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Extract from the Register of European Patents

EP About this file: EP3765452

EP3765452 - PREPARATIVE PROCESS OF TWO 4-{[(2S)-2-{4-[5-CHLORO-2-(1H-1,2,3-TRIAZOL-1-YL)PHENYL]-5-METHOXY-2-OXOPYRIDIN-1(2H)-YL}BUTANOYL]AMINO}-2-FLUOROBENZAMIDE DERIVATIVES [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  17.02.2023
Database last updated on 05.10.2024
FormerThe patent has been granted
Status updated on  11.03.2022
FormerGrant of patent is intended
Status updated on  16.12.2021
FormerRequest for examination was made
Status updated on  18.12.2020
FormerThe international publication has been made
Status updated on  21.09.2019
Formerunknown
Status updated on  15.03.2019
Most recent event   Tooltip27.10.2023Lapse of the patent in a contracting state
New state(s): MC
published on 29.11.2023  [2023/48]
Applicant(s)For all designated states
Bayer Aktiengesellschaft
Kaiser-Wilhelm-Allee 1
51373 Leverkusen / DE
For all designated states
Bayer Pharma Aktiengesellschaft
Müllerstrasse 178
13353 Berlin / DE
[2021/03]
Inventor(s)01 / EGGER, Julian
Anton-Küppers-Weg 15
42855 Remscheid / DE
02 / GÖTZ, Daniel
Martinstr. 46
40223 Düsseldorf / DE
03 / SOWA, Michal
Kempers Häuschen 10
42109 Wuppertal / DE
 [2021/03]
Representative(s)BIP Patents
c/o Bayer Intellectual Property GmbH
Alfred-Nobel-Straße 50
40789 Monheim am Rhein / DE
[N/P]
Former [2021/03]BIP Patents
c/o Bayer Intellectual Property GmbH
Alfred-Nobel-Straße 10
40789 Monheim am Rhein / DE
Application number, filing date19708556.608.03.2019
[2021/03]
WO2019EP55815
Priority number, dateEP2018016198315.03.2018         Original published format: EP 18161983
[2021/03]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2019175043
Date:19.09.2019
Language:EN
[2019/38]
Type: A1 Application with search report 
No.:EP3765452
Date:20.01.2021
Language:EN
The application published by WIPO in one of the EPO official languages on 19.09.2019 takes the place of the publication of the European patent application.
[2021/03]
Type: B1 Patent specification 
No.:EP3765452
Date:13.04.2022
Language:EN
[2022/15]
Search report(s)International search report - published on:EP19.09.2019
ClassificationIPC:C07D401/10, C07C233/00
[2021/03]
CPC:
C07D401/10 (EP,IL,KR,US); A61K31/4439 (IL,KR); A61P7/02 (KR);
C07C237/30 (IL,KR)
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   RS,   SE,   SI,   SK,   SM,   TR [2021/03]
Extension statesBA15.10.2020
Validation statesKHNot yet paid
MANot yet paid
MDNot yet paid
TNNot yet paid
TitleGerman:VERFAHREN ZUR HERSTELLUNG VON ZWEI 4-{[(2S)-2-{4-[5-CHLOR-2-(1H-1,2,3-TRIAZOL-1-YL)PHENYL]-5-METHOXY-2-OXOPYRIDIN-1(2H)-YL}BUTANOYL]AMINO}-2-FLUORBENZAMID-DERIVATEN[2021/03]
English:PREPARATIVE PROCESS OF TWO 4-{[(2S)-2-{4-[5-CHLORO-2-(1H-1,2,3-TRIAZOL-1-YL)PHENYL]-5-METHOXY-2-OXOPYRIDIN-1(2H)-YL}BUTANOYL]AMINO}-2-FLUOROBENZAMIDE DERIVATIVES[2021/03]
French:PROCÉDÉ DE PRÉPARATION DE DEUX DÉRIVÉS DE 4-{[(2S)-2-{4-[5-CHLORO-2-(1H-1,2,3-TRIAZOL-1-YL)PHÉNYL]-5-MÉTHOXY-2-OXOPYRIDIN-1(2H)-YL}BUTANOYL]AMINO}-2-FLUOROBENZAMIDE[2021/03]
Entry into regional phase15.10.2020National basic fee paid 
15.10.2020Designation fee(s) paid 
15.10.2020Examination fee paid 
Examination procedure15.10.2020Examination requested  [2021/03]
15.10.2020Date on which the examining division has become responsible
19.04.2021Amendment by applicant (claims and/or description)
17.12.2021Communication of intention to grant the patent
03.03.2022Fee for grant paid
03.03.2022Fee for publishing/printing paid
03.03.2022Receipt of the translation of the claim(s)
Divisional application(s)EP21169162.1  / EP3889147
Opposition(s)16.01.2023No opposition filed within time limit [2023/12]
Fees paidRenewal fee
12.03.2021Renewal fee patent year 03
02.03.2022Renewal fee patent year 04
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Lapses during opposition  TooltipAL13.04.2022
MC13.04.2022
SM13.04.2022
GR14.07.2022
[2023/48]
Former [2023/17]AL13.04.2022
SM13.04.2022
GR14.07.2022
Former [2023/10]SM13.04.2022
GR14.07.2022
Former [2022/49]GR14.07.2022
Cited inInternational search[IDA]WO2017005725  (BAYER PHARMA AG [DE]) [ID] 16,17 * scheme 1, page 44; example 234 + example 235, pages 355-356; example 171 + example 242, pages 317, 318 and 360; claim 4 and 5 *[A] 1-15
by applicantWO2014154794
 WO2017005725
    - P. S. DRAGOVICH et al., J. Med. Chem., (20030000), vol. 46, page 4572
    - L. CHEN et al., Organic Process Research & Development, (20060000), vol. 10, page 838
    - A. S. GURAM et al., Organic Letters, (20060000), vol. 8, page 1787
    - H. RAPOPORT et al., J. Org. Chem.,, (19860000), vol. 51, page 1713
    - J. R. DUNETZ et al., Org. Lett., (20110000), vol. 13, page 5048
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.