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Extract from the Register of European Patents

EP About this file: EP4208456

EP4208456 - HETEROCYCLIC COMPOUNDS [Right-click to bookmark this link]
StatusRequest for examination was made
Status updated on  09.06.2023
Database last updated on 26.06.2024
FormerThe international publication has been made
Status updated on  11.03.2022
Formerunknown
Status updated on  27.09.2021
Most recent event   Tooltip10.11.2023Change: Validation statespublished on 13.12.2023  [2023/50]
10.11.2023Change - extension statespublished on 13.12.2023  [2023/50]
Applicant(s)For all designated states
F. Hoffmann-La Roche AG
Grenzacherstrasse 124
4070 Basel / CH
[2023/28]
Inventor(s)01 / BENZ, Joerg
4070 Basel / CH
02 / GRETHER, Uwe
4070 Basel / CH
03 / HORNSPERGER, Benoit
4070 Basel / CH
04 / KROLL, Carsten
4070 Basel / CH
05 / KUHN, Bernd
4070 Basel / CH
06 / MARTIN, Rainer, E.
4070 Basel / CH
07 / O'HARA, Fionn
4070 Basel / CH
08 / PUELLMANN, Bernd
4070 Basel / CH
09 / RICHTER, Hans
4070 Basel / CH
10 / RITTER, Martin
4070 Basel / CH
 [2023/28]
Representative(s)Neuhaus, Christian Michel, et al
F. Hoffmann-La Roche AG
Grenzacherstrasse 124
4070 Basel / CH
[2023/28]
Application number, filing date21772763.501.09.2021
[2023/28]
WO2021EP74150
Priority number, dateEP2020019431803.09.2020         Original published format: EP 20194318
[2023/28]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2022049134
Date:10.03.2022
Language:EN
[2022/10]
Type: A1 Application with search report 
No.:EP4208456
Date:12.07.2023
Language:EN
The application published by WIPO in one of the EPO official languages on 10.03.2022 takes the place of the publication of the European patent application.
[2023/28]
Search report(s)International search report - published on:EP10.03.2022
ClassificationIPC:C07D403/06, C07D403/14, C07D413/04, C07D413/14, C07D487/04, A61K31/4192, A61K31/422, A61P25/00
[2023/28]
CPC:
C07D403/06 (EP,IL,KR,US); A61K31/4025 (KR); A61K31/407 (KR);
A61K9/2009 (IL,US); A61K9/2054 (IL,US); A61K9/2059 (IL,US);
A61K9/485 (IL,US); A61K9/4858 (IL,US); A61K9/4866 (IL,US);
A61P1/00 (KR); A61P25/00 (KR); A61P25/18 (KR);
A61P25/28 (KR); A61P29/00 (KR); A61P35/00 (KR);
C07D401/06 (KR); C07D401/14 (IL,KR,US); C07D403/12 (KR);
C07D403/14 (EP,IL); C07D413/04 (EP,IL); C07D413/06 (IL,KR,US);
C07D413/12 (KR); C07D413/14 (EP,IL,KR,US); C07D417/06 (KR);
C07D471/10 (KR); C07D487/04 (EP,IL,KR,US); C07D487/10 (KR) (-)
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   RS,   SE,   SI,   SK,   SM,   TR [2023/28]
Validation statesMA03.04.2023
TitleGerman:HETEROCYCLISCHE VERBINDUNGEN[2023/28]
English:HETEROCYCLIC COMPOUNDS[2023/28]
French:COMPOSÉS HÉTÉROCYCLIQUES[2023/28]
Entry into regional phase03.04.2023National basic fee paid 
03.04.2023Designation fee(s) paid 
03.04.2023Examination fee paid 
Examination procedure03.04.2023Examination requested  [2023/28]
03.04.2023Date on which the examining division has become responsible
02.10.2023Amendment by applicant (claims and/or description)
Fees paidRenewal fee
20.09.2023Renewal fee patent year 03
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Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Cited inInternational search[A]US4632925  (MULLIN JR JOHN G [US], et al) [A] 1-27 * abstract *;
 [A]US4956359  (TAYLOR JR CHANDLER R [US], et al) [A] 1-27 * table 1, examples 11, 17; column 1 *;
 [A]WO0107043  (VERNALIS RES LTD [GB], et al) [A] 1-27 * page 22, examples 16, 17, 21;; claim - *;
 [A]WO2004096763  (VERNALIS RES LTD [GB], et al) [A] 1-15* example -; claim - *;
 [A]WO2009058347  (JANSSEN PHARMACEUTICA NV [BE], et al) [A] 1-27 * page 106, example 131;; claim - *;
 [A]WO2010106333  (MEDICAL RES COUNCIL TECHNOLOGY [GB], et al) [A] 1-27 * examples 257-260; claim - *;
 [A]  - VENKATESH RAMINENI ET AL, "Novel benzothiazine-piperazine derivatives by peptide-coupling as potential anti-proliferative agents", BIORGANIC & MEDICINAL CHEMISTRY LETTERS, ELSEVIER, AMSTERDAM , NL, (20161025), vol. 27, no. 2, doi:10.1016/J.BMCL.2016.10.071, ISSN 0960-894X, pages 354 - 359, XP029862571 [A] 1-27 * abstract *

DOI:   http://dx.doi.org/10.1016/j.bmcl.2016.10.071
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