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Extract from the Register of European Patents

EP About this file: EP0737232

EP0737232 - MODULAR DESIGN AND SYNTHESIS OF AMINIMIDE CONTAINING MOLECULES [Right-click to bookmark this link]
StatusThe application is deemed to be withdrawn
Status updated on  22.09.2000
Database last updated on 15.06.2024
Most recent event   Tooltip22.09.2000Application deemed to be withdrawnpublished on 08.11.2000 [2000/45]
Applicant(s)For all designated states
ARQULE, INC.
Suite 3600, 200 Boston Avenue
Medford, MA 02155 / US
[1996/42]
Inventor(s)01 / HOGAN, Joseph, C., Jr.
50 Oak Avenue
Belmont, MA 02178 / US
02 / CASEBIER, David
45 Priest Street
Hudson, MA 01749 / US
03 / FURTH, Paul
Apartment 13, 310 College Farm Road
Waltham, MA 01749 / US
04 / TU, Cheng
305 Memorial Drive
Cambridge, MA 02139 / US
[1996/42]
Representative(s)Lawrence, John
Barker Brettell LLP
100 Hagley Road
Edgbaston
Birmingham B16 8QQ / GB
[N/P]
Former [1996/42]Lawrence, John
Barker, Brettell & Duncan, 138, Hagley Road, Edgbaston
Birmingham B16 9PW / GB
Application number, filing date94906465.328.12.1993
[1996/42]
WO1993US12612
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO9518186
Date:06.07.1995
Language:EN
[1995/29]
Type: A1 Application with search report 
No.:EP0737232
Date:16.10.1996
Language:EN
The application published by WIPO in one of the EPO official languages on 06.07.1995 takes the place of the publication of the European patent application.
[1996/42]
Search report(s)International search report - published on:US06.07.1995
(Supplementary) European search report - dispatched on:EP09.10.1997
ClassificationIPC:A61K31/205
[1997/47]
CPC:
C07C245/00 (EP); C07D209/16 (EP); C07D211/52 (EP);
C07D213/89 (EP); C07D239/47 (EP); C07D239/54 (EP);
C07D461/00 (EP); C07D489/00 (EP); C07D489/02 (EP);
C07H13/04 (EP); C07H21/00 (EP); C07K1/047 (EP);
C07K14/005 (EP); C07K5/1013 (EP); C07K7/02 (EP);
C08G73/02 (EP); C12N2740/16222 (EP) (-)
Former IPC [1996/42]C09B44/00, C07C245/00
Designated contracting statesAT,   BE,   CH,   DE,   DK,   ES,   FR,   GB,   GR,   IE,   IT,   LI,   LU,   MC,   NL,   PT,   SE [1996/42]
TitleGerman:MODULARER ENTWURF UND SYNTHESE VON AMINIMID ENTHALTENDEN VERBINDUNGEN[1996/42]
English:MODULAR DESIGN AND SYNTHESIS OF AMINIMIDE CONTAINING MOLECULES[1996/42]
French:STRUCTURE ET SYNTHESE MODULAIRE DE MOLECULES CONTENANT L'AMINIMIDE[1996/42]
Entry into regional phase19.07.1996National basic fee paid 
19.07.1996Search fee paid 
19.07.1996Designation fee(s) paid 
19.07.1996Examination fee paid 
Examination procedure06.07.1995Request for preliminary examination filed
International Preliminary Examining Authority: US
19.07.1996Examination requested  [1996/42]
29.09.1999Despatch of a communication from the examining division (Time limit: M07)
10.02.2000Application deemed to be withdrawn, date of legal effect  [2000/45]
13.06.2000Despatch of communication that the application is deemed to be withdrawn, reason: reply to the communication from the examining division not received in time  [2000/45]
Fees paidRenewal fee
19.07.1996Renewal fee patent year 03
30.12.1996Renewal fee patent year 04
20.12.1997Renewal fee patent year 05
30.11.1998Renewal fee patent year 06
06.12.1999Renewal fee patent year 07
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See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Documents cited:Search[X]FR1478953  (FARBEWERKE HOECHST AG.) [X] 1 * page 8; example AS *;
 [X]DE1809950  (BADISCHE ANILIN- & SODA-FABRIK A.G.) [X] 1 * page 3 * * page 5 * * page 6 - page 7; examples 5,6 * * claim - *;
 [X]FR1558886  (FARBEWERKE HOECHST AG.) [X] 1,4 * page 6; example 16 *;
 [E]WO9401102  (LEGOMER PARTNERS LP ;HOGAN JOSEPH C JR (US)) [E] 1-21 * example -; claim - *
 [X]  - M. LILER ET AL., "Mono- and di-protonation sites in N-ammonio-amidates: a spectroscopic study", JOURNAL OF THE CHEMICAL SOCIETY, PERKIN TRANSACTIONS 2, LETCHWORTH GB, (1977), pages 909 - 914, XP002031550 [X] 1 * page 910; table 1 *

DOI:   http://dx.doi.org/10.1039/p29770000909
 [X]  - B. ZEEH ET AL., "Eine einfache isoindol-synthese", SYNTHESIS, STUTTGART DE, (1972), pages 45 - 46, XP002031551 [X] 1 * figure 5 *

DOI:   http://dx.doi.org/10.1055/s-1972-21830
 [X]  - W.J. MCKILLIP ET AL., "Aminimides. II- A one-step synthesis of aminimides from carboxylic acid esters", CANADIAN JOURNAL OF CHEMISTRY, OTTAWA CA, (1967), vol. 45, pages 2619 - 2623, XP002031748 [X] 1 * page 2620; table II *

DOI:   http://dx.doi.org/10.1139/v67-425
International search[A]US4012364
 [A]  - PROC. NATL. ACAD. SCI., Volume 89, issued October 1992, REYNA J. SIMON et al., "Peptoids: A Modular Approach to Drug Discovery", pages 9367-9371.
 [A]  - CHEMICAL ABSTRACTS, Volume 105, No. 19, issued 1986, MOULTON et al., "Studies on the Transverse Tubule Membrane Magnesium ATPase. Lectin-Induced Alterations of Kenetic Behaviour", Abstract No. 167889v.
 [A]  - THE FASEB JOURNAL, Volume 7, issued April 1993, STANLEY T. CROOKE, "Progress Toward Oligonucleotide Therapeutics: Pharmacodynamic Properties", pages 533-539.
 [A]  - CHEMICAL ABSTRACTS, Volume 120, No. 15, issued 1993, TOYOKUNI et al., "Multivalent Mimetics and Peptide Mimetics for Blocking Carbohydrate-Dependent Cellular Interaction and for Eliciting Anti-Carbohydrate T-Cell Response", Abstract No. 183041c.
 [A]  - CHEMICAL ABSTRACTS, Volume 111, No. 5, issued 31 July 1989, GHOSH et al., "Synthesis of 5'-Oligonucleotide Hydrazide Derivatives and their Use in Preparation of Enzyme-Nucleic Acid Hybridization Probes", Abstract No. 36183m.
 [A]  - CHEMICAL ABSTRACTS, Volume 115, No. 11, issued 16 September 1991, WRASIDLO, "Interfacial Condensation of Bioactive Compounds and Site Specific Compounds Such as Monoclonal Antibodies and Conjugates Thereof", Abstract No. 112642k.
 [A]  - CHEMICAL ABSTRACTS, Volume 105, No. 6, issued 11 August 1986, KROSCHWITZ, "Aminimide Polymers", Abstract No. 43373e.
 [A]  - CHEMICAL ABSTRACTS, Volume 89, No. 14, issued 1989, MIRON et al., "Unsaturated Aminimide for Anaerobic Hardening", Abstract No. 111205c.
 [A]  - CHEMICAL ABSTRACTS, Volume 93, No. 6, issued 1980, KUWAMURA, "Surface-Active Agents and Detergents", Abstract No. 48,980s.
 [A]  - CHEMICAL ABSTRACTS, Volume 108, No. 28, issued 1988, INOKUMA, "Surface Active Crown Ethers, XI, Synthesis and Properties of Aminimides and their Crown Derivatives Bearing an L-Alinine Residue", Abstract No. 223506u.
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.