019
GR08.02.2019
IS07.03.2019
Former [2019/23]AT07.11.2018
FI07.11.2018
LT07.11.2018
LV07.11.2018
BG07.02.2019
IS07.03.2019
Former [2019/22]FI07.11.2018
LT07.11.2018
BG07.02.2019
IS07.03.2019
Former [2019/21]FI07.11.2018
LT07.11.2018
IS07.03.2019
Former [2019/20]LT07.11.2018
Documents cited:Search[XI]WO9413695  (BASF AG [DE]) [X] 1-4 * the whole document * * page 3; compound 70 * [I] 1-14;
 [I]US5767237  (SAKAKIBARA KYOICHI [JP], et al) [I] 1-14 * the whole document *;
 [XI]WO0118032  (BASF AG [DE], et al) [X] 1-4 * the whole document * [I] 1-14;
 [XI]WO2004010957  (SEATTLE GENETICS INC [US], et al) [X] 1-14 * the whole document * * pages 20-28 * [I] 1-14;
 [XI]WO2004073656  (SEATTLE GENETICS INC [US], et al) [X] 1-14 * the whole document * * pages 62-65 * [I] 1-14;
 [XI]WO2005001038  (SEATTLE GENETICS INC [US], et al) [X] 1-4 * the whole document * [I] 1-14;
 [XP]WO2005081711  (SEATTLE GENETICS INC [US], et al) [XP] 1-14 * the whole document *;
 [A]  - G Valle ET AL, "Constrained phenylalanine analogues. Preferred conformation of the 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid (Tic) residue", International journal of peptide and protein research, DENMARK, (19920901), pages 222 - 232, URL: http://www.ncbi.nlm.nih.gov/pubmed/1335996, XP055105311 [A] 1-14 * the whole document *
 [A]  - MIYAZAKI ET AL, "Synthesis and antitumor activity of novel dolastatin 10 analogs", CHEMICAL AND PHARMACEUTICAL BULLETIN, PHARMACEUTICAL SOCIETY OF JAPAN, TOKYO, JP, (19950101), vol. 43, no. 10, ISSN 0009-2363, pages 1706 - 1718, XP002080987 [A] 1-14 * the whole document * * page 1714; table 6; compounds 1,28b *
by applicantEP0012023
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