| EP3215142 - IMMUNOREGULATORY AGENTS [Right-click to bookmark this link] | Status | No opposition filed within time limit Status updated on 04.02.2022 Database last updated on 11.04.2026 | |
| Former | The patent has been granted Status updated on 19.02.2021 | ||
| Former | Grant of patent is intended Status updated on 28.10.2020 | ||
| Former | Examination is in progress Status updated on 07.09.2019 | ||
| Former | Request for examination was made Status updated on 11.08.2017 | ||
| Former | The international publication has been made Status updated on 28.04.2017 | Most recent event Tooltip | 19.12.2025 | Lapse of the patent in a contracting state New state(s): TR | published on 21.01.2026 [2026/04] | Applicant(s) | For all designated states Flexus Biosciences, Inc. Route 206 and Province Line Road Princeton, New Jersey 08540 / US | [2021/12] |
| Former [2017/37] | For all designated states Flexus Biosciences, Inc. Route 206 and Province Line Road Princeton, New Jersey 08540 / US | Inventor(s) | 01 /
BECK, Hilary Plake 115 Springdale Way Emerald Hills, California 94062 / US | 02 /
JAEN, Juan Carlos 154 Los Robles Drive Burlingame, California 94010 / US | 03 /
OSIPOV, Maksim 200 Irene Court Apt. 35 Belmont, California 94002 / US | 04 /
POWERS, Jay Patrick 745 Rockaway Beach Avenue Pacifica, California 94044 / US | 05 /
REILLY, Maureen Kay 2151 Carlmont Drive Apt. 301 Belmont, California 94002 / US | 06 /
SHUNATONA, Hunter Paul 79 Melrose Avenue San Francisco, California 94131 / US | 07 /
WALKER, James Ross 123 Newbridge Street Menlo Park, California 94025 / US | 08 /
ZIBINSKY, Mikhail 324 Ravenwood Way Lodi, California 95240 / US | 09 /
BALOG, James Aaron c/o Flexus Biosciences Inc. Route 206 and Province Line Road Princeton, New Jersey 08540 / US | 10 /
WILLIAMS, David K. c/o Flexus Biosciences Inc. Route 206 and Province Line Road Princeton, New Jersey 08540 / US | 11 /
MARKWALDER, Jay A. c/o Flexus Biosciences Inc. Route 206 and Province Line Road Princeton, New Jersey 08540 / US | 12 /
SEITZ, Steven P. c/o Flexus Biosciences Inc. Route 206 and Province Line Road Princeton, New Jersey 08540 / US | 13 /
CHERNEY, Emily Charlotte c/o Flexus Biosciences Inc. Route 206 and Province Line Road Princeton, New Jersey 08540 / US | 14 /
ZHANG, Liping c/o Flexus Biosciences Inc. Route 206 and Province Line Road Princeton, New Jersey 08540 / US | 15 /
SHAN, Weifang c/o Flexus Biosciences Inc. Route 206 and Province Line Road Princeton, New Jersey 08540 / US | 16 /
GUO, Weiwei c/o Flexus Biosciences Inc. Route 206 and Province Line Road Princeton, New Jersey 08540 / US | 17 /
HUANG, Audris c/o Flexus Biosciences Inc. Route 206 and Province Line Road Princeton, New Jersey 08540 / US | [2017/37] | Representative(s) | Mewburn Ellis LLP Aurora Building Counterslip Bristol BS1 6BX / GB | [2021/12] |
| Former [2017/37] | Reitstötter Kinzebach Patentanwälte Sternwartstrasse 4 81679 München / DE | Application number, filing date | 15857810.4 | 05.11.2015 | [2017/37] | WO2015US59316 | Priority number, date | US201462075678P | 05.11.2014 Original published format: US 201462075678 P | [2017/37] | Filing language | EN | Procedural language | EN | Publication | Type: | A2 Application without search report | No.: | WO2016073774 | Date: | 12.05.2016 | Language: | EN | [2016/19] | Type: | A2 Application without search report | No.: | EP3215142 | Date: | 13.09.2017 | Language: | EN | The application published by WIPO in one of the EPO official languages on 12.05.2016 takes the place of the publication of the European patent application. | [2017/37] | Type: | B1 Patent specification | No.: | EP3215142 | Date: | 24.03.2021 | Language: | EN | [2021/12] | Search report(s) | International search report - published on: | US | 07.07.2016 | (Supplementary) European search report - dispatched on: | EP | 07.08.2018 | Classification | IPC: | A61K45/06, A61K31/136, A61K31/166, A61K31/277, A61K31/4412, A61K31/445, A61K31/47, A61K31/4709, A61K31/496, A61K31/497, A61K31/506, A61K31/519, A61K31/5377, A61K31/381, A61P35/00 | [2020/47] | CPC: |
A61K31/166 (EP,KR,US);
C07C255/60 (KR);
A61K31/00 (US);
A61K31/136 (EP,US);
A61K31/277 (EP,US);
A61K31/381 (EP,US);
A61K31/4412 (EP,US);
A61K31/445 (EP,KR,US);
A61K31/47 (EP,KR,US);
A61K31/4709 (EP,US);
A61K31/496 (EP,US);
A61K31/497 (EP,US);
A61K31/506 (EP,US);
A61K31/519 (EP,US);
A61K31/5377 (EP,US);
A61K45/06 (EP,US);
A61P35/00 (EP,US);
C07C211/45 (US);
C07C217/80 (EP,US);
C07C233/10 (EP,US);
C07C233/59 (EP,US);
C07C233/60 (EP,US);
C07C233/65 (US);
C07C233/74 (EP,US);
C07C255/50 (US);
C07C255/58 (EP,US);
C07C275/30 (EP,US);
C07D211/08 (EP,US);
C07D211/16 (EP);
C07D211/46 (EP);
C07D213/40 (EP);
C07D213/68 (EP,US);
C07D213/81 (EP);
C07D215/04 (EP,US);
C07D215/12 (EP);
C07D215/233 (EP,US);
C07D401/04 (EP);
C07D401/12 (EP);
C07D413/06 (EP);
C07D417/12 (EP);
C07D487/04 (EP,US);
A61K2300/00 (US);
| C-Set: |
A61K31/136, A61K2300/00 (US,EP);
A61K31/166, A61K2300/00 (US,EP);
A61K31/277, A61K2300/00 (US,EP);
A61K31/381, A61K2300/00 (US,EP);
A61K31/4412, A61K2300/00 (US,EP);
A61K31/445, A61K2300/00 (US,EP);
A61K31/4709, A61K2300/00 (US,EP);
A61K31/47, A61K2300/00 (US,EP);
A61K31/496, A61K2300/00 (US,EP);
A61K31/497, A61K2300/00 (EP,US);
A61K31/506, A61K2300/00 (EP,US);
A61K31/519, A61K2300/00 (EP,US); |
| Former IPC [2017/37] | A61K31/16, C07C13/02, C07C13/16 | Designated contracting states | AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR [2017/37] | Extension states | BA | 27.04.2017 | ME | 27.04.2017 | Validation states | MA | Not yet paid | MD | Not yet paid | Title | German: | IMMUNREGULATORISCHE WIRKSTOFFE | [2017/37] | English: | IMMUNOREGULATORY AGENTS | [2017/37] | French: | AGENTS IMMUNORÉGULATEURS | [2017/37] | Entry into regional phase | 27.04.2017 | National basic fee paid | 27.04.2017 | Search fee paid | 27.04.2017 | Designation fee(s) paid | 27.04.2017 | Examination fee paid | Examination procedure | 27.04.2017 | Examination requested [2017/37] | 27.04.2017 | Date on which the examining division has become responsible | 04.03.2019 | Amendment by applicant (claims and/or description) | 11.09.2019 | Despatch of a communication from the examining division (Time limit: M04) | 21.01.2020 | Reply to a communication from the examining division | 16.04.2020 | Despatch of a communication from the examining division (Time limit: M02) | 01.06.2020 | Reply to a communication from the examining division | 29.10.2020 | Communication of intention to grant the patent | 02.02.2021 | Fee for grant paid | 02.02.2021 | Fee for publishing/printing paid | 02.02.2021 | Receipt of the translation of the claim(s) | Opposition(s) | 04.01.2022 | No opposition filed within time limit [2022/10] | Fees paid | Renewal fee | 13.11.2017 | Renewal fee patent year 03 | 14.11.2018 | Renewal fee patent year 04 | 14.11.2019 | Renewal fee patent year 05 | 13.11.2020 | Renewal fee patent year 06 |
| Opt-out from the exclusive Tooltip competence of the Unified Patent Court | See the Register of the Unified Patent Court for opt-out data | ||
| Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Lapses during opposition Tooltip | HU | 05.11.2015 | AL | 24.03.2021 | AT | 24.03.2021 | CY | 24.03.2021 | CZ | 24.03.2021 | DK | 24.03.2021 | EE | 24.03.2021 | FI | 24.03.2021 | HR | 24.03.2021 | LT | 24.03.2021 | LV | 24.03.2021 | MC | 24.03.2021 | MK | 24.03.2021 | MT | 24.03.2021 | NL | 24.03.2021 | PL | 24.03.2021 | RO | 24.03.2021 | RS | 24.03.2021 | SE | 24.03.2021 | SI | 24.03.2021 | SK | 24.03.2021 | SM | 24.03.2021 | TR | 24.03.2021 | BG | 24.06.2021 | NO | 24.06.2021 | GR | 25.06.2021 | IS | 24.07.2021 | PT | 26.07.2021 | IE | 05.11.2021 | LU | 05.11.2021 | BE | 30.11.2021 | CH | 30.11.2021 | LI | 30.11.2021 | [2026/04] |
| Former [2024/41] | HU | 05.11.2015 | |
| AL | 24.03.2021 | ||
| AT | 24.03.2021 | ||
| CY | 24.03.2021 | ||
| CZ | 24.03.2021 | ||
| DK | 24.03.2021 | ||
| EE | 24.03.2021 | ||
| FI | 24.03.2021 | ||
| HR | 24.03.2021 | ||
| LT | 24.03.2021 | ||
| LV | 24.03.2021 | ||
| MC | 24.03.2021 | ||
| MK | 24.03.2021 | ||
| MT | 24.03.2021 | ||
| NL | 24.03.2021 | ||
| PL | 24.03.2021 | ||
| RO | 24.03.2021 | ||
| RS | 24.03.2021 | ||
| SE | 24.03.2021 | ||
| SI | 24.03.2021 | ||
| SK | 24.03.2021 | ||
| SM | 24.03.2021 | ||
| BG | 24.06.2021 | ||
| NO | 24.06.2021 | ||
| GR | 25.06.2021 | ||
| IS | 24.07.2021 | ||
| PT | 26.07.2021 | ||
| IE | 05.11.2021 | ||
| LU | 05.11.2021 | ||
| BE | 30.11.2021 | ||
| CH | 30.11.2021 | ||
| LI | 30.11.2021 | ||
| Former [2024/22] | HU | 05.11.2015 | |
| AL | 24.03.2021 | ||
| AT | 24.03.2021 | ||
| CY | 24.03.2021 | ||
| CZ | 24.03.2021 | ||
| DK | 24.03.2021 | ||
| EE | 24.03.2021 | ||
| FI | 24.03.2021 | ||
| HR | 24.03.2021 | ||
| LT | 24.03.2021 | ||
| LV | 24.03.2021 | ||
| MC | 24.03.2021 | ||
| MK | 24.03.2021 | ||
| NL | 24.03.2021 | ||
| PL | 24.03.2021 | ||
| RO | 24.03.2021 | ||
| RS | 24.03.2021 | ||
| SE | 24.03.2021 | ||
| SI | 24.03.2021 | ||
| SK | 24.03.2021 | ||
| SM | 24.03.2021 | ||
| BG | 24.06.2021 | ||
| NO | 24.06.2021 | ||
| GR | 25.06.2021 | ||
| IS | 24.07.2021 | ||
| PT | 26.07.2021 | ||
| IE | 05.11.2021 | ||
| LU | 05.11.2021 | ||
| BE | 30.11.2021 | ||
| CH | 30.11.2021 | ||
| LI | 30.11.2021 | ||
| Former [2023/30] | HU | 05.11.2015 | |
| AL | 24.03.2021 | ||
| AT | 24.03.2021 | ||
| CY | 24.03.2021 | ||
| CZ | 24.03.2021 | ||
| DK | 24.03.2021 | ||
| EE | 24.03.2021 | ||
| FI | 24.03.2021 | ||
| HR | 24.03.2021 | ||
| LT | 24.03.2021 | ||
| LV | 24.03.2021 | ||
| MC | 24.03.2021 | ||
| NL | 24.03.2021 | ||
| PL | 24.03.2021 | ||
| RO | 24.03.2021 | ||
| RS | 24.03.2021 | ||
| SE | 24.03.2021 | ||
| SI | 24.03.2021 | ||
| SK | 24.03.2021 | ||
| SM | 24.03.2021 | ||
| BG | 24.06.2021 | ||
| NO | 24.06.2021 | ||
| GR | 25.06.2021 | ||
| IS | 24.07.2021 | ||
| PT | 26.07.2021 | ||
| IE | 05.11.2021 | ||
| LU | 05.11.2021 | ||
| BE | 30.11.2021 | ||
| CH | 30.11.2021 | ||
| LI | 30.11.2021 | ||
| Former [2023/28] | HU | 05.11.2015 | |
| AL | 24.03.2021 | ||
| AT | 24.03.2021 | ||
| CZ | 24.03.2021 | ||
| DK | 24.03.2021 | ||
| EE | 24.03.2021 | ||
| FI | 24.03.2021 | ||
| HR | 24.03.2021 | ||
| LT | 24.03.2021 | ||
| LV | 24.03.2021 | ||
| MC | 24.03.2021 | ||
| NL | 24.03.2021 | ||
| PL | 24.03.2021 | ||
| RO | 24.03.2021 | ||
| RS | 24.03.2021 | ||
| SE | 24.03.2021 | ||
| SI | 24.03.2021 | ||
| SK | 24.03.2021 | ||
| SM | 24.03.2021 | ||
| BG | 24.06.2021 | ||
| NO | 24.06.2021 | ||
| GR | 25.06.2021 | ||
| IS | 24.07.2021 | ||
| PT | 26.07.2021 | ||
| IE | 05.11.2021 | ||
| LU | 05.11.2021 | ||
| BE | 30.11.2021 | ||
| CH | 30.11.2021 | ||
| LI | 30.11.2021 | ||
| Former [2022/48] | AL | 24.03.2021 | |
| AT | 24.03.2021 | ||
| CZ | 24.03.2021 | ||
| DK | 24.03.2021 | ||
| EE | 24.03.2021 | ||
| FI | 24.03.2021 | ||
| HR | 24.03.2021 | ||
| LT | 24.03.2021 | ||
| LV | 24.03.2021 | ||
| MC | 24.03.2021 | ||
| NL | 24.03.2021 | ||
| PL | 24.03.2021 | ||
| RO | 24.03.2021 | ||
| RS | 24.03.2021 | ||
| SE | 24.03.2021 | ||
| SI | 24.03.2021 | ||
| SK | 24.03.2021 | ||
| SM | 24.03.2021 | ||
| BG | 24.06.2021 | ||
| NO | 24.06.2021 | ||
| GR | 25.06.2021 | ||
| IS | 24.07.2021 | ||
| PT | 26.07.2021 | ||
| IE | 05.11.2021 | ||
| LU | 05.11.2021 | ||
| BE | 30.11.2021 | ||
| CH | 30.11.2021 | ||
| LI | 30.11.2021 | ||
| Former [2022/37] | AL | 24.03.2021 | |
| AT | 24.03.2021 | ||
| CZ | 24.03.2021 | ||
| DK | 24.03.2021 | ||
| EE | 24.03.2021 | ||
| FI | 24.03.2021 | ||
| HR | 24.03.2021 | ||
| LT | 24.03.2021 | ||
| LV | 24.03.2021 | ||
| MC | 24.03.2021 | ||
| NL | 24.03.2021 | ||
| PL | 24.03.2021 | ||
| RO | 24.03.2021 | ||
| RS | 24.03.2021 | ||
| SE | 24.03.2021 | ||
| SI | 24.03.2021 | ||
| SK | 24.03.2021 | ||
| SM | 24.03.2021 | ||
| BG | 24.06.2021 | ||
| NO | 24.06.2021 | ||
| GR | 25.06.2021 | ||
| IS | 24.07.2021 | ||
| PT | 26.07.2021 | ||
| LU | 05.11.2021 | ||
| BE | 30.11.2021 | ||
| CH | 30.11.2021 | ||
| LI | 30.11.2021 | ||
| Former [2022/34] | AL | 24.03.2021 | |
| AT | 24.03.2021 | ||
| CZ | 24.03.2021 | ||
| DK | 24.03.2021 | ||
| EE | 24.03.2021 | ||
| FI | 24.03.2021 | ||
| HR | 24.03.2021 | ||
| LT | 24.03.2021 | ||
| LV | 24.03.2021 | ||
| MC | 24.03.2021 | ||
| NL | 24.03.2021 | ||
| PL | 24.03.2021 | ||
| RO | 24.03.2021 | ||
| RS | 24.03.2021 | ||
| SE | 24.03.2021 | ||
| SI | 24.03.2021 | ||
| SK | 24.03.2021 | ||
| SM | 24.03.2021 | ||
| BG | 24.06.2021 | ||
| NO | 24.06.2021 | ||
| GR | 25.06.2021 | ||
| IS | 24.07.2021 | ||
| PT | 26.07.2021 | ||
| LU | 05.11.2021 | ||
| BE | 30.11.2021 | ||
| Former [2022/33] | AL | 24.03.2021 | |
| AT | 24.03.2021 | ||
| CZ | 24.03.2021 | ||
| DK | 24.03.2021 | ||
| EE | 24.03.2021 | ||
| FI | 24.03.2021 | ||
| HR | 24.03.2021 | ||
| LT | 24.03.2021 | ||
| LV | 24.03.2021 | ||
| MC | 24.03.2021 | ||
| NL | 24.03.2021 | ||
| PL | 24.03.2021 | ||
| RO | 24.03.2021 | ||
| RS | 24.03.2021 | ||
| SE | 24.03.2021 | ||
| SI | 24.03.2021 | ||
| SK | 24.03.2021 | ||
| SM | 24.03.2021 | ||
| BG | 24.06.2021 | ||
| NO | 24.06.2021 | ||
| GR | 25.06.2021 | ||
| IS | 24.07.2021 | ||
| PT | 26.07.2021 | ||
| BE | 30.11.2021 | ||
| Former [2022/23] | AL | 24.03.2021 | |
| AT | 24.03.2021 | ||
| CZ | 24.03.2021 | ||
| DK | 24.03.2021 | ||
| EE | 24.03.2021 | ||
| FI | 24.03.2021 | ||
| HR | 24.03.2021 | ||
| LT | 24.03.2021 | ||
| LV | 24.03.2021 | ||
| NL | 24.03.2021 | ||
| PL | 24.03.2021 | ||
| RO | 24.03.2021 | ||
| RS | 24.03.2021 | ||
| SE | 24.03.2021 | ||
| SI | 24.03.2021 | ||
| SK | 24.03.2021 | ||
| SM | 24.03.2021 | ||
| BG | 24.06.2021 | ||
| NO | 24.06.2021 | ||
| GR | 25.06.2021 | ||
| IS | 24.07.2021 | ||
| PT | 26.07.2021 | ||
| Former [2022/13] | AL | 24.03.2021 | |
| AT | 24.03.2021 | ||
| CZ | 24.03.2021 | ||
| DK | 24.03.2021 | ||
| EE | 24.03.2021 | ||
| FI | 24.03.2021 | ||
| HR | 24.03.2021 | ||
| LT | 24.03.2021 | ||
| LV | 24.03.2021 | ||
| NL | 24.03.2021 | ||
| PL | 24.03.2021 | ||
| RO | 24.03.2021 | ||
| RS | 24.03.2021 | ||
| SE | 24.03.2021 | ||
| SI | 24.03.2021 | ||
| SK | 24.03.2021 | ||
| SM | 24.03.2021 | ||
| BG | 24.06.2021 | ||
| NO | 24.06.2021 | ||
| GR | 25.06.2021 | ||
| PT | 26.07.2021 | ||
| IS | 24.12.2021 | ||
| Former [2022/10] | AL | 24.03.2021 | |
| AT | 24.03.2021 | ||
| CZ | 24.03.2021 | ||
| DK | 24.03.2021 | ||
| EE | 24.03.2021 | ||
| FI | 24.03.2021 | ||
| HR | 24.03.2021 | ||
| LT | 24.03.2021 | ||
| LV | 24.03.2021 | ||
| NL | 24.03.2021 | ||
| PL | 24.03.2021 | ||
| RO | 24.03.2021 | ||
| RS | 24.03.2021 | ||
| SE | 24.03.2021 | ||
| SK | 24.03.2021 | ||
| SM | 24.03.2021 | ||
| BG | 24.06.2021 | ||
| NO | 24.06.2021 | ||
| GR | 25.06.2021 | ||
| PT | 26.07.2021 | ||
| IS | 24.12.2021 | ||
| Former [2022/08] | AL | 24.03.2021 | |
| AT | 24.03.2021 | ||
| CZ | 24.03.2021 | ||
| DK | 24.03.2021 | ||
| EE | 24.03.2021 | ||
| FI | 24.03.2021 | ||
| HR | 24.03.2021 | ||
| LT | 24.03.2021 | ||
| LV | 24.03.2021 | ||
| NL | 24.03.2021 | ||
| PL | 24.03.2021 | ||
| RO | 24.03.2021 | ||
| RS | 24.03.2021 | ||
| SE | 24.03.2021 | ||
| SK | 24.03.2021 | ||
| SM | 24.03.2021 | ||
| BG | 24.06.2021 | ||
| NO | 24.06.2021 | ||
| GR | 25.06.2021 | ||
| IS | 24.07.2021 | ||
| PT | 26.07.2021 | ||
| Former [2022/07] | AL | 24.03.2021 | |
| AT | 24.03.2021 | ||
| CZ | 24.03.2021 | ||
| EE | 24.03.2021 | ||
| FI | 24.03.2021 | ||
| HR | 24.03.2021 | ||
| LT | 24.03.2021 | ||
| LV | 24.03.2021 | ||
| NL | 24.03.2021 | ||
| PL | 24.03.2021 | ||
| RO | 24.03.2021 | ||
| RS | 24.03.2021 | ||
| SE | 24.03.2021 | ||
| SK | 24.03.2021 | ||
| SM | 24.03.2021 | ||
| BG | 24.06.2021 | ||
| NO | 24.06.2021 | ||
| GR | 25.06.2021 | ||
| IS | 24.07.2021 | ||
| PT | 26.07.2021 | ||
| Former [2021/52] | AT | 24.03.2021 | |
| CZ | 24.03.2021 | ||
| EE | 24.03.2021 | ||
| FI | 24.03.2021 | ||
| HR | 24.03.2021 | ||
| LT | 24.03.2021 | ||
| LV | 24.03.2021 | ||
| NL | 24.03.2021 | ||
| PL | 24.03.2021 | ||
| RO | 24.03.2021 | ||
| RS | 24.03.2021 | ||
| SE | 24.03.2021 | ||
| SK | 24.03.2021 | ||
| SM | 24.03.2021 | ||
| BG | 24.06.2021 | ||
| NO | 24.06.2021 | ||
| GR | 25.06.2021 | ||
| IS | 24.07.2021 | ||
| PT | 26.07.2021 | ||
| Former [2021/51] | AT | 24.03.2021 | |
| CZ | 24.03.2021 | ||
| EE | 24.03.2021 | ||
| FI | 24.03.2021 | ||
| HR | 24.03.2021 | ||
| LT | 24.03.2021 | ||
| LV | 24.03.2021 | ||
| NL | 24.03.2021 | ||
| RO | 24.03.2021 | ||
| RS | 24.03.2021 | ||
| SE | 24.03.2021 | ||
| SK | 24.03.2021 | ||
| SM | 24.03.2021 | ||
| BG | 24.06.2021 | ||
| NO | 24.06.2021 | ||
| GR | 25.06.2021 | ||
| IS | 24.07.2021 | ||
| PT | 26.07.2021 | ||
| Former [2021/50] | AT | 24.03.2021 | |
| CZ | 24.03.2021 | ||
| EE | 24.03.2021 | ||
| FI | 24.03.2021 | ||
| HR | 24.03.2021 | ||
| LT | 24.03.2021 | ||
| LV | 24.03.2021 | ||
| NL | 24.03.2021 | ||
| RO | 24.03.2021 | ||
| RS | 24.03.2021 | ||
| SE | 24.03.2021 | ||
| SK | 24.03.2021 | ||
| SM | 24.03.2021 | ||
| BG | 24.06.2021 | ||
| NO | 24.06.2021 | ||
| GR | 25.06.2021 | ||
| PT | 26.07.2021 | ||
| Former [2021/48] | AT | 24.03.2021 | |
| CZ | 24.03.2021 | ||
| EE | 24.03.2021 | ||
| FI | 24.03.2021 | ||
| HR | 24.03.2021 | ||
| LT | 24.03.2021 | ||
| LV | 24.03.2021 | ||
| NL | 24.03.2021 | ||
| RS | 24.03.2021 | ||
| SE | 24.03.2021 | ||
| SM | 24.03.2021 | ||
| BG | 24.06.2021 | ||
| NO | 24.06.2021 | ||
| GR | 25.06.2021 | ||
| Former [2021/46] | AT | 24.03.2021 | |
| FI | 24.03.2021 | ||
| HR | 24.03.2021 | ||
| LT | 24.03.2021 | ||
| LV | 24.03.2021 | ||
| NL | 24.03.2021 | ||
| RS | 24.03.2021 | ||
| SE | 24.03.2021 | ||
| SM | 24.03.2021 | ||
| BG | 24.06.2021 | ||
| NO | 24.06.2021 | ||
| GR | 25.06.2021 | ||
| Former [2021/43] | FI | 24.03.2021 | |
| HR | 24.03.2021 | ||
| LV | 24.03.2021 | ||
| NL | 24.03.2021 | ||
| RS | 24.03.2021 | ||
| SE | 24.03.2021 | ||
| BG | 24.06.2021 | ||
| NO | 24.06.2021 | ||
| GR | 25.06.2021 | ||
| Former [2021/38] | FI | 24.03.2021 | |
| HR | 24.03.2021 | ||
| LV | 24.03.2021 | ||
| RS | 24.03.2021 | ||
| SE | 24.03.2021 | ||
| BG | 24.06.2021 | ||
| NO | 24.06.2021 | ||
| GR | 25.06.2021 | ||
| Former [2021/37] | FI | 24.03.2021 | |
| HR | 24.03.2021 | ||
| LV | 24.03.2021 | ||
| RS | 24.03.2021 | ||
| BG | 24.06.2021 | ||
| NO | 24.06.2021 | ||
| GR | 25.06.2021 | ||
| Former [2021/36] | FI | 24.03.2021 | |
| HR | 24.03.2021 | ||
| BG | 24.06.2021 | ||
| NO | 24.06.2021 | ||
| GR | 25.06.2021 | ||
| Former [2021/35] | FI | 24.03.2021 | |
| HR | 24.03.2021 | ||
| NO | 24.06.2021 | ||
| Former [2021/33] | FI | 24.03.2021 | |
| NO | 24.06.2021 | Documents cited: | Search | [A] WO2007095050 (INCYTE CORP et al.) [A] 1-3,5-12 * pages 30-32 * | [X] WO2010094126 (MERCK FROSST CANADA LTD et al.) [X] 1,2,5-12 * page 1; example -; claim 1 * | [X] WO2013086002 (CELLWORKS RES INDIA PRIVATE LTD et al.) [X] 1,2,5-12 * page 22; claim 4 * | [X] WO2012158784 [X] 1,2,5-12 * example -; claim 1 * | [X] WO2008077554 (SANOFI AVENTIS et al.) [X] 1,2,5-12 * page 75; claim 1 * | [X] US2005176764 (MATAKI CHIKAGE et al.) [X] 1,2,5-12 * pages 34,54,55; claim 1 * | [X] WO2008133975 (AVALON PHARMACEUTICALS et al.) [X] 1,2,5-12 * example -; claim - * | [X] US2009023773 (VOHRA RAHUL et al.) [X] 1,2,5-12 * paragraph [0029]; example -; claim 1 * | [X] WO2007082079 [X] 1,2,5-12 * example -; claim - * | [X] WO2007044085 (XENON PHARMACEUTICALS INC et al.) [X] 1,2,5-12 * page 32; example -; claim 1 * | [X] WO2014007998 (UNIV CALIFORNIA et al.) [X] 1,2,5-12 * example -; claim - * | [X] WO2014001247 (BAYER PHARMA AG et al.) [X] 1,2,5-12 * example -; claim - * | [X] WO2004047755 (TULARIK INC et al.) [X] 1,2,5-12 * page 120; example 129 * * claim 27 * | [X] WO2006135649 (JANSSEN PHARMACEUTICA NV et al.) [X] 1,2,5-12 * example -; claim - * | [X] WO03076421 (JANSSEN PHARMACEUTICA NV et al.) [X] 1,2,5-12 * example -; claim - * | [X] WO2013041457 (MSD OSS BV et al.) [X] 1,2,5-12 * example -; claim 9 * | [X] WO0220474 (PFIZER PROD INC et al.) [X] 1,2,5-12 * example - * | [X] EP1884510 (DAINIPPON SUMITOMO PHARMA CO et al.) [X] 1,2,5-12 * page 39 * | [X] WO2008156717 (MERCK & CO INC et al.) [X] 1,2,5-12 * example - * | [X] WO2009052320 (UNIV NORTHEASTERN et al.) [X] 1,2,5-12 * pages 44-45 * | [X] WO2007137107 (ABBOTT LAB et al.) [X] 1,2,5-12 * page 30; example - * | [X] US6291499 (THOMPSON WAYNE et al.) [X] 1,2,5-12 * example - * | [X] US2008221175 (YUAN CHESTER CHENGUANG et al.) [X] 1,2,5-12 * example - * | [X] WO2005110976 (GRUENENTHAL GMBH et al.) [X] 1,2,5-12 * example - * | [X] WO2009151800 (MERCK & CO INC et al.) [X] 1,2,5-12 * page 11; example -; claim - * | [X] EP0497303 (KYORIN SEIYAKU KK et al.) [X] 1,2,5-12 * example -; claim - * | [X] WO0071171 (UNIV WAKE FOREST et al.) [X] 1,2,5-12 * example -; claim - * | [X] EP1217000 (AVENTIS PHARMA GMBH et al.) [X] 1,2,5-12 * example -; claim - * | [E] WO2015188085 (FLEXUS BIOSCIENCES INC et al.) [E] 1-3 * pages 59,74 * * pages 79-81; example - * | [X] HUANG ET AL: "Synthesis and quantitative structure-activity relationships of N-(1-benzylpiperidin-4-yl)phenylacetamides and related analogues as potent and selective sigma1 receptors", JOURNAL OF MEDICINAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY, vol. 41, 1 January 1998 (1998-01-01), pages 2361 - 2370, XP002154246, ISSN: 0022-2623, DOI: 10.1021/JM980032L [X] 1,2,5-12 * table 1 * DOI: http://dx.doi.org/10.1021/jm980032l | International search | [X] US2003190298 (BRADLEY STUART E et al.) [X] 1, 15 * ; paragraph [0109] * | [X] US2013197095 (NOLTE BERT et al.) [X] 1, 17-18 * ; paragraphs [0436]-[0437] * | [X] WO2004054974 (SMITHKLINE BEECHAM CORP et al.) [X] 1, 19 * ; page 50, lines 10-15 * | [XY] WO2009052320 (UNIV NORTHEASTERN et al.) [X] 1, 20, 23, 30-31 * ; abstract; paragraphs [0012], [0020], [0024] [0078], [0102], [0360]-[0361] *[Y] 26-29, 32-33, 34/32-33 | [X] EP0596298 (BAYER AG et al.) [X] 1, 21 * ; paragraph [0110] * | [X] EP1781656 (SANOFI AVENTIS DEUTSCHLAND et al.) [X] 1, 22 * ; paragraph [0125] * | [XY] WO2005080317 (PFIZER JAPAN INC et al.) [X] 1-8, 25 * ; abstract; page 15, paragraph 2; page 16, paragraph 1; page 17, paragraph 3; page 29, paragraphs 4-5; page 78, paragraphs 4-5; page 85, paragraphs 2-3 *[Y] 9-14, 16, 24 | [Y] US5455273 (MAIER ROLAND et al.) [Y] 9-13 * ; column 11, lines 50-55; column 22, lines 15-20 * | [Y] WO2010015655 (NOVARTIS AG et al.) [Y] 1, 14 * ; page 26, lines 10-15; page 97, lines 1-20; * | [Y] US2013217706 (TRAN THUY-ANH et al.) [Y] 1, 16 * ; paragraphs [0049], [0643] * | [Y] WO2014150677 (BRISTOL MYERS SQUIBB CO et al.) [Y] 26-29 * ; abstract; page 1, lines 20-30; page 107, lines 15-22 * | [Y] WO2014160967 (BIOMED VALLEY DISCOVERIES INC et al.) [Y] 32-33, 34/32-33 * ; paragraphs [0032], [0052], [0079], [0101]; claim 31 * | [Y] DATABASE PUBCHEM 22 May 2013 (2013-05-22), Database accession no. SID162741420 [Y] 1, 24 * ; page 3 * | by applicant | WO9929310 | WO2004094409 | WO2007095050 | WO2005080317 | WO0192204 | SERAFINI, P. ET AL., SEMIN. CANCER BIOL., vol. 16, no. 1, February 2006 (2006-02-01), pages 53 - 65 | BALL, H.J. ET AL., GENE, vol. 396, no. 1, 1 July 2007 (2007-07-01), pages 203 - 213 [Y] 9-14, 16, 24 | BRANDACHER, G. ET AL., CLIN. CANCER RES., vol. 12, no. 4, 15 February 2006 (2006-02-15), pages 1144 - 1151 | YAMAMOTO, T. ET AL., J. ORGANOMET. CHEM., vol. 694, 2009, pages 1325 - 1332 | LI, G. ET AL., BIOORG. MED. CHEM. LETT., vol. 18, 2008, pages 1146 - 1150 | BIOORG. MED. CHEM. LETT., vol. 24, 2014, pages 5377 [Y] 1, 24 * ; page 3 * |