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Extract from the Register of European Patents

EP About this file: EP3327016

EP3327016 - PREPARATION OF MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  22.04.2022
Database last updated on 26.06.2024
FormerThe patent has been granted
Status updated on  14.05.2021
FormerGrant of patent is intended
Status updated on  16.06.2020
FormerExamination is in progress
Status updated on  12.04.2019
FormerRequest for examination was made
Status updated on  23.11.2018
FormerThe application has been published
Status updated on  27.04.2018
Most recent event   Tooltip12.04.2024Lapse of the patent in a contracting state
New state(s): CY		published on 15.05.2024  [2024/20]
Applicant(s)For all designated states
Vertex Pharmaceuticals Incorporated
50 Northern Avenue
Boston, MA 02210 / US
[2018/22]
Inventor(s)01 / RUAH, Sara S. Hadida
2356 Torrey Pines Road 16
La Jolla, CA 92037 / US
02 / GROOTENHUIS, Peter D.J.
1955 Jimmy Durante Boulevard
Del Mar, CA 92104 / US
03 / VAN GOOR, Fredrick
832 Ormond Court
San Diego, CA 92109 / US
04 / ZHOU, Jinglan
4466 Shorepointe Way
San Diego, CA 92109 / US
05 / BEAR, Brian
7010 Sitio Corazon
Carlsbad, CA 92109 / US
06 / MILLER, Mark T.
5075 La Jolla Blvd. 9
San Diego, CA 92109 / US
07 / MCCARTNEY, Jason
1428 Kings Cross Drive
Cardiff By The Sea, CA 92007 / US
08 / NUMA, Mehdi, Michel, Jamel
4664 36th Street
San Diego, CA 92116 / US
09 / YANG, Xiaoqing
4526 Vareda Mar de Ponderosa
San Diego, CA 92130 / US
 [2018/26]
Former [2018/22]01 / RUAH, Sara S. Hadida
2356 Torrey Pines Road 16
La Jolla, CA 92037 / US
02 / GROOTENHUIS, Peter D.J.
4801 Riding Ridge Road
San Diego, CA 92130 / US
03 / VAN GOOR, Fredrick
832 Ormond Court
San Diego, CA 92109 / US
04 / ZHOU, Jinglan
4466 Shorepointe Way
San Diego, CA 92109 / US
05 / BEAR, Brian
7010 Sitio Corazon
Carlsbad, CA 92109 / US
06 / MILLER, Mark T.
5075 La Jolla Blvd. 9
San Diego, CA 92109 / US
07 / MCCARTNEY, Jason
1429 Kings Cross Drive
Cardiff By The Sea, CA 92007 / US
08 / NUMA, Mehdi, Michel, Jamel
4664 36th Street
San Diego, CA 92116 / US
09 / YANG, Xiaoqing
4526 Vareda Mar de Ponderosa
San Diego, CA 92130 / US
Representative(s)Carpmaels & Ransford LLP
One Southampton Row
London WC1B 5HA / GB
[2018/22]
Application number, filing date17209175.309.04.2007
[2018/22]
Priority number, dateUS20060790459P07.04.2006         Original published format: US 790459 P
[2018/22]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report 
No.:EP3327016
Date:30.05.2018
Language:EN
[2018/22]
Type: B1 Patent specification 
No.:EP3327016
Date:16.06.2021
Language:EN
[2021/24]
Search report(s)(Supplementary) European search report - dispatched on:EP23.02.2018
ClassificationIPC:C07D405/12, C07D405/14, C07D471/04
[2018/22]
CPC:
C07D405/12 (EP,US); A61K31/445 (US); A61K31/496 (US);
A61K31/5377 (US); A61P1/18 (EP); A61P11/00 (EP);
A61P11/08 (EP); A61P11/12 (EP); A61P13/02 (EP);
A61P13/12 (EP); A61P15/00 (EP); A61P19/08 (EP);
A61P21/00 (EP); A61P21/02 (EP); A61P25/00 (EP);
A61P25/14 (EP); A61P25/16 (EP); A61P25/28 (EP);
A61P27/02 (EP); A61P27/04 (EP); A61P29/00 (EP);
A61P3/00 (EP); A61P3/06 (EP); A61P3/10 (EP);
A61P31/00 (EP); A61P35/00 (EP); A61P43/00 (EP);
A61P5/00 (EP); A61P5/06 (EP); A61P5/14 (EP);
A61P5/18 (EP); A61P5/48 (EP); A61P7/00 (EP);
A61P7/02 (EP); A61P7/10 (EP); A61P7/12 (EP);
A61P9/14 (EP); C07B59/002 (US); C07D209/08 (EP);
C07D403/12 (EP,US); C07D405/14 (EP,US); C07D471/04 (EP,US);
C07D487/04 (EP,US); G01N33/5008 (US); G01N33/6872 (US);
C07B2200/05 (US); G01N2333/705 (US); G01N2500/02 (US);
G01N2500/10 (US) (-)
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MT,   NL,   PL,   PT,   RO,   SE,   SI,   SK,   TR [2018/52]
Former [2018/22]AT,  BE,  BG,  CH,  CY,  CZ,  DE,  DK,  EE,  ES,  FI,  FR,  GB,  GR,  HU,  IE,  IS,  IT,  LI,  LT,  LU,  LV,  MC,  MT,  NL,  PL,  PT,  RO,  SE,  SI,  SK,  TR 
TitleGerman:HERSTELLUNG VON MODULATOREN VON ATP-BINDENDEN KASSETTENTRANSPORTERN[2018/22]
English:PREPARATION OF MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS[2018/22]
French:PRÉPARATION DES MODULATEURS DE TRANSPORTEURS DE CASSETTE À LIAISON ATP[2018/22]
Examination procedure20.11.2018Amendment by applicant (claims and/or description)
20.11.2018Examination requested  [2018/52]
20.11.2018Date on which the examining division has become responsible
16.04.2019Despatch of a communication from the examining division (Time limit: M06)
31.01.2020Reply to a communication from the examining division
17.06.2020Communication of intention to grant the patent
17.11.2020Despatch of communication that the application is deemed to be withdrawn, reason: fee for grant / fee for printing not paid in time
26.01.2021Fee for grant paid
26.01.2021Fee for publishing/printing paid
26.01.2021Receipt of the translation of the claim(s)
Parent application(s)   TooltipEP07755298.2  / EP2007756
EP13167785.8  / EP2674428
EP16155334.2  / EP3091011
Divisional application(s)EP21156114.7  / EP3882245
Opposition(s)17.03.2022No opposition filed within time limit [2022/21]
Request for further processing for:The application is deemed to be withdrawn due to failure to fulfill actions required for granting the patent
26.01.2021Request for further processing filed
26.01.2021Full payment received (date of receipt of payment)
Request granted
02.02.2021Decision despatched
The application is deemed to be withdrawn due to failure to reply to the examination report
31.01.2020Request for further processing filed
31.01.2020Full payment received (date of receipt of payment)
Request granted
13.02.2020Decision despatched
Fees paidRenewal fee
20.12.2017Renewal fee patent year 03
20.12.2017Renewal fee patent year 04
20.12.2017Renewal fee patent year 05
20.12.2017Renewal fee patent year 06
20.12.2017Renewal fee patent year 07
20.12.2017Renewal fee patent year 08
20.12.2017Renewal fee patent year 09
20.12.2017Renewal fee patent year 10
20.12.2017Renewal fee patent year 11
11.04.2018Renewal fee patent year 12
15.04.2019Renewal fee patent year 13
27.04.2020Renewal fee patent year 14
27.04.2021Renewal fee patent year 15
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Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipAT16.06.2021
CY16.06.2021
DK16.06.2021
EE16.06.2021
FI16.06.2021
LT16.06.2021
LV16.06.2021
MC16.06.2021
SE16.06.2021
GR17.09.2021
PT18.10.2021
[2024/20]
Former [2023/06]AT16.06.2021
DK16.06.2021
EE16.06.2021
FI16.06.2021
LT16.06.2021
LV16.06.2021
MC16.06.2021
SE16.06.2021
GR17.09.2021
PT18.10.2021
Former [2022/21]AT16.06.2021
DK16.06.2021
EE16.06.2021
FI16.06.2021
LT16.06.2021
LV16.06.2021
SE16.06.2021
GR17.09.2021
PT18.10.2021
Former [2022/11]AT16.06.2021
EE16.06.2021
FI16.06.2021
LT16.06.2021
LV16.06.2021
SE16.06.2021
GR17.09.2021
PT18.10.2021
Former [2022/07]AT16.06.2021
FI16.06.2021
LT16.06.2021
LV16.06.2021
SE16.06.2021
GR17.09.2021
Former [2021/49]FI16.06.2021
LT16.06.2021
LV16.06.2021
SE16.06.2021
GR17.09.2021
Former [2021/46]FI16.06.2021
LT16.06.2021
Documents cited:Search[X]WO03002533  (PFIZER PROD INC [US], et al) [X] 1-7 * page 75; example 122 * * page 16, line 11 - line 27 *;
 [I]EP1380576  (EISAI CO LTD [JP]) [I] 1-7 * pages 171,175,, column 182; examples I-85,I-159,II-25 *;
 [X]WO2004035571  (RIGEL PHARMACEUTICALS INC [US], et al) [X] 1-7 * pages 26,33; claims 1,25; compounds 5D,231 ** paragraph [00104] - paragraph [00110] *;
 [I]WO2004041277  (MERCK & CO INC [US], et al) [I] 1-7 * pages 83,89; examples 3-78,5; claims 1,15,18 *;
 [I]WO2004056745  (JANSSEN PHARMACEUTICA NV [BE], et al) [I] 1-7 * page 2, line 31 * *Scheme 2*; page 5, paragraph 1; example -; claims 1,13,16 *;
 [X]WO2005016884  (LUNDBECK & CO AS H [DK], et al) [X] 1-7 * page 7, line 30; claims 1,113,114 *;
 [X]WO2005075435  (VERTEX PHARMA [US], et al) [X] 1-7 * page 95, paragraphs 67,72; claims 1,129,131; table 1; compound 245 *
by applicantUS5304121
 US5886026
 US6099562
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