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Extract from the Register of European Patents

EP About this file: EP3762423

EP3762423 - CHEMOSELECTIVE THIOL-CONJUGATION WITH ALKENE OR ALKYNE-PHOSPHONOTHIOLATES AND -PHOSPHONATES [Right-click to bookmark this link]
Status	Examination is in progress Status updated on 07.07.2023 Database last updated on 19.03.2026
Former	Request for examination was made Status updated on 11.12.2020
Former	The international publication has been made Status updated on 14.09.2019
Former	unknown Status updated on 08.04.2019
Most recent event Tooltip	12.03.2026	Change - representative
Applicant(s)	For all designated states Forschungsverbund Berlin E.V. Rudower Chaussee 17 12489 Berlin / DE
	For all designated states Ludwig-Maximilians-Universität München Geschwister-Scholl-Platz 1 80539 München / DE
	[2021/02]
Inventor(s)	01 / HACKENBERGER, Christian Klausenerplatz 22 14059 Berlin / DE
	02 / BAUMANN, Alice Leonie Scherenbergstraße 22 10439 Berlin / DE
	03 / KASPER, Marc-André Pettenkoferstrasse 14 10247 Berlin / DE
	04 / BYRNE, Stephen 524 Mourne road Drimnagh Dublin 12, D12 XW01 / IE
	05 / HELMA-SMETS, Jonas Preysingstrasse 40 81667 Muenchen / DE
	06 / LEONHARDT, Heinrich Klenzestr. 4 80469 Muenchen / DE
	07 / STOSCHECK, Tina Oetztaler Strasse 25 81373 Muenchen / DE
	08 / GERLACH, Marcus Kornwegerstrasse 54 81375 Muenchen / DE
	09 / SCHUMACHER, Dominik Gottfried-Keller-Str. 13 81245 Muenchen / DE
	[2021/02]
Representative(s)	Dörries, Hans Ulrich df-mp Patentanwälte Rechtsanwälte PartG mbB Theatinerstraße 16 80333 München / DE
	[N/P]
Former [2021/02]	Schiweck Weinzierl Koch Patentanwälte Partnerschaft mbB Ganghoferstraße 68 B 80339 München / DE
Application number, filing date	19713707.8	06.03.2019
	[2021/02]
	WO2019EP55509
Priority number, date	EP20180160384	07.03.2018 Original published format: EP 18160384
	[2021/02]
Filing language	EN
Procedural language	EN
Publication	Type:	A2 Application without search report
	No.:	WO2019170710
	Date:	12.09.2019
	Language:	EN
	[2019/37]
	Type:	A2 Application without search report
	No.:	EP3762423
	Date:	13.01.2021
	Language:	EN
	The application published by WIPO in one of the EPO official languages on 12.09.2019 takes the place of the publication of the European patent application.
	[2021/02]
Search report(s)	International search report - published on:	EP	24.10.2019
	(Supplementary) European search report - dispatched on:	EP	05.07.2023
Classification	IPC:	C07K16/28, C07F9/40, A61K47/68	[2021/02]
	CPC:	A61K47/6849 (EP,IL,KR,US); A61K47/6803 (IL); C07F9/4071 (EP,IL,KR,US); C07K14/76 (CN,IL,KR); A61K47/68031 (EP,KR,US); A61K47/6889 (EP,IL,KR,US); (+) C07F9/4006 (CN); C07F9/4015 (EP,CN,IL,KR,US); C07F9/4075 (CN); C07F9/4087 (CN); C07F9/572 (CN); C07F9/6561 (CN); C07K16/2863 (EP,CN,IL); C07K16/2878 (EP,CN,IL); C07K16/42 (CN,IL,KR); C07K5/0215 (CN); C07K7/06 (CN) (-)
Designated contracting states	AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR [2021/02]
Title	German:	CHEMOSELEKTIVE THIOLKONJUGATION MIT ALKEN- ODER ALKYN-PHOSPHONOTHIOLATEN UND -PHOSPHONATEN	[2021/02]
	English:	CHEMOSELECTIVE THIOL-CONJUGATION WITH ALKENE OR ALKYNE-PHOSPHONOTHIOLATES AND -PHOSPHONATES	[2021/02]
	French:	CONJUGAISON CHIMIOSÉLECTIVE D'UN THIOL AVEC DES ALCÈNE- OU ALCYNE-PHOSPHONOTHIOLATES ET -PHOSPHONATES	[2021/02]
Entry into regional phase	07.10.2020	National basic fee paid
	07.10.2020	Designation fee(s) paid
	07.10.2020	Examination fee paid
Examination procedure	07.10.2020	Examination requested [2021/02]
	07.10.2020	Date on which the examining division has become responsible
	06.05.2021	Amendment by applicant (claims and/or description)
	05.07.2023	Despatch of a communication from the examining division to which search results under Rule 164(2) EPC are annexed (Time limit: M04) [2023/32]
	05.07.2023	Despatch of a communication from the examining division (Time limit: M04)
	14.11.2023	Reply to a communication from the examining division
Fees paid	Renewal fee
	24.03.2021	Renewal fee patent year 03
	25.03.2022	Renewal fee patent year 04
	23.03.2023	Renewal fee patent year 05
	27.03.2024	Renewal fee patent year 06
	26.03.2025	Renewal fee patent year 07
Opt-out from the exclusive Tooltip competence of the Unified Patent Court	See the Register of the Unified Patent Court for opt-out data
	Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Cited in	International search	[T] WO2009051025 (KATAYAMA CHEMICAL IND CO LTD et al.)
		[IP] WO2018041985 (FORSCHUNGSVERBUND BERLIN EV et al.)
		[XI] FENG GAO ET AL: "Synthesis of a Phosphonate-Linked Aminoglycoside-Coenzyme A Bisubstrate and Use in Mechanistic Studies of an Enzyme Involved in Aminoglycoside Resistance", CHEMISTRY - A EUROPEAN JOURNAL, vol. 15, no. 9, 16 February 2009 (2009-02-16), pages 2064 - 2070, XP055092919, ISSN: 0947-6539, DOI: 10.1002/chem.200802172 DOI: http://dx.doi.org/10.1002/chem.200802172
		[T] DATABASE CA [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; KOLOMNIKOVA, G. D. ET AL: "Vinylic esters of phosphorus acids. 32. Phosphorus-containing isothiuronium salts", XP002792670, retrieved from STN Database accession no. 1993:124641
		[XI] QUN DANG ET AL: "Fructose-1,6-bisphosphatase Inhibitors. 1. Purine Phosphonic Acids as Novel AMP Mimics", JOURNAL OF MEDICINAL CHEMISTRY, vol. 52, no. 9, 14 May 2009 (2009-05-14), US, pages 2880 - 2898, XP055602023, ISSN: 0022-2623, DOI: 10.1021/jm900078f DOI: http://dx.doi.org/10.1021/jm900078f
		[XI] KHUSAINOVA N G ET AL: "Reactions of 1,2-ethanedithiol and 2-mercaptoethanol with unsaturated derivatives of four-coordinate phosphorus acids", RUSSIAN CHEMICAL BULLETIN, KLUWER ACADEMIC PUBLISHERS-PLENUM PUBLISHERS, NE, vol. 53, no. 10, 1 October 2004 (2004-10-01), pages 2253 - 2256, XP019224174, ISSN: 1573-9171, DOI: 10.1007/S11172-005-0109-7 DOI: http://dx.doi.org/10.1007/s11172-005-0109-7
		[XI] DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; 2016, "S-[2-(diethoxyphosphinyl)ethyl]-D-Cysteine", XP002792671, retrieved from STN Database accession no. 2002527-58-2
		[XI] DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; 21 September 2016 (2016-09-21), "S-[2-(diethoxyphosphinyl)ethyl]-L-Cysteine,", XP002792672, retrieved from STN Database accession no. 1997361-25-7
		[XI] KRZYSZTOF FELCZAK ET AL: "Cofactor-type inhibitors of inosine monophosphate dehydrogenase via modular approach: Targeting the pyrophosphate binding sub-domain", BIOORGANIC & MEDICINAL CHEMISTRY : A TETRAHEDRON PUBLICATION FOR THE RAPID DISSEMINATION OF FULL ORIGINAL RESEARCH PAPERS AND CRITICAL REVIEWS ON BIOMOLECULAR CHEMISTRY, MEDICINAL CHEMISTRY AND RELATED DISCIPLINES, ELSEVIER, NL, vol. 19, no. 5, 21 January 2011 (2011-01-21), pages 1594 - 1605, XP028382307, ISSN: 0968-0896, [retrieved on 20110127], DOI: 10.1016/J.BMC.2011.01.042 DOI: http://dx.doi.org/10.1016/j.bmc.2011.01.042
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