EP2925737 - TRICYCLIC COMPOUNDS FOR USE IN THE TREATMENT AND/OR CONTROL OF OBESITY [Right-click to bookmark this link] | Status | No opposition filed within time limit Status updated on 20.04.2018 Database last updated on 14.06.2024 | |
Former | The patent has been granted Status updated on 12.05.2017 | ||
Former | Grant of patent is intended Status updated on 11.01.2017 | Most recent event Tooltip | 17.07.2020 | Lapse of the patent in a contracting state New state(s): AL | published on 19.08.2020 [2020/34] | Applicant(s) | For all designated states Zafgen, Inc. 175 Portland Street 4th Floor Boston, MA 02114 / US | [2016/07] |
Former [2015/41] | For all designated states Zafgen, Inc. One Broadway, 8th Floor Cambridge, MA 02142 / US | Inventor(s) | 01 /
PALLIN, Thomas, David 8/9 Spire Green Centre Flex Meadow Harlow Essex CM19 5TR / GB | 02 /
CRAMP, Susan, Mary 8/9 Spire Green Centre Flex Meadow Harlow Essex CM19 5TR / GB | 03 /
DYKE, Hazel, Joan 8/9 Spire Green Centre Flex Meadow Harlow Essex CM19 5TR / GB | 04 /
ZAHLER, Robert 5 East Welling Avenue Pennington, NJ 08534 / US | [2015/41] | Representative(s) | Harris, Jennifer Lucy Kilburn & Strode LLP Lacon London 84 Theobalds Road London WC1X 8NL / GB | [N/P] |
Former [2015/41] | Harris, Jennifer Lucy Kilburn & Strode LLP 20 Red Lion Street London WC1R 4PJ / GB | Application number, filing date | 13792204.3 | 05.11.2013 | [2015/41] | WO2013US68492 | Priority number, date | US201261722449P | 05.11.2012 Original published format: US 201261722449 P | [2015/41] | Filing language | EN | Procedural language | EN | Publication | Type: | A1 Application with search report | No.: | WO2014071369 | Date: | 08.05.2014 | Language: | EN | [2014/19] | Type: | A1 Application with search report | No.: | EP2925737 | Date: | 07.10.2015 | Language: | EN | The application published by WIPO in one of the EPO official languages on 08.05.2014 takes the place of the publication of the European patent application. | [2015/41] | Type: | B1 Patent specification | No.: | EP2925737 | Date: | 14.06.2017 | Language: | EN | [2017/24] | Search report(s) | International search report - published on: | EP | 08.05.2014 | Classification | IPC: | C07D405/12, C07D451/02, C07D453/02, C07D487/04, C07D311/94 | [2017/03] | CPC: |
C07D311/94 (EP,CN,US);
A61P3/04 (EP);
A61P43/00 (EP);
A61P9/00 (EP);
C07D405/12 (EP,CN,US);
C07D451/02 (EP,US);
|
Former IPC [2015/41] | C07D311/94, A61K31/353, A61P3/04 | Designated contracting states | AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR [2015/41] | Extension states | BA | 05.06.2015 | ME | 05.06.2015 | Title | German: | TRICYCLISCHE VERBINDUNGEN ZUR VERWENDUNG BEI DER BEHANDLUNG UND/ODER KONTROLLE VON ADIPOSITAS | [2015/41] | English: | TRICYCLIC COMPOUNDS FOR USE IN THE TREATMENT AND/OR CONTROL OF OBESITY | [2015/41] | French: | COMPOSÉS TRICYCLIQUES À UTILISER DANS LE TRAITEMENT ET/OU LA LUTTE CONTRE L'OBÉSITÉ | [2015/41] | Entry into regional phase | 05.06.2015 | National basic fee paid | 05.06.2015 | Designation fee(s) paid | 05.06.2015 | Examination fee paid | Examination procedure | 05.06.2015 | Examination requested [2015/41] | 18.02.2016 | Amendment by applicant (claims and/or description) | 20.04.2016 | Despatch of a communication from the examining division (Time limit: M06) | 25.10.2016 | Reply to a communication from the examining division | 12.01.2017 | Communication of intention to grant the patent | 08.05.2017 | Fee for grant paid | 08.05.2017 | Fee for publishing/printing paid | 08.05.2017 | Receipt of the translation of the claim(s) | Divisional application(s) | The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is 20.04.2016 | Opposition(s) | 15.03.2018 | No opposition filed within time limit [2018/21] | Fees paid | Renewal fee | 30.11.2015 | Renewal fee patent year 03 | 28.11.2016 | Renewal fee patent year 04 |
Opt-out from the exclusive Tooltip competence of the Unified Patent Court | See the Register of the Unified Patent Court for opt-out data | ||
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Lapses during opposition Tooltip | HU | 05.11.2013 | AL | 14.06.2017 | AT | 14.06.2017 | CY | 14.06.2017 | CZ | 14.06.2017 | DK | 14.06.2017 | EE | 14.06.2017 | ES | 14.06.2017 | FI | 14.06.2017 | HR | 14.06.2017 | IT | 14.06.2017 | LT | 14.06.2017 | LV | 14.06.2017 | MC | 14.06.2017 | MK | 14.06.2017 | NL | 14.06.2017 | PL | 14.06.2017 | PT | 14.06.2017 | RO | 14.06.2017 | RS | 14.06.2017 | SE | 14.06.2017 | SI | 14.06.2017 | SK | 14.06.2017 | SM | 14.06.2017 | TR | 14.06.2017 | BG | 14.09.2017 | NO | 14.09.2017 | GR | 15.09.2017 | IS | 14.10.2017 | LU | 05.11.2017 | MT | 05.11.2017 | BE | 30.11.2017 | [2020/34] |
Former [2020/28] | HU | 05.11.2013 | |
AT | 14.06.2017 | ||
CY | 14.06.2017 | ||
CZ | 14.06.2017 | ||
DK | 14.06.2017 | ||
EE | 14.06.2017 | ||
ES | 14.06.2017 | ||
FI | 14.06.2017 | ||
HR | 14.06.2017 | ||
IT | 14.06.2017 | ||
LT | 14.06.2017 | ||
LV | 14.06.2017 | ||
MC | 14.06.2017 | ||
MK | 14.06.2017 | ||
NL | 14.06.2017 | ||
PL | 14.06.2017 | ||
PT | 14.06.2017 | ||
RO | 14.06.2017 | ||
RS | 14.06.2017 | ||
SE | 14.06.2017 | ||
SI | 14.06.2017 | ||
SK | 14.06.2017 | ||
SM | 14.06.2017 | ||
TR | 14.06.2017 | ||
BG | 14.09.2017 | ||
NO | 14.09.2017 | ||
GR | 15.09.2017 | ||
IS | 14.10.2017 | ||
LU | 05.11.2017 | ||
MT | 05.11.2017 | ||
BE | 30.11.2017 | ||
Former [2020/15] | HU | 05.11.2013 | |
AT | 14.06.2017 | ||
CY | 14.06.2017 | ||
CZ | 14.06.2017 | ||
DK | 14.06.2017 | ||
EE | 14.06.2017 | ||
ES | 14.06.2017 | ||
FI | 14.06.2017 | ||
HR | 14.06.2017 | ||
IT | 14.06.2017 | ||
LT | 14.06.2017 | ||
LV | 14.06.2017 | ||
MC | 14.06.2017 | ||
MK | 14.06.2017 | ||
NL | 14.06.2017 | ||
PL | 14.06.2017 | ||
RO | 14.06.2017 | ||
RS | 14.06.2017 | ||
SE | 14.06.2017 | ||
SI | 14.06.2017 | ||
SK | 14.06.2017 | ||
SM | 14.06.2017 | ||
TR | 14.06.2017 | ||
BG | 14.09.2017 | ||
NO | 14.09.2017 | ||
GR | 15.09.2017 | ||
IS | 14.10.2017 | ||
LU | 05.11.2017 | ||
MT | 05.11.2017 | ||
BE | 30.11.2017 | ||
Former [2019/51] | HU | 05.11.2013 | |
AT | 14.06.2017 | ||
CY | 14.06.2017 | ||
CZ | 14.06.2017 | ||
DK | 14.06.2017 | ||
EE | 14.06.2017 | ||
ES | 14.06.2017 | ||
FI | 14.06.2017 | ||
HR | 14.06.2017 | ||
IT | 14.06.2017 | ||
LT | 14.06.2017 | ||
LV | 14.06.2017 | ||
MC | 14.06.2017 | ||
MK | 14.06.2017 | ||
NL | 14.06.2017 | ||
PL | 14.06.2017 | ||
RO | 14.06.2017 | ||
RS | 14.06.2017 | ||
SE | 14.06.2017 | ||
SI | 14.06.2017 | ||
SK | 14.06.2017 | ||
SM | 14.06.2017 | ||
BG | 14.09.2017 | ||
NO | 14.09.2017 | ||
GR | 15.09.2017 | ||
IS | 14.10.2017 | ||
LU | 05.11.2017 | ||
MT | 05.11.2017 | ||
BE | 30.11.2017 | ||
Former [2019/47] | HU | 05.11.2013 | |
AT | 14.06.2017 | ||
CY | 14.06.2017 | ||
CZ | 14.06.2017 | ||
DK | 14.06.2017 | ||
EE | 14.06.2017 | ||
ES | 14.06.2017 | ||
FI | 14.06.2017 | ||
HR | 14.06.2017 | ||
IT | 14.06.2017 | ||
LT | 14.06.2017 | ||
LV | 14.06.2017 | ||
MC | 14.06.2017 | ||
NL | 14.06.2017 | ||
PL | 14.06.2017 | ||
RO | 14.06.2017 | ||
RS | 14.06.2017 | ||
SE | 14.06.2017 | ||
SI | 14.06.2017 | ||
SK | 14.06.2017 | ||
SM | 14.06.2017 | ||
BG | 14.09.2017 | ||
NO | 14.09.2017 | ||
GR | 15.09.2017 | ||
IS | 14.10.2017 | ||
LU | 05.11.2017 | ||
MT | 05.11.2017 | ||
BE | 30.11.2017 | ||
Former [2019/31] | HU | 05.11.2013 | |
AT | 14.06.2017 | ||
CZ | 14.06.2017 | ||
DK | 14.06.2017 | ||
EE | 14.06.2017 | ||
ES | 14.06.2017 | ||
FI | 14.06.2017 | ||
HR | 14.06.2017 | ||
IT | 14.06.2017 | ||
LT | 14.06.2017 | ||
LV | 14.06.2017 | ||
MC | 14.06.2017 | ||
NL | 14.06.2017 | ||
PL | 14.06.2017 | ||
RO | 14.06.2017 | ||
RS | 14.06.2017 | ||
SE | 14.06.2017 | ||
SI | 14.06.2017 | ||
SK | 14.06.2017 | ||
SM | 14.06.2017 | ||
BG | 14.09.2017 | ||
NO | 14.09.2017 | ||
GR | 15.09.2017 | ||
IS | 14.10.2017 | ||
LU | 05.11.2017 | ||
MT | 05.11.2017 | ||
BE | 30.11.2017 | ||
Former [2018/50] | AT | 14.06.2017 | |
CZ | 14.06.2017 | ||
DK | 14.06.2017 | ||
EE | 14.06.2017 | ||
ES | 14.06.2017 | ||
FI | 14.06.2017 | ||
HR | 14.06.2017 | ||
IT | 14.06.2017 | ||
LT | 14.06.2017 | ||
LV | 14.06.2017 | ||
MC | 14.06.2017 | ||
NL | 14.06.2017 | ||
PL | 14.06.2017 | ||
RO | 14.06.2017 | ||
RS | 14.06.2017 | ||
SE | 14.06.2017 | ||
SI | 14.06.2017 | ||
SK | 14.06.2017 | ||
SM | 14.06.2017 | ||
BG | 14.09.2017 | ||
NO | 14.09.2017 | ||
GR | 15.09.2017 | ||
IS | 14.10.2017 | ||
LU | 05.11.2017 | ||
MT | 05.11.2017 | ||
BE | 30.11.2017 | ||
Former [2018/43] | AT | 14.06.2017 | |
CZ | 14.06.2017 | ||
DK | 14.06.2017 | ||
EE | 14.06.2017 | ||
ES | 14.06.2017 | ||
FI | 14.06.2017 | ||
HR | 14.06.2017 | ||
IT | 14.06.2017 | ||
LT | 14.06.2017 | ||
LV | 14.06.2017 | ||
MC | 14.06.2017 | ||
NL | 14.06.2017 | ||
PL | 14.06.2017 | ||
RO | 14.06.2017 | ||
RS | 14.06.2017 | ||
SE | 14.06.2017 | ||
SI | 14.06.2017 | ||
SK | 14.06.2017 | ||
SM | 14.06.2017 | ||
BG | 14.09.2017 | ||
NO | 14.09.2017 | ||
GR | 15.09.2017 | ||
IS | 14.10.2017 | ||
LU | 05.11.2017 | ||
MT | 05.11.2017 | ||
Former [2018/40] | AT | 14.06.2017 | |
CZ | 14.06.2017 | ||
DK | 14.06.2017 | ||
EE | 14.06.2017 | ||
ES | 14.06.2017 | ||
FI | 14.06.2017 | ||
HR | 14.06.2017 | ||
IT | 14.06.2017 | ||
LT | 14.06.2017 | ||
LV | 14.06.2017 | ||
MC | 14.06.2017 | ||
NL | 14.06.2017 | ||
PL | 14.06.2017 | ||
RO | 14.06.2017 | ||
RS | 14.06.2017 | ||
SE | 14.06.2017 | ||
SI | 14.06.2017 | ||
SK | 14.06.2017 | ||
SM | 14.06.2017 | ||
BG | 14.09.2017 | ||
NO | 14.09.2017 | ||
GR | 15.09.2017 | ||
IS | 14.10.2017 | ||
LU | 05.11.2017 | ||
Former [2018/33] | AT | 14.06.2017 | |
CZ | 14.06.2017 | ||
DK | 14.06.2017 | ||
EE | 14.06.2017 | ||
ES | 14.06.2017 | ||
FI | 14.06.2017 | ||
HR | 14.06.2017 | ||
IT | 14.06.2017 | ||
LT | 14.06.2017 | ||
LV | 14.06.2017 | ||
MC | 14.06.2017 | ||
NL | 14.06.2017 | ||
PL | 14.06.2017 | ||
RO | 14.06.2017 | ||
RS | 14.06.2017 | ||
SE | 14.06.2017 | ||
SK | 14.06.2017 | ||
SM | 14.06.2017 | ||
BG | 14.09.2017 | ||
NO | 14.09.2017 | ||
GR | 15.09.2017 | ||
IS | 14.10.2017 | ||
Former [2018/21] | AT | 14.06.2017 | |
CZ | 14.06.2017 | ||
DK | 14.06.2017 | ||
EE | 14.06.2017 | ||
ES | 14.06.2017 | ||
FI | 14.06.2017 | ||
HR | 14.06.2017 | ||
IT | 14.06.2017 | ||
LT | 14.06.2017 | ||
LV | 14.06.2017 | ||
NL | 14.06.2017 | ||
PL | 14.06.2017 | ||
RO | 14.06.2017 | ||
RS | 14.06.2017 | ||
SE | 14.06.2017 | ||
SK | 14.06.2017 | ||
SM | 14.06.2017 | ||
BG | 14.09.2017 | ||
NO | 14.09.2017 | ||
GR | 15.09.2017 | ||
IS | 14.10.2017 | ||
Former [2018/11] | AT | 14.06.2017 | |
CZ | 14.06.2017 | ||
EE | 14.06.2017 | ||
ES | 14.06.2017 | ||
FI | 14.06.2017 | ||
HR | 14.06.2017 | ||
IT | 14.06.2017 | ||
LT | 14.06.2017 | ||
LV | 14.06.2017 | ||
NL | 14.06.2017 | ||
PL | 14.06.2017 | ||
RO | 14.06.2017 | ||
RS | 14.06.2017 | ||
SE | 14.06.2017 | ||
SK | 14.06.2017 | ||
SM | 14.06.2017 | ||
BG | 14.09.2017 | ||
NO | 14.09.2017 | ||
GR | 15.09.2017 | ||
IS | 14.10.2017 | ||
Former [2018/10] | AT | 14.06.2017 | |
CZ | 14.06.2017 | ||
EE | 14.06.2017 | ||
FI | 14.06.2017 | ||
HR | 14.06.2017 | ||
LT | 14.06.2017 | ||
LV | 14.06.2017 | ||
NL | 14.06.2017 | ||
RO | 14.06.2017 | ||
RS | 14.06.2017 | ||
SE | 14.06.2017 | ||
SK | 14.06.2017 | ||
BG | 14.09.2017 | ||
NO | 14.09.2017 | ||
GR | 15.09.2017 | ||
Former [2018/09] | EE | 14.06.2017 | |
FI | 14.06.2017 | ||
HR | 14.06.2017 | ||
LT | 14.06.2017 | ||
LV | 14.06.2017 | ||
NL | 14.06.2017 | ||
RS | 14.06.2017 | ||
SE | 14.06.2017 | ||
BG | 14.09.2017 | ||
NO | 14.09.2017 | ||
GR | 15.09.2017 | ||
Former [2017/52] | FI | 14.06.2017 | |
HR | 14.06.2017 | ||
LT | 14.06.2017 | ||
LV | 14.06.2017 | ||
NL | 14.06.2017 | ||
RS | 14.06.2017 | ||
SE | 14.06.2017 | ||
BG | 14.09.2017 | ||
NO | 14.09.2017 | ||
GR | 15.09.2017 | ||
Former [2017/50] | FI | 14.06.2017 | |
HR | 14.06.2017 | ||
LT | 14.06.2017 | ||
LV | 14.06.2017 | ||
RS | 14.06.2017 | ||
SE | 14.06.2017 | ||
BG | 14.09.2017 | ||
NO | 14.09.2017 | ||
GR | 15.09.2017 | ||
Former [2017/49] | FI | 14.06.2017 | |
HR | 14.06.2017 | ||
LT | 14.06.2017 | ||
NO | 14.09.2017 | ||
GR | 15.09.2017 | Cited in | International search | [A]WO2012012642 (ZAFGEN CORP [US], et al) [A] 1-13 * example 20; claims 1, 18-30 *; | [XP]WO2012154676 (ZAFGEN CORP [US], et al) [XP] 1-13 * claims 1, 32-41 * | by applicant | US2004167128 | - O'BRIEN ET AL., AMER J SURGERY, (2002), vol. 184, pages 4S - 8S | - HILL ET AL., SCIENCE, (1998), vol. 280, page 1371 | - WARDER ET AL., J PROTEOME RES, (2008), vol. 7, page 4807 | - WANG ET AL., CANCER RES., (2003), vol. 63, page 7861 | - ZHANG ET AL., J. BIOMED. SCI., (2002), vol. 9, page 34 | - RUPNICK ET AL., PROC. NATL. ACAD. SCI. USA, (2002), vol. 99, page 10730 | - RAUTIO, KUMPULAINEN ET AL., NATURE REVIEWS DRUG DISCOVERY, (2008), vol. 7, page 255 | - SIMPLICIO ET AL., MOLECULES, (2008), vol. 13, page 519 | - MIYAURA, SUZUKI, CHEM. REV., (1995), vol. 95, page 2457 | - SUZUKI, MODEM ARENE CHEMISTRY, (2002), pages 53 - 106 | - SMITH, MARCH, March's Advanced Organic Chemistry, WILEY, (2001), pages 931 - 932 | - DE SOUZA, CURRENT ORGANIC SYNTHESIS, (2006), vol. 3, no. 3, pages 313 - 326 | - MARSHALL, CHEMTRACTS, (2000), vol. 13, no. 4, pages 219 - 222 | - ASTRUP, A, PUB HEALTH NUTR, (2001), vol. 4, pages 499 - 515 | - CARR ET AL., THE JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM, (2004), vol. 89, no. 6, pages 2601 - 2607 | - ECKEL, CIRCULATION, (1997), vol. 96, pages 3248 - 3250 | - WONG ET AL., NATURE CLINICAL PRACTICE CARDIOVASCULAR MEDICINE, (2007), vol. 4, pages 436 - 443 | - YUSEF ET AL., LANCET, (2005), vol. 366, no. 9497, pages 1640 - 1649 | - SUK ET AL., STROKE, (2003), vol. 34, pages 1586 - 1592 | - STEIN ET AL., THE AMERICAN JOURNAL OF MEDICINE, (2005), vol. 18, no. 9, pages 978 - 980 | - SZTRYMF ET AL., REV PNEUMOL CLIN, (2002), vol. 58, no. 2, pages 104 - 10 | - ELAMIN, CHEST, (2004), vol. 125, pages 1972 - 1974 | - KESSLER ET AL., EUR RESPIR J, (1996), vol. 9, pages 787 - 794 | - TOLMAN ET AL., THER CLIN RISK MANAG, (2007), vol. 6, pages 1153 - 1163 | - VAN SAASE, J RHEUMATOL, (1988), vol. 15, no. 7, pages 1152 - 1158 | - PRADER-WILLI SYNDROME, "polycystic ovary syndrome, have been linked to being overweight or obese. Cassidy", JOURNAL OF MEDICAL GENETICS, (1997), vol. 34, pages 917 - 923 | - HOEGER, OBSTETRICS AND GYNECOLOGY CLINICS OF NORTH AMERICA, (2001), vol. 28, no. 1, pages 85 - 97 | - LARSEN ET AL., INT J OBES (LOND, (2007), vol. 8, pages 1189 - 1198 | - CHUNG ET AL., EUR UROL, (1999), vol. 36, no. 1, pages 68 - 70 | - PASQUALI ET AL., HUM REPROD, (1997), vol. 1, pages 82 - 87 | - WEISS ET AL., AMERICAN JOURNAL OF OBSTETRICS AND GYNECOLOGY, (2004), vol. 190, no. 4, pages 1091 - 1097 | - DIXSON ET AL., ARCH INTERN MED, (2003), vol. 163, pages 2058 - 2065 | - SIMON ET AL., ARCHIVES OF GENERAL PSYCHIATRY, (2006), vol. 63, no. 7, pages 824 - 830 |