Extract from the Register of European Patents

EP About this file: EP2838888

EP2838888 - THIADIAZOLIDINEDIONES AS GSK-3 INHIBITORS [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  16.02.2018
Database last updated on 11.04.2026
FormerThe patent has been granted
Status updated on  10.03.2017
FormerGrant of patent is intended
Status updated on  06.11.2016
Most recent event   Tooltip28.09.2018Lapse of the patent in a contracting state
New state(s): MC
published on 31.10.2018  [2018/44]
Applicant(s)For all designated states
ASD Therapeutics Partners LLC
5 Rose Court
Warren, NJ 07059 / US
[2015/09]
Inventor(s)01 / MEDINA PADILLA, Miguel
C/ La Baneza, 42 C, 6° D
E-28035 Madrid / ES
02 / DOMÍNGUEZ CORREA, Juan Manuel
C/ Arturo Soria, 333 - 10 F
E-28033 Madrid / ES
03 / DE CRISTOBAL BLANCO, Javier
C/ Doctor Gómez Ulla, 20 - 4° B
E-28028 Madrid / ES
04 / FUERTES HUERTA, Ana
C/ Alenza, 9 - 5° D
E-28003 Madrid / ES
05 / SÁNCHEZ-QUESADA, Jorge
C/ Vital Aza, 96 - 2° B
E-28017 Madrid / ES
06 / LÓPEZ OGALLA, Javier
C/ Isabel Colbrand 16, Portal H, 2°, 2
E-28050 Madrid / ES
07 / HERRERO SANTOS, Susana
C/ San José, 9 Esc. Izq. - 2° C
E-28921 Alcorcón - Madrid / ES
08 / PÉREZ DE LA CRUZ MORENO, María Ángeles
Ctra. del Plantío, 100 - 2° B
E-28221 Majadahonda - Madrid / ES
09 / MARTÍNEZ MONTERO, Olga
Av. de los Artesanos, 64 - 2, 7° 3
E-28760 Tres Cantos -Madrid / ES
10 / RODRÍGUEZ SALGUERO, Beatriz
Av. Oliva, 67 - 3° B
E-28222 Majadahonda - Madrid / ES
11 / PALOMO NICOLAU, Francisco
C/ Félix Yuste, 22
E-28804 Alcalá de Henares / ES
 [2015/35]
Former [2015/09]01 / MEDINA PADILLA, Miguel
Noscira S.A.
Avda. de la Industria 52
E-28760 Tres Cantos - Madrid / ES
02 / DOMÍNGUEZ CORREA, Juan Manuel
Noscira S.A.
Avda. de la Industria 52
E-28760 Tres Cantos - Madrid / ES
03 / DE CRISTOBAL BLANCO, Javier
Noscira S.A.
Avda. de la Industria 52
E-28760 Tres Cantos - Madrid / ES
04 / FUERTES HUERTA, Ana
Noscira S.A.
Avda. de la Industria 52
E-28760 Tres Cantos - Madrid / ES
05 / SÁNCHEZ-QUESADA, Jorge
Noscira S.A.
Avda. de la Industria 52
E-28760 Tres Cantos - Madrid / ES
06 / LÓPEZ OGALLA, Javier
Noscira S.A.
Avda. de la Industria 52
E-28760 Tres Cantos - Madrid / ES
07 / HERRERO SANTOS, Susana
Noscira S.A.
Avda. de la Industria 52
E-28760 Tres Cantos - Madrid / ES
08 / PÉREZ DE LA CRUZ MORENO, María Ángeles
Noscira S.A.
Avda. de la Industria 52
E-28760 Tres Cantos - Madrid / ES
09 / MARTÍNEZ MONTERO, Olga
Noscira S.A.
Avda. de la Industria 52
E-28760 Tres Cantos -Madrid / ES
10 / RODRÍGUEZ SALGUERO, Beatriz
Noscira S.A.
Avda. de la Industria 52
E-28760 Tres Cantos - Madrid / ES
11 / PALOMO NICOLAU, Francisco
Noscira S.A.
Avda. de la Industria 52
E-28760 Tres Cantos - Madrid / ES
Representative(s)ABG Intellectual Property Law, S.L.
Avenida de Burgos, 16D
Edificio Euromor
28036 Madrid / ES
[N/P]
Former [2015/09]ABG Patentes, S.L.
Avenida de Burgos, 16D
Edificio Euromor
28036 Madrid / ES
Application number, filing date13705492.022.02.2013
[2017/15]
WO2013EP53554
Priority number, dateEP2012038206624.02.2012         Original published format: EP 12382066
[2015/09]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2013124413
Date:29.08.2013
Language:EN
[2013/35]
Type: A1 Application with search report 
No.:EP2838888
Date:25.02.2015
Language:EN
The application published by WIPO in one of the EPO official languages on 29.08.2013 takes the place of the publication of the European patent application.
[2015/09]
Type: B1 Patent specification 
No.:EP2838888
Date:12.04.2017
Language:EN
[2017/15]
Search report(s)International search report - published on:EP29.08.2013
ClassificationIPC:C07D285/08, C07D417/06, A61K31/433, A61P25/28, A61P3/10
[2015/09]
CPC:
C07D285/08 (EP,US); A61P11/00 (EP); A61P19/10 (EP);
A61P25/00 (EP); A61P25/02 (EP); A61P25/28 (EP);
A61P27/06 (EP); A61P29/00 (EP); A61P3/00 (EP);
A61P3/10 (EP); A61P31/12 (EP); A61P37/02 (EP);
A61P43/00 (EP); A61P9/02 (EP); C07D417/06 (EP,US) (-)
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   RS,   SE,   SI,   SK,   SM,   TR [2015/09]
Extension statesBA22.09.2014
ME22.09.2014
TitleGerman:THIADIAZOLIDINDIONE ALS GSK-3-INHIBITOREN[2016/17]
English:THIADIAZOLIDINEDIONES AS GSK-3 INHIBITORS[2015/09]
French:THIADIAZOLIDINEDIONES EN TANT QU'INHIBITEURS DE GSK-3[2016/17]
Former [2015/09]THIADIAZOLIDINDIONE ALS GSK-3-HEMMER
Former [2015/09]THIADIAZOLIDINEDIONES SOUS FORME D'INHIBITEURS DE GSK-3
Entry into regional phase22.09.2014National basic fee paid 
22.09.2014Designation fee(s) paid 
22.09.2014Examination fee paid 
Examination procedure23.12.2013Request for preliminary examination filed
International Preliminary Examining Authority: EP
22.09.2014Amendment by applicant (claims and/or description)
22.09.2014Examination requested  [2015/09]
23.09.2015Despatch of a communication from the examining division (Time limit: M04)
09.12.2015Reply to a communication from the examining division
22.01.2016Despatch of a communication from the examining division (Time limit: M02)
09.03.2016Reply to a communication from the examining division
02.05.2016Despatch of a communication from the examining division (Time limit: M04)
02.09.2016Reply to a communication from the examining division
30.09.2016Despatch of a communication from the examining division (Time limit: M01)
19.10.2016Reply to a communication from the examining division
07.11.2016Communication of intention to grant the patent
06.03.2017Fee for grant paid
06.03.2017Fee for publishing/printing paid
06.03.2017Receipt of the translation of the claim(s)
Divisional application(s)The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is  23.09.2015
Opposition(s)15.01.2018No opposition filed within time limit [2018/12]
Fees paidRenewal fee
22.01.2015Renewal fee patent year 03
18.01.2016Renewal fee patent year 04
16.01.2017Renewal fee patent year 05
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Lapses during opposition  TooltipMC12.04.2017
RS12.04.2017
SM12.04.2017
IS12.08.2017
[2018/44]
Former [2018/13]RS12.04.2017
SM12.04.2017
IS12.08.2017
Former [2017/51]RS12.04.2017
IS12.08.2017
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 [XI]   MARTINEZ A ET AL: "First Non-ATP Competitive Glycogen Synthase Kinase 3.beta. (GSK-3.beta.) Inhibitors: Thiadiazolidinones (TDZD) as Potential Drugs for the Treatment of Alzheimer's Disease", JOURNAL OF MEDICINAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY, US, vol. 45, no. 6, 1 January 2002 (2002-01-01), pages 1292 - 1299, XP002292084, ISSN: 0022-2623, DOI: 10.1021/JM011020U

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 [XI]   EMMA M. TURNER ET AL: "Small Molecule Inhibitors of Regulators of G Protein Signaling (RGS) Proteins", ACS MEDICINAL CHEMISTRY LETTERS, vol. 3, no. 2, 9 February 2012 (2012-02-09), pages 146 - 150, XP055026893, ISSN: 1948-5875, DOI: 10.1021/ml200263y

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