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Extract from the Register of European Patents

EP About this file: EP3415515

EP3415515 - METHOD FOR THE PREPARATION OF METHYL-{4,6-DIAMINO-2-[1-(2-FLUOROBENZYL)-1H-PYRAZOLO[3,4-B]PYRIDIN-3-YL]PYRIMIDIN-5-YL}METHYLCARBAMATE [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  30.10.2020
Database last updated on 02.07.2024
FormerThe patent has been granted
Status updated on  22.11.2019
FormerGrant of patent is intended
Status updated on  31.07.2019
FormerRequest for examination was made
Status updated on  16.11.2018
Most recent event   Tooltip15.07.2022Lapse of the patent in a contracting state
New state(s): MK		published on 17.08.2022  [2022/33]
Applicant(s)For all designated states
Adverio Pharma GmbH
Willy-Brandt-Platz 2
12529 Schönefeld / DE
[2018/51]
Inventor(s)01 / MAIS, Franz-Josef
Otto-Hahn-Str. 164
40591 Düsseldorf / DE
02 / REHSE, Joachim
Am Kloster 12
42799 Leichlingen / DE
03 / JOENTGEN, Winfried
Sprengelstrasse 1
50735 Köln / DE
04 / SIEGEL, Konrad
Augsburger Strasse 11
40597 Düsseldorf / DE
 [2018/51]
Representative(s)BIP Patents
c/o Bayer Intellectual Property GmbH
Alfred-Nobel-Straße 50
40789 Monheim am Rhein / DE
[N/P]
Former [2018/51]BIP Patents
c/o Bayer Intellectual Property GmbH
Alfred-Nobel-Straße 10
40789 Monheim am Rhein / DE
Application number, filing date18178602.122.11.2010
[2018/51]
Priority number, dateEP2009017737127.11.2009         Original published format: EP 09177371
[2018/51]
Previously filed application, dateEP2014015476222.11.2010
[2018/51]
Filing languageDE
Procedural languageDE
PublicationType: A1 Application with search report 
No.:EP3415515
Date:19.12.2018
Language:DE
[2018/51]
Type: B1 Patent specification 
No.:EP3415515
Date:25.12.2019
Language:DE
[2019/52]
Search report(s)(Supplementary) European search report - dispatched on:EP08.10.2018
ClassificationIPC:C07D471/04
[2018/51]
CPC:
A61P1/04 (EP); C07D471/04 (EP,CN,EA,IL,KR,US); A61K31/437 (KR);
A61K31/506 (KR); A61P11/06 (EP); A61P13/02 (EP);
A61P13/08 (EP); A61P15/00 (EP); A61P15/10 (EP);
A61P19/02 (EP); A61P19/10 (EP); A61P27/06 (EP);
A61P7/02 (EP); A61P9/00 (EP); A61P9/04 (EP);
A61P9/06 (EP); A61P9/10 (EP); A61P9/12 (EP);
C07C325/02 (IL,KR,US); C07D239/48 (IL,KR,US); C07D239/50 (IL,KR,US);
C07D403/04 (IL,KR,US); C07D487/04 (IL,KR,US) (-)
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   RS,   SE,   SI,   SK,   SM,   TR [2018/51]
Extension statesBA19.06.2018
ME19.06.2018
TitleGerman:VERFAHREN ZUR HERSTELLUNG VON METHYL-{4,6-DIAMINO-2-[1-(2-FLUOROBENZYL)-1H-PYRAZOLO[3,4-B]PYRIDIN-3-YL]PYRIMIDIN-5-YL}METHYLCARBAMAT[2018/51]
English:METHOD FOR THE PREPARATION OF METHYL-{4,6-DIAMINO-2-[1-(2-FLUOROBENZYL)-1H-PYRAZOLO[3,4-B]PYRIDIN-3-YL]PYRIMIDIN-5-YL}METHYLCARBAMATE[2018/51]
French:PROCÉDÉ DE PRODUCTION DE MÉTHYL{4,6-DIAMINO-2-[1-(2-FLUOROBENZYL)-1H-PYRAZOLO [3,4-B]PYRIDIN-3-YL]PYRIMIDIN-5-YL}MÉTHYLCARBAMATE[2018/51]
Examination proceduredeletedDate on which the examining division has become responsible
19.06.2018Examination requested  [2018/51]
01.08.2019Communication of intention to grant the patent
31.10.2019Fee for grant paid
31.10.2019Fee for publishing/printing paid
31.10.2019Receipt of the translation of the claim(s)
Parent application(s)   TooltipEP10781686.0  / EP2504334
EP13151569.4  / EP2604608
EP14154762.0  / EP2733142
Divisional application(s)EP19214991.2  / EP3699180
Opposition(s)28.09.2020No opposition filed within time limit [2020/49]
Fees paidRenewal fee
19.06.2018Renewal fee patent year 03
19.06.2018Renewal fee patent year 04
19.06.2018Renewal fee patent year 05
19.10.2018Renewal fee patent year 06
19.10.2018Renewal fee patent year 07
19.10.2018Renewal fee patent year 08
14.11.2018Renewal fee patent year 09
14.11.2019Renewal fee patent year 10
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court		 See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipAL25.12.2019
CY25.12.2019
MC25.12.2019
MK25.12.2019
SM25.12.2019
GR26.03.2020
[2022/33]
Former [2022/28]AL25.12.2019
CY25.12.2019
MC25.12.2019
SM25.12.2019
GR26.03.2020
Former [2021/31]AL25.12.2019
MC25.12.2019
SM25.12.2019
GR26.03.2020
Former [2020/38]AL25.12.2019
SM25.12.2019
GR26.03.2020
Former [2020/32]AL25.12.2019
GR26.03.2020
Former [2020/25]GR26.03.2020
Documents cited:Search[AD]WO03095451  (BAYER AG [DE], et al) [AD] 1,2 * the whole document * * insbesondere Beispiele 8a, 5, 8 *;
 [A]WO2005046725  (BAYER HEALTHCARE AG [DE], et al) [A] 1,2 * the whole document ** Insbesondere Beipiele 8A, 1, 5 und 8 *;
 [AP]WO2010079120  (BAYER SCHERING PHARMA AG [DE], et al) [AP] 1,2 * the whole document *;
 [AD]  - CHEMMEDCHEM, (200905), vol. 4, no. 5, doi:10.1002/CMDC.200900014, ISSN 1860-7179, pages 853 - 865, XP002622814 [AD] 1,2 * the whole document * * Insbesondere Schemata 10 und 11, Seiten 860, 863-864, Verbindungen 51, 52 und 20 *

DOI:   http://dx.doi.org/10.1002/CMDC.200900014
 [A]  - SCHWOCH S ET AL, "2,3-DIHYDROSPIRO[1H-4- AND 5-AZABENZIMIDAZOLE-2.1'-CYCLOHEXANE] (= SPIRO[CYCLOHEXANE-1,2'(3'H)-1'H-IMIDAZO[4,5-B]PYRIDINE] AND SPIRO[CYCLOHEXANE-1,2'(3'H)-1'H-IMIDAZO[4,5-C]PYRIDINE]): REACTIONS WITH NUCLEOPHILES", HELVETICA CHIMICA ACTA, VERLAG HELVETICA CHIMICA ACTA, BASEL, CH, (19940101), vol. 77, no. 8, doi:10.1002/HLCA.19940770811, ISSN 0018-019X, pages 2175 - 2190, XP002073789 [A] 1 * page 2182; figure 6 * * page 2189 - page 2190; compounds 39,40 *

DOI:   http://dx.doi.org/10.1002/hlca.19940770811
 [A]  - BARRACLOUGH P ET AL, "Mono-arylation of 2,3- and 3,4-diaminopyridine and 4,5-diaminopyrimidine, and syntheses of putative inotrope/beta-adrenoceptor antagonists", JOURNAL OF CHEMICAL RESEARCH, SCIENCE REVIEWS LTD, GB, (19960101), vol. 9, no. 9, ISSN 0308-2342, pages 2316 - 2335, XP002103810 [A] 1 * page 407; figures 3,4 *
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.