EP3013814 - SUBSTITUTED TETRAHYDROCARBAZOLE AND CARBAZOLE CARBOXAMIDE COMPOUNDS USEFUL AS KINASE INHIBITORS [Right-click to bookmark this link] | Status | No opposition filed within time limit Status updated on 20.04.2018 Database last updated on 17.05.2024 | |
Former | The patent has been granted Status updated on 12.05.2017 | ||
Former | Grant of patent is intended Status updated on 10.05.2017 | ||
Former | Request for examination was made Status updated on 05.04.2017 | ||
Former | Grant of patent is intended Status updated on 21.11.2016 | Most recent event Tooltip | 20.04.2018 | No opposition filed within time limit | published on 23.05.2018 [2018/21] | Applicant(s) | For all designated states Bristol-Myers Squibb Company Route 206 and Province Line Road Princeton, NJ 08543 / US | [2016/18] | Inventor(s) | 01 /
TINO, Joseph A. c/o Bristol-Myers Squibb Company Route 206 & Province Line Road Princeton, New Jersey 08543 / US | 02 /
SRIVASTAVA, Anurag S. c/o Bristol-Myers Squibb Company Route 206 & Province Line Road Princeton, New Jersey 08543 / US | 03 /
KO, Soo Sung 7 Aston Circle Hockessin, Delaware 19707 / US | 04 /
GALELLA, Michael A. c/o Bristol-Myers Squibb Company Route 206 & Province Line Road Princeton, New Jersey 08543 / US | 05 /
LANGEVINE, Charles M. 580 Flatbush Avenue, 1M Brooklyn, New York 11225 / US | 06 /
DELUCCA, George V. c/o Bristol-Myers Squibb Company Route 206 & Province Line Road Princeton, New Jersey 08543 / US | 07 /
LIU, Qingjie c/o Bristol-Myers Squibb Company Route 206 & Province Line Road Princeton, New Jersey 08543 / US | 08 /
BATT, Douglas G. c/o Bristol-Myers Squibb Company Route 206 & Province Line Road Princeton, New Jersey 08543 / US | 09 /
WATTERSON, Scott Hunter c/o Bristol-Myers Squibb Company Route 206 & Province Line Road Princeton, New Jersey 08543 / US | 10 /
SHI, Qing c/o Bristol-Myers Squibb Company Route 206 & Province Line Road Princeton, New Jersey 08543 / US | 11 /
BERTRAND, Myra Beaudoin c/o Bristol-Myers Squibb Company Route 206 & Province Line Road Princeton, New Jersey 08543 / US | [2017/24] |
Former [2016/18] | 01 /
TINO, Joseph A. c/o Bristol-Myers Squibb Company Route 206 & Province Line Road Princeton, New Jersey 08543 / US | ||
02 /
SRIVASTAVA, Anurag S. c/o Bristol-Myers Squibb Company Route 206 & Province Line Road Princeton, New Jersey 08543 / US | |||
03 /
KO, Soo Sung 7 Aston Circle Hockessin, Delaware 19707 / US | |||
04 /
GALELLA, Michael A. c/o Bristol-Myers Squibb Company Route 206 & Province Line Road Princeton, New Jersey 08543 / US | |||
05 /
LANGEVINE, Charles M. 580 Flatbush Avenue, 1M Brooklyn, New York 11225 / US | |||
06 /
DELUCCA, George V. c/o Bristol-Myers Squibb Company Route 206 & Province Line Road Princeton, New Jersey 08543 / US | |||
07 /
LIU, Qingjie c/o Bristol-Myers Squibb Company Route 206 & Province Line Road Princeton, New Jersey 08543 / US | |||
08 /
BATT, Douglas G. c/o Bristol-Myers Squibb Company Route 206 & Province Line Road Princeton, New Jersey 08543 / US | |||
09 /
WATTERSON, Scott Hunter c/o Bristol-Myers Squibb Company Route 206&Province Line Road Princeton New Jersey 08543 / US | |||
10 /
SHI, Qing c/o Bristol-Myers Squibb Company Route 206 & Province Line Road Princeton, New Jersey 08543 / US | |||
11 /
BERTRAND, Myra Beaudoin c/o Bristol-Myers Squibb Company Route 206 & Province Line Road Princeton, New Jersey 08543 / US | Representative(s) | Beacham, Annabel Rose Dehns St Bride's House 10 Salisbury Square London EC4Y 8JD / GB | [2016/18] | Application number, filing date | 14740094.9 | 25.06.2014 | [2016/18] | WO2014US43978 | Priority number, date | US201361839141P | 25.06.2013 Original published format: US 201361839141 P | [2016/18] | Filing language | EN | Procedural language | EN | Publication | Type: | A1 Application with search report | No.: | WO2014210085 | Date: | 31.12.2014 | Language: | EN | [2014/53] | Type: | A1 Application with search report | No.: | EP3013814 | Date: | 04.05.2016 | Language: | EN | The application published by WIPO in one of the EPO official languages on 31.12.2014 takes the place of the publication of the European patent application. | [2016/18] | Type: | B1 Patent specification | No.: | EP3013814 | Date: | 14.06.2017 | Language: | EN | [2017/24] | Search report(s) | International search report - published on: | EP | 31.12.2014 | Classification | IPC: | C07D403/10, C07D471/04, C07D513/04, A61K31/429, A61K31/513, A61K31/517, A61K31/522, A61P37/00, A61P29/00 | [2016/18] | CPC: |
C07D513/04 (EP,US);
A61K31/517 (US);
A61P19/02 (EP);
A61P25/28 (EP);
A61P29/00 (EP);
A61P35/00 (EP);
A61P37/00 (EP);
A61P37/02 (EP);
A61P37/06 (EP);
A61P43/00 (EP);
C07D209/88 (EP,US);
C07D239/70 (EP,US);
C07D403/10 (EP,US);
C07D471/04 (EP,US);
C07B2200/07 (EP,US);
C07B2200/13 (EP,US)
(-)
| C-Set: |
C07D209/88, C07B2200/07 (US);
C07D209/88, C07B2200/13 (US);
C07D239/70, C07B2200/07 (US);
C07D239/70, C07B2200/13 (US) | Designated contracting states | AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR [2016/18] | Extension states | BA | Not yet paid | ME | Not yet paid | Title | German: | ALS KINASEHEMMER GEEIGNETE SUBSTITUIERTE TETRAHYDROCARBAZOL- UND CARBAZOL-CARBOXAMID-VERBINDUNGEN | [2016/18] | English: | SUBSTITUTED TETRAHYDROCARBAZOLE AND CARBAZOLE CARBOXAMIDE COMPOUNDS USEFUL AS KINASE INHIBITORS | [2016/18] | French: | COMPOSÉS CARBOXAMIDE DE CARBAZOLE ET DE TÉTRAHYDROCARBAZOLE SUBSTITUÉS CONVENANT COMME INHIBITEURS DE KINASES | [2016/18] | Entry into regional phase | 20.01.2016 | National basic fee paid | 20.01.2016 | Designation fee(s) paid | 20.01.2016 | Examination fee paid | Examination procedure | 20.01.2016 | Examination requested [2016/18] | 18.08.2016 | Amendment by applicant (claims and/or description) | 22.11.2016 | Communication of intention to grant the patent | 31.03.2017 | Disapproval of the communication of intention to grant the patent by the applicant or resumption of examination proceedings by the EPO | 31.03.2017 | Fee for grant paid | 31.03.2017 | Fee for publishing/printing paid | 09.05.2017 | Information about intention to grant a patent | 09.05.2017 | Receipt of the translation of the claim(s) | Opposition(s) | 15.03.2018 | No opposition filed within time limit [2018/21] | Fees paid | Renewal fee | 10.06.2016 | Renewal fee patent year 03 |
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Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Cited in | International search | [A]WO2011159857 (BRISTOL MYERS SQUIBB CO [US], et al) [A] 1-13 * example - *; | [A]US8084620 (LIU QINGJIE [US], et al) [A] 1-13 * example - *; | [A] - YAN LOU ET AL, "Bruton's Tyrosine Kinase Inhibitors: Approaches to Potent and Selective Inhibition, Preclinical and Clinical Evaluation for Inflammatory Diseases and B Cell Malignancies", JOURNAL OF MEDICINAL CHEMISTRY, (20120524), vol. 55, no. 10, doi:10.1021/jm300035p, ISSN 0022-2623, pages 4539 - 4550, XP055080230 [A] 1-13 * example - * DOI: http://dx.doi.org/10.1021/jm300035p | by applicant | US4200750 | WO2011159857 | US8084620 | US8242260 | - LAPLANTE ET AL., J. MED. CHEM., (2011), vol. 54, pages 7005 - 7022 | - WHITE ET AL., J. CHROMATOGRAPHY A, (2005), vol. 1074, pages 175 - 185 | - "Design and Application of Prodrugs", BUNDGAARD, H. ET AL., A Textbook of Drug Design and Development, HARWOOD ACADEMIC PUBLISHERS, (1991), pages 113 - 191 | - CHOU ET AL., ADV. ENZYME REGUL., (1984), vol. 22, pages 27 - 55 | - HERAVI, M.M. ET AL., TETRAHEDRON, (2012), vol. 68, page 9145 | - ISHIYAMA, T. ET AL., TETRAHEDRON, (2001), vol. 57, page 9813 | - CAO, J. ET AL., SYNTHETIC COMMUN., (2009), vol. 39, page 205 | - WU, F. ET AL., J. ORG. CHEM., (2004), vol. 69, page 9307 | - JACOBSEN, M.F. ET AL., J. ORG. CHEM., (2006), vol. 71, page 9183 | - HIRSCH, J. ET AL., J. ORG. CHEM., (1986), vol. 51, page 2218 | - KAMATA, J. ET AL., CHEM. PHARM. BULL., (2004), vol. 52, page 1071 | - STILL, W.C. ET AL., J. ORG. CHEM., (1978), vol. 43, page 2923 | - COSIER, J. ET AL., J. APPL. CRYST., (1986), vol. 19, page 105 | - PARDANANI, A, LEUKEMIA, (2012), vol. 26, pages 1449 - 1451 | - UETRECHT, CHEM. RES. TOXICOL., (1999), vol. 12, pages 387 - 395 | - NAKAYAMA, DRUG METABOLISM AND DISPOSITION, (2009), vol. 37, no. 9, pages 1970 - 1977 |