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Extract from the Register of European Patents

EP About this file: EP3653611

EP3653611 - INHIBITORS OF METALLO-BETA-LACTAMASES [Right-click to bookmark this link]
StatusThe application is deemed to be withdrawn
Status updated on  26.03.2021
Database last updated on 19.10.2024
FormerThe application has been published
Status updated on  17.04.2020
Most recent event   Tooltip26.03.2021Application deemed to be withdrawnpublished on 28.04.2021  [2021/17]
Applicant(s)For all designated states
CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE
3, rue Michel Ange
75016 Paris / FR
For all designated states
Universite de Sienne
Policlinico "Le Scotte" II piano
V lotto Viale Braci 16
53100 Siena / IT
For all designated states
Ecole Nationale Supérieure de Chimie de Montpellier
240 Avenue du Professeur Emile Jeanbrau
34090 Montpellier / FR
For all designated states
UNIVERSITE DE MONTPELLIER
163, rue Auguste Broussonnet
34090 Montpellier / FR
[2020/21]
Inventor(s)01 / HERNANDEZ, Jean-François
6 rue Pierre Curie
34150 Gignac / FR
02 / GAVARA, Laurent
3 Impasse Camille Claudel
34920 Le Cres / FR
03 / DOCQUIER, Jean-Denis
15 Via Alcide de Gasperi
53018 Sovicille / IT
04 / SEVAILLE, Laurent
145 Impasse de la voie Romaine
34090 Montpellier / FR
 [2020/21]
Representative(s)Cabinet Becker et Associés
25, rue Louis le Grand
75002 Paris / FR
[2020/21]
Application number, filing date18306493.015.11.2018
[2020/21]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report 
No.:EP3653611
Date:20.05.2020
Language:EN
[2020/21]
Search report(s)(Supplementary) European search report - dispatched on:EP21.10.2019
ClassificationIPC:C07D249/10, C07D401/04, C07D401/06, C07D401/12, C07D405/06, C07D409/04, C07D417/04, A61P31/04, A61K31/4196
[2020/21]
CPC:
A61P31/04 (EP); A61K31/4196 (US); A61K31/433 (US);
A61K31/4709 (US); A61K31/496 (US); A61K31/5377 (US);
A61K31/655 (US); A61K45/06 (US); C07D249/10 (EP);
C07D249/12 (US); C07D401/04 (EP,US); C07D401/06 (EP);
C07D401/12 (EP,US); C07D403/04 (US); C07D405/06 (EP,US);
C07D409/04 (EP,US); C07D417/04 (EP,US) (-)
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   RS,   SE,   SI,   SK,   SM,   TR [2020/21]
Extension statesBANot yet paid
MENot yet paid
Validation statesKHNot yet paid
MANot yet paid
MDNot yet paid
TNNot yet paid
TitleGerman:METALLO-BETA-LACTAMASE INHIBITOREN[2020/21]
English:INHIBITORS OF METALLO-BETA-LACTAMASES[2020/21]
French:INHIBITEURS DE METALLO-BETA-LACTAMASES[2020/21]
Examination procedure21.11.2020Application deemed to be withdrawn, date of legal effect  [2021/17]
11.12.2020Despatch of communication that the application is deemed to be withdrawn, reason: examination fee not paid in time  [2021/17]
Fees paidPenalty fee
Additional fee for renewal fee
30.11.202003   M06   Not yet paid
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Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Documents cited:Search[X]US2012330009  (YING WEIWEN [US], et al) [X] 1,3 * claim 1; table 1; compounds 1,3,4,10-19 *;
 [X]US2007155809  (YING WEIWEN [US], et al) [X] 1,3 * examples 35,37; claim 1; table 1; compounds 15,38 *;
 [X]US2012064175  (VUKOVIC VOJO [US], et al) [X] 1,3,4 * examples 2,3,4,5,7; claim 1; table 1 *;
 [X]FR2546887  (PARIS 7 UNIVERSITE [FR]) [X] 1,3 * claim 1; table II *;
 [X]DE2321218  (FUJI PHOTO FILM CO LTD) [X] 1,3 * examples 4,8,9; claim 1 *;
 [X]EP2527335  (UNIV KING SAUD [SA]) [X] 1 * Scheme 1; paragraph [0017] *;
 [X]EP1906245  (FUJIFILM CORP [JP]) [X] 1,3 * SH8-SH11, SH16; paragraph [0082] *
 [I]  - FRANCESCA SPYRAKIS ET AL, "Structure-Based Virtual Screening for the Discovery of Novel Inhibitors of New Delhi Metallo-[beta]-lactamase-1", ACS MEDICINAL CHEMISTRY LETTERS, (20171130), vol. 9, no. 1, doi:10.1021/acsmedchemlett.7b00428, ISSN 1948-5875, pages 45 - 50, XP055574723 [I] 1-6,11,13,14,16,18-22 * abstract *

DOI:   http://dx.doi.org/10.1021/acsmedchemlett.7b00428
 [I]  - OLSEN L ET AL, "New leads of metallo-@b-lactamase inhibitors from structure-based pharmacophore design", BIOORGANIC & MEDICINAL CHEMISTRY, PERGAMON, GB, vol. 14, no. 8, ISSN 0968-0896, (20060415), pages 2627 - 2635, (20060415), XP027992523 [I] 1-6,11,13,14,16,18-22 * abstract *
 [XI]  - LAURENT SEVAILLE ET AL, "1,2,4-Triazole-3-thione Compounds as Inhibitors of Dizinc Metallo-[beta]-lactamases", CHEMMEDCHEM, DE, (20170621), vol. 12, no. 12, doi:10.1002/cmdc.201700186, ISSN 1860-7179, pages 972 - 985, XP055575617 [X] 1-4 * abstract * [I] 1-6,11,13,14,16,18-22

DOI:   http://dx.doi.org/10.1002/cmdc.201700186
 [XI]  - AGATA SIWEK ET AL, "Molecular Properties Prediction, Docking Studies, and Antimicrobial Screening of 1,3,4-Thiadiazole and s-Triazole Derivatives", CURRENT COMPUTER-AIDED DRUG DESIGN, AE, (20140531), vol. 10, no. 1, doi:10.2174/15734099113096660033, ISSN 1573-4099, pages 3 - 14, XP055574720 [X] 1,3 * Scheme 1, series II;; table 4 * [I] 1-6,11,13,14,16,18-22

DOI:   http://dx.doi.org/10.2174/15734099113096660033
by applicant   - MAINGOT L.; LEROUX F.; LANDRY V.; DUMONT J.; NAGASE H.; VILLOUTREIX B.; SPERANDIO O.; DEPREZ-POULAIN R.; DEPREZ B., Bioorg. Med. Chem. Letters, (20100000), vol. 20, pages 6213 - 6
    - DOCQUIER J.D.; LAMOTTE-BRASSEUR J.; GALLENI M.; AMICOSANTE G.; FRERE J.M.; ROSSOLINI G.M., J. Antimicrob. Chemother., (20030000), vol. 51, pages 257 - 266
    - BORGIANNI L.; VANDENAMEELE J.; MATAGNE A.; BINI L.; BONOMO R.A.; FRERE J.M.; ROSSOLINI G.M.; DOCQUIER J.D., Antimicrob. Agents Chemother., (20100000), vol. 54, pages 3197 - 3204
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.