Extract from the Register of European Patents

EP About this file: EP0520320

EP0520320 - Tetrahydropyrrolo[1,2-a]pyrazine-4-spiro-3'-pyrrolidine derivatives, processes for the preparation thereof and pharmaceutical compositions containing the same [Right-click to bookmark this link]
Former [1993/01]Tetrahydropyrrolo 1,2-a pyrazine-4-spiro-3'-pyrrolidine derivatives, processes for the preparation thereof and pharaceutical compositions containing the same
[1997/37]
StatusNo opposition filed within time limit
Status updated on  17.07.1998
Database last updated on 09.04.2026
Most recent event   Tooltip17.07.1998No opposition filed within time limitpublished on 02.09.1998 [1998/36]
Applicant(s)For all designated states
Dainippon Pharmaceutical Co., Ltd.
6-8, Dosho-machi 2-chome, Chuo-ku
Osaka-shi, Osaka-fu / JP
[1997/01]
Former [1993/01]For all designated states
DAINIPPON PHARMACEUTICAL CO., LTD.
6-8, Doshomachi 2-chome, Chuo-ku
Osaka / JP
Inventor(s)01 / Negoro, Toshiyuki
1495-1, Oaza-Noda, Kumatori-cho
Sennan-gun, Osaka-fu / JP
02 / Murata, Makoto
1-13-37-803, Shin-machi
Hirakata-shi, Osaka-fu / JP
03 / Ueda, Shòzò
6-26, Hattori-dai 3-chome, Kanmaki-cho
Kitakatsuragi-gun, Nara-ken / JP
04 / Fujitani, Buichi
13-20, Mihra-dai 3-cho
Sakai-shi, Osaka-fu / JP
05 / Ono, Yoshiyuki
14-10, Katagiharashihata-cho
Nishikyo-ku, Kyoto-shi, Kyoto-fu / JP
[1993/01]
Representative(s)Kraus, Walter, et al
Patentanwälte Kraus, Weisert & Partner Thomas-Wimmer-Ring 15
80539 München / DE
[N/P]
Former [1993/01]Kraus, Walter, Dr., et al
Patentanwälte Kraus, Weisert & Partner Thomas-Wimmer-Ring 15
D-80539 München / DE
Application number, filing date92110270.317.06.1992
[1993/01]
Priority number, dateJP1991018318526.06.1991         Original published format: JP 18318591
[1993/01]
Filing languageEN
Procedural languageEN
PublicationType: A2 Application without search report 
No.:EP0520320
Date:30.12.1992
Language:EN
[1992/53]
Type: A3 Search report 
No.:EP0520320
Date:24.03.1993
Language:EN
[1993/12]
Type: B1 Patent specification 
No.:EP0520320
Date:10.09.1997
Language:EN
[1997/37]
Search report(s)(Supplementary) European search report - dispatched on:EP29.01.1993
ClassificationIPC:C07D487/20, A61K31/495, // (C07D487/20, 241:00, 209:00, 209:00)
[1993/01]
CPC:
C07D487/20 (EP,KR,US); A61P27/00 (EP); A61P3/08 (EP);
A61P3/10 (EP); Y02P20/55 (EP,US)
Designated contracting statesAT,   BE,   CH,   DE,   DK,   ES,   FR,   GB,   GR,   IT,   LI,   LU,   NL,   PT,   SE [1993/01]
TitleGerman:Tetrahydropyrrolo[1,2-a]Pyrazin-4-Spiro-3'-Pyrrolidin-Derivate, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Zubereitungen[1997/37]
English:Tetrahydropyrrolo[1,2-a]pyrazine-4-spiro-3'-pyrrolidine derivatives, processes for the preparation thereof and pharmaceutical compositions containing the same[1997/37]
French:Dérivés de la tétrahydropyrrolo[1,2-a]pyrazine-4-spiro-3'-pyrrolidine, procédés pour leur préparation et compositions pharmaceutiques les contenant[1997/37]
Former [1993/01]Tetrahydropyrrolo(1,2-a)Pyrazin-4-Spiro-3'-Pyrrolidinderivate, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Zubereitungen
Former [1993/01]Tetrahydropyrrolo 1,2-a pyrazine-4-spiro-3'-pyrrolidine derivatives, processes for the preparation thereof and pharaceutical compositions containing the same
Former [1993/01]Dérivés de la tétrahydropyrrolo(1,2-a)pyrazine-4-spiro-3'-pyrrolidine, procédé pour leur préparation et compositions pharmaceutiques les contenant
Examination procedure18.08.1993Examination requested  [1993/42]
20.09.1996Despatch of communication of intention to grant (Approval: No)
18.11.1996Despatch of communication of intention to grant (Approval: later approval)
25.11.1996Communication of intention to grant the patent
19.02.1997Fee for grant paid
19.02.1997Fee for publishing/printing paid
Opposition(s)11.06.1998No opposition filed within time limit [1998/36]
Fees paidRenewal fee
23.06.1994Renewal fee patent year 03
26.06.1995Renewal fee patent year 04
21.06.1996Renewal fee patent year 05
18.06.1997Renewal fee patent year 06
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Documents cited:Search[A] EP0147805  (KYORIN SEIYAKU KK et al.) [A]
 [A] EP0173497  (PFIZER et al.) [A]
 [AD] EP0365324  (AMERICAN HOME PROD et al.) [AD]
 [A]   CHEMICAL ABSTRACTS, vol. 82, no. 23, 9 June 1975, Columbus, Ohio, US; abstract no. 156398q, A. MORITOMO ET AL. 'Pyrrole lactame derivatives with antiprotozoa antitrichomonas blood sugar decreasing and gastric juice apoleptic activity' page 621 ; [A]
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