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Extract from the Register of European Patents

EP About this file: EP3949963

EP3949963 - NOVEL COMPOUND AND COMPOSITION FOR PREVENTION OR TREATMENT OF RESPIRATORY DISEASES COMPRISING SAME AS ACTIVE INGREDIENT [Right-click to bookmark this link]
StatusRequest for examination was made
Status updated on  07.01.2022
Database last updated on 14.06.2024
FormerThe international publication has been made
Status updated on  09.10.2020
Most recent event   Tooltip13.03.2024New entry: Renewal fee paid 
Applicant(s)For all designated states
Yonsei University, University-Industry Foundation(UIF).
50, Yonsei-ro
Seodaemun-gu
Seoul 03722 / KR
[2022/06]
Inventor(s)01 / CHOI, Jae Young
Gireum New Town, Gireum-dong) 201-701, 119,
Gireum-ro, Seongbuk-gu
Seoul 02714 / KR
02 / HAN, Gyoonhee
Sinwon-dong) 3, 8-19, Cheonggyesan-ro 11-gil,
Seocho-gu
Seoul 06802 / KR
03 / NAMKUNG, Wan
Hanyang 1cha Apt., Dongchun-dong) 103-1905, 124
Woninjae-ro, Yeonsu-gu
Incheon 21974 / KR
04 / PARK, Sung Ha
Hyundai Apt., Apgujeong-dong) 202-1208, 69,
Apgujeong-ro 29-gil, Gangnam-gu
Seoul 06005 / KR
05 / PARK, Moo Suk
Gaepo 1, 2cha Woosung Apt., Daechi-dong) 11-1005
120, Seolleung-ro, Gangnam-gu
Seoul 06289 / KR
[N/P]
Former [2022/06]01 / CHOI, Jae Young
Seoul 02714 / KR
02 / HAN, Gyoonhee
Seoul 06802 / KR
03 / NAMKUNG, Wan
Incheon 21974 / KR
04 / PARK, Sung Ha
Seoul 06005 / KR
05 / PARK, Moo Suk
Seoul 06289 / KR
Representative(s)Bates, Philip Ian
Reddie & Grose LLP The White Chapel Building
10 Whitechapel High Street
London E1 8QS / GB
[2022/06]
Application number, filing date20782123.201.04.2020
[2022/06]
WO2020KR04464
Priority number, dateKR2019003824602.04.2019         Original published format: KR 20190038246
[2022/06]
Filing languageKO
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2020204602
Date:08.10.2020
Language:KO
[2020/41]
Type: A1 Application with search report 
No.:EP3949963
Date:09.02.2022
Language:EN
[2022/06]
Search report(s)International search report - published on:KR08.10.2020
(Supplementary) European search report - dispatched on:EP02.12.2022
ClassificationIPC:C07D207/337, C07D231/12, C07D413/10, A61K31/422, A61K31/427, A61P11/00
[2022/50]
CPC:
C07D413/06 (EP,US); A61K31/422 (KR,US); A61K31/341 (US);
A61K31/381 (US); A61K31/40 (US); A61K31/415 (US);
A61K31/421 (US); A61K31/426 (US); A61K31/427 (KR,US);
A61K31/4439 (US); A61K31/454 (US); A61K31/4709 (US);
A61K31/519 (US); A61K9/0056 (US); A61P11/00 (EP,KR);
A61P11/06 (US); C07D207/337 (EP,US); C07D209/18 (EP);
C07D209/20 (US); C07D231/12 (EP,US); C07D263/38 (EP);
C07D263/42 (US); C07D277/30 (EP,US); C07D307/54 (EP,US);
C07D333/24 (EP,US); C07D333/60 (EP,US); C07D413/04 (EP,US);
C07D413/10 (EP,US); C07D413/12 (EP,US); C07D413/14 (EP,US);
C07D417/06 (EP,US); C07D495/04 (EP,US) (-)
Former IPC [2022/06]A61K31/422, A61K31/427, A61P11/00
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   RS,   SE,   SI,   SK,   SM,   TR [2022/06]
TitleGerman:VERBINDUNG UND ZUSAMMENSETZUNG ZUR VORBEUGUNG ODER BEHANDLUNG VON ATEMWEGSERKRANKUNGEN, DIE DIESE ALS AKTIVEN BESTANDTEIL ENTHALTEN[2022/06]
English:NOVEL COMPOUND AND COMPOSITION FOR PREVENTION OR TREATMENT OF RESPIRATORY DISEASES COMPRISING SAME AS ACTIVE INGREDIENT[2022/06]
French:NOUVEAU COMPOSÉ ET COMPOSITION POUR LA PRÉVENTION OU LE TRAITEMENT DE MALADIES RESPIRATOIRES COMPRENANT CELUI-CI COMME PRINCIPE ACTIF[2022/06]
Entry into regional phase04.10.2021Translation filed 
04.10.2021National basic fee paid 
04.10.2021Search fee paid 
04.10.2021Designation fee(s) paid 
04.10.2021Examination fee paid 
Examination procedure04.10.2021Examination requested  [2022/06]
26.06.2023Amendment by applicant (claims and/or description)
Fees paidRenewal fee
23.03.2022Renewal fee patent year 03
12.04.2023Renewal fee patent year 04
13.03.2024Renewal fee patent year 05
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Documents cited:Search[XA]EP0422900  (TOSHIBA KK [JP]) [X] 1 * claim -; tables 4-6; compound A12 * [A] 2-10;
 [XA]US2004180943  (AUGELLI-SZAFRAN CORINNE ELIZAB [US], et al) [X] 1 * claim - * [A] 2-10;
 [XA]EP1695968  (SHANGHAI INST MATERIA MEDICA [CN]) [X] 1 * compound 2f -paragraph [0047];; claim - * [A] 2-10;
 [XA]WO2008056356  (PROTEOLOGICS LTD [IL], et al) [X] 1 * scheme 2-inntermediate 2; page 65 * [A] 2-10;
 [XA]WO2010094009  (CHILDRENS HOSP MEDICAL CENTER [US], et al) [X] 1 * page 101; claim -; table 7 * [A] 2-10;
 [XPA]WO2019231935  (OMEROS CORP [US], et al) [XP] 1 * compound with rn:369637-37-6 *[A] 2-10;
 [XA]  - TOPUZYAN V O ET AL, "Derivatives of [alpha],[beta]-dehydro amino acids: III. Reaction of 4-arylmethylidene-4,5-dihydro-1,3-oxazol-5-ones with hexamethyldisilazane", RUSSIAN JOURNAL OF ORGANIC CHEMISTRY, M A I K NAUKA - INTERPERIODICA, RU, (20070101), vol. 43, doi:10.1134/S1070428007060127, ISSN 1070-4280, pages 868 - 871, XP009169535 [X] 1 * schemes 1-2;; compound 9 * [A] 2-10

DOI:   http://dx.doi.org/10.1134/S1070428007060127
 [XA]  - ALAN R KATRITZKY ET AL, "Synthesis and photochemistry of pH-sensitive GFP chromophore analogs", TETRAHEDRON LETTERS, vol. 52, no. 17, doi:10.1016/J.TETLET.2010.12.082, ISSN 0040-4039, (2011), pages 2224 - 2227, (20101224), XP028159081 [X] 1 * schemes 1 to 4;; table 1; compound 6d * [A] 2-10

DOI:   http://dx.doi.org/10.1016/j.tetlet.2010.12.082
 [XA]  - CATIVIELA, C.; DIAZ DE VILLEGAS, M. D.; MAYORAL, J. A.; MELEN, "Synthesis and stereospecific ring opening of the (Z/E)-isomers of 2-methyl(phenyl)-4-(thienylmethylene)-5(4H)-oxazolone", SYNTHESIS, (1983), vol. 11, doi::10.1055/s-1983-30556, ISSN 0039-7881, pages 899 - 902, XP055977796 [X] 1 * table 1; compound 3bb * [A] 2-10

DOI:   http://dx.doi.org/10.1055/s-1983-30556
 [X]  - EIDEN F. ET AL, "4-Pyranyliden-oxazolone-(5)", ARCHIV DER PHARMAZIE, Weinheim, (19670101), vol. 300, no. 3, doi:10.1002/ardp.19673000305, ISSN 0365-6233, pages 211 - 225, XP055977626 [X] 1 * table 1; compounds III-l *

DOI:   http://dx.doi.org/10.1002/ardp.19673000305
 [XA]  - Singhal, O. P.; Ittyerah, P. I., "2-Thiophenecarboxaldehyde: Condensation with some acyl glycines", CAPLUS, CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US, (1965), Database accession no. 1965:498270, URL: STN, XP002807902 [X] 1 * compounds with rn: 4211-92-1; 4211-98-7; 4211-99-8; 4211-93-2 and 4466-61-9 * [A] 2-10
 [XA]  - REGBERG TOR ET AL, "Novel Affinity Ligands for Chromatography Using Combinatorial Chemistry", COMBINATORIAL CHEMISTRY AND HIGH THROUGHPUT SCREENING, NL, (20110501), vol. 14, no. 4, doi:10.2174/138620711795222482, ISSN 1386-2073, pages 267 - 278, XP055977642 [X] 1 * figures 3, 6 * [A] 2-10

DOI:   http://dx.doi.org/10.2174/138620711795222482
International search[X]JP2006096708  (MOCHIDA PHARM CO LTD) [X] 1-10 * See abstract; paragraph [0022]; claim 1. *;
 [X]KR20150126687  (TAKEDA PHARMACEUTICAL [JP]) [X] 1 * See abstract; paragraph [0248]. *;
 [X]  - Dayana Abboud, Daubeuf François, Do Quoc Tuan, Utard Valérie, Villa Pascal, Haiech Jacques, Bonnet Dominique, Hibert Marcel, Bernard Philippe, Galzi Jean-Luc, Frossard Nelly, "A strategy to discover decoy chemokine ligands with an anti-inflammatory activity", Scientific Reports, (20151007), vol. 5, doi:10.1038/srep14746, ISSN 2045-2322, pages 1 - 14, XP055744972 [X] 1-10 * See abstract; compound GPN251 of figure 3; inner page 9. *

DOI:   http://dx.doi.org/10.1038/srep14746
 [X]  - Sanjay D Sawant, Barvrkar Atul A, Chabukswar Anirudh R, Sarak Swati D, "Molecular docking and synthesis of 8-substituted 3,4-dihydro-6-methyl-4-(2,4-dinitrophenyl)imidazo[1,5-b][1,2,4]triazin-2(8H)-one derivatives as novel antiasthmatic agents", Journal of Applicable Chemistry, (20130428), vol. 2, no. 3, ISSN 2278-1862, pages 372 - 384, XP055744973 [X] 1 * See compounds 3a-3g. *
 [X]  - Elena Serrano, Juan Alberto, García-Montero Angel, Soler Tatiana, Jiménez-Márquez Francisco, Cativiela Carlos, Gomez M. Victoria, Urriolabeitia Esteban P., "Stereoselective synthesis of 1,3-diaminotmxillic acid derivatives: an advantageous combination of C-H-oitho-Palladation and on-flow [2+2]-photocycloaddition in microreactors", Chemistry- A European Journal, (20151124), vol. 22, no. 1, doi:10.1002/chem.201503742, ISSN 0947-6539, pages 144 - 152, XP055744974 [X] 1 * See figure 4. *

DOI:   http://dx.doi.org/10.1002/chem.201503742
by applicant   - GRAZIANO, Tetrahedron, (20060000), vol. 62, pages 1165 - 1170
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.